Regioselective Hydroarylation of Protected Allylic Amines

doi:10.1055/s-0030-1257903

Subscribe to RSS

Please copy the URL and add it into your RSS Feed Reader.

https://www.thieme-connect.de/rss/thieme/en/10.1055-s-00000131.xml

Share / Bookmark

Facebook Linkedin Weibo

Download PDF

Synfacts 2010(9): 1062-1062
DOI: 10.1055/s-0030-1257903

Metal-Mediated Synthesis

Regioselective Hydroarylation of Protected Allylic Amines

Contributor(s): Paul Knochel, Thomas Kunz
G. C. Tsui, F. Menard, M. Lautens*
University of Toronto, Canada

Further Information

Publication History

Publication Date:
23 August 2010 (online)

Permissions and Reprints

Significance

A rhodium(I)-catalyzed hydroarylation of unactivated alkenes with arylboronic acids is reported. The regioselectivity of the addition is highly dependent on the protecting group and the carbon chain length of the allylic amine.