Synfacts, Table of Contents Synfacts 2025; 21(09): 883DOI: 10.1055/a-2653-4980 Synthesis of Heterocycles Synthesis of Functionalized Bicyclic Heterocycles as Bioisosteres for meta-Substituted (Hetero)arenes Authors Contributor(s): Paul Richardson (Pfizer) Recommend Article Abstract Buy Article(opens in new window)Keywords Keywordsbioisosteres - bromocyclization - oxazines - oxazepanes - high-throughput experimentation - exit vectors Full Text