Subscribe to RSS
Please copy the URL and add it into your RSS Feed Reader.
https://www.thieme-connect.de/rss/thieme/en/10.1055-s-00000131.xml
Synfacts 2006(10): 0992-0992
DOI: 10.1055/s-2006-949346
DOI: 10.1055/s-2006-949346
Synthesis of Heterocycles
© Georg Thieme Verlag Stuttgart · New York
Palladium- and Copper-Catalyzed Arylation of Azoles
F. Bellina*, S. Cauteruccio, R. Rossi*
University of Pisa, Italy
Further Information
Publication History
Publication Date:
21 September 2006 (online)
Significance
A C-H activation type Pd- and Cu- catalyzed arylation of azoles is reported. The reaction proceeds regioselectively under ligandless and base-free conditions on oxazole, thiazole, and imidazoles, including derivatives without N-protection.