Synthesis 2022; 54(19): 4347-4352
DOI: 10.1055/s-0040-1719933
paper

Enantioselective Synthesis of (+)-Agelasidine A Using Thio-Claisen Rearrangement

Yoshiyasu Ichikawa
a   Faculty of Science, Kochi University, Akebono-cho Kochi 780-8520, Japan
,
Rika Ochi
a   Faculty of Science, Kochi University, Akebono-cho Kochi 780-8520, Japan
,
Toshiya Masuda
b   Graduate School of Human Life Science, Osaka City University, Osaka 558-8585, Japan
› Author Affiliations
Generous financial support provided by a Grant-in-Aid for Scientific Research (C) (16K01916) from MEXT is gratefully acknowledged.


Dedicated to the memory of Hideshi Nakamura (1952–2000)

Abstract

Enantioselective synthesis of the marine natural product (+)-agelasidine A has been achieved by taking advantage of [1,3]-chirality transfer from enantiomerically enriched α-silyl farnesol through a key thio-Claisen rearrangement. The optical rotation of the hydrochloride salt of the synthetic substance confirmed that natural (+)-agelasidine A has the S-configuration at its C-10 stereogenic center.

Supporting Information



Publication History

Received: 21 April 2022

Accepted after revision: 09 May 2022

Article published online:
28 June 2022

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