DOI: 10.1055/s-00000105

Zentralblatt für Gynäkologie

References

Jones CD, Jevnikar MG, Pike AJ, Peters MK, Black LJ, Thompson AR. et al.
Antiestrogens. 2. Structure-activity studies in a series of 3-aroyl-2-arylbenzo[b]thiophene derivatives leading to [6-hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3- yl] [4-[2-(1-piperidinyl)ethoxy]-phenyl]methanone hydrochloride (LY156758), a remarkably effective estrogen antagonist with only minimal intrinsic estrogenicity. 
J Med Chem 1984; 27: 1057-66  

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