DOI: 10.1055/s-00000083

Synlett

eFirst

Publication Date: 17 August 2017

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Do, Jean-Louis; Friščić, Tomislav: Chemistry 2.0: Developing a New, Solvent-Free System of Chemical Synthesis Based on Mechanochemistry
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Yasui, Kosuke; Higashino, Masaya; Chatani, Naoto; Tobisu, Mamoru: Rhodium-Catalyzed Reductive Cleavage of Aryl Carbamates Using Isopropanol as a Reductant
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Supporting Information

letter

Aeyad, Tahani; Williams, Jason D.; Meijer, Anthony J. H. M.; Coldham, Iain: Lithiation–Substitution of N-Boc-2-phenylazepane
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letter

Afsar, Ashfaq; Cowell, Joseph; Distler, Petr; Harwood, Laurence M.; John, Jan; Westwood, James: Synthesis of Novel BTPhen-Functionalized Silica-Coated Magnetic Nanoparticles for Separating Trivalent Actinides and Lanthanides
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letter

Banan, Alireza; Valizadeh, Hassan; Heydari, Akbar; Moghimi, Abolghasem: Selective Oxidation of Secondary Amines to N,N-Disubstituted Hydroxylamines by Choline Peroxydisulfate
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letter

Calvo, Beatriz C.; Minnaard, Adriaan J.: Copper-Catalyzed Asymmetric 1,2-Addition of Grignard Reagents to 3-Acyl 2H-chromenes
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letter

Chaabouni, S.; Pinkerton, N. M.; Abid, S.; Galaup, C.; Chassaing, S.: Photochemistry of ortho-Azidocinnamoyl Derivatives: Facile and Modular Synthesis of 2-Acylated Indoles and 2-Substituted Quinolines under Solvent Control
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letter

Chittimalla, Santhosh Kumar; Nakka, Srinuvasu; Koodalingam, Manikandan; Bandi, Chennakesavulu: N-Arylation of Heterocycles by a Tandem Aza-Michael Addition Reaction and Aromatization Sequence
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letter

Gao, Ke; Yamamoto, Keita; Nogi, Keisuke; Yorimitsu, Hideki: Palladium-Catalyzed Arylation of Benzylic C–H Bonds of Azaarylmethanes with Aryl Sulfides
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letter

Jopp, Stefan; Liesegang, Marko; Ehlers, Peter; Frank, Eva; Schneider, Gyula; Wölfling, János; Villinger, Alexander; Langer, Peter: Palladium-Catalysed Sonogashira Reactions of 16-(Hydroxymethylidene)-3-methoxy-α-estrone
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letter

Liang, Honggang; Bao, Lingxiang; Du, Yao; Zhang, Yiying; Pang, Siping; Sun, Chenghui: Synthesis of Cyanamides from Cyanogen Bromide under Mild Conditions through N-Cyanation of Allylic Tertiary Amines
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letter

Mandal, Samir K.; Sarkar, Apurba; Chakraborty, Puskin; Chattopadhyay, Ashoke P.: Synthetic Studies Towards the Synthesis of 6-Substituted 3-Fluoro-5,6-dihydropyran-2-ones
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letter

Onge, Brent St.; Green, James R.: Nicholas Reactions of Alkynyl- and Alkenyltrifluoroborates
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letter

Tanwar, Dinesh Kumar; Surendrabhai, Vaghela Ravikumar; Gill, Manjinder Singh: An Efficient and Practical Process for the Synthesis of Glimepiride
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letter

Xu, Lanting; Tan, Lushi; Ma, Dawei: Rhodium-Catalyzed Regioselective C7-Functionalization of Indole Derivatives with Acrylates by Using an N-Imino Directing Group
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Supporting Information

synpacts

Jacobse, Peter H.; Moret, Marc-Etienne; Klein Gebbink, Robertus J. M.; Swart, Ingmar: Tracking On-Surface Chemistry with Atomic Precision
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Publication Date: 16 August 2017

cluster

Hossain, Asik; Pagire, Santosh K.; Reiser, Oliver: Visible-Light-Mediated Synthesis of Pyrazines from Vinyl Azides Utilizing a Photocascade Process
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Supporting Information

cluster

Moyer, Brandon S.; Gagné, Michel R.: Taming Silylium Ions for Synthesis: N-Heterocycle Synthesis via Stereoselective C–C Bond Formation
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letter

Corbett, Michael T.; Caille, Seb: A Bench-Stable Vilsmeier Reagent for in situ Alcohol Activation: Synthetic Application in the Synthesis of 2-Amino-2-Thiazolines
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letter

Mai, Duy N.; Uchenik, Dmitriy; Vanderwal, Christopher D.: Efforts Toward a Synthesis of Crotogoudin and Crotobarin
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letter

Mei, Ruhuai; Zhang, Shou-Kun; Ackermann, Lutz: Concise Synthesis of Lamellarin Alkaloids by C–H/N–H Activation: Evaluation of Metal Catalysts in Oxidative Alkyne Annulation
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Supporting Information

Publication Date: 15 August 2017

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May, Jeremy A.; Nguyen, Thien S.; Nguyen, Truong N.; Le, Phong Q.; Chen, Po-An; Vallakati, Ravikrishna: Pursuit of Enantioselective Synthesis of Heterocycle-Bearing ­Stereocenters: The Development of a Stereocontrolled BINOL-­Catalyzed Conjugate Addition of Organoboron Nucleophiles
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Talero, Alexánder G.; Burtoloso, Antonio C. B.: Sharpless Asymmetric Dihydroxylation on α,β-Unsaturated Diazoketones: A New Entry for the Synthesis of Disubstituted Furanones
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letter

Parra, Claudio; Solís, Pablo; Bonjoch, Josep; Bradshaw, Ben: A One-Pot Methodology for the Synthesis of the Yohimban Skeleton
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Publication Date: 14 August 2017

letter

Cooze, Christopher; Manchoju, Amarender; Pansare, Sunil V.: Synthesis of (–)-Muricatacin and (–)-(R,R)-L-Factor Involving an Organocatalytic Direct Vinylogous Aldol Reaction
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letter

Wang, Qing-Dong; Zhou, Bin; Yang, Jin-Ming; Fang, Dong; Ren, Jiangmeng; Zeng, Bu-Bing: Iron-Catalyzed C3-Formylation of Indoles with Formaldehyde and Aqueous Ammonia under Air
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Publication Date: 11 August 2017

letter

Dos Santos, Aurélie; Cordier, Marie; El Kaïm, Laurent: Nef–Perkow–Mumm Cascade towards Imido Phosphate Derivatives
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letter

Matsuo, Yosuke; Oowatashi, Ryosuke; Saito, Yoshinori; Tanaka, Takashi: Nonenzymatic Biomimetic Synthesis of Black Tea Pigment Theaflavins
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letter

Singh, Amandeep; Shalini; Kaur, Harleen; Sharma, Palak; Anand, Amit; Kumar, Vipan: β-Lactam-Synthon-Interceded Metal/Acid-Free Diastereoselective Access to Highly Functionalized Oxazol-5-ones and Dihydroimidazoles
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Supporting Information

Publication Date: 08 August 2017

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Davies, Stephen G.; Fletcher, Ai M.; Roberts, Paul M.; Thomson, James E.: Asymmetric Synthesis of Pyrrolizidines, Indolizidines and Quinolizidines via a Double Reductive Cyclisation Protocol
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Wang, Jian; Zhang, Ru-Yan; Wang, Ya-Cong; Chen, Xiang-Zhao; Yin, Xu-Guang; Du, Jing-Jing; Lei, Ze; Xin, Ling-Ming; Gao, Xiao-Fei; Liu, Zheng; Guo, Jun: Polyfluorophenyl Ester-Terminated Homobifunctional Cross-Linkers for Protein Conjugation
https://www.thieme-connect.de/media/synlett/EFirst/i_w0310_ga_10-1055_s-0036-1590974.gif
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letter

Dobrowolski, Jeremy C.; Fraser, Benjamin H.; Bhadbhade, Mohan; Black, David StC.; Kumar, Naresh: Efficient Access to Chromeno[4,3-b]quinolines Related to Dependensin
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letter

Fahandej-Sadi, Anis; Lundgren, Rylan J.: Copper-Mediated Synthesis of Monofluoro Aryl Acetates via Decarboxylative Cross-Coupling
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letter

Kobayashi, Yuichi; Saeki, Ryohei; Nanba, Yutaro; Suganuma, Yuta; Morita, Masao; Nishimura, Keita: Synthesis of the Verapamil Intermediate through the Quaternary Carbon-Constructing Allylic Substitution
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letter

Ng, Wing Hin; Shing, Tony K. M.; Yeung, Ying-Yeung: Mild and Efficient Vicinal Dibromination of Olefins Mediated by Aqueous Ammonium Fluoride
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letter

Nguyen, Thi Ha; Ma, Eunsook: Chemoselective Synthesis of N-(Aminoalkyl/amidino)phenyl Naphthalene-1-carboxamides and 5,6,7,8-Tetrahydronaphthalene-1-carboxamides and Their Anticoagulant Screening
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letter

Wang, Liangguang; Ma, Juan; Chen, Xia; Zhou, Xiaoyu: Synthesis of Enaminones by a Palladium-Catalyzed Four-Component Carbonylative Addition Reaction
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letter

Yamamoto, Yasutomo; Yamaguchi, Tatsuya; Kaneshige, Atsunori; Hashimoto, Aiko; Kaibe, Sachiho; Miyawaki, Akari; Yamada, Ken-ichi; Tomioka, Kiyoshi: Consecutive Aminolithiation–Carbolithiation of a Linear Aminoalkene Bearing Terminal Vinyl Sulfide Moiety to Give Hydro­indolizine
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synpacts

Wan, Liqiang; Tian, Lan; Liu, Jie; Niu, Dawen: Iridium-Catalyzed Asymmetric Umpolung Allylation of N-Fluor­enyl Imines to Prepare 1,4-Disubstituted Homoallylic Amines
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Publication Date: 04 August 2017

letter

Qiao, Shuo; Wu, Jianbin; Mo, Junming; Spigener, Preston T.; Zhao, Brian Nlong; Jiang, Bo; Li, Guigen: Chiral Phosphinyl Enamines and Their Asymmetric Reduction through Group-Assisted Purification Chemistry Leading to Enantiopure β-Amino Esters/Amides
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Supporting Information CIF File

Publication Date: 03 August 2017

letter

Dileep, Kommula; Murty, M. S. R.: Aqueous, One-Pot, Three-Component Reaction for Efficient Synthesis of 2-[4-(Arylsulfonyl)piperazin-1-yl]-1,3-benzothiazole, ‑1H-benzimidazole, or -1,3-benzoxazole Derivatives
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letter

Lapinskaite, Ringaile; Ghavre, Mukund; Rintelmann, Chelsea L.; Bedard, Korey; Dela Paz, Helen E.; Hudlicky, Tomas: Chemoenzymatic Formal Total Synthesis of Pancratistatin from Narciclasine-Type Compounds via Myers Transposition: Model Study for a Short Conversion of Narciclasine to Pancratistatin
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letter

Tanwar, Dinesh Kumar; Ratan, Anjali; Gill, Manjinder Singh: Facile One-Pot Synthesis of Substituted Hydantoins from Carbamates
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letter

Wang, Yunxia; Cui, Na; Zhao, Yu: Catalyst-Free Oxidative [3+2] Cycloaddition of Phenols and Styrenes in the Presence of a 2,3-Dichloro-5,6-dicyano-1,4-benzoquinone/1,1,1,3,3,3-hexafluoropropan-2-ol System
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synpacts

Feng, Quanyou; Zhong, Yongliang; Xie, Linghai; Tong, Rong: Recent Advances in Ring-Opening Polymerization of O-Carboxyanhydrides
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Publication Date: 02 August 2017

letter

Guo, Tao; Wei, Xu-Ning: Ammonium Iodide-Mediated Sulfenylation of 4-Hydroxycoumarins or 4-Hydroxyquinolinones with a Sulfonyl Chloride as a Sulfur Source
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synpacts

Gurak, John A.; Engle, Keary M.: Regioselective Hydroamination Using a Directed Nucleopalladation/Protodepalladation Strategy
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Publication Date: 27 July 2017

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Wang, Qiang; Shi, Min: Synthesis of Cyclic and Heterocyclic Compounds via Gold-Catalyzed Reactions
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letter

Matsumoto, Kenji; Mizushina, Naoyuki; Yoshida, Masahiro; Shindo, Mitsuru: Stereocontrolled Synthesis of Multisubstituted 1,3-Dienes via an Allene–Claisen Rearrangement
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letter

Matsumoto, Nobuyuki; Nakazaki, Atsuo; Nishikawa, Toshio: Concise Synthesis of a Cyclopentane Intermediate Possessing All Nitrogen Functionalities for Pactamycin
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letter

Stairs, Shaun; Powner, Matthew W.: Scalable Synthesis of 2,2′-Anhydro-arabinofuranosyl Imidazoles
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synpacts

Hullaert, Jan; Denoo, Bram; Christiaens, Mien; Callebaut, Brenda; Winne, Johan M.: Heterocycles as Moderators of Allyl Cation Cycloaddition Reactivity
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Publication Date: 24 July 2017

cluster

Patil, Pravin C.; Luzzio, Frederick A.: Unnatural Amino Acid Derivatives through Click Chemistry: Synthesis of Triazolylalanine Analogues
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Supporting Information

cluster

Yamamoto, Eiji; Ukigai, Satoshi; Ito, Hajime: Formal Nucleophilic Silyl Substitution of Aryl Halides with Silyllithium Reagents via Halogenophilic Attack of Silyl Nucleophiles
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letter

Han, Jusung; Kim, Yo-Han; Jung, Byeong Yeon; Hwang, Seung Hyun; Jegal, Jonggon; Kim, Jung Won; Lee, Yoon-Sik: Highly Selective Catalytic Hydrogenation and Etherification of 5-Hydroxymethyl-2-furaldehyde to 2,5-Bis(alkoxymethyl)furans for Potential Biodiesel Production
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letter

Lessing, Timo; Müller, Thomas J. J.: One-Pot Coupling–Cyclization–Alkylation Synthesis of 1,2,5-Trisubstituted 7-Azaindoles in a Consecutive Three-component Fashion
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new tools

Richert, Clemens; Krupp, Felix: Encapsulating Organic Crystals (EnOCs)
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Publication Date: 21 July 2017

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Quiclet-Sire, Béatrice; Zard, Samir Z.: Convergent Routes to Pyrroles Exploiting the Unusual Radical Chemistry of Xanthates – An Overview
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Flinker, Mathias; Lopez, Sara; Nielsen, Dennis U.; Daasbjerg, Kim; Jensen, Frank; Skrydstrup, Troels: Experimental and Theoretical Studies on the Reduction of CO2 to CO with Chloro(methyl)disilane Components from the Direct Process
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letter

Wei, Wen-Ting; Ying, Wei-Wei; Zhu, Wen-Ming; Wu, Yi; Huang, Yi-Ling; Cao, Yi-Qi; Wang, Yi-Ning; Liang, Hongze: Convenient and Clean Synthesis of Isatins by Metal-Free Oxidation of Oxindoles
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Publication Date: 20 July 2017

cluster

Guan, Xiaoyang; Chaffey, Patrick K.; Ruan, Yuan; Hurd, Connor K.; Taatjes, Dylan J.; Tan, Zhongping: Chemical Synthesis of the Multiply Phosphorylated and Biotinylated N-Terminal Transactivation Domain of Human p53 (p53TAD)
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cluster

Lee, Yong Ho; Morandi, Bill: Ether Synthesis through Reductive Cross-Coupling of Ketones with Alcohols Using Me2SiHCl as both Reductant and Lewis Acid
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cluster

Swartz, Brett D.; Brennessel, William W.; Jones, William D.: Lewis Acid Assisted C–CN Cleavage of Benzonitrile Using [(dippe)NiH]2
https://www.thieme-connect.de/media/synlett/EFirst/i_u0304_ga_10-1055_s-0036-1590801.gif
Supporting Information CIF File

letter

Ma, Teng; Li, Changwei; Liang, Haijing; Wang, Zhaoyan; Yu, Lan; Xue, Weihua: InBr3-Catalyzed Synthesis of Aryl 1,2-trans-Thio(seleno)glycosides
https://www.thieme-connect.de/media/synlett/EFirst/i_w0399_ga_10-1055_s-0036-1588507.gif
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letter

Stockdale, Trevor F.; O’Neil, Gregory W.: Regio- and Diastereoselective Samarium-Mediated Allylic Benzoate Reductions
https://www.thieme-connect.de/media/synlett/EFirst/i_r0421_ga_10-1055_s-0036-1590831.gif
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synpacts

Hou, Zhong-Wei; Mao, Zhong-Yi; Xu, Hai-Chao: Recent Progress on the Synthesis of (Aza)indoles through Oxidative Alkyne Annulation Reactions
https://www.thieme-connect.de/media/synlett/EFirst/i_p0452_ga_10-1055_s-0036-1590842.gif

Publication Date: 19 July 2017

cluster

Rohrbacher, Florian; Baldauf, Simon; Wucherpfennig, Thomas G.; Bode, Jeffrey W.: Product Selectivity in KAHA Ligations: Ester vs. Amide Formation with Cyclic Hydroxylamines
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Xie, Hengmu; Lu, Ji; Gui, Yingying; Gao, Lu; Song, Zhenlei: (HMe2SiCH2)2: A Useful Reagent for B(C6F5)3-Catalyzed Reduction–Lactonization of Keto Acids: Concise Syntheses of (–)-cis-Whisky and (–)-cis-Cognac Lactones
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letter

Benoit, Emeline; Dansereau, Julien; Gagnon, Alexandre: Palladium-Catalyzed Carbonylative Cross-Coupling Reaction between Aryl(Heteroaryl) Iodides and Tricyclopropylbismuth: Expedient Access to Aryl Cyclopropylketones
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letter

Dumitrescu, Denisa; Georgescu, Emilian; Caira, Mino R.; Draghici, Constantin; Dumitrascu, Florea: A New Synthesis of Pyrroles from Benzimidazolium N-Cyanomethyl Ylides and Alkyne Dipolarophiles
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letter

Schleper, A. Lennart; Voll, Constantin-Christian A.; Engelhart, Jens U.; Swager, Timothy M.: Iptycene-Containing Azaacenes with Tunable Luminescence
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Supporting Information

letter

Someshwar, Nagamalla; Karthick, Muthupandi; Ramanathan, Chinnasamy Ramaraj: Desymmetrization of Symmetrical Triarylcarbinols: Synthesis of 7-Arylfluorenes and a C2-Symmetric Chiral BIFOL Phosphoric Acid
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Publication Date: 18 July 2017

letter

Aitken, R. Alan; Harper, Andrew D; Slawin, Alexandra M. Z.: Base-Induced Cyclisation of ortho-Substituted 2-Phenyloxazolines to Give 3-Aminobenzofurans and Related Heterocycles
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letter

Kaddour, Alaa; Toumieux, Sylvestre; Wadouachi, Anne: Efficient Synthesis of N-Alkyl Polyhydroxylated Pipecolamide Compounds from d-Glucurono-6,3-lactone
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Supporting Information

letter

Lühning, Lars H.; Rosien, Michael; Doye, Sven: Thieme Chemistry Journals Awardees – Where Are They Now?
Titanium-Catalyzed Hydroaminoalkylation of Vinylsilanes and a One-Pot Procedure for the Synthesis of 1,4-Benzoazasilines
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Supporting Information

letter

Mennen, Steven M.; Arunachalampillai, Athimoolam; Choquette, Deborah M.; Muppalla, Harikrishna; Sheena, Krishna: Scalable Synthesis of 6,6-Dimethylbicyclo[3.1.0]hexan-3-one
https://www.thieme-connect.de/media/synlett/EFirst/i_r0291_ga_10-1055_s-0036-1588484.gif
Supporting Information

letter

Rabet, Pauline; Wagschal, Simon; Lemaire, Sébastien: Ferrier Rearrangement of 1,2-Dihydropyrans with Organozinc Species in Toluene/n-Dibutyl Ether
https://www.thieme-connect.de/media/synlett/EFirst/i_d0403_ga_10-1055_s-0036-1588485.gif

letter

Xue, Hongyu; Jing, Bing; Liu, Shasha; Chae, Junghyun; Liu, Yajun: Copper-Catalyzed Direct Synthesis of Aryl Thiols from Aryl Iodides Using Sodium Sulfide Aided by Catalytic 1,2-Ethanedithiol
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Supporting Information

Publication Date: 14 July 2017

cluster

Castillo-Pazos, Durbis J.; Macmillan, Derek: Investigation of Cysteine as an Activator of Side-Chain N→S Acyl Transfer and Tail-to-Side-Chain Cyclization
https://www.thieme-connect.de/media/synlett/EFirst/i_w0322_ga_10-1055_s-0036-1590797.gif
Supporting Information

cluster

Mao, Wenbin; Zhu, Chen: Rhodium-Catalyzed C–C Bond Olefination of Ring-Fused Benzocyclobutenols and Application in the Construction of Polycyclic Compounds
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Supporting Information

letter

Bagdžiūnas, Gintautas; Stončius, Sigitas; Butkus, Eugenijus: Synthesis of Star-Shaped Aromatic Derivatives with Chirality Predetermined by Bicyclo[3.3.1]nonane Framework
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Supporting Information

letter

Rajan, Blessy; Bedekar, Ashutosh V.: Synthesis of Unsymmetrical Aza[7]helicenes by One-Pot Wittig–Heck and Photodehydrogenation Sequence
https://www.thieme-connect.de/media/synlett/EFirst/i_b0306_ga_10-1055_s-0036-1590820.gif
Supporting Information

letter

Samzadeh-Kermani, Alireza: Ethynylation of Isoquinoline and Quinoline Derivatives with Calcium Carbide
https://www.thieme-connect.de/media/synlett/EFirst/i_d0206_ga_10-1055_s-0036-1590815.gif
Supporting Information

Publication Date: 13 July 2017

letter

Cherfaoui, Brahim; Lakhdari, Houria; Bennamane, Norah; Ameraoui, Rachid; Talhi, Oualid; Almeida Paz, Filipe A.; Bachari, Khaldoun; Kirsch, Gilbert; Nejar-Bellara, Kolli; Silva, Artur M. S.: Dibenzo[b,e][1,4]diazepin-1-ones and their Ring-Opened Derivatives: Revisited Synthesis, 2D NMR and Crystal Structure
https://www.thieme-connect.de/media/synlett/EFirst/i_d0318_ga_10-1055_s-0036-1590306.gif
Supporting Information CIF File

letter

Jiang, Qijian; Yang, Luo; Zhou, Wang: Copper-Catalyzed Cleavage of Unstrained C–C Bonds for the Synthesis of 1-Acyloxy-2,2,6,6-tetramethylpiperidines from Cyclic or Acyclic Ketones
https://www.thieme-connect.de/media/synlett/EFirst/i_w0266_ga_10-1055_s-0036-1590805.gif
Supporting Information

letter

Kolita, Sinki; Dutta, Leema; Das, Pankaj; Bhuyan, Pulak J: One-Pot Synthesis of Unsymmetrical Bis(4-Hydroxycoumarin-3-yl)methanes
https://www.thieme-connect.de/media/synlett/EFirst/i_d0288_ga_10-1055_s-0036-1589065.gif
Supporting Information

letter

Rajeev, Narasimhamurthy; Swaroop, Toreshettahally R.; Anil, Seegehalli M.; Bommegowda, Yadaganahalli K.; Rangappa, Kanchugarakoppal S.; Sadashiva, Marilinganadoddi P.: Base-Induced Cyclization of Active Methylene Isocyanides with Xanthate Esters: An Efficient Method for the Synthesis of 5-Alkoxy-4-(tosyl/ethoxycarbonyl)-1,3-thiazoles
https://www.thieme-connect.de/media/synlett/EFirst/i_b0262_ga_10-1055_s-0036-1590811.jpg
Supporting Information

letter

Yang, Zan; Li, Jiao; Hua, Jie; Yang, Tao; Yi, Jianmin; Zhou, Congshan: KI/K2S2O8-Mediated α-C–H Sulfenylation of Carbonyl Compounds with (Hetero)Aryl Thiols
https://www.thieme-connect.de/media/synlett/EFirst/i_r0233_ga_10-1055_s-0036-1588483.gif
Supporting Information

letter

Zhi, Ying; Zhao, Kun; von Essen, Carolina; Rissanen, Kari; Enders, Dieter: Thiourea-Catalyzed Domino Michael–Mannich [3+2] Cycloadditions: A Strategy for the Asymmetric Synthesis of 3,3′-Pyrrolidinyl-dispirooxindoles
https://www.thieme-connect.de/media/synlett/EFirst/i_r0387_ga_10-1055_s-0036-1589070.gif
Supporting Information

Publication Date: 12 July 2017

cluster

Denmark, Scott E.; Ambrosi, Andrea: Understanding Site Selectivity in the Palladium-Catalyzed Cross-Coupling of Allenylsilanolates
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Supporting Information

letter

Eljo, Jasmin; Carle, Myriam S.; Murphy, Graham K.: Hypervalent Iodine-Based Activation of Triphenylphosphine for the Functionalization of Alcohols
https://www.thieme-connect.de/media/synlett/EFirst/i_r0272_ga_10-1055_s-0036-1589069.gif
Supporting Information

letter

Hu, Xiao-Si; Du, Yi; Yu, Jin-Sheng; Liao, Fu-Min; Ding, Pei-Gang; Zhou, Jian: A Highly Efficient Gold(I)-Catalyzed Mukaiyama–Mannich Reaction of α-Amino Sulfones with Fluorinated Silyl Enol Ethers To Give β-Amino α-Fluorinated Ketones
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Supporting Information

letter

Pietrasiak, Ewa; Schade, Grit; Baalouch, Myriam; Emery, Daniel; Beaudegnies, Renaud: Synthesis of 2-Substituted Aziridine-2-Carboxylic Esters via Michael-Induced Ring-Closure Strategy
https://www.thieme-connect.de/media/synlett/EFirst/i_b0275_ga_10-1055_s-0036-1590806.gif
Supporting Information

Publication Date: 11 July 2017

cluster

Qi, Yun-Kun; He, Qiao-Qiao; Ai, Hua-Song; Li, Jia-Bin; Zheng, Ji-Shen: Convergent Total Synthesis of Histone H2B Protein with Site-Specific Ubiquitination at Lys120
https://www.thieme-connect.de/media/synlett/EFirst/i_w0257_ga_10-1055_s-0036-1590794.gif
Supporting Information

letter

Adhikari, Arijit A.; Radal, Léa; Chisholm, John D.: Synthesis of 3,3′-Disubstituted Indolenines Utilizing the Lewis Acid Catalyzed Alkylation of 2,3-Disubstituted Indoles with Trichloroacetimidates
https://www.thieme-connect.de/media/synlett/EFirst/i_r0343_ga_10-1055_s-0036-1588491.gif
Supporting Information

letter

Inagaki, Fuyuhiko; Hira, Shisen; Mukai, Chisato: Silver(I)-Catalyzed Deprenylation of Allylsulfonamide Derivatives
https://www.thieme-connect.de/media/synlett/EFirst/i_u0355_ga_10-1055_s-0036-1589066.gif
Supporting Information

letter

Leslie, Ray; Tseke, Kavnen; Vitkute, Agneta; Benjamin, Sophie L.; Seetohul, L. Nitin: Fluoropyridyl Sugars – Masked Imidate Glycosyl Donors that Display Reactivity, Selectivity, and Stability
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Supporting Information

letter

Ramulu, Bokka Venkat; Kumar, Devarapalli Ravi; Satyanarayana, Gedu: Superacid-Mediated Intramolecular Cyclization/Condensation: Facile One-Pot Synthesis of Spirotetracyclic Indanones and ­Indenes
https://www.thieme-connect.de/media/synlett/EFirst/i_d0323_ga_10-1055_s-0036-1590816.gif
Supporting Information

letter

Tang, Ruotian; Jiang, Chunfeng; Li, Hongliang; Li, Wei; Xu, Youjun: Facile Synthesis of N-Substituted 4-Amino-6-methyl Resorcinols from Polysubstituted Cyclohexanone
https://www.thieme-connect.de/media/synlett/EFirst/i_w0263_ga_10-1055_s-0036-1590817.gif
Supporting Information

Publication Date: 06 July 2017

cluster

Aihara, Keisuke; Inokuma, Tsubasa; Jichu, Takahisa; Lin, Zhenjian; Fu, Feixue; Yamaoka, Kosuke; Shigenaga, Akira; Hutchins, David A.; Schmidt, Eric W.; Otaka, Akira: Cysteine-Free Intramolecular Ligation of N-Sulfanylethylanilide Peptide Using 4-Mercaptobenzylphosphonic Acid: Synthesis of Cyclic Peptide Trichamide
https://www.thieme-connect.de/media/synlett/EFirst/i_u0286_ga_10-1055_s-0036-1589055.gif
Supporting Information

cluster

Chen, Pu-Guang; Huang, Zhi-Hua; Sun, Zhan-Yi; Li, Qian-Qian; Chen, Yong-Xiang; Zhao, Yu-Fen; Li, Yan-Mei: Synthesis of an MUC1 Glycopeptide Dendrimer Based on β-Cyclodextrin by Click Chemistry
https://www.thieme-connect.de/media/synlett/EFirst/i_w0259_ga_10-1055_s-0036-1590796.gif
Supporting Information

cluster

Ren, Xiaoyu; Han, Caifang; Feng, Xiangqing; Du, Haifeng: A Borane-Catalyzed Metal-Free Hydrosilylation of Chromones and Flavones
https://www.thieme-connect.de/media/synlett/EFirst/i_b0302_ga_10-1055_s-0036-1588474.gif
Supporting Information

letter

Hamel, Jean-Denys; Beaudoin, Meggan; Cloutier, Mélissa; Paquin, Jean-François: Hydrogen-Bond-Promoted Friedel–Crafts Reaction of Secondary Propargylic Fluorides: Preparation of 1-Alkyl-1-aryl-2-alkynes
https://www.thieme-connect.de/media/synlett/EFirst/i_r0278_ga_10-1055_s-0036-1589057.gif
Supporting Information

letter

Han, Jianwei; Qian, Xiaofei; Xu, Bowen; Wang, Limin: Potassium tert-Butoxide Mediated Arylation of 2-Substituted Malononitriles Using Diaryliodonium Salts
https://www.thieme-connect.de/media/synlett/EFirst/i_u0285_ga_10-1055_s-0036-1589061.gif
Supporting Information

letter

Kudoh, Takayuki; Fujisawa, Syo; Kitamura, Megumi; Sakakura, Akira: Heat Versus Basic Conditions: Intramolecular Dehydro-Diels–Alder Reaction of 1-Indolyl-1,6-heptadiynes for the Selective Synthesis of Substituted Carbazoles
https://www.thieme-connect.de/media/synlett/EFirst/i_u0315_ga_10-1055_s-0036-1588461.gif
Supporting Information

letter

Li, Yang; Wang, Yu; Xu, Dawen; Jin, Ruiwen; Gu, Guangxin; Guo, Hao: AlCl3-Catalyzed Intramolecular Hydroarylation of Arenes with Alkynes
https://www.thieme-connect.de/media/synlett/EFirst/i_w0250_ga_10-1055_s-0036-1588479.gif
Supporting Information

letter

Mase, Nobuyuki; Nishina, Yuki; Isomura, Shogo; Sato, Kohei; Narumi, Tetsuo; Watanabe, Naoharu: Fine-Bubble-Based Strategy for the Palladium-Catalyzed Hydrogenation of Nitro Groups: Measurement of Ultrafine Bubbles in Organic Solvents
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Supporting Information

letter

Wakamatsu, Hideaki; Yanagisawa, Rika; Kimura, Sho; Osawa, Nao; Natori, Yoshihiro; Yoshimura, Yuichi: Palladium-Catalyzed Regioselective Hydroarylation of Ynamides with Aryl Iodides: Easy Synthesis of Various Substituted Enamides Containing Stilbene Derivatives
https://www.thieme-connect.de/media/synlett/EFirst/i_u0276_ga_10-1055_s-0036-1588874.gif
Supporting Information

letter

Zhou, Manxi; Zhu, Lei; Sun, Zhimin; Yang, Zhenqing; Cao, Dapeng; Li, Qifang: Tri-Petal Lilac-Like Perylene: Asymmetrical Substituted Platform for Regioselective Ether-Exchange Reaction
https://www.thieme-connect.de/media/synlett/EFirst/i_w0307_ga_10-1055_s-0036-1590808.jpg
Supporting Information

Publication Date: 05 July 2017

account

Deng, Yongming; Cheng, Qing-Qing; Doyle, Michael P.: Asymmetric [3+3] Cycloaddition for Heterocycle Synthesis
https://www.thieme-connect.de/media/synlett/EFirst/i_a0230_ga_10-1055_s-0036-1588453.gif

cluster

Li, Kaicheng; Gao, Jianmin: Iminoboronate-Mediated Peptide Cyclization with Lysine Homologues
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Supporting Information

cluster

Shima, Yusuke; Igarashi, Emiko; Yoshimura, Tomoyuki; Matsuo, Jun-ichi: Reactions of Nitrosobenzenes with Cyclobutanones by Activation with a Lewis Acid
https://www.thieme-connect.de/media/synlett/EFirst/i_u0293_ga_10-1055_s-0036-1588469.gif
Supporting Information

letter

Chittimalla, Santhosh Kumar; Bandi, Chennakesavulu; Gadi, Vinod Kumar; Gunturu, Siva Ramakrishna: Facile Synthesis of 2-Arylindoles through Plancher-Type Rearrangement of 3-Alkyl-3-Arylindolenines
https://www.thieme-connect.de/media/synlett/EFirst/i_b0247_ga_10-1055_s-0036-1588448.gif
Supporting Information

letter

Sato, Shogo; Kawada, Takuma; Takikawa, Hiroshi; Suzuki, Keisuke: Preparation of 2-Substituted 3-Methoxycarbonyl-4-methoxyfurans that Allow Access to Highly Functionalized Naphthalenes via Regioselective Cycloaddition with Alkoxybenzyne
https://www.thieme-connect.de/media/synlett/EFirst/i_b0332_ga_10-1055_s-0036-1590825.gif
Supporting Information

Publication Date: 04 July 2017

letter

Feng, Ruokun; Gao, Yuan; Liu, Zhanxiang; Zhang, Yuhong: Rhodium(III)-Catalyzed Sequential Cleavage of Two C–H Bonds for the Synthesis of Polyarylated Naphthols
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Supporting Information

letter

Igawa, Kazunobu; Aoyama, Shin; Kawasaki, Yuuya; Kashiwagi, Takeru; Seto, Yuki; Ni, Runyan; Mitsuda, Naoto; Tomooka, Katsuhiko: Thieme Chemistry Journals Awardees: Where Are They Now? One-Pot Synthesis of Versatile Buckle Units for Click Chemistry: 4,8-Diazacyclononynes (DACNs)
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Supporting Information

Publication Date: 29 June 2017