DOI: 10.1055/s-00000083

Synlett

eFirst

Publication Date: 27 June 2017

cluster

Jarrige, Lucie; Zaied, Siwar; Merad, Jeremy; Blanchard, Florent; Masson, Géraldine: Easy Access to Quinolin-2(1H)-ones via a One-Pot Tandem Oxa-Michael–Aldol Sequence
https://www.thieme-connect.de/media/synlett/EFirst/i_b0305_ga_10-1055_s-0036-1588470.gif
Supporting Information

errata

Guo, Yongbiao; Gao, Zhenhua; Meng, Xiangyan; Huang, Guilan; Zhong, Hui; Yu, Huilan; Ding, Xiaoqin; Tang, Hui; Zou, Chuanpin: Highly Enantioselective Biginelli Reaction of Aliphatic Aldehydes Catalyzed by Chiral Phosphoric Acids

Publication Date: 21 June 2017

account

Morimoto, Koji; Dohi, Toshifumi; Kita, Yasuyuki: Metal-free Oxidative Cross-Coupling Reaction of Aromatic Compounds Containing Heteroatoms
https://www.thieme-connect.de/media/synlett/EFirst/i_a0218_ga_10-1055_s-0036-1588455.gif

cluster

Sanzone, Jillian R.; Woerpel, K. A.: Reactivity of Seven-Membered-Ring trans-Alkenes with Electrophiles
https://www.thieme-connect.de/media/synlett/EFirst/i_b0248_ga_10-1055_s-0036-1588451.gif
Supporting Information

cluster

Tsuda, Shugo; Uemura, Tsuyoshi; Mochizuki, Masayoshi; Nishio, Hideki; Yoshiya, Taku: Preparation of Peptide o-Aminoanilides Using a Modified Dawson's Linker for Microwave-Assisted Peptide Synthesis
https://www.thieme-connect.de/media/synlett/EFirst/i_w0227_ga_10-1055_s-0036-1588862.gif
Supporting Information

letter

Kumari, P.; Sharma, N.; Kumar, A.; Mohapatra, S. C.; Bhagat, S.: A Highly Efficient Approach for the Synthesis of Novel Trifluoroacetylated Enaminones using DBU as a Base
https://www.thieme-connect.de/media/synlett/EFirst/i_d0251_ga_10-1055_s-0036-1588865.gif
Supporting Information

letter

Wei, Wen-Ting; Zhu, Wen-Ming; Liang, Weida; Wu, Yi; Huang, Hui-Yan; Huang, Yi-Ling; Luo, Junfei; Liang, Hongze: Room-Temperature, Water-Promoted, Radical-Coupling Reactions of Phenols with tert-Butyl Nitrite
https://www.thieme-connect.de/media/synlett/EFirst/i_w0241_ga_10-1055_s-0036-1589038.gif
Supporting Information

letter

Xiong, Xiaoyu; Zhu, Ranran; Huang, Lin; Chang, Shuqin; Huang, Jianhui: Direct ortho Arylation of Anisoles via the Formation of Four-Membered Lithiumcycles/Palladacycles
https://www.thieme-connect.de/media/synlett/EFirst/i_w0237_ga_10-1055_s-0036-1588863.gif
Supporting Information

Publication Date: 08 June 2017

account

Biafora, Agostino; Gooßen, Lukas J.: Thieme Chemistry Journals Awardees – Where Are They Now? New Reaction Mode in Carboxylate-Directed C–H Functionalizations: Carboxylates as Deciduous Directing Groups
https://www.thieme-connect.de/media/synlett/EFirst/i_a0238_ga_10-1055_s-0036-1588450.gif

Publication Date: 07 June 2017

letter

Guo, Yongbiao; Gao, Zhenhua; Meng, Xiangyan; Huang, Guilan; Zhong, Hui; Yu, Huilan; Ding, Xiaoqin; Tang, Hui; Zou, Chuanpin: Highly Enantioselective Biginelli Reaction of Aliphatic Aldehydes Catalyzed by Chiral Phosphoric Acids
https://www.thieme-connect.de/media/synlett/EFirst/i_w0235_ga_10-1055_s-0036-1588853.gif
Supporting Information

letter

Rhoné, Benoît; Semetey, Vincent: Base-Catalyzed Transcarbamoylation
https://www.thieme-connect.de/media/synlett/EFirst/i_d0172_ga_10-1055_s-0036-1588866.gif
Supporting Information

letter

Seio, Kohji; Tokugawa, Munefumi; Kaneko, Kazuhei; Shiozawa, Takashi; Masaki, Yoshiaki: A Systematic Study of the Synthesis of 2ʹ-Deoxynucleosides by Mitsunobu Reaction
https://www.thieme-connect.de/media/synlett/EFirst/i_u0217_ga_10-1055_s-0036-1588445.gif
Supporting Information

Publication Date: 06 June 2017

account

Saha, Mrinmoy; Carter, Rich G.: Lycopodium Alkaloids: An Intramolecular Michael Reaction Approach
https://www.thieme-connect.de/media/synlett/EFirst/i_a0150_ga_10-1055_s-0036-1588851.jpg

letter

Ketels, Marthe; Ziegler, Dorothée S.; Knochel, Paul: Selective Zincation of 1,2-Dicyanobenzene and Related Benzonitriles in Continuous Flow Using In Situ Trapping Metalations
https://www.thieme-connect.de/media/synlett/EFirst/i_r0246_ga_10-1055_s-0036-1588837.gif
Supporting Information

letter

Schmidt, Stephan; Hanelt, Sven; Canitz, Carsten; Hoffmann, Holger; Garbe, Leif-Alexander; Schneider, Rudolf J.: Synthetic Strategies for the Modification of Diclofenac
https://www.thieme-connect.de/media/synlett/EFirst/i_b0210_ga_10-1055_s-0036-1588858.gif

synpacts

Lu, Dapeng; Cui, Shengsheng; Du, Pingwu: Large π-Extension of Carbon Nanorings by Incorporating Hexa-peri-hexabenzocoronenes
https://www.thieme-connect.de/media/synlett/EFirst/i_p0201_ga_10-1055_s-0036-1588830.gif

Publication Date: 31 May 2017

cluster

Wübbolt, Simon; Oestreich, Martin: Exhaustive Chemoselective Reduction of Nitriles by Catalytic Hydrosilylation Involving Cooperative Si–H Bond Activation
https://www.thieme-connect.de/media/synlett/EFirst/i_b0170_ga_10-1055_s-0036-1588441.gif
Supporting Information

letter

Gao, Hongjie; Xu, Xiangsheng; Xu, Jianfeng: Sc(OTf)3-Catalyzed Aza-Friedel–Crafts Reaction of Electron-Rich Arenes with Isatin-Derived Ketimines: Access to 3-Amino-3-Aryl-2-Oxindoles
https://www.thieme-connect.de/media/synlett/EFirst/i_w0202_ga_10-1055_s-0036-1588432.gif
Supporting Information

letter

Puentes, Alfredo R.; Neves Filho, Ricardo A. W.; Rivera, Daniel G.; Wessjohann, Ludger A.: Total Synthesis of Cordyheptapeptide A
https://www.thieme-connect.de/media/synlett/EFirst/i_d0209_ga_10-1055_s-0036-1588433.gif
Supporting Information

letter

Sun, Pengcheng; Tang, Wenli; Huang, Yu; Hu, Bi-Huang: Improved Fmoc Solid-Phase Peptide Synthesis of Oxytocin with High Bioactivity
https://www.thieme-connect.de/media/synlett/EFirst/i_w0240_ga_10-1055_s-0036-1589037.gif
Supporting Information

letter

Tang, Hai-Tao; Zeng, Jia-Hao; Chen, Jun-Jia; Chen, Yi-Hui; Zhan, Zhuang-Ping: Synthesis of (E)-4,5-Dihydro-1H-Pyrazoles via Tandem Intermolecular Addition–Cyclization of N-Propargylic Sulfonylhydrazones
https://www.thieme-connect.de/media/synlett/EFirst/i_w0219_ga_10-1055_s-0036-1588844.gif
Supporting Information

Publication Date: 24 May 2017

cluster

Tornøe, Christian W.; Johansson, Eva; Wahlund, Per-Olof: Divergent Protein Synthesis of Bowman–Birk Protease Inhibitors, their Hydrodynamic Behavior and Co-crystallization with α-Chymotrypsin
https://www.thieme-connect.de/media/synlett/EFirst/i_w0211_ga_10-1055_s-0036-1588840.jpg
Supporting Information

letter

Shen, Guodong; Wang, Yichen; Zhao, Xiliang; Huangfu, Xinlei; Tian, Yanmeng; Zhang, Tongxin; Yang, Bingchuan: Pd/C-Catalyzed Homocoupling Reaction for the Synthesis of Symmetrical Biaryl Diamides
https://www.thieme-connect.de/media/synlett/EFirst/i_w0197_ga_10-1055_s-0036-1588437.gif
Supporting Information

letter

Yuan, Wenjiao; Liu, Yali; Li, Chunbao: A Rapid and Diastereoselective Synthesis of 2-Deoxy-2-iodo-α-glycosides and its Mechanism for Diastereoselectivity
https://www.thieme-connect.de/media/synlett/EFirst/i_w0212_ga_10-1055_s-0036-1588440.gif
Supporting Information

synpacts

Zhu, Feng; Yang, Tianyi; Walczak, Maciej A.: Glycosyl Stille Cross-Coupling with Anomeric Nucleophiles – A General Solution to a Long-Standing Problem of Stereocontrolled Synthesis of C-Glycosides
https://www.thieme-connect.de/media/synlett/EFirst/i_p0176_ga_10-1055_s-0036-1589020.gif

Publication Date: 23 May 2017

cluster

Gandhamsetty, Narasimhulu; Park, Sehoon; Chang, Sukbok: Boron-Catalyzed Hydrogenative Reduction of Substituted Quinolines to Tetrahydroquinolines with Hydrosilanes
https://www.thieme-connect.de/media/synlett/EFirst/i_b0216_ga_10-1055_s-0036-1588442.gif
Supporting Information

Publication Date: 19 May 2017

letter

Szantai-Kis, D. Miklos; Walters, Christopher R.; Barrett, Taylor M.; Hoang, Eileen M.; Petersson, E. James: Thieme Chemistry Journals Awardees – Where Are They Now?
Improved Fmoc Deprotection Methods for the Synthesis of Thioamide-Containing Peptides and Proteins
https://www.thieme-connect.de/media/synlett/EFirst/i_r0178_ga_10-1055_s-0036-1589027.gif
Supporting Information

Publication Date: 18 May 2017

letter

Chavan, Sujit P.; K., Adithyaraj; Bhanage, Bhalchandra M.: In situ Generation and Utilization of CO: An Efficient Route towards N-Substituted Saccharin via Carbonylative Cyclization of 2-Iodosulfonamides
https://www.thieme-connect.de/media/synlett/EFirst/i_d0143_ga_10-1055_s-0036-1588422.gif
Supporting Information

Publication Date: 17 May 2017

letter

Kazem-Rostami, Masoud: Facile Preparation of Λ-Shaped Building Blocks: Hünlich Base Derivatization
https://www.thieme-connect.de/media/synlett/EFirst/i_b0194_ga_10-1055_s-0036-1588180.gif
Supporting Information

letter

Yoshimura, Fumihiko; Saito, Hiroki; Abe, Taiki; Tanino, Keiji: Nucleophilic Addition of Alkanenitriles to Aldehydes via N-Silyl Ketene Imines Generated In Situ
https://www.thieme-connect.de/media/synlett/EFirst/i_u0185_ga_10-1055_s-0036-1588424.gif
Supporting Information

letter

Yuan, Yan-qin; Kumar, Pailla Santhosh; Guo, Sheng-rong: Metal-Free Ammonium Iodide Catalyzed Oxidative Dehydrocoupling of Silanes with Alcohols
https://www.thieme-connect.de/media/synlett/EFirst/i_w0110_ga_10-1055_s-0036-1588816.gif
Supporting Information

Publication Date: 16 May 2017

letter

Shao, Tongle; Fang, Xiang; Zhou, Jun; Jin, Chen; Yang, Xueyan; Wu, Fanhong: I2/TBHP-Promoted Approach to α-Keto Esters from Trifluoromethyl β-Diketones and Alcohols via C–C Bond Cleavage
https://www.thieme-connect.de/media/synlett/EFirst/i_w0151_ga_10-1055_s-0036-1588833.gif
Supporting Information

synpacts

Ludwig, Jacob R.; Schindler, Corinna S.: Lewis Acid Catalyzed Carbonyl–Olefin Metathesis
https://www.thieme-connect.de/media/synlett/EFirst/i_p0146_ga_10-1055_s-0036-1588827.gif

Publication Date: 12 May 2017

letter

Ho, Son Long; Dao, Pham Duy Quang; Cho, Chan Sik: Microwave-Assisted Synthesis of Benzo[4,5]imidazo[1,2-a]pyrimidines from β-Bromo-α,β-unsaturated Aldehydes and 2-Aminobenzimidazoles
https://www.thieme-connect.de/media/synlett/EFirst/i_u0161_ga_10-1055_s-0036-1588834.gif

Publication Date: 11 May 2017

letter

Inamori, Daiki; Miwa, Takuya; Fujihara, Tetsuaki; Tsuji, Yasushi; Terao, Jun: Thieme Chemistry Journals Awardees – Where Are They Now?
Synthesis of a Dinuclear Copper NHC Complex Bearing a Rigid π-Conjugated Cyclic Framework
https://www.thieme-connect.de/media/synlett/EFirst/i_u0199_ga_10-1055_s-0036-1588824.gif
Supporting Information

Publication Date: 10 May 2017

letter

Cai, Yuguo; Zhang, Ronghua; Sun, Deli; Xu, Song; Zhou, Qiguang: Eosin Y-Sensitized Photocatalytic Reaction of Tertiary Aliphatic Amines with Arenesulfonyl Chlorides under Visible-Light Irradiation
https://www.thieme-connect.de/media/synlett/EFirst/i_w0167_ga_10-1055_s-0036-1588828.gif
Supporting Information

letter

Chen, Zhengkai; Cao, Gangjian; Zhang, Fengjin; Li, Hongli; Xu, Jianfeng; Miao, Maozhong; Ren, Hongjun: Metal-Free Mediated C-3 Methylsulfanylation of Imidazo[1,2-a]-pyridines with Dimethyl Sulfoxide as a Methylsulfanylating Agent
https://www.thieme-connect.de/media/synlett/EFirst/i_w0152_ga_10-1055_s-0036-1588419.gif
Supporting Information

letter

Chen, Xiang-Xiang; Wang, Jia-Xin; Ren, Jiang-Tao; Xie, Hu; Zhao, Yanxia; Li, Ya-Min; Sun, Meng: A Convenient Strategy for Remote C–H Bond Halogenation of 8-Aminoquinolines in the C5 Position
https://www.thieme-connect.de/media/synlett/EFirst/i_w0174_ga_10-1055_s-0036-1588420.gif
Supporting Information Primary Data

letter

Zhang, Xiao-Ru; Zhou, Su-Lan; Yuan, Yi; Du, Wei; Chen, Ying-Chun: Chemo- and Regioselective Asymmetric Friedel–Crafts Reaction of Furans and Thiophenes with α,β-Unsaturated Aldehydes through Dual Activation
https://www.thieme-connect.de/media/synlett/EFirst/i_w0173_ga_10-1055_s-0036-1588831.gif
Supporting Information

Publication Date: 08 May 2017

cluster

Minami, Yasunori; Komiyama, Takeshi; Shimizu, Kenta; Uno, Shu-ichi; Hiyama, Tamejiro; Goto, Osamu; Ikehira, Hideyuki: Nickel-Catalyzed N-Arylation Using N-Trimethylsilyl-carbazole
https://www.thieme-connect.de/media/synlett/EFirst/i_b0163_ga_10-1055_s-0036-1588417.gif
Supporting Information

letter

Abronina, Polina I.; Zinin, Alexander I.; Malysheva, Nelly N.; Stepanova, Elena V.; Chizhov, Alexander O.; Torgov, Vladimir I.; Kononov, Leonid O.: A Novel Glycosyl Donor with a Triisopropylsilyl Nonparticipating Group in Benzyl-Free Stereoselective 1,2-cis-Galactosylation
https://www.thieme-connect.de/media/synlett/EFirst/i_d0159_ga_10-1055_s-0036-1589028.gif
Supporting Information

letter

Yavari, Issa; Khajeh-Khezri, Aliyeh; Bahemmat, Samira; Halvagar, Mohammad Reza: A Synthesis of Novel Dioxapropellanes from the Knoevenagel Adducts of Acenaphthoquinone and 3-Oxo-3-arylpropionitriles in Aqueous Methanol
https://www.thieme-connect.de/media/synlett/EFirst/i_d0023_ga_10-1055_s-0036-1588822.gif
Supporting Information

letter

Zhao, Mingzhu; Tian, Yawei; Zhao, Xiaoming: Thieme Chemistry Journals Awardees – Where Are They Now?
Chiral Sulfinamide Ligands and Pd-Catalyzed Asymmetric Allylic Alkylations of Ethyl 2-Fluoroacetoacetate
https://www.thieme-connect.de/media/synlett/EFirst/i_w0191_ga_10-1055_s-0036-1589033.gif
Supporting Information

Publication Date: 04 May 2017

account

Komiyama, Takeshi; Minami, Yasunori; Hiyama, Tamejiro: Recent Progress in the Cross-Coupling Reaction Using Triorgano­silyl-Type Reagents
https://www.thieme-connect.de/media/synlett/EFirst/i_a0142_ga_10-1055_s-0036-1589008.gif

letter

Gang, Fangli; Che, Yang; Du, Zhengyin; Feng, Hua; Fu, Ying: Palladium-Catalyzed Regioselective C-5 Arylation of 1,2,3-Triazoles with Diaryliodonium Salts
https://www.thieme-connect.de/media/synlett/EFirst/i_w0112_ga_10-1055_s-0036-1588815.gif
Supporting Information

letter

Guo, Tao; Wang, Hongyan: Copper-Mediated Direct Sulfenylation of 4-Hydroxyquinolinones and 4-Hydroxypyridones with Aryl Thiols via a C−H Functionalization Process
https://www.thieme-connect.de/media/synlett/EFirst/i_w0177_ga_10-1055_s-0036-1588829.gif
Supporting Information

letter

Peng, Zhihua; Yu, Zhi; Chen, Dong-Huang; Liang, Shuyuan; Zhang, Liwei; Zhao, Dezhi; Song, Linhua; Jiang, Cuiyu: Efficient C(sp3)–H Bond Arylation of Tetrahydroisoquinolines with Knochel-Type Arylzinc Reagents under Oxidative Conditions
https://www.thieme-connect.de/media/synlett/EFirst/i_w0113_ga_10-1055_s-0036-1589029.gif
Supporting Information

letter

Wang, Xiaodong; Wang, Huihong; Wu, Xia; Yu, Tianqun; Gao, Weiwei; Shi, Tao; Peng, Xue; He, Dian; Wang, Zhen: Total Synthesis of (+)-Mintlactone and (–)-Isomintlactone via SmI2-Induced Radical Cyclization
https://www.thieme-connect.de/media/synlett/EFirst/i_w0134_ga_10-1055_s-0036-1588418.gif
Supporting Information

letter

Zhu, Yi-Fan; Geng, Xin-Le; Guan, Yong-Hong; Teng, Wei; Fan, Xiaohui: Poly(phosphoric acid) (PPA)-Promoted 5-exo-Cyclization of Iminium Ions Generated In Situ: A Facile Access to Functionalized Indene Derivatives
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Supporting Information

Publication Date: 02 May 2017

cluster

Das, Manas; Manvar, Atul; Fox, Ian; Roberts, Dilwyn J.; O’Shea, Donal F.: Bu4N+-Controlled Addition and Olefination with Ethyl 2-(Trimethylsilyl)acetate via Silicon Activation
https://www.thieme-connect.de/media/synlett/EFirst/i_b0077_ga_10-1055_s-0036-1588805.gif
Supporting Information

cluster

Sterckx, Hans; Sambiagio, Carlo; Lemière, Filip; Tehrani, Kourosch Abbaspour; Maes, Bert U. W.: Iron-Catalyzed Aerobic Oxidation of (Alkyl)(aryl)azinylmethanes
https://www.thieme-connect.de/media/synlett/EFirst/i_r0149_ga_10-1055_s-0036-1589014.gif
Supporting Information

letter

Brocklehurst, Cara E.; Koch, Guido; Rothe-Pöllet, Stephanie; La Vecchia, Luigi: In Situ Preparation and Consumption of O-Mesitylsulfonylhydroxylamine (MSH) in Continuous Flow for the Amination of Pyridines
https://www.thieme-connect.de/media/synlett/EFirst/i_b0095_ga_10-1055_s-0036-1588799.gif
Supporting Information

letter

Grigor’ev, Arthur A.; Karpov, Sergey V.; Kayukov, Yakov S.; Gracheva, Iuliia A.; Tafeenko, Victor A.: Cascade Regioselective Heterocyclization of 2-Acyl-1,1,3,3-tetracyanopropenides: Synthesis of Pyrrolo[3,4-c]pyridine and Pyrrolo[3,4-d]thieno[2,3-b]pyridine Derivatives
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Supporting Information

letter

Hofsäß, Robert; Rombach, David; Wagenknecht, Hans-Achim: Thieme Chemistry Journal Awardees – Where are They Now?
The Influence of Electron-Withdrawing Groups at the 2- and 2′-Positions of Dibenzothienylethenes on Molecular Switching
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letter

Maurya, Chandra Kant; Gupta, Pradeep Kumar: Phosphorus Pentasulfide Mediated Conversion of Primary Carbamates into Thiols
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letter

Sawatzky, Ryan S.; Ferguson, Michael J.; Stradiotto, Mark: Thieme Chemistry Journals Awardees – Where Are They Now?
Efficient Cross-Coupling of Secondary Amines/Azoles and Activated (Hetero)Aryl Chlorides Using an Air-Stable DPEPhos/Nickel Pre-Catalyst
https://www.thieme-connect.de/media/synlett/EFirst/i_r0188_ga_10-1055_s-0036-1588806.gif
Supporting Information CIF File

letter

Vásquez-Céspedes, Suhelen; Holtkamp, Michael; Karst, Uwe; Glorius, Frank: Reusable and Magnetic Palladium and Copper Oxide Catalysts in Direct ortho and meta Arylation of Anilide Derivatives
https://www.thieme-connect.de/media/synlett/EFirst/i_r0147_ga_10-1055_s-0036-1589007.gif
Supporting Information

letter

Yang, Seung-Hye; Jo, Seohyun; Shin, Dongyun: AlCl3-Mediated Synthesis of 4-Aryl-2-quinolone-3-carboxylates
https://www.thieme-connect.de/media/synlett/EFirst/i_u0119_ga_10-1055_s-0036-1588798.gif

Publication Date: 27 April 2017

account

Macmillan, Derek: Going Round in Circles with N→S Acyl Transfer
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letter

Fan, Yuanyuan; Zhou, Bei; Chen, Kun; Wang, Bingtao; Li, Xiaoqing; Xu, Xiangsheng: A Facile Synthesis of β-Iodonitro Alkenes via Iodonitration of Alkynes with tert-Butyl Nitrite and Iodine
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Supporting Information

letter

He, Jie; Kimani, Flora W.; Jewett, John C.: Rapid in Situ Generation of Benzene Diazonium Ions under Basic Aqueous Conditions from Bench-Stable Triazabutadienes
https://www.thieme-connect.de/media/synlett/EFirst/i_r0097_ga_10-1055_s-0036-1588797.gif
Supporting Information

letter

Tanii, Saori; Arisawa, Mieko; Tougo, Takaya; Horiuchi, Kiyofumi; Yamaguchi, Masahiko: Thieme Chemistry Journals Awardees – Where Are They Now?
Rhodium-Catalyzed Synthesis of Unsymmetric Di(heteroaryl) Ethers Using Heteroaryl Exchange Reaction
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Supporting Information

Publication Date: 26 April 2017

letter

Onda, Kai; Hayakawa, Ichiro; Sakakura, Akira: Reinvestigation of the Biomimetic Cyclization of 3,5-Diketo Esters: Application to the Total Synthesis of Cyercene A, an α-Methoxy-γ-Pyrone-Containing Polypropionate
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Supporting Information

letter

Shahsavari, Fatemeh; Abbasi, Alireza; Ghazanfarpour-Darjani, Majid; Ghafelebashi, Seyed Mehdi; Daftari-Besheli, Majid: Synthesis of Allylbenzene Derivatives through sp3 C–H Bond Functionalization of Toluene Derivatives
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Supporting Information

Publication Date: 20 April 2017

cluster

Jiang, Yan-Hong; Zhao, Hui; Tian, Yuan; Li, Zi-Gang: Lipid–Cell-Penetrating-Peptide Conjugates as Effective Delivery Systems
https://www.thieme-connect.de/media/synlett/EFirst/i_w0118_ga_10-1055_s-0036-1588807.gif
Supporting Information

Publication Date: 19 April 2017

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Caruana, Lorenzo; Fochi, Mariafrancesca; Bernardi, Luca: Enantioselective Approaches to 3,4-Annulated Indoles Using Organocatalytic Domino Reactions
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cluster

Li, Ziyuan; Wang, Xiaoyang; Ma, Lifang; Jiao, Ning: Copper-Catalyzed Aerobic Oxidation and Oxygenation of Anilines and Acetaldehydes with Dioxygen for the Concise Synthesis of 2-Aroylquinolines
https://www.thieme-connect.de/media/synlett/EFirst/i_r0074_ga_10-1055_s-0036-1588171.gif
Supporting Information

cluster

Matveenko, Maria; Becker, Christian F. W.: Synthetic Approach to Argpyrimidine as a Tool for Investigating Nonenzymatic Posttranslational Modification of Proteins
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Supporting Information

letter

Adib, Mehdi; Pashazadeh, Rahim; Gohari, Seyed Jamal Adin; Shahsavari, Fatemeh: Metal-Free Oxidative C=C Bond Cleavage of Electron-Deficient Enamines Promoted by tert-Butyl Hydroperoxide
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Supporting Information

letter

Guethner, Thomas; Huber, Eva; Sans, Juergen; Thalhammer, Franz: Direct Introduction of an N,N′-Nonsubstituted Carboxamidine Group by Grignard Addition to Silylated Cyanamide
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letter

Pilkington, Lisa I.; Song, Soo Min; Fedrizzi, Bruno; Barker, David: Efficient Total Synthesis of (±)-Isoguaiacin and (±)-Isogalbulin
https://www.thieme-connect.de/media/synlett/EFirst/i_d0162_ga_10-1055_s-0036-1588788.gif

Publication Date: 18 April 2017

letter

Wu, Yen-Ku; Lin, Rongrong; West, F. G.: Intercepting the Nazarov Oxyallyl Intermediate with α-Formyl­vinyl Anion Equivalents to Access Formal Morita–Baylis–Hillman Alkylation Products
https://www.thieme-connect.de/media/synlett/EFirst/i_r0080_ga_10-1055_s-0036-1588769.gif
Supporting Information

Publication Date: 11 April 2017

account

Shaaban, Saad; Maulide, Nuno: Metal-Free Redox Transformations for C–C and C–N Bond Construction
https://www.thieme-connect.de/media/synlett/EFirst/i_r0098_ga_10-1055_s-0036-1588776.gif

letter

Chen, Zhiwei; Chen, Hao; Yang, Xiaofeng; Chang, Xiangqing: Novel One-Pot Cyclization of the Blaise Reaction Intermediate and Arylglyoxals: The Synthesis of Substituted NH-Pyrroles
https://www.thieme-connect.de/media/synlett/EFirst/i_w0001_ga_10-1055_s-0036-1588168.gif
Supporting Information

letter

Dengiz, Cagatay; Swager, Timothy M.: Homoconjugated and Spiro Push–Pull Systems: Cycloadditions of Naphtho- and Anthradiquinones with Electron-Rich Alkynes
https://www.thieme-connect.de/media/synlett/EFirst/i_r0078_ga_10-1055_s-0036-1588771.gif
Supporting Information CIF File

letter

Fang, Jizhong; Xu, Lige; Fang, Bowen; Huo, Xing: Synergistic Oxidative Coupling–[3+2] Cyclization of Quinones with Olefins Promoted by Cerium(IV) Sulfate Tetrahydrate
https://www.thieme-connect.de/media/synlett/EFirst/i_w0073_ga_10-1055_s-0036-1588781.gif
Supporting Information

letter

Ichioka, Fumiki; Itai, Yuhei; Nishii, Yuji; Miura, Masahiro: Palladium-Catalyzed Direct C2-Arylation of Benzo[b]thiophenes with Electron-Rich Aryl Halides: Facile Access to Thienoacene Derivatives
https://www.thieme-connect.de/media/synlett/EFirst/i_r0128_ga_10-1055_s-0036-1588994.gif
Supporting Information

letter

Lee, Sunggi; Kaib, Philip S. J.; List, Benjamin: N-Triflylphosphorimidoyl Trichloride: A Versatile Reagent for the Synthesis of Strong Chiral Brønsted Acids
https://www.thieme-connect.de/media/synlett/EFirst/i_d0137_ga_10-1055_s-0036-1588782.gif
Supporting Information

letter

Lin, Yan; Ma, Wei-Yang; Sun, Qiao-Ying; Cui, Yu-Ming; Xu, Li-Wen: Catalytic Synthesis of Chiral Phosphole Oxides via Desymmetric C–H Arylation of o-Bromoaryl Phosphine Oxides
https://www.thieme-connect.de/media/synlett/EFirst/i_w0094_ga_10-1055_s-0036-1588983.gif
Supporting Information

letter

Liu, Yaowen; Zhang, Wensheng; Xie, Kai; Jiang, Yubo: Silver-Catalyzed Intramolecular C(5)–H Acyloxylation of 1,4-Di­substituted 1,2,3-Triazoles
https://www.thieme-connect.de/media/synlett/EFirst/i_w0129_ga_10-1055_s-0036-1588779.gif
Supporting Information

letter

Nematpour, Manijeh; Rezaee, Elham; Tabatabai, Sayyed Abbas; Jahani, Mehdi: A Copper-Catalyzed Synthesis of Functionalized Quinazolines from Isocyanides and Aniline Tri- and Dichloroacetonitrile Adducts through Intramolecular C–H Activation
https://www.thieme-connect.de/media/synlett/EFirst/i_d0018_ga_10-1055_s-0036-15588166.gif
Supporting Information

letter

Yu, Haifeng; Zhao, Lijuan; Diao, Quanping; Li, Tiechun; Liao, Peiqiu; Hou, Dongyan; Xin, Guang: FeCl3·6H2O-Catalyzed Tandem Alkylation–Hydrolysis Reaction of Chain α-Oxo Ketene Dithioacetals with Alcohols: Efficient ­Synthesis of α-Alkylated β-Oxo Thioesters
https://www.thieme-connect.de/media/synlett/EFirst/i_w0079_ga_10-1055_s0036-1588982.gif
Supporting Information

Publication Date: 10 April 2017

account

Amyes, Tina L.; Richard, John P.: Substituent Effects on Carbon Acidity in Aqueous Solution and at Enzyme Active Sites
https://www.thieme-connect.de/media/synlett/EFirst/i_a0092_ga_10-1055_s-0036-1588778.gif

letter

Ito, Takatoshi; Inoue, Yuta; Iwasawa, Tetsuo; Sumino, Shuhei; Matsumoto, Fukashi; Iwai, Toshiyuki; Moriwaki, Kazuyuki; Takao, Yuko; Mizuno, Takumi; Ohno, Toshinobu: Regioselective Synthesis of [6,6]-Phenyl-C71-Butyric Acid Methyl Esters via Sulfur Ylides for Use in Bulk Heterojunction Solar Cells
https://www.thieme-connect.de/media/synlett/EFirst/i_u0069_ga_10-1055_s-0036-1588770.gif
Supporting Information

letter

Jha, Ajit Kumar; Inani, Heena; Easwar, Srinivasan: A Nucleophilic Activation of Carboxylic Acids by Proline: Oxa-Michael Addition to Methyl Vinyl Ketone under Solvent-Free Conditions
https://www.thieme-connect.de/media/synlett/EFirst/i_b0090_ga_10-1055_s-0036-1588172.jpg
Supporting Information

letter

Khalaj, Mehdi; Ghazanfarpour-Darjani, Majid; Barat-Seftejani, Forugh; Nouri, Azita: Novel Catalytic Three-Component Reaction between a Terminal Alkyne, Sulfonyl Azide, and O-Methyl Oxime
https://www.thieme-connect.de/media/synlett/EFirst/i_d0070_ga_10-1055_s-0036-1588989.gif

Publication Date: 07 April 2017

letter

Zhu, Jia-Liang; Wu, Yung-Peng: Rhodium-Catalyzed Intramolecular Cyclopropanation of α-Diazo β-Keto Nitriles Containing an Unsaturated Substituted Cycloalkyl Group
https://www.thieme-connect.de/media/synlett/EFirst/i_w0103_ga_10-1055_s-0036-1588174.gif
Supporting Information

Publication Date: 06 April 2017

account

Du, Guangyan; Wang, Gaopeng; Ma, Wenjing; Yang, Qianqian; Bao, Wenli; Liang, Xuefeng; Zhu, Lizhi; Lee, Chi-Sing: Syntheses of Diverse Natural Products via Dual-Mode Lewis Acid Induced Cascade Cyclization Reactions
https://www.thieme-connect.de/media/synlett/EFirst/i_a0083_ga_10-1055_s-0036-1588777.gif

letter

Bananezhad, Behjat; Islami, Mohammad Reza: Stereoselective Synthesis of 3-(5-Benzoyl-1-methyl-1H-pyrrol-2-yl)-2-azetidinone Derivatives via an in Situ Generated Ketene
https://www.thieme-connect.de/media/synlett/EFirst/i_d0867_ga_10-1055_s-0036-1558974.gif
Supporting Information

Publication Date: 28 March 2017

cluster

Kwon, Ohhyeon; Esguerra, Kenneth Virgel N.; Glazerman, Michael; Petitjean, Laurène; Xu, Yalun; Ottenwaelder, Xavier; Lumb, Jean-Philip: Development of 3,5-Di-tert-butylphenol as a Model Substrate for Biomimetic Aerobic Copper Catalysis
https://www.thieme-connect.de/media/synlett/EFirst/i_r0048_ga_10-1055_s-0036-1588761.gif
Supporting Information

Publication Date: 21 March 2017

synpacts

Mousa, Reem; Reddy, Post Sai; Metanis, Norman: Chemical Protein Synthesis through Selenocysteine Chemistry
https://www.thieme-connect.de/media/synlett/EFirst/i_p0089_ga_10-1055_s-0036-1588762.gif

Publication Date: 20 March 2017

synpacts

Luan, Yi; Cong, Huan: Recent Synthetic Advances on π-Extended Carbon Nanohoops
https://www.thieme-connect.de/media/synlett/EFirst/i_p0002_ga_10-1055_s-0036-1588978.gif

Publication Date: 09 March 2017

cluster

He, Qiaoqiao; Qi, Yunkun; Liu, Chao; Li, Jiabin; Hu, Honggang: Synthesis of a Ubiquitinated Histone Mimic Bearing a New Thioether Linkage
https://www.thieme-connect.de/media/synlett/EFirst/i_w0047_ga_10-1055_s-0036-1588744.gif
Supporting Information

Publication Date: 08 March 2017

cluster

Shibuya, Masatoshi; Furukawa, Keisuke; Yamamoto, Yoshihiko: Selective Aerobic Oxidation of Primary Alcohols to Aldehydes
https://www.thieme-connect.de/media/synlett/EFirst/i_r0025_ga_10-1055_s-0036-1588155.gif
Supporting Information

cluster

Tanaka, Hirotaka; Oisaki, Kounosuke; Kanai, Motomu: Ligand-Free, Copper-Catalyzed Aerobic Benzylic sp3 C–H Oxygenation
https://www.thieme-connect.de/media/synlett/EFirst/i_r0042_ga_10-1055_s-0036-1588969.gif
Supporting Information

Publication Date: 28 February 2017

cluster

Singh, Atul K.; Yi, Hong; Zhang, Guoting; Bian, Changliang; Pei, Pengkun; Lei, Aiwen: Photoinduced Oxidative Cross-Coupling for O–S Bond Formation: A Facile Synthesis of Alkyl Benzenesulfonates
https://www.thieme-connect.de/media/synlett/EFirst/i_r0028_ga_10-1055_s-0036-1588728.gif
Supporting Information

Publication Date: 15 March 2013

letter

Fernandes, Rodney A.; Chavan, Vijay P.: A Concise Total Synthesis of (±)-Asteriscunolide C