Synlett

eFirst

• Accepted Manuscripts
• eFirst
• Issue
• Most Read

Publication Date: 24 April 2025

account

Kumar, Sundaravel Vivek; Guiry, Patrick J: Enantioselective Zinc-Catalyzed [3+2] Azomethine Ylide Cycloaddition: Developing Planar Chiral [2.2]Paracyclophane-Imidazoline N,O-Ligands

• Full Text
• HTML
• PDF (695 kb)

account

Paul, Suvam; Choudhuri, Tathagata; Das, Sourav; Sikdar, Papiya; Bagdi, Avik Kumar: Recent Advances in the Synthesis of Functionalized Pyrazolo[1,5-a]pyrimidines via C–H Functionalization

• Full Text
• HTML
• PDF (925 kb)

letter > Emerging Trends in Organic Chemistry: A Focus on India

Joshi, Ashish; Chavada, Lilesh Rambhai; Choudhary, Mridula; Patel, Dhruvilkumar; Mishra, Priyanka; Patil, Sneha; Sridhar, Balasubramanian; Singh, Saurabh Kumar; Pandey, Ashok Kumar: Synthesis of Cytogenin Analogues by C(sp²)–H Functionalization under Ruthenium(II) Catalysis, and DFT Analysis

• Full Text
• HTML
• PDF (1400 kb)

Supporting Information

letter > Emerging Trends in Organic Chemistry: A Focus on India

Yaragorla, Srinivasarao; Kumar, Avinash; Ali, Liyaqat: Regioselective Formal (3+2) Cyclization of Propargylic para-Quinone Methides (p-QMs) with β-Keto Carbonyls: Direct Access to (Fused)-Furans

• Full Text
• HTML
• PDF (1102 kb)

Supporting Information

Publication Date: 23 April 2025

account > Small Molecules in Medicinal Chemistry

Pal, Deepti; Yadav, Shruti; Verma, Abhishek Kumar; Maurya, Sushil K.: Recent Developments in the Synthesis of Triazoles and Their Applications in Antibacterial Drug Discovery

• Full Text
• HTML
• PDF (886 kb)

Publication Date: 22 April 2025

letter

Zhang, Jinlong; Huang, Zening; Zuo, Kaicheng; Zhang, Chengyang; Jiang, Gaoxi: Synthesis of Indolo[1,2-a]quinoxalines and 2-Arylquinazolinones by Oxidative Aromatization from Aromatic Aldehydes or Benzyl Alcohols

• Full Text
• HTML
• PDF (271 kb)

Supporting Information

perspectives > Small Molecules in Medicinal Chemistry

Goel, Kapil Kumar; Singhal, Peeush; Sathish, Elagandhula; Babu, M. Arockia; Pandey, Sarvesh Kumar; Tyagi, Yogita; Kumar, Roshan; Singh, Thakur Gurjeet; Puri, Sarthak: A Minireview on the Morpholine-Ring-Containing U.S. FDA Approved Drugs: A Medicinal-Chemistry-Based Analysis from 2013 to 2023

• Full Text
• HTML
• PDF (1618 kb)

Publication Date: 17 April 2025

letter > Emerging Trends in Organic Chemistry: A Focus on India

Mahato, Frenki; Ghosh, Asim Kumar; Hajra, Alakananda: Synthesis of Silylated Azauracil 1-Oxides by Metal-Free Direct Silylation

• Full Text
• HTML
• PDF (183 kb)

Supporting Information

Publication Date: 15 April 2025

letter > Small Molecules in Medicinal Chemistry

Beveridge, Julia; Söderström, Marcus; Balestri, Lorenzo Jacopo Ilic; Prieto-Díaz, Rubén; Gutierrez-de-Teran, Hugo; Odell, Luke R; Hallberg, Mathias; Larhed, Mats; Gising, Johan: Benzylhydroxamic Acids as IRAP Inhibitors: Sulfonamide Variations

• HTML
• PDF (665 kb)

Supporting Information

letter > Small Molecules in Medicinal Chemistry

Ito, Toshiya; Kinoshita, Kazutomo; Tomizawa, Masaki; Shinohara, Shojiro; Nishii, Hiroki; Tanaka, Hiroshi; Kuramoto, Shino; Oikawa, Nobuhiro: Development of a Novel Tropomyosin Receptor Kinase Inhibitor Based on Structure–Activity Relationships: Identification of a Promising Clinical Candidate

• Full Text
• HTML
• PDF (1850 kb)

Supporting Information

Publication Date: 14 April 2025

account

Zhang, Yuanyuan; Ding, Shuai; Meng, Limin; Tao, Chuanzhou; Wang, Huiyan; Xu, Song: Catalytic Enantioselective Friedel–Crafts Reactions of Arenes Enabled by Iranium/Irenium-Ion-Triggered Electrophilic Functionalization

• Full Text
• HTML
• PDF (887 kb)

letter > Hydrogen Atom Transfer Reactions

Fang, Yi; Fan, Pei; Wang, Chuan: Palladium/TBADT-Cocatalyzed Acyl C–H Alkenylation of Aldehydes with Alkenyl Triflates

• Full Text
• HTML
• PDF (230 kb)

Supporting Information

letter

Yazzaf, Rozita; Sayahi, Mohammad Hosein; Mahdavi, Mohammad: Potassium Carbonate Catalyzed Intramolecular Post-Ugi Hydroamination Reaction Leading to N-Aryl Piperazine Derivatives

• Full Text
• HTML
• PDF (162 kb)

Supporting Information

letter > First-Row Transition-Metal Catalysis for Organic Synthesis

Zhang, Zhaolun; Chen, Sanxia; Tian, Haitao; Tang, Conghui: Synthesis of Alkenyl Nitriles by Bidentate Cobalt-Catalyzed Acceptorless Dehydrogenation Coupling of Alcohols and Nitriles

• Full Text
• HTML
• PDF (281 kb)

Supporting Information

Publication Date: 11 April 2025

letter

Ma, Shi-Wei; Huang, Jin; Ma, Long-jun; Li, Guang-xun: One-Pot Efficient Synthesis of Sulfonimidamides from Sulfonyl Chloride

• Full Text
• HTML
• PDF (281 kb)

Supporting Information

letter

Wang, Yan; Wang, Zongkang; Fei, Nana; He, Peng; Kong, Lingkai; Li, Yanzhong: Synthesis of Pyrano[2,3-b]indol-4-ones Fused with Medium-Sized Rings: A Base-Induced C–C σ-Bond Insertion and Subsequent I₂-Mediated 1,2-Acyl Migration/Cyclization Reaction

• Full Text
• HTML
• PDF (236 kb)

Supporting Information

synpacts

Bayer, Eva A.; Sekiguchi, Yoshiya; Onnuch, Polpum; Liu, Richard Y.: ‘Ring-Walking’ Aryl Cross-Coupling Reactions Involving Palladium Aryne Intermediates

• Full Text
• HTML
• PDF (202 kb)

Publication Date: 10 April 2025

letter > Hydrogen Atom Transfer Reactions

Chi, Zhiyong; Huang, Siyuan; Tang, Guo; Zhao, Qianyi; Gong, Lei: Visible-Light-Induced Hydrogen-Atom-Transfer Catalysis for the Regioselective Hydroacylation of N-Sulfonylimine Esters with Aldehydes

• Full Text
• HTML
• PDF (352 kb)

Supporting Information CIF File

letter > Emerging Trends in Organic Chemistry: A Focus on India

Nookaraju, U.; Danve, Shivam S.; Kumar, Pradeep: Tetrahydrofuran Ring Construction through Tandem Iodocyclizations: Synthesis of Hagen’s Gland Lactones, a Pheromone of Idea leuconoe, an Oxylipid, and Related Compounds

• Full Text
• HTML
• PDF (206 kb)

Supporting Information

letter

Stell, Matthew; Sandoval, Marissa; Ramirez, Santiago; Darragh, Kathy; Schulz, Stefan: A Simplified Synthesis of HNDB (Albiducin A) and Calidiol A

• Full Text
• HTML
• PDF (273 kb)

Supporting Information Movie File

Show more