DOI: 10.1055/s-00000083

Synlett

eFirst

Publication Date: 25 September 2017

letter

Khan, Raysa; Felix, Robert; Kemmitt, Paul D.; Coles, Simon J.; Tizzard, Graham J.; Spencer, John: N1-Arylation of 1,4-Benzodiazepine-2-ones with Diaryliodonium Salts
https://www.thieme-connect.de/media/synlett/EFirst/i_d0556_ga_10-1055_s-0036-1590920.gif
Supporting Information

Publication Date: 21 September 2017

letter

Chernichenko, Nataliya M.; Shevchuk, Vadim N.; Averin, Alexei D.; Maloshitskaya, Olga A.; Beletskaya, Irina P.: Synthesis of Dansyl-Substituted Cryptands Containing Triaza­cycloalkane Moieties and their Evaluation as Fluorescent Chemosensors
https://www.thieme-connect.de/media/synlett/EFirst/i_r0525_ga_10-1055_s-0036-1590883.gif
Supporting Information

letter

Gorepatil, Amarsinha; Gorepatil, Pratapsinha; Gaikwad, Mahadev; Mhamane, Dattakumar; Phadkule, Ajit; Ingle, Vilas: Zirconyl Nitrate as an Efficient Catalyst for Facile Synthesis of 2-Aryl-2,3-dihydroquinolin-4(1H)-one Derivatives in Aqueous ­Medium
https://www.thieme-connect.de/media/synlett/EFirst/i_d0585_ga_10-1055_s-0036-1589110.gif

letter

Irwin, Lauren C.; Kerr, Michael A.: One-Pot Michael Addition/Radical Cyclization Reaction of N-Acryloyl Indoles
https://www.thieme-connect.de/media/synlett/EFirst/i_r0529_ga_10-1055_s-0036-1589105.gif
Supporting Information

letter

Mangaonkar, Saeesh R.; Kole, Priyanka B.; Singh, Fateh V.: Oxidation of Organosulfides to Organosulfones with Trifluoromethyl 3-Oxo-1λ3,2-benziodoxole-1(3H)-carboxylate as an Oxidant
https://www.thieme-connect.de/media/synlett/EFirst/i_d0596_ga_10-1055_s-0036-1588575.gif
Supporting Information

letter

Obst, Martin; Srivastava, Akriti; Baskaran, Sundarababu; König, Burkhard: Preparation of Propargyl Amines in a ZnCl2–Dimethylurea Deep-Eutectic Solvent
https://www.thieme-connect.de/media/synlett/EFirst/i_b0580_ga_10-1055_s-0036-1588571.gif
Supporting Information

Publication Date: 19 September 2017

letter

Jiang, Xinpeng; Liu, Yong; Zhang, Lei; Chen, Jinkang; Cheng, Kang; Yu, Chuanming: Palladium-Catalyzed Allylation of Polyfluoroarenes with Allylic Pivalates
https://www.thieme-connect.de/media/synlett/EFirst/i_w0541_ga_10-1055_s-0036-1590914.gif
Supporting Information

letter

Talaei, Bahareh; Heravi, Majid M.; Oskooie, Hossein A.; Rezvanian, Atieh: An Approach to the Diastereoselective Synthesis of Cyclohexane-1,3-dicarboxamide Derivatives via a Pseudo Five-Component ­Reaction Based on Diketene
https://www.thieme-connect.de/media/synlett/EFirst/i_d0523_ga_10-1055_s-0036-1590980.gif
Supporting Information

Publication Date: 15 September 2017

letter

Adib, Mehdi; Pashazadeh, Rahim: TBHP/n-Bu4PBr-Promoted Oxidative Cross-Dehydrogenative Coupling of Aryl Methanols: A Facile Synthesis of Symmetrical Carboxylic Anhydride Derivatives
https://www.thieme-connect.de/media/synlett/EFirst/i_d0480_ga_10-1055_s-0036-1590905.jpg
Supporting Information

letter

Khalaj, Mehdi; Taherkhani, Mahboubeh; Mousavi-Safavi, Seyed Mahmoud; Akbari, Jafar: Synthesis of Benzamide Derivatives by the Reaction of Arenes and Isocyanides through a C–H Bond Activation Strategy
https://www.thieme-connect.de/media/synlett/EFirst/i_d0550_ga_10-1055_s-0036-1588565.gif

Publication Date: 14 September 2017

account

Liu, Wenbo; Li, Chao-Jun: Recent Synthetic Applications of Catalyst-Free Photochemistry
https://www.thieme-connect.de/media/synlett/EFirst/i_r0490_ga_10-1055_s-0036-1590900.gif

cluster

Tang, Jinghua; Luo, Meiming; Zeng, Xiaoming: Chromium-Catalyzed, Regioselective Cross-Coupling of C–O Bonds by Using Organic Bromides as Reactants
https://www.thieme-connect.de/media/synlett/EFirst/i_s0536_ga_10-1055_s-0036-1588568.gif
Supporting Information

letter

Bhagat, Ujjawal Kumar; Peddinti, Rama Krishna: Regiospecific Aza-Michael Addition of 4-Aryl-1H-1,2,3-triazoles to Chalcones: Synthesis of 2,4-Disubstituted 1,2,3-Triazoles in Basic Medium
https://www.thieme-connect.de/media/synlett/EFirst/i_d0572_ga_10-1055_s-0036-1588567.gif
Supporting Information

letter

Ji, Yuan; Zhong, Ning; Kang, Zinan; Yan, Guobing; Zhao, Ming: Synthesis of Internal Alkynes through an Effective Tandem ­Elimination–Hydrodebromination–Cross-Coupling of gem-­Dibromoalkenes with Halobenzenes
https://www.thieme-connect.de/media/synlett/EFirst/i_w0486_ga_10-1055_s-0036-1590907.gif
Supporting Information

letter

Ying, Wei-Wei; Zhu, Wen-Ming; Liang, Hongze; Wei, Wen-Ting: Synthesis of Indoline-2,3-diones by Radical Coupling of Indolin-2-ones with tert-Butyl Hydroperoxide
https://www.thieme-connect.de/media/synlett/EFirst/i_w0574_ga_10-1055_s-0036-1589106.gif
Supporting Information

Publication Date: 13 September 2017

account

Prabagar, B.; Ghosh, Nayan; Sahoo, Akhila K.: Cyclization and Cycloisomerization of π-Tethered Ynamides: An Expedient Synthetic Method to Construct Carbo- and Heterocycles
https://www.thieme-connect.de/media/synlett/EFirst/i_a0397_ga_10-1055_s-0036-1590877.gif

Publication Date: 12 September 2017

synpacts

Hu, Jiadong; Yu, Xin; Xie, Weiqing: New Strategy for Forging Contiguous Quaternary Carbon Centers via H2O2-Mediated Ring Contraction
https://www.thieme-connect.de/media/synlett/EFirst/i_p0581_ga_10-1055_s-0036-1590979.gif

Publication Date: 05 September 2017

account

Bull, James A.; Degennaro, Leonardo; Luisi, Renzo: Straightforward Strategies for the Preparation of NH-Sulfox­imines: A Serendipitous Story
https://www.thieme-connect.de/media/synlett/EFirst/i_a0415_ga_10-1055_s-0036-1590874.gif

cluster

Bo, Yingjian; Sieburth, Scott McN.: A Quantitative NMR Method for Silyllithium Analysis
https://www.thieme-connect.de/media/synlett/EFirst/i_b0517_ga_10-1055_s-0036-1590902.gif
Supporting Information

letter

Balalaie, Saeed; Derakhshan-Panah, Fatemeh; Zolfigol, Mohammad Ali; Rominger, Frank: A Convenient Method for the Synthesis of Imidazo[1,2-a]pyridines with a New Approach
https://www.thieme-connect.de/media/synlett/EFirst/i_d0543_ga_10-1055_s-0036-1590906.gif
Supporting Information

Publication Date: 01 September 2017

letter

Ma, Zhi-Xiong; Fang, Li-Chao; Haugen, Bryan J.; Bruckbauer, Daniel; Feltenberger, John B.; Hsung, Richard P.: Facile Synthesis of 3-Amido-Dienynes via a Tandem α-Propargylation–Isomerization of Chiral Allenamides and their Applications in Diels–Alder Cycloadditions
https://www.thieme-connect.de/media/synlett/EFirst/i_r0444_ga_10-1055_s-0036-1590899.gif
Supporting Information

letter

Piras, Monica; Andriu, Alexandra; Testa, Andrea; Wienecke, Paul; Fleming, Ian N.; Zanda, Matteo: Design and Synthesis of an RGD Peptidomimetic-Paclitaxel Conjugate Targeting αvβ3 Integrin for Tumour-Directed Drug Delivery
https://www.thieme-connect.de/media/synlett/EFirst/i_r0479_ga_10-1055_s-0036-1590898.gif
Supporting Information

Publication Date: 31 August 2017

account

Husain, Syed Masood; Müller, Michael: Fungal Dihydroxynaphthalene-Melanin: Diversity-Oriented Biosynthesis through Enzymatic and Non-enzymatic Transformations
https://www.thieme-connect.de/media/synlett/EFirst/i_a0382_ga_10-1055_s-0036-1588526.gif

letter

Mohr, Lisa-Marie; Bach, Thorsten: Intermolecular [2+2] Photocycloaddition of β-Nitrostyrenes to Olefins upon Irradiation with Visible Light
https://www.thieme-connect.de/media/synlett/EFirst/i_r0492_ga_10-1055_s-0036-1588524.gif
Supporting Information Primary Data

Publication Date: 30 August 2017

cluster

De, Chandra Kanta; Mitra, Raja; List, Benjamin: Design and Synthesis of Enantiopure Tetrakis(pentafluorophenyl) Borate Analogues for Asymmetric Counteranion Directed Catalysis
https://www.thieme-connect.de/media/synlett/EFirst/i_d0462_ga_10-1055_s-0036-1590903.gif

letter

Hofmayer, Maximilian S.; Hammann, Jeffrey M.; Cahiez, Gérard; Knochel, Paul: Iron-Catalyzed C(sp2)–C(sp3) Cross-Coupling Reactions of Di(hetero)arylmanganese Reagents and Primary and Secondary Alkyl Halides
https://www.thieme-connect.de/media/synlett/EFirst/i_b0542_ga_10-1055_s-0036-1590891.gif
Supporting Information

Publication Date: 29 August 2017

letter

Ouyang, Banlai; Liu, Deming; Xia, Kejian; Zheng, Yanxia; Mei, Hongxin; Qiu, Guanyinsheng: Synthesis of N-Arylsulfonamides by a Copper-Catalyzed Reaction of Chloramine-T and Arylboronic Acids at Room Temperature
https://www.thieme-connect.de/media/synlett/EFirst/i_w0473_ga_10-1055_s-0036-1590978.gif
Supporting Information

letter

Yamasaki, Naoto; Kanno, Marina; Sakamoto, Kyohei; Kasai, Yusuke; Imagawa, Hiroshi; Yamamoto, Hirofumi: m-C2B10H11HgCl/AgOTf-Catalyzed Reaction for Reductive Deoxygenation
https://www.thieme-connect.de/media/synlett/EFirst/i_u0535_ga_10-1055_s-0036-1588554.gif
Supporting Information

Publication Date: 28 August 2017

letter

Muddam, Bhooshan; Venkanna, P.; Venkateswarlu, M.; Satish Kumar, M.; Rajanna, K. C.: Symmetrical Trichlorotriazine Derivatives as Efficient Reagents for One-Pot Synthesis of 3-Acetyl-2-chloroquinolines from Acetanilides under Vilsmeier–Haack Conditions
https://www.thieme-connect.de/media/synlett/EFirst/i_d0454_ga_10-1055_s-0036-1589099.gif
Supporting Information

Publication Date: 25 August 2017

cluster

Cornelissen, Loïc; Nagy, Audric; Leyssens, Tom; Riant, Olivier: Tetrabutylammonium Bifluoride as an Efficient Activating Agent for Copper-Catalyzed Vinylsilane Cross-Coupling Reactions
https://www.thieme-connect.de/media/synlett/EFirst/i_b0337_ga_10-1055_s-0036-1588504.gif
Supporting Information

cluster

Igawa, Kazunobu; Kuroo, Akihiro; Yoshihiro, Daisuke; Yamanaka, Yuki; Tomooka, Katsuhiko: Synthesis of Stereoselectively Functionalized Silacyclopentanes
https://www.thieme-connect.de/media/synlett/EFirst/i_b0368_ga_10-1055_s-0036-1590826.gif
Supporting Information

cluster

Yang, Ze-Kun; Wang, Chao; Uchiyama, Masanobu: DFT Studies Provide Mechanistic Insight into Nickel-Catalyzed Cross-Coupling Involving Organoaluminum-Mediated C–O Bond Cleavage
https://www.thieme-connect.de/media/synlett/EFirst/i_s0411_ga_10-1055_s-0036-1590863.gif
Supporting Information

letter

Chui, Tin-Ki; Chow, Hak-Fun: New Triazole-Containing Branched Bis(dipeptidomimetic) – Switching from Self-Dimerization to Anion-Binding Properties
https://www.thieme-connect.de/media/synlett/EFirst/i_r0531_ga_10-1055_s-0036-1590884.gif
Supporting Information

letter

Ramadhar, Timothy R.; Kawakami, Jun-ichi; Batey, Robert A.: Sequential O-Arylation/Lanthanide(III)-Catalyzed [3,3]-Sigmatropic Rearrangement of Bromo-Substituted Allylic Alcohols
https://www.thieme-connect.de/media/synlett/EFirst/i_r0540_ga_10-1055_s-0036-1590890.gif
Supporting Information

letter

Ren, Zhi-Lin; Sun, Mei; Guan, Zhi-Rong; Ding, Ming-Wu: New Efficient Synthesis of 1,2,4-Trisubstituted Furans by a ­Sequential Passerini/Wittig/Isomerization Reaction Starting from Baylis–Hillman β-Bromo Aldehydes
https://www.thieme-connect.de/media/synlett/EFirst/i_w0460_ga_10-1055_s-0036-1588564.gif
Supporting Information

letter

Salvanna, N.; Reddy, P. Raghavendar; Das, Biswanath: Palladium-Catalyzed Cross-Coupling of 1,3,4-Oxadiazoles and Styrenes: An Efficient Method to Synthesize 2-Alkenyl-1,3,4- Oxadiazoles§
https://www.thieme-connect.de/media/synlett/EFirst/i_d0511_ga_10-1055_s-0036-1588561.gif

letter

Yavari, Issa; Amirahmadi, Asiyeh; Halvagar, Mohammad Reza: A Synthesis of Functionalized Thiazoles and Pyrimidine-4(3H)-thiones from 1,1,3,3-Tetramethylguanidine, Acetylenic Esters, and Aryl Isothiocyanates
https://www.thieme-connect.de/media/synlett/EFirst/i_d0327_ga_10-1055_s-0036-1590862.gif
Supporting Information

synpacts

Zhang, Ze-Xin; Chen, Si-Cong; Jiao, Lei: Asymmetric Total Synthesis of (+)-Minfiensine by an Asymmetric Cascade Cyclization Strategy
https://www.thieme-connect.de/media/synlett/EFirst/i_p0404_ga_10-1055_s-0036-1589075.gif

Publication Date: 24 August 2017

letter

Joo, Seong-Ryu; Youn, Young-Jin; Hwang, Young-Ran; Kim, Seung-Hoi: Highly Active Manganese-Mediated Acylation of Alcohols with Acid Chlorides or Anhydrides
https://www.thieme-connect.de/media/synlett/EFirst/i_u0429_ga_10-1055_s-0036-1590973.gif

Publication Date: 23 August 2017

letter

Gao, Ang; Liu, Xiu-Yan; Ding, Chang-Hua; Hou, Xue-Long: Diastereoselective Palladium-Catalyzed Conjugate Addition of Arylboronic Acids to α-Substituted Cyclic Enones
https://www.thieme-connect.de/media/synlett/EFirst/i_r0385_ga_10-1055_s-0036-1590742.gif
Supporting Information

letter

Hurtak, Jessica A.; McDonald, Frank E.: Regioselectivity of Mercury-Promoted Oxacyclizations of Alkynyl Diols
https://www.thieme-connect.de/media/synlett/EFirst/i_r0506_ga_10-1055_s-0036-1588562.gif
Supporting Information

letter

Jia, Zhi-Jun; Merten, Christian; Knauer, Lena; Murarka, Sandip; Strohmann, Carsten; Waldmann, Herbert: Biology-Oriented Synthesis of Decahydro-4,8-epoxyazulene Scaffolds
https://www.thieme-connect.de/media/synlett/EFirst/i_r0463_ga_10-1055_s-0036-1588558.gif
Supporting Information

letter

Papatzimas, James W.; Gorobets, Evgueni; Brownsey, Duncan K.; Maity, Ranjan; Bahlis, Nizar J.; Derksen, Darren J.: A General Strategy for the Preparation of Thalidomide-Conjugate Linkers
https://www.thieme-connect.de/media/synlett/EFirst/i_r0401_ga_10-1055_s-0036-1588539.gif
Supporting Information

Publication Date: 22 August 2017

account

Paraja, Miguel; Plaza, Manuel; Valdés, Carlos: Transition-Metal-Free Reactions Between Boronic Acids and N-Sulfonylhydrazones or Diazo Compounds: Reductive Coupling Processes and Beyond
https://www.thieme-connect.de/media/synlett/EFirst/i_a0494_ga_10-1055_s-0036-1590868.gif

letter

Liu, Wenjie; Wang, Shaohua; Cai, Zhihao; Li, Ziying; Liu, Jianwen; Wang, Anda: Iodine-Catalyzed Regioselective Sulfenylation of 4H-Pyrido[1,2-a]pyrimidin-4-ones with Sulfonyl Hydrazides
https://www.thieme-connect.de/media/synlett/EFirst/i_w0478_ga_10-1055_s-0036-1588549.gif
Supporting Information

letter

Morozzi, Chiara; Rosati, Ornelio; Curini, Massimo; Lanari, Daniela: A Solvent-Free Reaction for Silyl Enol Ethers Synthesis
https://www.thieme-connect.de/media/synlett/EFirst/i_b0386_ga_10-1055_s-0036-1590876.gif
Supporting Information

letter

Narayanappa, Arkesh; Hurem, David; McNulty, James: Regioselective Ylide Formation on Acetal-Functionalized Trialkyl Phosphonium Salts: Extending the Scope of Carbonyl Homologation
https://www.thieme-connect.de/media/synlett/EFirst/i_r0528_ga_10-1055_s-0036-1588551.gif
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letter

Qian, Hua; Gu, Guoxian; Zhou, Qinghai; Lu, Jiaxiang; Chung, Lung Wa; Zhang, Xumu: Enantioselective Palladium-Catalyzed Decarboxylative Allylation of β-Keto Esters Assisted by a Thiourea
https://www.thieme-connect.de/media/synlett/EFirst/i_w0477_ga_10-1055_s-0036-1590869.gif
Supporting Information

letter

Sommer, Heiko; Braun, Max; Schröder, Benjamin; Kirschning, Andreas: 4-Ethoxy-1,1,1-trifluoro-3-buten-2-one (ETFBO), a Versatile Precursor for Trifluoromethyl-Substituted Heteroarenes – a Short Synthesis of Celebrex® (Celecoxib)
https://www.thieme-connect.de/media/synlett/EFirst/i_b0101_ga_10-1055_s-0036-1589097.gif
Supporting Information

letter

Wang, Tao; Oswood, Christian J.; Hoye, Thomas R.: Trapping of Hexadehydro-Diels–Alder Benzynes with Exocyclic, Conjugated Enals as a Route to Fused Spirocyclic Benzopyran Motifs
https://www.thieme-connect.de/media/synlett/EFirst/i_r0467_ga_10-1055_s-0036-1589091.gif
Supporting Information

letter

Zhang, Xiao; Huang, Binbin; Yang, Chao; Xia, Wujiong: Photoinduced Regioselective Lactonization of ortho-Iodobenzoic Acids with Alkenes: Synthesis of 3,4-Dihydroisocoumarin Derivatives
https://www.thieme-connect.de/media/synlett/EFirst/i_w0461_ga_10-1055_s-0036-1588541.gif
Supporting Information

synpacts

Jeon, Sangbin; Park, Joonoh; Han, Sunkyu: Syntheses of Dimeric Securinega Alkaloids
https://www.thieme-connect.de/media/synlett/EFirst/i_p0455_ga_10-1055_s-0036-1590864.gif

synpacts

Mitra, Nirmal K.; Merryman, Caroline P.; Merner, Bradley L.: Highly Strained para-Phenylene-Bridged Macrocycles from Unstrained 1,4-Diketo Macrocycles
https://www.thieme-connect.de/media/synlett/EFirst/i_p0417_ga_10-1055_s-0036-1589081.gif

Publication Date: 21 August 2017

letter

Barraza, Scott J.; Denmark, Scott E.: Unexpected Rearrangement of 2-Bromoaniline under Biphasic Alkylation Conditions
https://www.thieme-connect.de/media/synlett/EFirst/i_r0502_ga_10-1055_s-0036-1590882.gif
Supporting Information

letter

Emberson, Kassandra; Tran, Ngan; Metallinos, Costa: Diastereoselective Lithiation of N-Benzyl Pyrroloimidazolones Derived from l-Proline Hydantoin
https://www.thieme-connect.de/media/synlett/EFirst/i_r0443_ga_10-1055_s-0036-1591206.gif
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letter

Isbrandt, Eric S.; Vandavasi, Jaya Kishore; Zhang, Wanying; Jamshidi, Mohammad P.; Newman, Stephen G.: Catalytic Deuteration of Aldehydes with D2O
https://www.thieme-connect.de/media/synlett/EFirst/i_r0495_ga_10-1055_s-0036-1588540.gif
Supporting Information

letter

Labes, Ricardo; González-Calderón, Davir; Battilocchio, Claudio; Mateos, Carlos; Cumming, Graham R.; de Frutos, Oscar; Rincón, Juan A.; Ley, Steven V.: Rapid Continuous Ruthenium-Catalysed Transfer Hydrogenation of Aromatic Nitriles to Primary Amines
https://www.thieme-connect.de/media/synlett/EFirst/i_r0508_ga_10-1055_s-0036-1589096.gif
Supporting Information

Publication Date: 17 August 2017

cluster

Yasui, Kosuke; Higashino, Masaya; Chatani, Naoto; Tobisu, Mamoru: Rhodium-Catalyzed Reductive Cleavage of Aryl Carbamates Using Isopropanol as a Reductant
https://www.thieme-connect.de/media/synlett/EFirst/i_s0413_ga_10-1055_s-0036-1589093.gif
Supporting Information

letter

Aeyad, Tahani; Williams, Jason D.; Meijer, Anthony J. H. M.; Coldham, Iain: Lithiation–Substitution of N-Boc-2-phenylazepane
https://www.thieme-connect.de/media/synlett/EFirst/i_r0412_ga_10-1055_s-0036-1590857.gif
Supporting Information

letter

Afsar, Ashfaq; Cowell, Joseph; Distler, Petr; Harwood, Laurence M.; John, Jan; Westwood, James: Synthesis of Novel BTPhen-Functionalized Silica-Coated Magnetic Nanoparticles for Separating Trivalent Actinides and Lanthanides
https://www.thieme-connect.de/media/synlett/EFirst/i_r0433_ga_10-1055_s-0036-1590865.gif
Supporting Information

letter

Banan, Alireza; Valizadeh, Hassan; Heydari, Akbar; Moghimi, Abolghasem: Selective Oxidation of Secondary Amines to N,N-Disubstituted Hydroxylamines by Choline Peroxydisulfate
https://www.thieme-connect.de/media/synlett/EFirst/i_d0281_ga_10-1055_s-0036-1589089.gif
Supporting Information

letter

Calvo, Beatriz C.; Minnaard, Adriaan J.: Copper-Catalyzed Asymmetric 1,2-Addition of Grignard Reagents to 3-Acyl 2H-chromenes
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Supporting Information

letter

Chaabouni, S.; Pinkerton, N. M.; Abid, S.; Galaup, C.; Chassaing, S.: Photochemistry of ortho-Azidocinnamoyl Derivatives: Facile and Modular Synthesis of 2-Acylated Indoles and 2-Substituted Quinolines under Solvent Control
https://www.thieme-connect.de/media/synlett/EFirst/i_d0321_ga_10-1055_s-0036-1590861.gif
Supporting Information

letter

Chittimalla, Santhosh Kumar; Nakka, Srinuvasu; Koodalingam, Manikandan; Bandi, Chennakesavulu: N-Arylation of Heterocycles by a Tandem Aza-Michael Addition Reaction and Aromatization Sequence
https://www.thieme-connect.de/media/synlett/EFirst/i_b0426_ga_10-1055_s-0036-1588538.gif
Supporting Information

letter

Gao, Ke; Yamamoto, Keita; Nogi, Keisuke; Yorimitsu, Hideki: Palladium-Catalyzed Arylation of Benzylic C–H Bonds of Azaarylmethanes with Aryl Sulfides
https://www.thieme-connect.de/media/synlett/EFirst/i_r0514_ga_10-1055_s-0036-1589098.gif
Supporting Information

letter

Jopp, Stefan; Liesegang, Marko; Ehlers, Peter; Frank, Eva; Schneider, Gyula; Wölfling, János; Villinger, Alexander; Langer, Peter: Palladium-Catalysed Sonogashira Reactions of 16-(Hydroxymethylidene)-3-methoxy-α-estrone
https://www.thieme-connect.de/media/synlett/EFirst/i_d0422_ga_10-1055_s-0036-1588537.gif
Supporting Information

letter

Liang, Honggang; Bao, Lingxiang; Du, Yao; Zhang, Yiying; Pang, Siping; Sun, Chenghui: Synthesis of Cyanamides from Cyanogen Bromide under Mild Conditions through N-Cyanation of Allylic Tertiary Amines
https://www.thieme-connect.de/media/synlett/EFirst/i_w0431_ga_10-1055_s-0036-1588533.gif
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letter

Mandal, Samir K.; Sarkar, Apurba; Chakraborty, Puskin; Chattopadhyay, Ashoke P.: Synthetic Studies Towards the Synthesis of 6-Substituted 3-Fluoro-5,6-dihydropyran-2-ones
https://www.thieme-connect.de/media/synlett/EFirst/i_d0518_ga_10-1055_s-0036-1588534.gif
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letter

Onge, Brent St.; Green, James R.: Nicholas Reactions of Alkynyl- and Alkenyltrifluoroborates
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Supporting Information

letter

Tanwar, Dinesh Kumar; Surendrabhai, Vaghela Ravikumar; Gill, Manjinder Singh: An Efficient and Practical Process for the Synthesis of Glimepiride
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Supporting Information

letter

Xu, Lanting; Tan, Lushi; Ma, Dawei: Rhodium-Catalyzed Regioselective C7-Functionalization of Indole Derivatives with Acrylates by Using an N-Imino Directing Group
https://www.thieme-connect.de/media/synlett/EFirst/i_r0441_ga_10-1055_s-0036-1588530.gif
Supporting Information

synpacts

Jacobse, Peter H.; Moret, Marc-Etienne; Klein Gebbink, Robertus J. M.; Swart, Ingmar: Tracking On-Surface Chemistry with Atomic Precision
https://www.thieme-connect.de/media/synlett/EFirst/i_p0425_ga_10-1055_s-0036-1590867.jpg

Publication Date: 16 August 2017

cluster

Moyer, Brandon S.; Gagné, Michel R.: Taming Silylium Ions for Synthesis: N-Heterocycle Synthesis via Stereoselective C–C Bond Formation
https://www.thieme-connect.de/media/synlett/EFirst/i_b0339_ga_10-1055_s-0036-1590967.gif
Supporting Information

letter

Corbett, Michael T.; Caille, Seb: A Bench-Stable Vilsmeier Reagent for in situ Alcohol Activation: Synthetic Application in the Synthesis of 2-Amino-2-Thiazolines
https://www.thieme-connect.de/media/synlett/EFirst/i_r0476_ga_10-1055_s-0036-1589086.gif
Supporting Information

Publication Date: 14 August 2017

letter

Cooze, Christopher; Manchoju, Amarender; Pansare, Sunil V.: Synthesis of (–)-Muricatacin and (–)-(R,R)-L-Factor Involving an Organocatalytic Direct Vinylogous Aldol Reaction
https://www.thieme-connect.de/media/synlett/EFirst/i_r0466_ga_10-1055_s-0036-1590858.gif
Supporting Information

letter

Wang, Qing-Dong; Zhou, Bin; Yang, Jin-Ming; Fang, Dong; Ren, Jiangmeng; Zeng, Bu-Bing: Iron-Catalyzed C3-Formylation of Indoles with Formaldehyde and Aqueous Ammonia under Air
https://www.thieme-connect.de/media/synlett/EFirst/i_w0388_ga_10-1055_s-0036-1589079.gif
Supporting Information

Publication Date: 11 August 2017

letter

Dos Santos, Aurélie; Cordier, Marie; El Kaïm, Laurent: Nef–Perkow–Mumm Cascade towards Imido Phosphate Derivatives
https://www.thieme-connect.de/media/synlett/EFirst/i_d0375_ga_10-1055_s-0036-1590856.gif
Supporting Information

letter

Matsuo, Yosuke; Oowatashi, Ryosuke; Saito, Yoshinori; Tanaka, Takashi: Nonenzymatic Biomimetic Synthesis of Black Tea Pigment Theaflavins
https://www.thieme-connect.de/media/synlett/EFirst/i_u0442_ga_10-1055_s-0036-1588529.gif
Supporting Information

letter

Singh, Amandeep; Shalini; Kaur, Harleen; Sharma, Palak; Anand, Amit; Kumar, Vipan: β-Lactam-Synthon-Interceded Metal/Acid-Free Diastereoselective Access to Highly Functionalized Oxazol-5-ones and Dihydroimidazoles
https://www.thieme-connect.de/media/synlett/EFirst/i_d0380_ga_10-1055_s-0036-1588531.gif
Supporting Information

Publication Date: 08 August 2017

account

Davies, Stephen G.; Fletcher, Ai M.; Roberts, Paul M.; Thomson, James E.: Asymmetric Synthesis of Pyrrolizidines, Indolizidines and Quinolizidines via a Double Reductive Cyclisation Protocol
https://www.thieme-connect.de/media/synlett/EFirst/i_r0464_ga_10-1055_s-0036-1590975.gif

letter

Fahandej-Sadi, Anis; Lundgren, Rylan J.: Copper-Mediated Synthesis of Monofluoro Aryl Acetates via Decarboxylative Cross-Coupling
https://www.thieme-connect.de/media/synlett/EFirst/i_r0405_ga_10-1055_s-0036-1588516.gif
Supporting Information

letter

Kobayashi, Yuichi; Saeki, Ryohei; Nanba, Yutaro; Suganuma, Yuta; Morita, Masao; Nishimura, Keita: Synthesis of the Verapamil Intermediate through the Quaternary Carbon-Constructing Allylic Substitution
https://www.thieme-connect.de/media/synlett/EFirst/i_u0341_ga_10-1055_s-0036-1588518.gif
Supporting Information

letter

Ng, Wing Hin; Shing, Tony K. M.; Yeung, Ying-Yeung: Mild and Efficient Vicinal Dibromination of Olefins Mediated by Aqueous Ammonium Fluoride
https://www.thieme-connect.de/media/synlett/EFirst/i_w0372_ga_10-1055_s-0036-1588506.gif
Supporting Information

letter

Nguyen, Thi Ha; Ma, Eunsook: Chemoselective Synthesis of N-(Aminoalkyl/amidino)phenyl Naphthalene-1-carboxamides and 5,6,7,8-Tetrahydronaphthalene-1-carboxamides and Their Anticoagulant Screening
https://www.thieme-connect.de/media/synlett/EFirst/i_u0359_ga_10-1055_s-0036-1588517.gif
Supporting Information

letter

Wang, Liangguang; Ma, Juan; Chen, Xia; Zhou, Xiaoyu: Synthesis of Enaminones by a Palladium-Catalyzed Four-Component Carbonylative Addition Reaction
https://www.thieme-connect.de/media/synlett/EFirst/i_w0436_ga_10-1055_s-0036-1590976.gif
Supporting Information

letter

Yamamoto, Yasutomo; Yamaguchi, Tatsuya; Kaneshige, Atsunori; Hashimoto, Aiko; Kaibe, Sachiho; Miyawaki, Akari; Yamada, Ken-ichi; Tomioka, Kiyoshi: Consecutive Aminolithiation–Carbolithiation of a Linear Aminoalkene Bearing Terminal Vinyl Sulfide Moiety to Give Hydro­indolizine
https://www.thieme-connect.de/media/synlett/EFirst/i_r0445_ga_10-1055_s-0036-1588522.gif
Supporting Information

Publication Date: 04 August 2017

letter

Qiao, Shuo; Wu, Jianbin; Mo, Junming; Spigener, Preston T.; Zhao, Brian Nlong; Jiang, Bo; Li, Guigen: Chiral Phosphinyl Enamines and Their Asymmetric Reduction through Group-Assisted Purification Chemistry Leading to Enantiopure β-Amino Esters/Amides
https://www.thieme-connect.de/media/synlett/EFirst/i_b0353_ga_10-1055_s-0036-1589080.gif
Supporting Information CIF File

Publication Date: 03 August 2017

letter

Dileep, Kommula; Murty, M. S. R.: Aqueous, One-Pot, Three-Component Reaction for Efficient Synthesis of 2-[4-(Arylsulfonyl)piperazin-1-yl]-1,3-benzothiazole, ‑1H-benzimidazole, or -1,3-benzoxazole Derivatives
https://www.thieme-connect.de/media/synlett/EFirst/i_d0360_ga_10-1055_s-0036-1590972.gif
Supporting Information

letter

Lapinskaite, Ringaile; Ghavre, Mukund; Rintelmann, Chelsea L.; Bedard, Korey; Dela Paz, Helen E.; Hudlicky, Tomas: Chemoenzymatic Formal Total Synthesis of Pancratistatin from Narciclasine-Type Compounds via Myers Transposition: Model Study for a Short Conversion of Narciclasine to Pancratistatin
https://www.thieme-connect.de/media/synlett/EFirst/i_r0439_ga_10-1055_s-0036-1588515.gif
Supporting Information

letter

Tanwar, Dinesh Kumar; Ratan, Anjali; Gill, Manjinder Singh: Facile One-Pot Synthesis of Substituted Hydantoins from Carbamates
https://www.thieme-connect.de/media/synlett/EFirst/i_d0256_ga_10-1055_s-0036-1588468.gif
Supporting Information

letter

Wang, Yunxia; Cui, Na; Zhao, Yu: Catalyst-Free Oxidative [3+2] Cycloaddition of Phenols and Styrenes in the Presence of a 2,3-Dichloro-5,6-dicyano-1,4-benzoquinone/1,1,1,3,3,3-hexafluoropropan-2-ol System
https://www.thieme-connect.de/media/synlett/EFirst/i_u0336_ga_10-1055_s-0036-1589082.gif
Supporting Information

Publication Date: 02 August 2017

letter

Guo, Tao; Wei, Xu-Ning: Ammonium Iodide-Mediated Sulfenylation of 4-Hydroxycoumarins or 4-Hydroxyquinolinones with a Sulfonyl Chloride as a Sulfur Source
https://www.thieme-connect.de/media/synlett/EFirst/i_w0410_ga_10-1055_s-0036-1589083.gif
Supporting Information

Publication Date: 27 July 2017

account

Wang, Qiang; Shi, Min: Synthesis of Cyclic and Heterocyclic Compounds via Gold-Catalyzed Reactions
https://www.thieme-connect.de/media/synlett/EFirst/i_a0345_ga_10-1055_s-0036-1590827.gif

letter

Matsumoto, Kenji; Mizushina, Naoyuki; Yoshida, Masahiro; Shindo, Mitsuru: Stereocontrolled Synthesis of Multisubstituted 1,3-Dienes via an Allene–Claisen Rearrangement
https://www.thieme-connect.de/media/synlett/EFirst/i_u0300_ga_10-1055_s-0036-1590970.gif
Supporting Information

letter

Matsumoto, Nobuyuki; Nakazaki, Atsuo; Nishikawa, Toshio: Concise Synthesis of a Cyclopentane Intermediate Possessing All Nitrogen Functionalities for Pactamycin
https://www.thieme-connect.de/media/synlett/EFirst/i_u0389_ga_10-1055_s-0036-1588495.gif
Supporting Information

letter

Stairs, Shaun; Powner, Matthew W.: Scalable Synthesis of 2,2′-Anhydro-arabinofuranosyl Imidazoles
https://www.thieme-connect.de/media/synlett/EFirst/i_d0449_ga_10-1055_s-0036-1590968.gif
Supporting Information

synpacts

Hullaert, Jan; Denoo, Bram; Christiaens, Mien; Callebaut, Brenda; Winne, Johan M.: Heterocycles as Moderators of Allyl Cation Cycloaddition Reactivity
https://www.thieme-connect.de/media/synlett/EFirst/i_p0408_ga_10-1055_s-0036-1588511.gif

Publication Date: 24 July 2017

cluster

Yamamoto, Eiji; Ukigai, Satoshi; Ito, Hajime: Formal Nucleophilic Silyl Substitution of Aryl Halides with Silyllithium Reagents via Halogenophilic Attack of Silyl Nucleophiles
https://www.thieme-connect.de/media/synlett/EFirst/i_b0342_ga_10-1055_s-0036-1590835.gif
Supporting Information

letter

Han, Jusung; Kim, Yo-Han; Jung, Byeong Yeon; Hwang, Seung Hyun; Jegal, Jonggon; Kim, Jung Won; Lee, Yoon-Sik: Highly Selective Catalytic Hydrogenation and Etherification of 5-Hydroxymethyl-2-furaldehyde to 2,5-Bis(alkoxymethyl)furans for Potential Biodiesel Production
https://www.thieme-connect.de/media/synlett/EFirst/i_u0338_ga_10-1055_s-0036-1589076.gif
Supporting Information

Publication Date: 21 July 2017

account

Quiclet-Sire, Béatrice; Zard, Samir Z.: Convergent Routes to Pyrroles Exploiting the Unusual Radical Chemistry of Xanthates – An Overview
https://www.thieme-connect.de/media/synlett/EFirst/i_r0364_ga_10-1055_s-0036-1590809.gif

cluster

Flinker, Mathias; Lopez, Sara; Nielsen, Dennis U.; Daasbjerg, Kim; Jensen, Frank; Skrydstrup, Troels: Experimental and Theoretical Studies on the Reduction of CO2 to CO with Chloro(methyl)disilane Components from the Direct Process
https://www.thieme-connect.de/media/synlett/EFirst/i_b0361_ga_10-1055_s-0036-1590840.gif
Supporting Information

letter

Wei, Wen-Ting; Ying, Wei-Wei; Zhu, Wen-Ming; Wu, Yi; Huang, Yi-Ling; Cao, Yi-Qi; Wang, Yi-Ning; Liang, Hongze: Convenient and Clean Synthesis of Isatins by Metal-Free Oxidation of Oxindoles
https://www.thieme-connect.de/media/synlett/EFirst/i_w0377_ga_10-1055_s-0036-1590965.gif
Supporting Information

Publication Date: 20 July 2017

cluster

Lee, Yong Ho; Morandi, Bill: Ether Synthesis through Reductive Cross-Coupling of Ketones with Alcohols Using Me2SiHCl as both Reductant and Lewis Acid
https://www.thieme-connect.de/media/synlett/EFirst/i_b0329_ga_10-1055_s-0036-1590838.gif
Supporting Information

cluster

Swartz, Brett D.; Brennessel, William W.; Jones, William D.: Lewis Acid Assisted C–CN Cleavage of Benzonitrile Using [(dippe)NiH]2
https://www.thieme-connect.de/media/synlett/EFirst/i_u0304_ga_10-1055_s-0036-1590801.gif
Supporting Information CIF File

letter

Ma, Teng; Li, Changwei; Liang, Haijing; Wang, Zhaoyan; Yu, Lan; Xue, Weihua: InBr3-Catalyzed Synthesis of Aryl 1,2-trans-Thio(seleno)glycosides
https://www.thieme-connect.de/media/synlett/EFirst/i_w0399_ga_10-1055_s-0036-1588507.gif
Supporting Information

letter

Stockdale, Trevor F.; O’Neil, Gregory W.: Regio- and Diastereoselective Samarium-Mediated Allylic Benzoate Reductions
https://www.thieme-connect.de/media/synlett/EFirst/i_r0421_ga_10-1055_s-0036-1590831.gif
Supporting Information

Publication Date: 19 July 2017