DOI: 10.1055/s-00000131

Synfacts

Ausgabe 03 · Volume 12 · März 2016 DOI: 10.1055/s-006-31012

Synform

A36
Zanda, Matteo: SYNFORM ISSUE 2016/03

Synthesis of Natural Products and Potential Drugs

z219
All PDFs of this category
0219
Synthesis of (–)-Chloramphenicol
0220
Synthesis of (S)-Baclofen
0221
Synthesis of Gelsenicine
0222
Total Synthesis of (+)-Cytosporolide A
0223
Synthesis of a CGRP Receptor Antagonist
0224
Synthesis of (–)-Hymenosetin
0225
Synthesis of a MCH1 Receptor Antagonist
0226
Synthesis of (R)-Lacosamide
0227
Synthesis of PF-04191834
0228
Synthesis of Enigmazole A
0229
Synthesis of (+)-Fastigiatine
0230
Synthesis of Cyclomarin A
0231
Synthesis of Vismodegib
0232
Synthesis of (+)-Chlorolissoclimide

Synthesis of Heterocycles

z233
All PDFs of this category
0233
Synthesis of Dihydrofurans from β-Ketocarbonyl Compounds and Olefins
0234
Synthesis of Oxazinanones from β-Lactams by Amide Bond Activation
0235
Tetrahydroquinolines by Michael Addition/Nitro-Mannich Reaction
0236
Palladium-Catalyzed Heteroannulation Route to (E)-Oxindolylideneacetates
0237
Aldehyde Allylation/Cyclization with Isocyanato Allylboronic Esters
0238
Enantiopure α-Substituted Piperazines by Asymmetric Lithiation−Trapping
0239
Gold-Catalyzed Synthesis of 7-Acylindoles from Anthranils
0240
Synthesis of Fluorinated Thiophenes by Ring Contraction of Thiopyrans
0241
Synthesis of 1-Benzyl- or 1-Benzoyliso-quinolines by Dehydrogenative Coupling
0242
Palladium-Catalyzed Synthesis of Difluoroalkylated Phenanthridines
0243
Pd-Catalyzed Arylation/[1,2]-Wittig Rearrangement of Pyridylmethyl Ethers
0244
Synthesis of Imidazo[1,2-a]pyridines by 1,3-Dipolar Cycloaddition
0245
Synthesis of Pyrrolopyridines from 3-Aminopyrrole
0246
Synthesis of Benzoxazoles by Copper/Palladium Catalysis
0247
Three-Component Synthesis of Oxazolidin-2-ones

Synthesis of Materials and Unnatural Products

z249
All PDFs of this category
0249
A Biphenyl Donor–Acceptor–Donor Ladder System
0250
Mind the ‘Band’ Gap
0251
A Solution for Dissolution of Polysaccharides
0252
Filling the Two-Coordinate, Acyclic Diaminosilylene Gap
0253
Adopting a Reductive Coupling Route to Grams of DOPT
0254
Potential Holey-Nanographene Precursor: A Pyrene-Based Macrocycle
0255
Good Things Come in Threes: Kabachnik–Fields Polycondensation
0256
Building Energetic Wheels for Hydrazine
0257
Got an Eye on Binding Anions? Better Put a (Rhenium-Capped) Ring on It
0258
Synthesis of Dibenzo[a,m]rubicenes and their Application in OTFTs
0259
Photochemical Cyclodehydrochlorination with Regioselectivity
0260
2 Se or Not 2 Se, That is the Question

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z261
All PDFs of this category
0261
Synthesis of Axially Chiral Vinyl Arenes by Palladium(0) Catalysis
0262
A New Ligand Design for Asymmetric Dehydrogenative Heck Arylation
0263
Asymmetric Hydrothiolation by Dynamic Kinetic Resolution
0264
Palladium-Catalyzed Regioselective 1,1-Difluoroallylation and Heck Cyclization
0265
Copper-Catalyzed Asymmetric Synthesis of Polysubstituted Cyclopropanes
0266
N–C Axial Chirality in Phenanthridine-6-ones by Palladium(0) Catalysis
0267
Iridium-Catalyzed Asymmetric Allylation of Silyl Enol Ethers
0268
Zinc-Catalyzed Diastereo- and Enantioselective Mannich-Type Reaction
0269
Enantioselective Aza-Michael Addition Catalyzed by a Chiral Boronic Acid
0270
A Copper-Catalyzed Enantioselective Hydroamination Sequence
0271
Copper-Catalyzed Nitroso-Diels–Alder Reaction
0272
A Bimetallic Titanium Catalyst for Asymmetric Epoxidation and Sulfoxidation
0273
Palladium-Catalyzed Asymmetric Decarboxylative Cycloaddition
0274
Asymmetric Domino Heck/Intermolecular C–H Bond Functionalization
0275
Metal Amide Catalyzed Asymmetric endo-Selective Cycloadditions
0276
Enantioselective 1,3-Dipolar Cycloaddition of Azomethine Ylides
0277
Synthesis of Chiral Tetrahydroquinolines by a Palladium–P,S Ligand Complex
0278
Hydrosilylation of Imines by a Chiral Zinc Catalyst
0279
Chiral α-Amino Acids by Palladium-Catalyzed Allylic Alkylation
0280
Scandium(III)-Catalyzed Asymmetric Synthesis of 1,2-Allenyl Ketones
0281
Copper-Catalyzed Asymmetric Cross-Aldol Reactions
0282
Copper-Catalyzed Synthesis of Chiral α-Hydroxy Amides and β-Amino Alcohols
0283
Iridium-Catalyzed Asymmetric Redox-Triggered Carbonyl Addition
0284
Asymmetric Hydrogenation of α-Oxyfunctionalized α,β-Unsaturated Acids
0285
Asymmetric Synthesis of α-Fluoromethylated Tertiary Alcohols
0286
Enantioselective Arylation of Isatin-Derived Ketimines
0287
Nonenzymatic Desymmetrization of Prochiral Allenic Diols
0288
Rhodium-Catalyzed C–C Bond Activation

Metal-Mediated Synthesis

z289
All PDFs of this category
0289
Catalytic Conjunctive Cross-Coupling
0290
Multicarbometalation of Alkynes
0291
Copper-Catalyzed Borylative Aromatization
0292
Synthesis of N-Boc-Propargylic and -Allylic Amines
0293
Copper-Catalyzed Asymmetric Allylic Arylation
0294
Transition-Metal-Free Cross-Couplings of Organoboron Reagents
0295
Ruthenium-Catalyzed C–O Activation/C–C Coupling Reactions
0296
Asymmetric Direct 1,2-Addition
0297
Sulfonylation of Aryl C(sp2)–H Bonds
0298
Iridium-Catalyzed Borylation of Aromatic Aldehydes
0299
Palladacycle-Catalyzed Aqueous Lipshutz–Negishi Cross-Coupling
0300
Selective Activation of Isatin Carbonyls
0301
Stereoselective Synthesis of Z-α,β-Unsaturated Sulfones
0302
Chemoselective Addition of Halomethyllithiums to Isatins
0303
Construction of α-Aryl β-Substituted Cyclic Ketone Scaffolds

Organo- and Biocatalysis

z305
All PDFs of this category
0305
Strong Hydrogen-Bonding Organocatalysts Activated by Electrostatics
0306
Organocatalytic Enantioselective Desymmetrization of Oxetanes
0307
Whole-Cell Biocatalysts for Stereoselective C–H Amination Reactions
0308
C1-Symmetric Chiral Brønsted Acid Catalyzed Diels−Alder Reaction
0309
Regiodivergent Enantioselective Addition of Oxazolones

Polymer-Supported Synthesis

z311
All PDFs of this category
0311
Suzuki Coupling with an N-Heterocyclic Carbene–Palladium Catalyst
0312
Synthesis of Spirocyclic Pyrazoles on Sulfonated Silica Supported Fe3O4
0313
One-Pot Synthesis of Chiral Esters by Oxidation–Olefination–1,4-Addition
0314
Amination of Aryl Halides with Palladium on Magnetic Nanoparticles
0315
Titanium Superoxide Catalyzed Oxidative Esterification of Aldehydes
0316
Palladium/Al(OH)3-Catalyzed Stille and Kumada Coupling
0317
Asymmetric Suzuki–Miyaura Coupling with Biotin-Tagged Palladium
0318
Reduction of Hetarenes with a Rhodium Nanoparticle–Ionic Liquid Catalyst
0319
Hydrogenation of Nitroarenes with Polymer-Supported Ruthenium Nanoparticles
0320
Preparation of 3-Amino-1,4-Diynes by Using Copper Oxide Nanoparticles
0321
Mesoporous Silica-Supported Zirconium Catalyst for Carbonyl Hydroboration
0322
Hydrogenation of Carbonyl Groups with Ruthenium Nanoparticles on Graphene
0323
A Chiral Imidazolidinone Polymer for the Asymmetric Diels–Alder Reaction
0324
Oxidative Imine Formation with Vitamin B12-Derived Mesoporous Carbon
0325
Synthesis of Enol Carbamates and Amides with Copper Nanoparticles on Charcoal
0326
Synthesis of Perhydrotriazolotriazole Derivatives with Fe3O4@SiO2-TiO2

Erratum

327
Sundar, M. S.; Bedekar, A. V.: Synthesis and Study of 7,12,17-Trioxa[11]helicene
327
Cheng, H.; Zeng, F.-H.; Yang, X. B.; Meng, Y.-J.; Xu, L.; Wang, F.-P.: (±)-Spiramilactone B, (±)-Spiraminol, (±)-Dihydroajaconine, and (±)-Spiramines C and D