DOI: 10.1055/s-00000083

Synlett

Ausgabe 03 · Volume 24 · Februar 2013 DOI: 10.1055/s-003-24466

synform

A15
Zanda, Matteo: SYNFORM ISSUE 2013/2

synpacts

269
Lalic, Gojko; Rucker, Richard P.: Copper-Catalyzed Electrophilic Amination of Organoboron Compounds
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276
Streuff, Jan: An Update on Catalytic Strategies for the Synthesis of α-Hydroxyketones
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account

281
Gualandi, Andrea; Cozzi, Pier Giorgio: Stereoselective Organocatalytic Alkylations with Carbenium Ions
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cluster

297
Cluster Cover Page
298
Yasuda, Nobuyoshi: Cluster Preface: Process Chemistry
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301
Chen, Ying; Crockett, Richard D.; Wang, Xin; Larsen, Robert D.; Cui, Sheng; Faul, Margaret M.: Development of a Scalable Synthesis of a VEGFR Inhibitor
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Supporting Information
305
Mudryk, Boguslaw; Joshi, Amit; Ortiz, Adrian; Young, Ian S.; Sawyer, James R.; Zheng, Bin; Sugiyama, Masano; Shi, Zhongping; Müslehiddinoğlu, Jale; Corbett, R. Michael; Kronenthal, David R.; Conlon, David A.: Evolution of the Process for the Preparation of a Selective ErbB VEGF Receptor Inhibitor
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Supporting Information
313
Houpis, Ioannis N.; Lemaire, Sebastien; Farina, Vittorio; Xiao, Tingting; Liu, Renmao; Nettekoven, Ulrike; Wang, Youchu: New Synthesis of 2′,4′-Functionalized Nucleotides via Stereospecific Hydrogenation and Azidation Reactions
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317
Lu, Bruce Z.; Li, Guisheng; Rodriguez, Sonia; Liu, Jianxu; Eriksson, Magnus C.; Tan, Zhulin; Song, Jinhua J.; Yee, Nathan K.; Farina, Vittorio; Senanayake, Chris H.: Development of a Practical Synthesis of 4-[6-(Morpholinomethyl)-pyridin-3-yl]naphthalen-1-amine, a Key Intermediate for the Synthesis of BIRB 1017, a Potent p38 MAP Kinase Inhibitor
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323
Chase, Charles E.; Fang, Francis G.; Lewis, Bryan M.; Wilkie, Gordon D.; Schnaderbeck, Matthew J.; Zhu, Xiaojie: Process Development of Halaven®: Synthesis of the C1–C13 Fragment from d-(–)-Gulono-1,4-lactone
https://www.thieme-connect.de/media/synlett/201303/i_y0971_ga_10-1055_s-0032-1317919.gif
327
Austad, Brian C.; Benayoud, Farid; Calkins, Trevor L.; Campagna, Silvio; Chase, Charles E.; Choi, Hyeong-wook; Christ, William; Costanzo, Robert; Cutter, James; Endo, Atsushi; Fang, Francis G.; Hu, Yongbo; Lewis, Bryan M.; Lewis, Michael D.; McKenna, Shawn; Noland, Thomas A.; Orr, John D.; Pesant, Marc; Schnaderbeck, Matthew J.; Wilkie, Gordon D.; Abe, Taichi; Asai, Naoki; Asai, Yumi; Kayano, Akio; Kimoto, Yuichi; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Mizuno, Masanori; Nakamura, Taiju; Omae, Takao; Ozeki, Naoki; Suzuki, Taeko; Takigawa, Teiji; Watanabe, Tomohiro; Yoshizawa, Kazuhiro: Process Development of Halaven®: Synthesis of the C14–C35 Fragment via Iterative Nozaki–Hiyama–Kishi Reaction–Williamson Ether Cyclization
https://www.thieme-connect.de/media/synlett/201303/i_y0973_ga_10-1055_s-0032-1317920.gif
Primary Data
333
Austad, Brian C.; Calkins, Trevor L.; Chase, Charles E.; Fang, Francis G.; Horstmann, Thomas E.; Hu, Yongbo; Lewis, Bryan M.; Niu, Xiang; Noland, Thomas A.; Orr, John D.; Schnaderbeck, Matthew J.; Zhang, Huiming; Asakawa, Naoki; Asai, Naoki; Chiba, Hiroyuki; Hasebe, Takashi; Hoshino, Yorihisa; Ishizuka, Hiroyuki; Kajima, Takashi; Kayano, Akio; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Miyazawa, Mamoru; Tagami, Katsuya; Watanabe, Tomohiro: Commercial Manufacture of Halaven®: Chemoselective Transformations En Route to Structurally Complex Macrocyclic Ketones
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Supporting Information 10.4125/pd0040th

letter

338
Mayer, Marilyn Graziano; Nador, Fabiana; Volpe, María Alicia; Radivoy, Gabriel: High Surface Area CeO2 Promoted Suzuki–Miyaura Cross-Coupling of Arylboronic Acids and Aryl Iodides
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343
Spork, Anatol P.; Ducho, Christian: Stereocontrolled Synthesis of 5′- and 6′-Epimeric Analogues of Muraymycin Nucleoside Antibiotics
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Supporting Information
347
Dighe, Mahesh G.; Lonkar, Sachin L.; Degani, Mariam S.: Mechanistic Insights into Palladium Leaching in Novel Pd/C-Catalyzed Boron-Heck Reaction of Arylboronic Acid
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Supporting Information
351
Pereshivko, Olga P.; Peshkov, Vsevolod A.; Ermolat’ev, Denis S.; Van der Eycken, Erik V.: Fast Assembly of 1H-Imidazo[1,2-a]imidazol-5-amines via Groebke–Blackburn–Bienaymé Reaction with 2-Aminoimidazoles
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Supporting Information
355
Titanyuk, Igor D.; Beletskaya, Irina P.: Palladium-Catalyzed Hydroarylation of Diazoacetic Ester
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Supporting Information
359
Ehlers, Peter; Petrosyan, Andranik; Ghochikyan, Tariel V.; Saghyan, Ashot S.; Neubauer, Antje; Lochbrunner, Stefan; Langer, Peter: Suzuki–Miyaura Reactions of 2,7-Dichloro-1,8-naphthyridine
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Supporting Information
363
Craven, Philip G. E.; Taylor, Richard J. K.: Stereocontrolled Routes to 4-Methoxypentadienoates for Use in Natural Product Synthesis
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369
Varghese, Vimal; Hudlicky, Tomas: Total Synthesis of Dihydrocodeine and Hydrocodone via a Double Claisen Rearrangement and C-10/C-11 Closure Strategy
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375
Narayama, Akira; Shibatomi, Kazutaka; Soga, Yoshinori; Muto, Tsubasa; Iwasa, Seiji: Copper(II)-Catalyzed Enantioselective Fluorination of β-Keto Esters Using Chiral Spiro Oxazoline Ligands
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Supporting Information
379
Choi, Juhee; Kim, Hyunseok; Park, Sangyun; Tae, Jinsung: Asymmetric Total Synthesis of (–)-Galanthamine via Intramolecular Heck Reaction of Conjugated Diene
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Supporting Information
383
Xu, Xiangsheng; Li, Tao; Li, Xiaoqing; Shao, Jiangbin: Synthesis of Substituted Fluorenes by Cascade Allenylation, Electrocyclization and Intramolecular Friedel–Crafts Reaction of 1,3-Diene-Substituted Propargylic Alcohols
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Supporting Information
389
Gao, Detian; Back, Thomas G.: Synthesis of the Reverse Transcriptase Inhibitor L-737,126 and the CB2 Cannabinoid Receptor Agonist Pravadoline by a Copper-Catalyzed Intramolecular Cross-Coupling
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394
Voltrova, Svatava; Srogl, Jiri: Expedient Method for Samarium(II) Iodide Preparation Utilizing a Flow Approach
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spotlight

397
Fintelman Dias, Flaviana Rodrigues: Ethyl 2-Diazoacetoacetate
399
Gigant, Nicolas: Triflic Acid

erratum

e1
Chase, Charles E.; Fang, Francis G.; Lewis, Bryan M.; Wilkie, Gordon D.; Schnaderbeck, Matthew J.; Zhu, Xiaojie: Process Development of Halaven®: Synthesis of the C1–C13 Fragment from d-(–)-Gulono-1,4-lactone
e2
Austad, Brian C.; Benayoud, Farid; Calkins, Trevor L.; Campagna, Silvio; Chase, Charles E.; Choi, Hyeong-wook; Christ, William; Costanzo, Robert; Cutter, James; Endo, Atsushi; Fang, Francis G.; Hu, Yongbo; Lewis, Bryan M.; Lewis, Michael D.; McKenna, Shawn; Noland, Thomas A.; Orr, John D.; Pesant, Marc; Schnaderbeck, Matthew J.; Wilkie, Gordon D.; Abe, Taichi; Asai, Naoki; Asai, Yumi; Kayano, Akio; Kimoto, Yuichi; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Mizuno, Masanori; Nakamura, Taiju; Omae, Takao; Ozeki, Naoki; Suzuki, Taeko; Takigawa, Teiji; Watanabe, Tomohiro; Yoshizawa, Kazuhiro: Process Development of Halaven®: Synthesis of the C14–C35 Fragment via Iterative Nozaki–Hiyama–Kishi Reaction–Williamson Ether Cyclization
e3
Austad, Brian C.; Calkins, Trevor L.; Chase, Charles E.; Fang, Francis G.; Horstmann, Thomas E.; Hu, Yongbo; Lewis, Bryan M.; Niu, Xiang; Noland, Thomas A.; Orr, John D.; Schnaderbeck, Matthew J.; Zhang, Huiming; Asakawa, Naoki; Asai, Naoki; Chiba, Hiroyuki; Hasebe, Takashi; Hoshino, Yorihisa; Ishizuka, Hiroyuki; Kajima, Takashi; Kayano, Akio; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Miyazawa, Mamoru; Tagami, Katsuya; Watanabe, Tomohiro: Commercial Manufacture of Halaven®: Chemoselective Transformations En Route to Structurally Complex Macrocyclic Ketones