Synthesis

Issue eFirst

Porashar, Bikoshita; Saikia, Anil K.: Lewis Acid Mediated Synthesis of 4-Aminoquinoline Derivatives from 2-Aminobenzonitriles and Activated Alkynes via Aza-Michael and Annulation Reactions

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Sá, Marcus M.; Moro, Pedro A. M.; Russo, Theo V. C.; Port, Vinicius C.; Caramori, Giovanni F.: Mild and Stereoselective Synthesis of (1E,3E)-Dienes through Silver(I)-Catalyzed β-Hydride Migration from Allylic α-Diazo Esters

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Kumari, Sangeeta; Tomar, Vijesh; Soni, Aditi; Manisha, Manisha; Sharma, Charu; Joshi, Raj K.: Ru-Mediated and Sulfur-Directed ortho-C–H Activation of Benzyl Thioethers with Internal Alkynes and Selective Hydrothiolation of Acetylene Dicarboxylates

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Jiang, Yong; Li, Yajuan; Zhu, Chen; Shen, Tao: Electrochemical Trioxygenation of Allylarenes

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Martin, Brandon S.; Ma, Donghui; Saito, Takeru; Gallagher, Katelyn S.; Dai, Mingji: Concise Total Synthesis of Complanadine A Enabled by Pyrrole-to-Pyridine Molecular Editing

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Issue Accepted Manuscripts

Pospech, Jola; Fessler, Johannes; Dao Xuan, Huy; Brandt, Sina; Täufer, Tobias; Kruse, Ayla; Lochbrunner, Stefan: A General Synthesis of 3,7-Di(carboxyalkyl)-functionalized Pyrimidopteridine Photoredox Catalysts

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Mizobuchi, Eduardo F.; Burtoloso, Antonio C. B.: The acylation of α-carbonyl sulfoxonium ylides with N-hydroxyphthalimide esters

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Guo, Yonghong; Zhao, Jiayi; Zu, Bing; He, Chuan: Aza-BODIPY-Based Bifunctional Photocatalyst for Red-Light-Driven Asymmetric Hydroxylation of β‑Ketoesters

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Ali, Kashif; Cho, Eun Jin: Platinum-Catalyzed Deoxygenation Process of N-Acyloxyamines

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Issue 19/2024

Hu, Mengjie; Ru, Liying; Zhu, Mengjiao; Yang, Shengwen; Fan, Suojiang; Ji, Jiangtao; Zheng, Dingming; Peng, Bo: Tandem [5,5]-/[3,3]-Rearrangements of Aryl Sulfoxides with Allyl Nitriles

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Marrazzo, John-Paul R.; Huynh, Tish; Fleming, Fraser F.: Isocyanoalkene Addition–Cyclization–Decarboxylation Cascades

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Issue 18/2024

Chen, Joseph; Chao, Darrian; Tran, Uyen Phuong; Billingsley, Kelvin L.: Design, Synthesis, and Assessment of Tricarboxylic Acid Cycle Probes

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Issue 17/2024

Xie, Liang-Jun; Chen, Lili; Xu, Senmiao: Benzothiazole-Directed Enantioselective Borylation of Secondary Benzylic C–H Bonds Using Iridium Catalysis

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Issue 16/2024

Rai, Archana; Das, Utpal: Accessing meta-Enone-Substituted Anisoles using ArN₂BF₄ as Precatalyst via Rearrangement of Alkyne-Tethered Cyclohexadienones

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Issue 13/2024

Li, Kun; Luan, Runze; Du, Yu; Su, Weiping: Remote-Carbonyl-Directed Consecutive Arylation of Terminal Alkenes for the Synthesis of Tetrasubstituted Olefins

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Issue 11/2024

Qian, Dang-Wei; Yang, Jin; Wang, Gang-Wei; Yang, Shang-Dong: Synthesis of β-Hydroxyhydrophosphonic Acids from Inorganic Sodium Hypophosphite

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Ding, Cheng-Lin; Zhong, Jun-Song; Yan, Hong; Ye, Ke-Yin: Electrochemical Hydro- and Deuterocarboxylation of Allenes

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Chen, Ruiming; Jia, Shihu; Man, Yuning; Cheng, Hong-Gang; Zhou, Qianghui: A Concise Total Synthesis of (±)-Stepharine and (±)-Pronuciferine

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Issue 08/2024

Zhang, Yan; Chen, Yuye; Xu, Jing: Total Synthesis of Daphniphyllum Alkaloids: (+)-Daphlongamine E, (+)-Calyciphylline R, and (–)-10-Deoxydaphnipaxianine A

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Issue 06/2024

Tiwari, Bindu; Sharma, Manish K.; Pandey, Ram P.; Hussain, Nazar: Site-Selective Lewis Acid Mediated Transformation of Pseudo Glycals to 1-Deoxy-2-thioaryl/alkyl Glycosides

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Issue 05/2024

Manisha, Manisha; Gupta, Shiv Shankar; Sharma, Upendra: Cobalt Catalysis: C7 Alkynylation of Indolines with a Bromoalkyne

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Issue 03/2024

Kwak, Soojin; Choi, Jeongin; Lee, Sarah Yunmi: Boron Lewis Acid Catalyzed Hydrophosphorylation of N-Heteroaryl-Substituted Alkenes

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Sarnes, Dustin M.; Struck, Valentina; Jones, Peter G.; Lindel, Thomas: N-Oxide Route to the Marine Natural Product Cyanogramide D

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Issue 01/2024

Jiang, Lu; Gao, Lei; Li, Xiaofei; Shao, Tingting; Yao, Jinzhong; Miao, Maozhong; Zhou, Hongwei: Rh(III)-Catalyzed Synthesis of Isocoumarins via C–H Activation of Phenacyl Phosphoniums with Iodonium Ylides

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Issue 24/2023

Semleit, Nina; Haberhauer, Gebhard: Gold(I)-Catalyzed Dearomatization–Allenene Reaction for the Construction of Polycycles with Excellent Diastereoselectivity

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Issue 23/2023

Pinter, Piermaria; Soellner, Johannes; Strassner, Thomas: Platinum(II) Complexes with Phenylpyridine, Benzo[h]quinoline, and NHC Ligands: Exploration of Ligand Effects on Photophysical Properties

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Wagner, Raphael; Wollnitzke, Philipp; Essig, Sebastian; Gölz, Jan P.; Menche, Dirk: Studies on Selective Metalation and Cross-Coupling Reactions of Oxazoles

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Issue 22/2023

Thye, Hermann; Fornfeist, Felix; Geik, Dennis; Schlüschen, Levi L.; Schmidtmann, Marc; Doye, Sven: Titanium-Catalyzed Intermolecular Hydroaminoalkylation of Terminal Alkynes

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Yagci, Bilge Banu; Munir, Badar; Zorlu, Yunus; Türkmen, Yunus Emre: Access to Symmetrical and Unsymmetrical Cyclobutanes via Template-Directed [2+2]-Photodimerization Reactions of Cinnamic Acids

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Issue 20/2023

Homer, Amal; Seitz, Oliver: New Thiazole Orange Derivatives for Improved Fluorescence Signaling of DNA FIT Probes

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Issue 17/2023

Wei, Kai; Hu, Wen; Sun, Yucui; Zhu, Tuo; Chen, Wen; Zhang, Hongbin: Asymmetric Total Syntheses of Macroline-Type Alkaloids Alstomicine and Alstofolinine A

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Tran Ngoc, Trung; van der Welle, Jasper; Rüffer, Tobias; Teichert, Johannes F.: Synthesis of Stable Neutral Homoaromatic Hydrocarbons

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Issue 16/2023

Pfitzer, Lucca; Heitkämper, Juliane; Kästner, Johannes; Peters, René: Use of the N–O Bonds in N-Mesyloxyamides and N-Mesyloxyimides To Gain Access to 5-Alkoxy-3,4-dialkyloxazol-2-ones and 3-Hetero-Substituted Succinimides: A Combined Experimental and Theoretical Study

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Berking, Tim; Frey, Wolfgang; Richert, Clemens: Kinetic or Thermodynamic Product? Case Studies on the Formation of Regioisomers of Tetraphenyladamantanes

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Issue 13/2023

Ammermann, Jonas; Meyer, Janina; Donner, Jannik; Reck, Michael; Wagner-Döbler, Irene; Kirschning, Andreas: New Demethylated Derivatives of Carolacton and Structure–Activity Relationship (SAR) Studies on Their Biofilm Inhibitory Properties

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Issue 12/2023

Zhou, Wei; Zhao, Qing-Wei; Luo, Yun-Cheng; Zhang, Xingang: Synthesis of 1-(Trifluoromethyl)alkenes through Transition-Metal-Catalyzed Alkylation and Arylation of 1-Chloro-3,3,3-trifluoroprop-1-ene (HCFO-1233zd)

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Issue 10/2023

Zisopoulou, Stavroula A.; Andreou, Thanos; Koftis, Theocharis V.; Gallos, John K.; Stathakis, Christos I.: Hetero-Diels–Alder Addition of Ethyl 2-Nitrosoacrylate to (Z)-Prop-1-enyl Ethers. Stereoselective Synthesis of a Precursor to Sacubitril

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Issue 09/2023

Bauer, Maximilian; Heretsch, Philipp: Biogenesis-Inspired Synthesis of Penicillitone

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Issue 07/2023

Baek, Sekwang; Jen, Hyundug; Yoo, Eun Jeong: Silver-Catalyzed Ring Expansion of Activated N-Heteroarenes via 1,4-Dearomative Addition of Diazomethylphosphonates

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Issue 06/2023

Su, Xiao-Yu; Huang, Pei-Qiang: Tf₂O-Promoted Morgan–Walls Reaction: From a Flexible Approach to Functionalized Phenanthridines and Quinazolines to the Short and Divergent Total Syntheses of Alkaloids

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Tenberge, Marius; Wahl, Johannes M.: Lewis Acid Catalysed Asymmetric One-Carbon Ring-Expansion of Prochiral Cyclobutanones

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Issue 05/2023

Ding, Ruiqi; Wang, Yidong; Wang, Yi-Ming: Synthesis of 1,1-Disubstituted Allenylic Silyl Ethers through Iron-Catalyzed Regioselective C(sp²)–H Functionalization of Allenes

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Issue 04/2023

Grenet, Erwann; van der Lee, Arie; Salom-Roig, Xavier J.: Doubly Switchable Diastereodivergent Strategy Mediated by a Chiral Sulfoxide to Access Disubstituted Tetrahydrocyclopenta­pyranone and Hexahydrocyclopentapyranol Scaffolds via Nazarov Cyclization

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Issue 03/2023

Zhang, Zongnan; Xue, Ting; Han, Zhe; Zeng, Rong: A Neutral FeCl₃ Photocatalysis for C–C Bond Animation and Alkylation of Cyclic Alcohols

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Issue 01/2023

Fansher, Douglas J.; Ngwira, Niza; Salehi, Ahmad Reza; Woods, Jerome; Cascão, Amanda; Palmer, David R. J.: Biocatalytic Synthesis of α,β-Unsaturated 2-Keto Acids and Derivatives Using the Promiscuous Aldolase, NahE

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Issue 24/2022

Porcu, Stefania; Cabua, Maria Chiara; Velichko, Viktoria; Baltaze, Jean-Pierre; Frongia, Angelo; Carbonaro, Carlo Maria; Ricci, Pier Carlo; Parsons, Drew Francis; Carlone, Armando; Secci, Francesco: Insights into the Reactivity of 2-Hydroxycyclobutanones with Thiols Corroborated by Quantum Chemical DFT Investigations and NMR and Raman Analysis

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Shi, Dong; Zeng, Tao; Lei, Xin; Wu, Xiaotong; Li, Mansirun; Zhang, Yandong: Unexpected Pyridinyl Group Mediated Metal-Free Wacker-Type Oxidation en Route to Pyrido[2,1-a]isoindol-5-ium Salts

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Issue 23/2022

Kikushima, Kotaro; Morita, Aki; Elboray, Elghareeb E.; Bae, Taeho; Miyamoto, Naoki; Kita, Yasuyuki; Dohi, Toshifumi: Transition-Metal-Free N-Arylation of N-Methoxysulfonamides and N,O-Protected Hydroxylamines with Trimethoxyphenyliodonium (III) Acetates

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Wei, Kaijie; Jiang, Menglu; Liang, Siyu; Yu, Wei: Iron-Catalyzed Benzene Ring Expansion of α-Azido-N-phenylamides

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Issue 22/2022

Zhang, Ziyin; Jiang, Zhi-Jiang; Cao, Yiwei; Chen, Jia; Gao, Zhanghua: Palladium-Catalyzed Ligand-Free ortho-Deuteration of Aromatic Carboxylic Acids with D₂O

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Pal, Parul; Fragis, Meghan; Dharavath, Srinivas; Johnson, Jarrod W.; Magolan, Jakob: Use of Vinyl Sulfides in Fischer Indole Reactions

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Issue 21/2022

Corpas, Javier; Ponce, Alberto; Maclean, Ian; Adrio, Javier; Carretero, Juan C.: Catalyst-Controlled Chemodivergent [3+3] and [3+2] Formal Cycloadditions of Azomethine Ylides with Diphenylcyclopropenone

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Mouthaan, Marc L. M. C.; Pouwer, Kees; Borst, Mark L. G.; Witte, Martin D.; Minnaard, Adriaan J.: α-C–H Photoalkylation of a Glucose Derivative in Continuous Flow

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Issue 20/2022

Kim, Suho; Park, Heon Kyu; Kang, Ju Young; Mishra, Neeraj Kumar; Kim, In Su: Assembly of the Hydroxycinnoline Core via Hydrazide-Assisted Rh(III)-Catalyzed C–H Functionalization and Annulation

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Luo, Han; Lu, Qixing; Xu, Mingchuan; Gu, Mingxi; Li, Baosheng: Facile Access to α-Substituted β-Thio Enals from 1,2,3-Triazines and Thiols

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Issue 19/2022

Guan, Yong; Buivydas, Tadas; Lalisse, Remy F.; Ali, Rameez; Hadad, Christopher M.; Mattson, Anita E.: Enantioselective Dearomative Alkynylation of Chromanones: Opportunities and Obstacles

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Herzog, Stefan; Marten, Inka; Weiß, Aaron; Podlech, Joachim: Synthesis of Diaza[5]helicenes by ortho,ortho′-Fusion of ortho-Terphenyls

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Issue 18/2022

Xi, Shuang; Zhang, Jingyang; Guo, Zhen; Zu, Yumeng; Liu, Yang; Wang, Gelin; Tang, Yefeng: Facile Access to Spiro[4.5]decanes through Oxidative Dearomatization-Induced Ring Expansion of Cyclobutanes

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Niu, Jiapan; Liu, Bowen; Zhang, Chun: Metal-Free Thiolation and Hydroxylation of CF₃-Substituted Alkenes: A Practical Method to Synthesize Trifluoromethyl Tertiary Alcohols

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Issue 17/2022

Kang, Xiaokang; Lai, Shuyan; Liang, Xiayu; Zeng, Qingle: 1,1-Difunctionalization of α‑Carbonyl Sulfur Ylides with Thiosulfonates: Synthesis of β-Keto Thiosulfones

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Yu, Jia; Wen, Si; Tian, Qingyu; Chen, Yanhui; Cheng, Guolin: Rhodium(I)-Catalyzed Regioselective C–H Alkenylation of 2,2′-Bipyridine Derivatives with Alkynes

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Qiu, Huixin; Wen, Lirong; Lv, Jian: Visible-Light-Induced Catalysis: A Regioselectivity Switch between [2+1] and [2+2] Cycloaddition of Diazocarbonyls with Olefins

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Issue 16/2022

Lin, Yutong; Malins, Lara R.: Synthesis of Peptide N-Acylpyrroles via Anodically Generated N,O-Acetals

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Chan, Hwai-Chien; Gagnon, Alexandre: On the Copper-Promoted Backbone Arylation of Histidine-Containing Peptides Using Triarylbismuthines

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Issue 15/2022

Li, Jia-Yue; Li, Lun; Lin, Yun-Zhi; Shi, Hang: External-Ligand-Free, Nickel-Catalyzed Alkenylation of N-Sulfonylamines with Internal Alkynes

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Hillrichs, Kai; Namyslo, Jan C.; Lederle, Felix; Hübner, Eike G.; Schmidt, Andreas: Pyrazoles in the Intersection of Mesomeric Betaines and N-Heterocyclic Carbenes: Formation of NHC Selenium Adducts of Pyrazolium-4-aminides

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Issue 14/2022

Sabadasch, Viktor; Dachwitz, Steffen; Hannappel, Yvonne; Hellweg, Thomas; Sewald, Norbert: Acrylamide-Based Pd-Nanoparticle Carriers as Smart Catalysts for the Suzuki–Miyaura Cross-Coupling of Amino Acids

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Guo, Donghui; Wang, Jian: Cinchona Alkaloid Catalyzed Dynamic Kinetic Resolution of Biaryl Aldehydes via Asymmetric Decarboxylative Transamination

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Issue 13/2022

Yao, Jie; Huang, Chengjie; Wu, Fan; Zhao, Yufen; Ni, Feng: Synthesis of Phosphoramidate Prodrugs of Phenolic Natural Products and Drugs by Ester Exchange

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Issue 12/2022

Qiu, Ju; Hou, Jingwei; Sun, Zuolian; Xie, Peizhong: Dehydrative and Decarboxylative Coupling of Alkynoic Acids with Allylic Alcohols

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Abaid, Kmar; Erb, William; Blot, Marielle; Roisnel, Thierry; Mongin, Florence; Touil, Soufiane: Ferrocenephosphonates: Copper-Promoted Synthesis and Further Functionalization

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Jamey, Nicolas; Ferrié, Laurent: From Ring-Expansion to Ring-Contraction: Synthesis of γ-Lactones from Cyclobutanols and Relative Stability of Five- and Six-Membered Endoperoxides toward Organic Bases

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Issue 11/2022

Li, Xiaojie; Xie, Yuxin; Yin, Kaixin; Shen, Ruwei; Zhu, Dunru: p-Quinol Ethers and p-Quinone Monoacetals as Arylation and Oxidation Reagents: Tandem N-Arylation and α-Functionalization of Pyrrolidine via Redox-Neutral Three-Component Reaction

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Li, Yi; Hu, Tianbao; Gao, Lu; Song, Zhenlei: Addition/Substitution Approach of TsNHCH₂SiMe₂CH₂Cl with Isocyanates or Isothiocyanates To Construct 1,3,5-Diazasilinan-2-ones or 1,3,5-Thiazasilinan-2-imines

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Viviano, Monica; Trapasso, Giacomo; Annatelli, Mattia; Milite, Ciro; Castellano, Sabrina; Aricò, Fabio: Microwave-Assisted Aminoalkylation of Phenols via Mustard Carbonate Analogues

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Issue 10/2022

Ma, Yu; Tian, Ze-Yu; Zheng, Shuang-Yang; Zhang, Cheng-Pan: Copper-Catalyzed Allylation of Amines with Cyclopropyldiphenylsulfonium Trifluoromethanesulfonate

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Zeng, Dishu; Yang, Tianbao; Tang, Niu; Deng, Wei; Xiang, Jiannan; Yin, Shuang-Feng; Kambe, Nobuaki; Qiu, Renhua: UV-Light-Induced Dehydrogenative N-Acylation of Amines with 2-Nitrobenzaldehydes To Give 2-Aminobenzamides

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Tang, Yu; Yu, Biao: A Mild Heteroatom (O-, N-, and S-) Methylation Protocol Using Trimethyl Phosphate (TMP)–Ca(OH)₂Combination

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Issue 09/2022

He, Maosheng; Zhang, Jinlong; Zhang, Cong; Wang, Hao-Yang; Jiang, Gaoxi: Brønsted Acid Catalyzed Direct Annulation of Alkoxyallenes and Naphthols to Chroman Ketals

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Dahiya, Gaurav; Abboud, Khalil A.; Aponick, Aaron: Tuning StackPhim Ligands: Applications in Enantioselective Borylation and Alkynylation

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Chaminda Lakmal, Hetti Handi; Istre, Jacob; Qian, Xiaolin; Zhou, Hui; Valle, Henry U.; Xu, Xue; Cui, Xin: Catalytic Amidomethylative [2+2+2] Cycloaddition of Formaldimine and Styrenes toward N-Heterocycles

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Issue 08/2022

Zhang, Jie; Yan, Peng; Wang, Zhichao; Zhao, Jinbo; Chen, Qin; Lu, Ping: Total Synthesis of (+)-Kingianin A by Enantioselective Cycloaddition of Strained Cyclobutenone

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Su, Bo; Zhang, Hui; Wang, Qingmin: Total Synthesis of the Proposed Structure of Tyloindane and Its Diastereoisomer

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Han, Jun-Fa; Guo, Peng; Chen, Lin; Ye, Ke-Yin: Cobalt-Catalyzed Glaser-type Homocoupling Reaction

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Issue 07/2022

Primdahl, Karoline G.; Kaupang, Åsmund; Park, Jong-Duk; Seyedsayamdost, Mohammad R.; Nolsøe, Jens M. J.; Aursnes, Marius: On the Structure of Thailandene A: Synthetic Examination of the Cryptic Natural Product Aided by a Theoretical Approach

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Vetter, Anna C.; Müller-Bunz, Helge; Muldoon, Jimmy; Nikitin, Kirill: Quaternary Phosphonium Carboxylates: Structure, Dynamics and Intriguing Olefination Mechanism

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Shen, Wen; Cunningham, Laura; Evans, Paul: Asymmetric Synthesis of γ-Amino-Functionalised Vinyl Sulfones: De Novo Preparation of Cysteine Protease Inhibitors

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Issue 06/2022

Li, Ping; Lee, Boon Chong; Zhang, Xiaoxiang; Koh, Ming Joo: Base-Mediated Site-Selective Hydroamination of Alkenes

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Hu, Yue; Gu, He; Jia, Yuanliang; Luo, Guiyin; Chen, Xiaochuan: A Flexible Approach to the Synthesis of Type II and III Lepadin Alkaloids

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Keim, Michael; Jasarevic, Medina; Miller, Ines; Maas, Gerhard: 1,3-Bis(trifluoromethyl)prop-2-ene 1-Iminium Salts: Reactions with Alkoxybenzenes and Anilines

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Issue 05/2022

Kuang, Cuiwen; Ni, Chuanfa; Gu, Yucheng; Hu, Jinbo: Photoredox-Catalyzed Ring-Opening Addition Reaction between Benzyl Bromides and Cyclic Ethers

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Köring, Laura; Sitte, Nikolai A.; Paradies, Jan: Towards the Development of Frustrated Lewis Pair (FLP) Catalyzed Hydrogenations of Tertiary and Secondary Carboxylic Amides

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Tlustý, Martin; Eigner, Václav; Lhoták, Pavel: Azide Decomposition as a Pathway to Intramolecularly Upper-Rim-Bridged Calix[4]arenes

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Issue 04/2022

Sun, Meng-Meng; Liu, Haidong; Zhu, Chuan; Feng, Chao: S_N2′ Defluorinative Allylation of Trifluoromethylalkenes with Allylsilanes

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Govindan, Karthick; Duraisamy, Tamilselvan; Jayaram, Alageswaran; Senadi, Gopal Chandru; Lin, Wei-Yu: Copper-Catalyzed Oxidative Cyclization of 2-Aminobenzamide Derivatives: Efficient Syntheses of Quinazolinones and Indazolones

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Issue 03/2022

Sansores Peraza, Pablo M.; García López, Jesús; Navarro, Yolanda; Iglesias, María J.; López Ortiz, Fernando: Synthesis of Pentacoordinated Spiro[4.4]phosphoranes by Reaction of Cyclic Phosphazenyl Anions with Epoxides: Study of their P-Remote Functionalization and Hydrolysis

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De Dios Miguel, Thomas; Louvel, Dan; Onida, Killian; Lavoignat, Adeline; Picot, Stephane; Duguet, Nicolas: Synthesis of Fatty 1,2,4-Trioxanes by Peracetalization of β-Hydroxy Hydroperoxides

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Timelthaler, Daniel; Topf, Christoph: Heterogeneous Hydrogenation of Quinoline Derivatives Effected by a Granular Cobalt Catalyst

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Mayorquín-Torres, Martha C.; Maldonado-Domínguez, Mauricio; Flores-Álamo, Marcos; Iglesias-Arteaga, Martín A.: Synthesis and Characterization of Hybrid Dimeric Steroid Spiroketals

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Issue 02/2022

Beckers, Igor; O’Rourke, Galahad; De Vos, Dirk: Late-Stage C–H Arylation of Azepinoindole via Pd/Cu Catalysis: A Step Efficient and Convergent Synthesis of Rucaparib

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Chand-Thakuri, Pratibha; Alahakoon, Indunil; Liu, Daniel; Kapoor, Mohit; Kennedy, John F.; Jenkins, Kenneth W.; Rabon, Allison M.; Young, Michael C.: Native Amine-Directed ortho-C–H Halogenation and Acetoxylation /Condensation of Benzylamines

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El-Tunsi, Ashraf; Carter, Nicholas; Yeo, Song-Hee; Priest, Joshua D.; Choi, Anthony; Kobras, Carolin M.; Ndlovu, Soneni; Proietti Silvestri, Ilaria; Fenton, Andrew K.; Coldham, Iain: Kinetic Resolution by Lithiation: Highly Enantioselective Synthesis of Substituted Dihydrobenzoxazines and Tetrahydroquinoxalines

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Tatevosyan, Stepan S.; Kotovshchikov, Yury N.; Latyshev, Gennadij V.; Lukashev, Nikolay V.; Beletskaya, Irina P.: Facile Access to Triazole-Fused 3,1-Benzoxazines Enabled by Metal-Free Base-Promoted Intramolecular C–O Coupling

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Issue 01/2022

Yu, Tian-Yang; Lu, Hong; Shao, Peng-Cheng; Qi, Xiu-Juan; Wei, Hao: Rhodium-Catalyzed Aryl Migratory/Decarbonylation of Diaryl Ketones via the Activation of Unstrained C–C Bonds

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Proietti, Giampiero; Prathap, Kaniraj Jeya; Ye, Xinchen; Olsson, Richard T.; Dinér, Peter: Nickel Boride Catalyzed Reductions of Nitro Compounds and Azides: Nanocellulose-Supported Catalysts in Tandem Reactions

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Issue 24/2021

Zhou, Chuanjiang; Zeng, Xianghua: Iodosulfonylation of Alkynes under Ultrasound Irradiation

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Minamikawa, Ryo; Fukaya, Keisuke; Kobayashi, Akihiro; Komiya, Yukinori; Yamamoto, Shio; Urabe, Daisuke; Chida, Noritaka; Sato, Takaaki: Development of a Chiral N-Alkoxyamide Strategy and Application to the Asymmetric Total Synthesis of Fasicularin

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Issue 23/2021

Jeng, Wey-Chyng; Chien, Po-Chung; Vagh, Sandip Sambhaji; Edukondalu, Athukuri; Lin, Wenwei: Organophosphane-Catalyzed Construction of Functionalized 2-Ylideneoxindoles via Direct β-Acylation

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Russo, Camilla; Cannalire, Rolando; Luciano, Paolo; Brunelli, Francesca; Tron, Gian Cesare; Giustiniano, Mariateresa: Visible-Light Photocatalytic Ugi/Aza-Wittig Cascade towards 2-Aminomethyl-1,3,4-oxadiazole Derivatives

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Issue 21/2021

Wang, Fei; Yi, Junyi; Nishimoto, Yoshihiro; Yasuda, Makoto: Homologation of Alkyl Acetates, Alkyl Ethers, Acetals, and Ketals by Formal Insertion of Diazo Compounds into a Carbon–Carbon Bond

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Laher, Romain; Gentilini, Emilie; Marin, Christophe; Michelet, Véronique: Oxygen-Tethered 1,6-Enynes and [4.1.0]-Bicyclic Ether Skeletons as Hedonic Materials for the Fragrance Industry

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Shao, Jiru; An, Caiyun; Wang, Sunewang R.: Facile Synthesis of Polysubstituted 2-Pyrones via TfOH-Mediated Ring Expansion of 2-Acylcyclopropane-1-carboxylates

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Kayama, Ayane; Shimizu, Akihiro; Shintani, Ryo: Anthracene-Based Zwitterion with a Small HOMO–LUMO Energy Gap

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Issue 20/2021

Sedano, Carlos; Virumbrales, Cintia; Suárez-Pantiga, Samuel; Sanz, Roberto: Aldol–Tishchenko Reaction of α-Oxy Ketones: Diastereoselective Synthesis of 1,2,3-Triol Derivatives

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St-Gelais, Jacob; Giguère, Denis: Protecting-Group-Free Synthesis of GB1107: An Orally Active Galectin-3 Antagonist

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Zhu, Deng; Ye, Ai-Hui; Chen, Zhi-Min: N-Selenocyanato-Dibenzenesulfonimide: A New Electrophilic Selenocyanation Reagent

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Zhu, Shaoqun; Wang, Jiawei; Zhou, Bing; Hou, Hong: Copper/Di-tert-butyl Peroxide-Catalyzed Regioselective Hydroxyphosphorylation of 1,3-Enynes

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Issue 19/2021

Britten, Thomas K.; Basson, Ashley J.; Roberts, Dean D.; McLaughlin, Mark G.: Aza-Peterson Olefinations: Rapid Synthesis of (E)-Alkenes

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Pudnika, Linda; Domraceva, Ilona; Werner, Thomas; Zalubovskis, Raivis; Grandane, Aiga: Base-Free Catalytic Wittig-/Cross-Coupling Reaction Sequence as Short Synthetic Strategy for the Preparation of Highly Functionalized Arylbenzoxepinones

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Wang, Pengfei; Li, Yuli; Wang, Guangwei: Tetrahydroxydiboron-Initiated Atom-Transfer Radical Cyclization

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Fang, Yong; Hu, Xiaoling; Shi, Zhuangzhuang; Zhao, Xu; Gopireddy, Raveendra Reddy; Luo, Yunfei: Iron-Catalyzed Stereoselective Allylboration of 3,4-Dihydroisoquinolines with Potassium Allyltrifluoroborates

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Issue 16/2021

Jia, Zongbin; Yang, Qi; Luo, Sanzhong: Photoredox-Mediated Asymmetric Cross-Dehydrogenative Coupling of Enones and Tertiary Amines by Chiral Primary Amine Catalysis

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Xie, Xiu-Ying; Jiang, Wei-Tao; Xiao, Bin: Alkyl Carbagermatrane Enabled Synthesis of Seven-Membered Carbocycle-Fused Aromatics through Catellani Strategy

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Issue 15/2021

Wata, Chisato; Hashimoto, Takuya: Organoiodine-Catalyzed Enantioselective Intramolecular Oxy­aminations of Alkenes with N-(Fluorosulfonyl)carbamate

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Lupi, Michela; Menichetti, Stefano; Stagnaro, Paola; Utzeri, Roberto; Viglianisi, Caterina: Thia-Bridged Triarylamine[4]helicene-Functionalized Polynorbor­nenes as Redox-Active pH-Sensitive Polymers

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Issue 14/2021

Maximiano, Adrielle P.; Ramos, Giovana S.; Marques, Marcelo V.; Sá, Marcus M.: Functionalized Cyclopropanes as Versatile Intermediates for the Diversity-Oriented Synthesis of γ-Lactones, γ-Lactams and δ-Lactams

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Issue 13/2021

Shaaban, Saad; Li, Houhua; Merten, Christian; Antonchick, Andrey P.; Waldmann, Herbert: Rhodium(III)-Catalyzed Enantioselective Benzamidation of Cyclopropenes

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Issue 12/2021

Steinke, Tim; Wonner, Patrick; Engelage, Elric; Huber, Stefan M.: Catalytic Activation of a Carbon–Chloride Bond by Dicationic Tellurium-Based Chalcogen Bond Donors

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Issue 11/2021

Li, Fusheng; Lin, Shuangjie; Li, Xiyu; Shi, Lei: Photocatalytic Generation of π-Allyltitanium Complexes from Butadiene via a Radical Strategy

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Issue 10/2021

Sirvent, Ana; Hernández-Ibáñez, Sandra; Yus, Miguel; Foubelo, Francisco: Pyrrolidine and Indolizidine Alkaloids from Chiral N-tert-Butanesulfinyl Imines Derived from 4-Halobutanal

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Issue 09/2021

Ikari, Yuta; Kaihara, Takahito; Goto, Shimpei; Bovenkerk, Marcel; Grenz, David C.; Esser, Birgit; Ferreira, Marli; Stachelek, Patrycja; Data, Przemyslaw; Yoshida, Takumu; Ikai, Tomoyuki; Tohnai, Norimitsu; Minakata, Satoshi; Takeda, Youhei: Peripherally Donor-Installed 7,8-Diaza[5]helicenes as a Platform for Helical Luminophores

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Issue 08/2021

Bubyrev, Andrey; Kantin, Grigory; Dar’in, Dmitry; Krasavin, Mikhail: CH-Diazomethane Sulfonamides Generated in Situ for Intramolecular [3+2] Cycloaddition of Alkynes: An Entry into Novel Pyrazole-Fused Five-Membered Sultams

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Issue 07/2021

Ponce, Marian Blanco; Parpart, Silvio; Villinger, Alexander; Rodríguez, Eugenio Torres; Ehlers, Peter; Langer, Peter: Synthesis of Pyrrolo[1,2-a][1,6]- and [1,8]naphthyridines by Alkyne-Carbonyl Metathesis

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Pruteanu, Elena; Tappin, Nicholas D. C.; Gîrbu, Vladilena; Morarescu, Olga; Dénès, Fabrice; Kulciţki, Veaceslav; Renaud, Philippe: Forskolin Editing via Radical Iodo- and Hydroalkylation

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Issue 06/2021

Laktsevich-Iskryk, Marharyta V.; Krech, Anastasiya V.; Zhabinskii, Vladimir N.; Khripach, Vladimir A.; Hurski, Alaksiej L.: Photocatalytic Stoichiometric Oxidant-Free Synthesis of Linear Unsaturated Ketones from 1,2-Disubstituted Cyclopropanols

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Inishi, Tsukasa; Hirata, Goki; Nishikata, Takashi: Michael Addition of Indoles to Enones Catalyzed by a Cationic Iron Salt

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Issue 05/2021

Blériot, Yves: Contributing to the Study of Enzymatic and Chemical Glycosyl Transfer Through the Observation and Mimicry of Glycosyl Cations

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Porcu, Stefania; Rodriguez, Carla Aira; Frongia, Angelo; Secci, Francesco: A Catalytic One-Pot Synthesis of Indolyl Cyclobutanones

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Issue 04/2021

Wech, Felix; Müller, Tizian; Becker, Jonathan; Gellrich, Urs: Synthesis of 6-Adamantyl-2-pyridone and Reversible Hydrogen Activation by the Corresponding Bis(perfluorophenyl)borane Complex

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Serusi, Lorenzo; Cuccu, Federico; Secci, Francesco; Aitken, David J.; Frongia, Angelo: Synthesis of Tryptamines through a Novel Brønsted Acid Mediated Tandem Reaction Initiated by α-Iminol Rearrangement of Transient 2-Substituted 2-Hydroxycyclobutylimines

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Issue 03/2021

Johnson, Trevor C.; Christy, Mitchell P.; Siegel, Dionicio: Synthesis of the 26-Membered Core of Thiopeptide Natural Products by Scalable Thiazole-Forming Reactions of Cysteine Derivatives and Nitriles

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Rachwalak, Marta; Gołębiewska, Justyna; Jakubowski, Tomasz; Stawinski, Jacek: Synthesis of Pyridiniumboranephosphonate Diesters and Related Compounds using Trityl Cation as a Borane Hydride Acceptor

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Issue 02/2021

Hornink, Milene Macedo; Lopes, Alice Uva; Andrade, Leandro Helgueira: Biobased Spiroimides from Itaconic Acid and Formamides: Molecular Targets for a Novel Synthetic Application of Renewable Chemicals

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Saktura, Maciej; Frankowski, Sebastian; Joachim, Bartłomiej; Albrecht, Łukasz: Aminocatalytic Synthesis of Uracil Derivatives Bearing a Bicyclo[2.2.2]octane Scaffold via a Doubly Cycloadditive Reaction Cascade

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Issue 01/2021

Helmecke, Lucas; Spittler, Michael; Schmidt, Bernd M.; Czekelius, Constantin: Metal-Free Iodoperfluoroalkylation: Photocatalysis versus Frustrated Lewis Pair Catalysis

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Issue 24/2020

Banert, Klaus; Heck, Manuel; Ihle, Andreas; Michael, Erik; Weber, Richard: Record-Breaking Steric Crowding in Trialkylamines Prepared by Oxidative Ring Opening

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Issue 23/2020

Buonomo, Joseph A.; Cole, Malcolm S.; Eiden, Carter G.; Aldrich, Courtney C.: 1,3-Diphenyldisiloxane Enables Additive-Free Redox Recycling Reactions and Catalysis with Triphenylphosphine

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Issue 22/2020

Ivanov, Konstantin L.; Tukhtaev, Hamidulla B.; Tukhtaeva, Feruza O.; Bezzubov, Stanislav I.; Melnikov, Mikhail Ya.; Budynina, Ekaterina M.: One-Pot Synthesis of γ-Azidobutyronitriles and Their Intramolecular Cycloadditions

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Issue 21/2020

Rehan, Mohammad; Flegel, Jana; Heitkamp, Franziska; Pergomet, Jorgelina L.; Otte, Felix; Strohmann, Carsten; Kumar, Kamal: Asymmetric Synthesis of 3,3′-Piperidinoyl Spirooxindoles and Discovery of Stereospecific Cycloadducts as Novel Hedgehog Pathway Modulators

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Issue 20/2020

Debiais, Mégane; Vasseur, Jean-Jacques; Müller, Sabine; Smietana, Michael: Selective Chemical Modification of DNA with Boronic Acids by On-Column CuAAc Reactions

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Issue 19/2020

Wang, Shuai; Kraus, George A.: Annulations with Butenolides and Phthalides: New Entries to Isocoumarins, 3,4-Dihydroisocoumarins, and Benzofurans

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Issue 18/2020

Xu, Chang-Jiang; Du, Wei; Albrecht, Łukasz; Chen, Ying-Chun: Lewis Basic Amine Catalyzed Aza-Michael Reaction of Indole- and Pyrrole-3-carbaldehydes

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Issue 17/2020

Zhang, Yuannian; Yang, Xin; Wu, Jie; Huang, Dejiang: Aerobic C–H Functionalization Using Pyrenedione as the Photocatalyst

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Issue 16/2020

Afewerki, Samson; Palo-Nieto, Carlos; Córdova, Armando: Efficient Heterogeneous Palladium-Catalyzed Transfer Hydrogenolysis of Benzylic Alcohols by Formic Acid

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Issue 15/2020

Sakai, Kentaro; Oisaki, Kounosuke; Kanai, Motomu: A Bond-Weakening Borinate Catalyst that Improves the Scope of the Photoredox α-C–H Alkylation of Alcohols

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Issue 14/2020

Tejeda-Serrano, María; Sanz-Navarro, Sergio; Blake, Finn; Leyva-Pérez, Antonio: Zeolites Catalyze the Nazarov Reaction and the tert-Butylation of Alcohols by Stabilization of Carboxonium Intermediates

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Issue 13/2020

Levitskiy, Oleg A.; Magdesieva, Tatiana V.: Reductive Amination of Aryl Boronic Acids: Parallelism of the Catalytic Reactivity of Transition Metals and Main Group Elements in the C(sp²)–N Bond-Forming Reactions

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Issue 12/2020

Amri, Nasser; Wirth, Thomas: Automated Electrochemical Selenenylations

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Camedda, Nicola; Serafino, Andrea; Maggi, Raimondo; Bigi, Franca; Cera, Gianpiero; Maestri, Giovanni: Functionalization of Alkenyl C–H Bonds with D₂O via Pd(0)/Carboxylic Acid Catalysis

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Issue 11/2020

Keerthana, Meledath Sudhakaran; Manoharan, Ramasamy; Jeganmohan, Masilamani: Cobalt(III)-Catalyzed Redox-Neutral Coupling of Acrylamides with Activated Alkenes via C–H Bond Activation

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Issue 09/2020

Ong, Derek Yiren; Chiba, Shunsuke: Controlled Reduction of Nitriles by Sodium Hydride and Zinc Chloride

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Issue 08/2020

Li, Dong; Lv, Shujun; Qu, Jingping; Zhou, Yuhan: Oxidation of 4-Aryl-1,1,1-trifluorobut-2-en-2-yl Trifluoro­methanesulfonates by 4-Picoline-N-Oxide: A Novel Approach to β-Trifluoromethyl-α,β-enones

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Issue 07/2020

Zhan, Fuxu; Zhang, Wei; Zhao, Huaiqing: Copper/Silver Cocatalyzed Regioselective C5–H Functionalization of 8-Aminoquinoline Amides with 1,3-Dicarbonyl Compounds

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Issue 06/2020

Gao, Qianwen; Liu, Ze-Shui; Hua, Yu; Zhou, Siwei; Cheng, Hong-Gang; Zhou, Qianghui: Alkyl Tosylates as Alkylating Reagents in the Catellani Reaction

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Issue 03/2020

Jeong, Hye Jin; Chae, Suyeon; Jeong, Keunhong; Namgoong, Sung Keon: Diverse One-Pot Electrophilic Trapping Reactions of 2-Quinolyl­zincates with Acyl Chlorides and Allyl Iodide

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Issue 02/2020

Song, Xian-Rong; Yang, Tao; Ding, Haixin; Xiao, Qiang: Direct Transformation of Propargylic Alcohols and O,O-Diethyl Phosphorothioic Acid into S-(2H-Chromen-4-yl) Phosphorothioates

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Issue 01/2020

Chernov, Nikita M.; Shutov, Roman V.; Potapova, Anastasia E.; Yakovlev, Igor P.: Convenient Synthesis of Fluorescent Chromeno[4,3-d]pyrimidines from Electron-Deficient 3-Vinylchromones

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Tang, Shuang-Qi; Schmitt, Martine; Bihel, Frédéric: POxAP Precatalysts and the Negishi Cross-Coupling Reaction

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Issue 24/2019

Valachová, Dominika; Ferko, Branislav; Puchľová, Eva; Caletková, Oľga; Berkeš, Dušan; Kolarovič, Andrej; Jakubec, Pavol: Stereoselective Synthesis of syn-γ-Hydroxynorvaline and Related α-Amino Acids

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Issue 23/2019

Li, Fang; He, Feifei; Koenigs, Rene M.: Catalyst-Free [2,3]-Sigmatropic Rearrangement Reactions of Photochemically Generated Ammonium Ylides

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Issue 22/2019

Fingerle, Michael; Stocker, Simon; Bettinger, Holger F.: New Synthesis of a Dibenzoperylene Motif Featuring a Doubly Boron–Nitrogen-Doped Bay Region

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Issue 13/2019

Zhao, Zhensheng; Jameel, Islam; Murphy, Graham K.: Vicinal Dichlorination of o-Vinylbiphenyls and the Synthesis of 9-(Arylmethyl)fluorenes via Tandem Friedel–Crafts Alkylations

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Issue 12/2019

Huy, Peter Helmut: Formamide Catalysis Facilitates the Transformation of Aldehydes into Geminal Dichlorides

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Issue 11/2019

Talko, Alicja; Antoniak, Damian; Barbasiewicz, Michał: Directed ortho-Metalation of Arenesulfonyl Fluorides and Aryl Fluorosulfates

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Issue 10/2019

Attard, Jonathan W.; Osawa, Kohei; Guan, Yong; Hatt, Jessica; Kondo, Shin-ichi; Mattson, Anita: Silanediol Anion Binding and Enantioselective Catalysis

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Issue 09/2019

Iskryk, Marharyta; Barysevich, Maryia; Ošeka, Maksim; Adamson, Jasper; Kananovich, Dzmitry: Asymmetric Kulinkovich Hydroxycyclopropanation of Alkenes Mediated by Titanium(IV) TADDOLate Complexes

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Issue 08/2019

Musolino, Manuele; Aricò, Fabio: Benzo-Fused 1,4-Heterocycles via Dialkyl Carbonate Chemistry

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Issue 07/2019

Della-Felice, Franco; de Assis, Francisco F.; Sarotti, Ariel M.; Pilli, Ronaldo A.: Palladium-Catalyzed Formation of Substituted Tetrahydropyrans: Mechanistic Insights and Structural Revision of Natural Products

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Issue 06/2019

Caillé, Julien; Pantin, Mathilde; Boeda, Fabien; Pearson-Long, Morwenna S. M.; Bertus, Philippe: Zinc-Mediated Double Addition on Functionalized Nitriles

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Issue 05/2019

Krieck, Sven; Schüler, Philipp; Peschel, Jan M.; Westerhausen, Matthias: Straightforward One-Pot Syntheses of Silylamides of Magnesium and Calcium via an In Situ Grignard Metalation Method

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Stöckl, Yannick; Frey, Wolfgang; Lang, Johannes; Claasen, Birgit; Baro, Angelika; Laschat, Sabine: Asymmetric Organocatalysis Revisited: Taming Hydrindanes with Jørgensen–Hayashi Catalyst

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Radtke, M. Alex; Dudley, Caroline C.; O’Leary, Jacob M.; Lambert, Tristan H.: A Scalable, One-Pot Synthesis of 1,2,3,4,5-Pentacarbomethoxycyclopentadiene

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Matsuoka, Seiya; Nakamura, Kayo; Ohmori, Ken; Suzuki, Keisuke: General Synthetic Approach to Rotenoids via Stereospecific, Group-Selective 1,2-Rearrangement and Dual S_NAr Cyclizations of Aryl Fluorides

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Leonov, Artem I.; Timofeeva, Daria S.; Ofial, Armin R.; Mayr, Herbert: Metal Enolates – Enamines – Enol Ethers: How Do Enolate Equivalents Differ in Nucleophilic Reactivity?

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Ueda, Mitsuhiro; Maeda, Ayami; Hamaoka, Kanako; Sasano, Mika; Fukuyama, Takahide; Ryu, Ilhyong: Bromine-Radical-Mediated Site-Selective Allylation of C(sp³)–H Bonds

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Schober, Lukas; Ratnam, Shahilan; Yamashita, Yasunobu; Adebar, Niklas; Pieper, Matthias; Berkessel, Albrecht; Hessel, Volker; Gröger, Harald: An Asymmetric Organocatalytic Aldol Reaction of a Hydrophobic Aldehyde in Aqueous Medium Running in Flow Mode

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Dohi, Toshifumi; Sasa, Hirotaka; Dochi, Mio; Yasui, Chihiro; Kita, Yasuyuki: Oxidative Coupling of N-Methoxyamides and Related Compounds toward Aromatic Hydrocarbons by Designer μ-Oxo Hypervalent Iodine Catalyst

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Wiegand, Anja; Wiese, Vera; Glowacki, Britta; Iovkova, Ljuba; Schirrmacher, Ralf; Jurkschat, Klaus; Krause, Norbert: GlucoSiFA and LactoSiFA: New Types of Carbohydrate-Tagged Silicon-Based Fluoride Acceptors for ¹⁸F-Positron Emission Tomography (PET)

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McLellan, Ross; Uzelac, Marina; Bole, Leonie J.; Gil-Negrete, Jose María; Armstrong, David R.; Kennedy, Alan R.; Mulvey, Robert E.; Hevia, Eva: Alkali Metal Effects in Trans-Metal-Trapping (TMT): Comparing LiTMP with NaTMP in Cooperative MTMP/Ga(CH₂SiMe₃)₃ Meta­lation Reactions

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Cecchini, Chiara; Lanzi, Matteo; Cera, Gianpiero; Malacria, Max; Maestri, Giovanni: Complementary Reactivity of 1,6-Enynes with All-Metal Aromatic Trinuclear Complexes and Carboxylic Acids

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Issue 03/2019

Modemann, Daniel J.; Zlatopolskiy, Boris D.; Urusova, Elizaveta A.; Zischler, Johannes; Craig, Austin; Ermert, Johannes; Guliyev, Mehrab; Endepols, Heike; Neumaier, Bernd: 2-[¹⁸F]Fluorophenylalanine: Synthesis by Nucleophilic ¹⁸F-Fluorination and Preliminary Biological Evaluation

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Nitti, Andrea; Bianchi, Gabriele; Po, Riccardo; Pasini, Dario: Scalable Synthesis of Naphthothiophene and Benzodithiophene Scaffolds as π-Conjugated Synthons for Organic Materials

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Issue 02/2019

Fritze, Lars; Riensch, Nicolas A.; Helten, Holger: Catalytic Si/B Exchange Condensation: A Green B–C Coupling Method That Provides Access to Monodisperse (Het)arylborane ‘Trimers’

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Hein, Julia; Klett, Jan: The Preparation of Tetramethyl 1,1′,3,3′-Ruthenocenetetra­carboxylate and Tetramethyl 1,1′,3,3′-Osmocenetetracarboxylate, and a Simplified Synthesis for Tetramethyl 1,1′,3,3′-Ferrocene­tetracarboxylate

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Issue 01/2019

Stopka, Tobias; Adler, Pauline; Hagn, Gerhard; Zhang, Haoqi; Tona, Veronica; Maulide, Nuno: Electrophilic Activation of Amides for the Preparation of Poly­substituted Pyrimidines

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Bartlett, Samuel L.; Keiter, Kimberly M.; Zavesky, Blane P.; Johnson, Jeffrey S.: Formation of Complex α-Imino Esters via Multihetero-Cope Rearrangement­ of α-Keto Ester Derived Nitrones

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McCabe, Stephanie R.; Wipf, Peter: Asymmetric Total Synthesis and Biological Evaluation of (+)-Cycloclavine

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Endoma-Arias, Mary Ann A.; Makarova, Mariia; Dela Paz, Helen E.; Hudlicky, Tomas: Chemoenzymatic Total Synthesis of (+)-Oxycodone from Phenethyl Acetate

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Xue, Weichao; Oestreich, Martin: Silicon Grignard Reagents as Nucleophiles in Transition-Metal-Catalyzed Allylic Substitution

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Sato, Io; Yamashita, Yasuhiro; Kobayashi, Shū: Alkylpotassium-Catalyzed Benzylic C–H Alkylation of Alkylarenes with Alkenes

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Nitelet, Antoine; Kairouz, Vanessa; Lebel, Hélène; Charette, André B.; Evano, Gwilherm: Continuous Flow Chlorination of Alkenyl Iodides Promoted by Copper Tubing

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Issue 24/2018

Gao, Qiwen; Xu, Lianyan L.; Parise, Vincent P.; Mehta, Yash R.; Aldrich, Leslie N.: Enantioselective Synthesis of 4-Amino-3-hydroxybenzopyran Flavanol Derivatives from Chalcones

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Funt, Liya D.; Tomashenko, Olesya A.; Novikov, Mikhail S.; Khlebnikov, Alexander F.: An Azirine Strategy for the Synthesis of Alkyl 4-Amino-5-(trifluoromethyl)-1H-pyrrole-2-carboxylates

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Issue 23/2018

Okamoto, Haruka; Toh, Kohei; Mochizuki, Takuya; Nakatsuji, Hidefumi; Sakakura, Akira; Hatano, Manabu; Ishihara, Kazuaki: Chiral Pyrophosphoric Acid Catalysts for the para-Selective and Enantioselective Aza-Friedel–Crafts Reaction of Phenols

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Sun, Weitao; Trinchera, Piera; Kurdi, Nada; Palomas, David; Crespo-Otero, Rachel; Afshinjavid, Saeed; Javid, Farideh; Jones, Christopher R.: Aryne-Mediated Arylation of Hantzsch Esters: Access to Highly Substituted Aryl-dihydropyridines, Aryl-tetrahydropyridines and Spiro[benzocyclobutene-1,1′-(3′,4′-dihydropyridines)]

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Issue 21/2018

Denizot, Natacha; Lachkar, David; Kouklovsky, Cyrille; Poupon, Erwan; Evanno, Laurent; Vincent, Guillaume: Divergent Oxidative Couplings between Indoles and 2,3-Dihydroxybenzoic Acid Derivatives for the Biomimetic Synthesis of Voacalgine A and Bipleiophylline

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Asano, Keisuke; Matsubara, Seijiro: Asymmetric Cycloetherification by Bifunctional Organocatalyst

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Belkheira, Mokhtaria; El Abed, Douniazad; Pons, Jean-Marc; Bressy, Cyril: Chemoselective Organoclick–Click Sequence

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Kutsumura, Noriki; Okada, Takahiro; Imaide, Satomi; Fujii, Hideaki; Nagase, Hiroshi: Acetic Anhydride Mediated Retro-Ene Reaction via a [4.4.3]Propel­lane Skeleton Intermediate Containing a Quaternary Ammonium Linkage

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Issue 20/2018

Moreno-Yruela, Carlos; Olsen, Christian A.: Synthesis of Trifluoromethyl Ketone Containing Amino Acid Building Blocks for the Preparation of Peptide-Based Histone Deacetylase (HDAC) Inhibitors

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Roiser, Lukas; Zielke, Katharina; Waser, Mario: Formal (4+1) Cyclization of Ammonium Ylides with Vinylogous para-Quinone Methides

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Issue 19/2018

Camp, Jason E.; Bousfield, Thomas W.; Dunsford, Jay J.; Adams, James; Britton, Joshua; Fay, Michael W.; Angelis-Dimakis, Athanasios: Dehydrative Cross-Coupling of 1-Phenylethanol Catalysed by Palladium Nanoparticles Formed in situ Under Acidic Conditions

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Rode, Katharina; Palomba, Martina; Ortgies, Stefan; Rieger, Rene; Breder, Alexander: Aerobic Allylation of Alcohols with Non-Activated Alkenes Enabled by Light-Driven Selenium-π-Acid Catalysis

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Issue 18/2018

Rosenthal, Amos J.; Mallet-Ladeira, Sonia; Bouhadir, Ghenwa; Bourissou, Didier: Persistent P-Stabilized Boryl Radicals with Bulky Substituents at Boron

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Romanovs, Vitalijs; Spura, Jana; Jouikov, Viatcheslav: Synthesis and Electrochemical Study of 1,1′-Thienyl-Substituted Fused Bis-germatranes with a Core 5c-6e Hyperbond

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Issue 17/2018

Cabezas, Jorge A.; Poveda, Rebeca R.; Brenes, José A.: One-Pot Conversion of Aldehydes and Ketones into 1-Substituted and 1,4-Disubstituted 1,3-Enynes

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Jain, Nikita; Ciufolini, Marco A.: Oxidative Kinetic Resolution of Some Naphtholic Alcohols Mediated by a Chiral Hypervalent Iodine Reagent

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Issue 16/2018

Riefert, Alexander; Maier, Martin E.: Approach to the Core Structure of 15-epi-Exiguolide

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Issue 15/2018

Romero-Ibañez, Julio; Cruz-Gregorio, Silvano; Quintero, Leticia; Sartillo-Piscil, Fernando: Concise and Environmentally Friendly Asymmetric Total Synthesis of the Putative Structure of a Biologically Active 3-Hydroxy-2-piperidone Alkaloid

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Issue 13/2018

Yamashita, Yu; Hirano, Yoichi; Takada, Akiomi; Takikawa, Hiroshi; Suzuki, Keisuke: Total Synthesis of Bis-anthraquinone Antibiotic BE-43472B

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Issue 12/2018

Al-Jawaheri, Yassir; Turner, Matthew; Kimber, Marc C.: Enabling the Rearrangement of Unactivated Allenes to 1,3-Dienes by Use of a Palladium (0)/Boric Acid System

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Issue 09/2018

Kenny, Miles; Schröder, Sybrin P.; Taylor, Nicholas J.; Jackson, Paula; Kitson, Daniel J.; Franckevičius, Vilius: Palladium-Catalysed Construction of All-Carbon Quaternary Centres with Propargylic Electrophiles: Challenges in the Simultaneous Control of Regio-, Chemo- and Enantioselectivity

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Issue 08/2018

Sipos, Zoltán; Kónya, Krisztina: Synthesis of Benzopyran-Fused Flavone Derivatives via Microwave-Assisted Intramolecular C–H Activation

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Vaghi, Luca; Sanzone, Alessandro; Sassi, Mauro; Pagani, Simone; Papagni, Antonio; Beverina, Luca: Synthesis of Fluorinated Acridines via Sequential Micellar Buchwald–Hartwig Amination/Cyclization of Aryl Bromides

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Issue 07/2018

Pirola, Margherita; Compostella, Maria Elena; Raimondi, Laura; Puglisi, Alessandra; Benaglia, Maurizio: A Continuous-Flow, Two-Step, Metal-Free Process for the Synthesis of Differently Substituted Chiral 1,2-Diamino Derivatives

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Dao Thi, Hang; Le Nhat Thuy, Giang; Catak, Saron; Van Speybroeck, Veronique; Van Nguyen, Tuyen; D’hooghe, Matthias: Use of 3-Hydroxy-4-(trifluoromethyl)azetidin-2-ones as Building Blocks for the Preparation of Trifluoromethyl-Containing Aminopropanes, 1,3-Oxazinan-2-ones, Aziridines, and 1,4-Dioxan-2-ones

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Issue 06/2018

Preface: The SYNTHESIS–SYNLETT Lectureship

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Carlsen, Peter N.; Stoutenburg, Eric G.; Frontier, Alison J.: SYNTHESIS–SYNLETT Lecture: Toward the Asymmetric Synthesis of Tetrapetalone A: Preparation of an Enantioenriched Indane Intermediate and Strategy for Endgame Glycosylation

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Duymaz, Adile; Körber, Jochen; Hofmann, Carolin; Gerlach, Dorothea; Nubbemeyer, Udo: Synthesis of Optically Active 15-epi-9,14-Methylene Lipoxin A₄

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Issue 05/2018

Lavrard, Hubert; Popowycz, Florence: Regioselective Late-Stage C-3 Functionalization of Pyrazolo[3,4-b]pyridines

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Seifried, Marco; Knoll, Christian; Welch, Jan M.; Müller, Danny; Weinberger, Peter: Unsaturated Aryl and Heteroaryl N1-Tetrazoles from 1-Allyl-1H-tetrazole

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Issue 04/2018

Jäckel, Elisabeth; Kaufmann, Julia; Haak, Edgar: Complex Polycycles from Simple Propargyl Alcohols through Ruthenium-Catalyzed Cascade Reactions and One-Pot Procedures

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Baumann, Marcus; Baxendale, Ian R.: Diastereoselective Synthesis and Diversification of Highly Functionalized Cyclopentanones

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Issue 03/2018

Fuchibe, Kohei; Takayama, Ryo; Aono, Tatsuya; Hu, Ji; Hidano, Tomohiro; Sasagawa, Hisashi; Fujiwara, Masaki; Miyazaki, Shinji; Nadano, Ryo; Ichikawa, Junji: Regioselective Syntheses of Fluorinated Cyclopentanone Derivatives: Ring Construction Strategy Using Transition-Metal–Difluorocarbene Complexes and Free Difluorocarbene

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Li, Jun; Xing, Jun; Lücke, Daniel; Lübken, Dennis; Millbrodt, Lucas; Plentz, Ruben R.; Kalesse, Markus: The Structure Elucidation of Haprolid

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Issue 02/2018

Paul, Jérôme; Presset, Marc; Le Gall, Erwan; Léonel, Eric; Retailleau, Pascal: Insights into the Cobalt-Catalyzed Three-Component Coupling of Mixed Aromatic Organozinc Species, Carbonyl Compounds or Imines and Michael Acceptors: Synthetic and Mechanistic Aspects

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Mancuso, Raffaella; Veltri, Lucia; Russo, Patrizio; Grasso, Giuseppe; Cuocci, Corrado; Romeo, Roberto; Gabriele, Bartolo: Palladium-Catalyzed Carbonylative Synthesis of Functionalized Benzimidazopyrimidinones

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Issue 01/2018

Da Silva Pinto, Solange; Davies, Stephen G.; Fletcher, Ai M.; Roberts, Paul M.; Thomson, James E.: Stereoselective Ammonium-Directed Epoxidation in the Asymmetric Syntheses of Dihydroconduramines (–)-A-2, (–)-B-2, (–)-C-3 and (+)-F-3

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Parsons, Philip J.; Allen, Lewis A. T.; Jones, Daniel R.; Padgham, Alex C.; Pryke, James A.; McKenna, Joseph; O’Reilly, Daniel: Approaches to the Synthesis of Highly Substituted Aromatic and Fused Rings: Metal-Catalysed versus Thermal Cyclisation

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Issue 24/2017

Blaukopf, Markus; Atamanyuk, Dmytro; Xavier, Nuno M.; Gerusz, Vincent; Kosma, Paul: Synthesis of 1,5-Anhydro-d-glycero-d-gluco-heptitol Derivatives as Potential Inhibitors of Bacterial Heptose Biosynthetic Pathways

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Issue 22/2017

Záborský, Ondrej; Štadániová, Radka; Doháňošová, Jana; Moncol, Ján; Fischer, Róbert: Synthesis of Isoxazolidinyl Epoxides by Oxone Treatment of 2,3-Dihydroisoxazoles in Acetone–Water Solution: A New Stereoselective Approach to Hydroxy-Substituted Isoxazolidines

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Aitken, R. Alan; Garnett, Alasdair N.: Versatile Pyrolytic Synthesis of Fused Polycyclic Heteroaromatic Compounds

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Issue 21/2017

Eastabrook, Andrew S.; Sperry, Jonathan: Synthetic Access to 3,5,7-Trisubstituted Indoles Enabled by Iridium­-Catalyzed C–H Borylation

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Desroches, Justine; Gilbert, Audrey; Houle, Camille; Paquin, Jean-François: A Radical Access to CF₃- and SF₅-Containing Dihydrobenzofurans and Indolines

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Issue 20/2017

Arii, Hidekazu; Nakabayashi, Kenichi; Mochida, Kunio; Kawashima, Takayuki: Synthesis of π-Extended Siloles Using Intramolecular Chain Hydrosilylation

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López-Rodríguez, Alberto; Domínguez, Gema; Pérez-Castells, Javier: Synthesis of Novel Iminosugar Derivatives Based on a 2-Azabi­cyclo[4.1.0]heptane Skeleton

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Issue 19/2017

Naganawa, Yuki; Ito, Jun-ichi; Kawagishi, Mayu; Nishiyama, Hisao: Asymmetric Desymmetrization of Substituted Cyclohexadienones by Rhodium-Catalyzed Conjugate Hydrosilylation and Theoretical Calculations of Its Mechanistic Aspects

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López, Enol; Lonzi, Giacomo; López, Luis A.: Synthesis of Functionalized Cyclopentene Derivatives through Gold-Catalyzed Reaction of Stabilized Vinyldiazo Compounds and Styrenes

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Issue 18/2017

Panferova, Liubov I.; Struchkova, Marina I.; Dilman, Alexander D.: Vinylation of Iododifluoromethylated Alcohols via a Light-Promoted Intramolecular Atom-Transfer Reaction

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Issue 17/2017

An, Yu; He, Huan; Liu, Tiantian; Zhang, Yong; Lu, Xiaoyun; Cai, Qian: Diversified Synthesis of 2-(4-Oxo[1,2,3]triazolo[1,5-a]quinoxalin-5(4H)-yl)acetamide Derivatives through Ugi-4-CR and Copper-Catalyzed Tandem Reactions

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Geibel, Irina; Kahrs, Christoph; Christoffers, Jens: Formation of Bicyclic Cyclopentenone Derivatives by Robinson-Type Annulation of Cyclic β-Oxoesters Containing a 1,4-Diketone Moiety

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Issue 16/2017

Muraca, Ana Carolina A.; Perecim, Givago P.; Rodrigues, Alessandro; Raminelli, Cristiano: Convergent Total Synthesis of (±)-Apomorphine via Benzyne Chemistry: Insights into the Mechanisms Involved in the Key Step

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Sato, Yuki; Kawaguchi, Shin-ichi; Nomoto, Akihiro; Ogawa, Akiya: Photoinduced Coupling Reaction of Diphenyl(2,4,6-trimethylbenzoyl)phosphine Oxide with Interelement Compounds: Application to the Synthesis of Thio- or Selenophosphinates

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Issue 14/2017

Xu, Wan; Zeng, Meng-Tian; Liu, Min; Liu, Sha-Sha; Li, Yue-Sheng; Dong, Zhi-Bing: Palladium-Catalyzed Synthesis of 2-Aminobenzothiazoles through Tandem Reaction

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Sun, Wei; Wilson, Dharyl C.; Harrowven, David C.: Steric Buttressing Changes Torquospecificity in Thermal Cyclo­butenone Rearrangements, Providing New Opportunities for 5H-Furanone Synthesis

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Issue 13/2017

Rais, Eduard; Flörke, Ulrich; Wilhelm, René: Reactivity of Grubbs–Hoveyda II Complexes Including Extended N-Heterocyclic Carbenes with a Bicyclic Camphor-Based Framework

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Lee, Wan-Chen Cindy; Tehrani, Arya; Li, Jie Jack: Copper-Mediated sp² C–H Chlorination with Trichloroacetamide Using a Removable Directing Group

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Issue 12/2017

Heindl, Andreas H.; Schweighauser, Luca; Logemann, Christian; Wegner, Hermann A.: Azobenzene Macrocycles: Synthesis of a Z-Stable Azobenzenophane

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Afanasyev, Oleg I.; Tsygankov, Alexey A.; Usanov, Dmitry L.; Perekalin, Dmitry S.; Samoylova, Alexandra D.; Chusov, Denis: Some Aspects of Reductive Amination in the Presence of Carbon Monoxide: Cyclopropyl Ketones as Bifunctional Electrophiles

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Issue 11/2017

Sinai, Ádám; Mészáros, Ádám; Balogh, Ádám; Zwillinger, Márton; Novák, Zoltán: Hexafluorosilicic Acid as a Novel Reagent for the Desilylation of Silylacetylenes: Application in Sequential Sonogashira Coupling and Click Reaction

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Pelzer, Stefanie; Neumann, Beate; Stammler, Hans-Georg; Ignat’ev, Nikolai; Eujen, Reint; Hoge, Berthold: Synthesis and Characterization of Tetrakis(pentafluoroethyl)germane

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Issue 10/2017

Grzelak, Paulina; Utecht, Greta; Jasiński, Marcin; Mlostoń, Grzegorz: First (3+2)-Cycloadditions of Thiochalcones as C=S Dipolarophiles: Efficient Synthesis of 1,3,4-Thiadiazoles via Reactions with Fluorinated Nitrile Imines

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Chadda, Rekha; McArdle, Patrick; Murphy, Paul V.: Allylic Azide Rearrangement in Tandem with Intramolecular Huisgen Cycloaddition for Iminosugar and Glycomimetic Synthesis: Functionalized Piperidine, Pyrrolidine, and Pyrrolotriazoles from d-Mannose

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Issue 09/2017

Craig, Alexander J.; Hawkins, Bill C.: Metal-Free Synthesis of Oxazinones and Their Reductive Ring Opening to Provide Cyclopropyl Carbinols

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Issue 07/2017

Meninno, Sara; Overgaard, Jacob; Lattanzi, Alessandra: Amine Thiourea Catalysed Double Michael Reaction: An Approach for the Asymmetric Synthesis of Spiro[pyrazolone-4,3′-tetrahydrothiophenes]

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Di Iorio, Nicola; Soprani, Lorenzo; Crotti, Simone; Marotta, Emanuela; Mazzanti, Andrea; Righi, Paolo; Bencivenni, Giorgio: Michael Addition of Oxindoles to N-(2-tert-Butylphenyl)maleimides: Efficient Desymmetrization for the Synthesis of Atropisomeric Succinimides with Quaternary and Tertiary Stereocenters

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Issue 06/2017

Jung, Eun-Kyung; Pilkington, Lisa I.; Barker, David: Synthesis of Benzodioxane and Benzofuran Scaffolds Found in Neolignans via TMS Triflate Mediated Addition to 1,4-Benzo­dioxane Hemiacetals

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Ábrahámi, Renáta A.; Kiss, Loránd; Fustero, Santos; Fülöp, Ferenc: Functionalized Dialdehydes as Promising Scaffolds for Access to Heterocycles and β-Amino Acids: Synthesis of Fluorinated Piperidine and Azepane Derivatives

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Issue 05/2017

D’Alonzo, Daniele; De Fenza, Maria; Palumbo, Giovanni; Romanucci, Valeria; Zarrelli, Armando; Di Fabio, Giovanni; Guaragna, Annalisa: Synthesis of β-l-2′-Fluoro-3′-thiacytidine (F-3TC) Stereoisomers: Toward a New Class of Oxathiolanyl Nucleosides?

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Lavendomme, Roy; Malytskyi, Volodymyr; Vandermeersch, Jeremy; Luhmer, Michel; Jabin, Ivan: One-Step Synthesis of a Unique Molecular Platform for the Selective Functionalization of Calix[6]arenes

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Issue 04/2017

Fopp, Carolin; Isaac, Kevin; Romain, Elise; Chemla, Fabrice; Ferreira, Franck; Jackowski, Olivier; Oestreich, Martin; Perez-Luna, Alejandro: Stereodivergent Synthesis of β-Heteroatom-Substituted Vinyl­silanes by Sequential Silylzincation–Copper(I)-Mediated Electrophilic­ Substitution

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Richard, Jimmy; Birepinte, Mélodie; Charbonnier, Jean Baptiste; Liautard, Virginie; Pinet, Sandra; Pucheault, Mathieu: Borinic Acids via Direct Arylation of Amine–Borane Complexes: An Air- and Water-Stable Boron Source

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Issue 03/2017

Pantaine, Loïc; Laverny, Aragorn; Moreau, Xavier; Coeffard, Vincent; Greck, Christine: Stereoselective Multibond-Forming Process towards Functionalized Sulfamide-Containing Polycycles

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Griesbeck, Axel G.; Porschen, Björn; Kropf, Christian; Landes, Agnieszka; Hinze, Olga; Huchel, Ursula; Gerke, Thomas: Photocaged Hydrocarbons, Aldehydes, Ketones, Enones, and Carboxylic Acids and Esters that Release by the Norrish II Cleavage Protocol and Beyond: Controlled Photoinduced Fragrance Release

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Issue 02/2017

Riehl, Barbara; Dyballa, Katrin M.; Franke, Robert; Waldvogel, Siegfried R.: Electro-organic Synthesis as a Sustainable Alternative for Dehydrogenative Cross-Coupling of Phenols and Naphthols

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Issue 01/2017

Bier, Claus; Binder, Dennis; Drobietz, Dagmar; Loeschcke, Anita; Drepper, Thomas; Jaeger, Karl-Erich; Pietruszka, Jörg: Photocaged Carbohydrates: Versatile Tools for Controlling Gene Expression by Light

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Issue 20/2016

Du, Haiying; Dudognon, Yohan; Sanchez Duque, Maria del Mar; Goudedranche, Sébastien; Bonne, Damien; Rodriguez, Jean; Bugaut, Xavier; Constantieux, Thierry: Organocatalytic Multicomponent Reactions of 1,3-Dicarbonyls for the Synthesis of Enantioenriched Heterocycles

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Issue 18/2016

Chiarini, Marco; Del Vecchio, Luana; Marinelli, Fabio; Rossi, Leucio; Arcadi, Antonio: Synthesis of 3-Substituted 2,1-Benzisoxazoles by the Oxidative Cyclization of 2-Aminoacylbenzenes with Oxone

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Issue 17/2016

Diamanti, Eleonora; Bottegoni, Giovanni; Goldoni, Luca; Realini, Natalia; Pagliuca, Chiara; Bertozzi, Fabio; Piomelli, Daniele; Pizzirani, Daniela: Pyrazole-Based Acid Ceramidase Inhibitors: Design, Synthesis, and Structure–Activity Relationships

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Koch, Niklas; Seichter, Wilhelm; Mazik, Monika: Compounds Based on a Triethyl- or Trimethoxybenzene Scaffold Bearing Pyrazole, Pyridine, and Pyrimidine Groups: Syntheses and Representative Binding Studies towards Carbohydrates

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Issue 16/2016

Capel, E.; Vidal-Albalat, A.; Rodríguez, S.; González, F. V.: Preparation of Morpholines and Benzoxazines Starting from Nitroepoxides

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Issue 15/2016

Balaraman, Kaluvu; Moskowitz, Max; Liu, Yang; Wolf, Christian: Detrifluoroacetylative Generation of Halogenated Enolates: Practical Access to Perhalogenated Ketones and Alkenes

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Mori, Yasuyuki; Kawabata, Toshiki; Onodera, Gen; Kimura, Masanari: Remarkably Selective Formation of Allenyl and Dienyl Alcohols via Ni-Catalyzed Coupling Reaction of Conjugated Enyne, Aldehyde, and Organozinc Reagents

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Issue 14/2016

Bontemps, Alexis; Mariaule, Gaëlle; Desbène-Finck, Stéphanie; Helissey, Philippe; Giorgi-Renault, Sylviane; Michelet, Véronique; Belmont, Philippe: Silver-Catalyzed Domino Hydroarylation/Cycloisomerization Reactions of 2-Alkynylquinoline-3-carbaldehydes: Access to (Hetero)arylpyranoquinolines

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Yamashita, Yasunobu; Kurihara, Tohru; Horiguchi, Takanobu; Miki, Atsushi; Shoji, Mitsuru; Sugai, Takeshi; Hanaya, Kengo: Ex Situ Enantioconvergent Approaches for the Effective Use of Undesired­ Isomers: Stereochemical Convergence of a Substrate with Multiple Chiral Centers and Recycling of a Decarboxylated Byproduct

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Issue 13/2016

Jungk, Phillip; Täufer, Tobias; Thiel, Indre; Hapke, Marko: Synthesis of Chiral Indenylcobalt(I) Complexes and Their Evaluation in Asymmetric [2+2+2] Cycloaddition Reactions

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Hutchby, Marc; Sedgwick, Adam C.; Bull, Steven D.: Orthogonally Protected Schöllkopf’s Bis-lactim Ethers for the Asymmetric Synthesis of α-Amino Acid Derivatives and Dipeptide Esters

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Issue 12/2016

Machara, Aleš; Endoma-Arias, Mary Ann A.; Císařova, Ivana; Cox, D. Phillip; Hudlický, Tomáš: Synthesis of Nororipavine and Noroxymorphone via N- and O-Demethylation of Iron Tricarbonyl Complex of Thebaine

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Issue 11/2016

Liu, Wenbo; Zhu, Youquan; Li, Chao-Jun: Pd-Catalyzed Homo Cross-Dehydrogenative Coupling of 2-Arylpyridines by Using I₂ as the Sole Oxidant

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Issue 09/2016

Pletz, Jakob; Berg, Bernhard; Breinbauer, Rolf: A General and Direct Reductive Amination of Aldehydes and Ketones with Electron-Deficient Anilines

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Issue 08/2016

Riml, Christian; Micura, Ronald: Synthesis of 5-Hydroxymethylcytidine- and 5-Hydroxymethyl­uridine-Modified RNA

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Issue 07/2016

Panther, Jesco; Müller, Thomas J. J.: Three- and Four-Component Syntheses of 3-Arylmethylindoles by Microwave-Assisted One-Pot Heck Isomerization–Fischer Indolization (Alkylation) (HIFI and HIFIA) Sequences

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Korotvička, Aleš; Frejka, David; Hampejsová, Zuzana; Císařová, Ivana; Kotora, Martin: Synthesis of Phenanthridines via a Rhodium-Catalyzed C–C Bond Cleavage Reaction of Biphenylene with Nitriles

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Issue 06/2016

Wöste, Thorsten H.; Muñiz, Kilian: Enantioselective Vicinal Diacetoxylation of Alkenes under Chiral Iodine(III) Catalysis

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Lindemann, Chris; Schneider, Christoph: Quinolizidine-Based Alkaloids: A General Catalytic, Highly Enantio- and Diastereoselective Synthetic Approach

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Issue 05/2016

Bernardim, Barbara; Couch, Erica D.; Hardman-Baldwin, Andrea M.; Burtoloso, Antonio C. B.; Mattson, Anita E.: Divergent Roles of Urea and Phosphoric Acid Derived Catalysts in Reactions of Diazo Compounds

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Issue 04/2016

Thapa, Surendra; Vangala, Adarsh S.; Giri, Ramesh: Copper-Catalyzed Negishi Coupling of Diarylzinc Reagents with Aryl Iodides

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Zhang, Yanqing; Xiao, Yuanjing; Zhang, Junliang: Gold(I)-Catalyzed Stereospecific [4+3]-Cycloaddition Reaction of 1-(Alk-1-ynyl)cyclopropyl Ketones with Nitrones: A Modular Entry to Enantioenriched 5,7-Fused Bicyclic Furo[3,4-d][1,2]oxazepines

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Issue 03/2016

Heid, Berenice; Plietker, Bernd: Iron-Catalyzed C-Allylating Partial Dearomatization of Naphthols

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Issue 02/2016

Asad, Sharif A.; Hossain, M. Mahmun: First Example of Intermolecular Palladium-Catalyzed Asymmetric Allylic Alkylation of Hydroxyacrylates: Synthesis of All-Carbon α-Aryl Quaternary Carbonyl Compounds

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Issue 01/2016

Marui, Kuniaki; Nomoto, Akihiro; Akashi, Haruo; Ogawa, Akiya: Green Oxidation of Amines to Imines Based on the Development of Novel Catalytic Systems Using Molecular Oxygen or Hydrogen Peroxide

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Issue 21/2015

Vasu, Dhananjayan; Yorimitsu, Hideki; Osuka, Atsuhiro: Base-Free Palladium-Catalyzed Cross-Coupling of Arylsulfonium Salts with Sodium Tetraarylborates

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Issue 20/2015

Jarzebski, Andreas; Bannwarth, Christoph; Tenten, Christina; Benkhäuser, Christian; Schnakenburg, Gregor; Grimme, Stefan; Lützen, Arne: Synthesis, Chiral Resolution, and Absolute Configuration of Functionalized Tröger’s Base Derivatives: Part III

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Issue 19/2015

Zhang, Feng; Min, Qiao-Qiao; Zhang, Xingang: Palladium-Catalyzed Heck-Type Difluoroalkylation of Alkenes with Functionalized Difluoromethyl Bromides

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Issue 17/2015

Morin, Marie S. T.; Vives, Thomas; Baslé, Olivier; Crévisy, Christophe; Ratovelomanana-Vidal, Virginie; Mauduit, Marc: Efficiency of Industrially Relevant Atropisomeric Diphosphines in Copper-Catalyzed 1,4-Asymmetric Conjugate Addition of Dialkylzincs to Cyclic or Acyclic Enones or Dienones

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Issue 16/2015

Skiredj, Adam; Beniddir, Mehdi A.; Joseph, Delphine; Bernadat, Guillaume; Evanno, Laurent; Poupon, Erwan: Harnessing the Intrinsic Reactivity within the Aplysinopsin Series for the Synthesis of Intricate Dimers: Natural from Start to Finish

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Issue 14/2015

Astruc, Didier; Wang, Dong; Deraedt, Christophe; Liang, Liyuang; Ciganda, Roberto; Ruiz, Jaime: Catalysis Inside Dendrimers

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Issue 11/2015

Teijaro, Christiana N.; Zhao, Senzhi; Kokkonda, Praveen; Andrade, Rodrigo B.: Total Syntheses of (–)-Alstolucines A, B, and F, (–)-Echitamidine, and (–)-N-Demethylalstogucine

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Issue 09/2015

De Coen, Laurens M.; Jatczak, Martyna; Muylaert, Koen; Mangelinckx, Sven; Stevens, Christian V.: Straightforward Synthesis of Functionalized Furo[3,4-d]pyrimidine-2,4-diones

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Issue 08/2015

Schienebeck, Casi M.; Song, Wangze; Smits, Angela M.; Tang, Weiping: Rhodium-Catalyzed Intermolecular [5+1] and [5+2] Cycloadditions Using 1,4-Enynes with an Electron-Donating Ester on the 3-Position

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Issue 07/2015

Delvos, Lukas B.; Oestreich, Martin: Temperature-Dependent Direct Enantioconvergent Silylation of a Racemic Cyclic Allylic Phosphate by Copper(I)-Catalyzed Allylic Substitution

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Issue 02/2015

Barrios, Francis J.; Springer, Brannon C.; Hazlitt, Robert A.; Colby, David A.: Effect of Substituents and Stability of Transient Aluminum–Aminals­ in the Presence of Nucleophiles

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