Synthesis

Issue eFirst

Gu, Guangxing; Wang, Chenyang; Zhao, Yanchuan: ¹⁹F-Labeled NMR Probes for the Detection and Discrimination of Nitrogen-Containing Analytes

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Pellissier, Hélène: The Use of Domino Reactions for the Synthesis of Chiral Rings

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Wang, Sichang; Zhou, Chengxiang; Han, Yunzi; Li, Miao; Ke, Congyu; Huang, Shenlin: Applications of Sulfonyl Fluorides in Organic Transformations

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Oh, Eun Hye; Kim, Hyun Jin; Han, Soo Bong: Recent Developments in Visible-Light-Catalyzed Multicomponent Trifluoromethylation of Unsaturated Carbon–Carbon Bonds

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Wei, Ming-Kai; Willis, Michael C.: The Catalytic Synthesis of Aza-Sulfur Functional Groups

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Ni, Qian; Chen, Yaqi; Ma, Yuanhong: Recent Progress in Base-Metal-Catalyzed Dearomative Reaction of N-Heteroarenes

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Zhao, Baoli; Liu, Yunyun: Step-Economical C–H Activation Reactions Directed by In Situ Amidation

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Lam, Long Yin; Ma, Cong: Recent Advances in Deoxygenative Thioether Synthesis Using Oxygenated Sulfur Surrogates

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Chen, Xu; Zhou, Xuesi; He, Jiawei; Liu, Xiang: Recent Advances in Photoinduced Borylation via N-Heterocyclic Carbene Boryl Radicals

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Li, Jianye; Li, Sijia; Liu, Shuting; Cui, Guohao; Zhang, Guozhu; Guo, Rui: Recent Advances in Transition-Metal-Catalyzed Enantioconvergent Transformations of Epoxides

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Breunig, Jamie L.; Pierce, Joshua G.: Synthetic Approaches toward the Batzelladine Class of Guanidinium Alkaloids

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Aida, Kazuhiro; Ota, Eisuke; Yamaguchi, Junichiro: Recent Advances in Single Electron Reduction Induced Ring Opening of N-Acyl Cyclic Amines

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Serbetci, Defne; Marraffa, Laura; Natho, Philipp; Andresini, Michael; Luisi, Renzo: A Practical Guide to SuFEx Chemistry: An Overview of S(VI)-SuFEx Linkers and Their Reactivity

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Kang, Wen-Jie; Tung, Chen-Ho; Wu, Li-Zhu: Energy-Demanding Redox Transformations via Electrophotocatalysis

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Zhou, Wen-Jun; Zhang, Yi-Han; Gui, Yong-Yuan; Sun, Liang; Yu, Da-Gang: Merging Transition-Metal Catalysis with Photoredox Catalysis: An Environmentally Friendly Strategy for C–H Functionalization

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Gong, Yiwei; Mulks, Florian F.: Recent Applications of Triphenylmethyl (Trityl) Cations in Synthesis

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Xiong, Ting; Hu, Zi-Jun; Wang, Ya-Qi; Weng, Jiang: Enhanced Synthesis of Sulfonyl Fluorides and Sulfamoyl Fluorides Using Fluorosulfonyl-Containing Radical Reagents

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Burianova, Valeria K.; McErlain, Holly; Sutherland, Andrew: Transition-Metal-Mediated Radiohalogenation using Aryl Boron Reagents

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Li, Heyin; Wang, Yi: Progress in Radical Fluorosulfonyl Reagents

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Zhang, Qiao; Zhu, Shou-Fei: Transition-Metal-Catalyzed C(sp³)–C(sp³) Cross-Coupling to Construct All-Carbon Quaternary Carbon Centers

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Kim, Kyungmi; Chae, Junghyun: Synthetic Applications of Symmetrical Disulfides and Their Synthesis from Non-thiolic Substrates

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Kim, Min Pyeong; Sahoo, Manoj Kumar; Chun, Joong-Hyun; Hong, Sung You: The First Decade of SuFEx Chemistry: Advancements in SuFEx Polymerization, Non-Canonical SuFEx Reactions, and SuFEx Radiochemistry

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Xie, Yang; Xuan, Jun: Advances in the Light-Promoted Transformations of N-Heterocyclic Carbene Ligated Boryl Radicals

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Takebe, Hiyori; Matsubara, Seijiro: Cuneanes as Potential Benzene Bioisosteres Having Chirality

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Geniller, Lilian; Taillefer, Marc; Jaroschik, Florian; Prieto, Alexis: Photocatalytic Strategies for the Synthesis of Xanthates and Their Analogues

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Liu, Yuyu; Yang, Shanxiu; Li, Pan; Wang, Hao; Cui, Xinjiang; Qian, Bo; Shi, Feng: Zinc-Catalyzed Carbon Dioxide Based Biodegradable Polycarbonate Synthesis

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Wu, Xiaomei; Yan, Xin; Qian, Deyun: Stereoselective Construction of Glycosides Enabled by Glycosyl/ Glycal Metal Species

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Issue Accepted Manuscripts

Jana, Sayan K.; Maji, Biplab: Nickel-Catalyzed Cross-Electrophile Coupling Reactions of Alcohols and Derivatives

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Yadav, Pooja; Berry, Shiwani; Bhalla, Aman: Chemical Methods for Construction of Spirocyclic β-Lactams and their Biological Importance

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Jabbarpoor, Maryam; Le, Christine: Carbamoyl Fluorides: A Platform to Interrogate Fluoride-Enabled Reactivity

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Issue 07/2025

Li, Xiang; Tu, Yong-Liang; Chen, Xiang-Yu: Recent Advances in Combining Photo- and N-Heterocycle Nitrenium Catalysis

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Wenninger, Marvin; Poulsen, Martin L.; Larsen, Megan E.; Hauser, Nicole M.: Recent Progress in the Synthesis and Glycosylation of Rare Sugars

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Palone, Andrea; Bietti, Massimo; Costas, Miquel: Enzymatic and Bio-Inspired Enantioselective Oxidation of Non-Activated C(sp³)–H Bonds

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Issue 06/2025

Gerlach, Tabea; Turner, Nicholas J.: Biocatalytic Dearomatisation Reactions

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Abd El Sater, Mariam; Popek, Lucas; Blanchard, Nicolas; Bizet, Vincent: Recent Advances in the Chemistry and Application of SF₅-Compounds

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Miguélez, Rubén; Arto, Omar; Rodríguez-Arias, Carlos; Barrio, Pablo: Gold(I)-Catalyzed Intramolecular C(sp3)–H Bond Functionalization

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Nagasawa, Shota; Iwabuchi, Yoshiharu: Recent Progress in Accessing Multi-functionalized Caged Hydrocarbons: En Route to Highly Functionalized Saturated (Bio)isosteres of Benzene Rings

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Fang, Zhuohan; Xu, Qian; Lu, Xuehe; Wan, Nianfeng; Yang, Wu-Lin: The Application of Bicyclo[1.1.1]pentane as a Bioisostere of the Phenyl Ring in Pharmaceutical Chemistry

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Issue 05/2025

Liu, Xigong; Liu, Lei: Catalytic Asymmetric Syntheses of 3-Monosubstituted Oxindoles

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Horwitz, Matthew A.: Discovery Process Chemistry: An Innovation Hub at the Interface of Academia, the Pharmaceutical Industry, and Contract Research Organizations

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Xie, Ke; Li, Ao; Kong, Bao-Rui; Chen, Zhi-Chao; Du, Wei; Chen, Ying-Chun: Recent Advances in Asymmetric Addition Reactions to Isatins

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Atriardi, Shafrizal R.; Anita, Yulia; Woo, Sang Kook: Harnessing Photoredox and Weak Brønsted Base Dual Catalysis for Selective C(sp³)–H Bond Activation

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Issue 04/2025

Martos, Mario; Bosque, Irene; Gonzalez-Gomez, Jose C.: Advances in Photoinduced Minisci-like Reactions

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Dong, Jianyang; Liao, Huijuan; Xue, Dong: Recent Advances in the Synthesis of Bicyclo[3.1.1]heptanes

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Issue 03/2025

Zheng, Cameron H. M.; Schafer, Laurel L.: Recent Advances in Saturated N-Heterocycle C–H Bond Functionalization for Alkylated N-Heterocycle Synthesis

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Li, Fei; Song, Jia-Wei; Han, Xue; Zhang, Cheng-Pan: Progress in Photocatalyzed Trifluoromethylthiolation and Trifluoromethylselenolation Reactions

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Burns, Sean M.; McClure, Timothy J.; Parikh, Seren G.; Schindler, Corinna S.: Synthesis and Biological Activity of Penaresidins A and B, Penazetidine A, and Related Analogues

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Issue 02/2025

Pandit, Soumen; Majumdar, Nilanjana: Catalytic Intermolecular [4+2]-Cycloaddition toward the Stereo­selective C2–C3 Annulation of Indoles

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Issue 24/2024

Bernardo, Olaya; García-Martínez, Patricia; Santamaría, Javier; López, Luis A.: Recent Advances in Gold-Catalyzed Transformations of Vinyldiazo Reagents

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Ramirez, Nieves P.; Waser, Jerome: Merging the Reactivity of (Pseudo)cyclic Hypervalent Iodine Reagents and Carbenes or Carbenoids

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Zhan, Xuan; He, Heng-Xian; Peng, Quanxin; Feng, Jian-Jun: Synthesis of Cyclobutanes and Cyclobutenes by Strain-Release-Driven Ring-Opening of Bicyclo[1.1.0]butanes

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Issue 23/2024

Villemure, Elisia; Wang, Yong; Zhou, Yuebiao; Wong, Alice R.; Nilewski, Christian: Tactics and Strategies for the Synthesis of Cereblon Ligands

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Sen, Abhijit; Yamada, Yoichi M. A.: Latest Developments on Palladium- and Nickel-Catalyzed Cross-Couplings Using Aryl Chlorides: Suzuki–Miyaura and Buchwald–Hartwig Reactions

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Issue 22/2024

Wu, Zhenwei; Feng, Xiaoming; Liu, Yangbin: Asymmetric Allylic Substitution Reactions Based on Relay Catalysis

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Yang, Kai; Chen, Lu; Su, Bo: Dual-Catalysis-Enabled Construction of Vicinal Stereogenic Centers through Diastereo- and Enantioselective Allylic Substitution

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Dang, Luzhen; Zhu, Chuan; Feng, Chao: Photoactive Ni-Complexes in Metallaphotoredox Catalysis: A Successful Match in C–C Cross-Coupling Reactions

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Sakuraba, Mahiro; Hoshimoto, Yoichi: Recent Trends in Triarylborane Chemistry: Diversification of Structures and Reactivity via meta-Substitution of the Aryl Groups

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Issue 21/2024

Sumino, Shuhei; Ryu, Ilhyong; Robert, Frédéric; Landais, Yannick: 1,2-Bis(phenylsulfonyl)ethylene (BPSE): A Potent Radical C2 Synthon Available in the Radical and Electron-Transfer-Based Organic Synthesis

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Issue 20/2024

Arepally, Sagar; Park, Jin Kyoon: Synthesis and Utilization of 1H-Indazole N-Oxides in the Production of C3-Functionalized 1H-Indazoles

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Moreau, Xavier; Ghiazza, Clément: Modern Dearomative Enlargement of Heteroaromatic Rings

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Issue 19/2024

Chang, Yu; Xing, Yuyang; Deng, Jian; Yan, Zifei; Luo, Guangsheng: Gas–Liquid Microchemical Oxidation for Continuous Synthesis Processes: A Short Review

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Song, Geyang; Dong, Jianyang; Song, Jiameng; Li, Gang; Xue, Dong: Transition-Metal-Catalyzed Direct Arylation of Ammonia

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Issue 18/2024

Yao, Minghan; Dong, Shanliang; Yusuf, Abdulla; Xu, Xinfang: Stepwise Carbene Transfer Reaction with Alkenes beyond Cyclopropanation

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Okamoto, Kazuhiro; Nagaki, Aiichiro: Flow Chemistry of Metal Carbenoid Species towards Selective Organic Synthesis

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Issue 17/2024

Roh, Byeongdo; Lee, Hong Geun: Stereospecific Palladium-Catalyzed Cross-Coupling of Alkylboron Compounds: A Short Account

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Bhanja, Rosalin; Bera, Shyamal Kanti; Mal, Prasenjit: Transition-Metal- and Photocatalyst-Free Photoinduced Formation of Carbon–Pnictogen (–N, –P) Bonds

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Issue 16/2024

Palomo, Claudio; Landa, Aitor; Oiarbide, Mikel: Catalytic Asymmetric Synthesis of α-Mono and α,α-Disubstituted 5- and 6-Membered α-Aza-lactams

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Agbaria, Mohamed; Egbaria, Nwar; Nairoukh, Zackaria: Unveiling Novel Synthetic Pathways through Brook Rearrangement

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Issue 15/2024

Zhang, Zhi-Xin; Hu, Tian-Qi; Ye, Long-Wu; Zhou, Bo: Organocatalytic Atroposelective Reactions of Alkynes

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Deshmukh, Dewal; Vagadiya, Nikunjkumar; Jagtap, Samadhan; Malasane, Pravin: Revolutionizing C–H Activation Reactions: Harnessing Green Solvents for Sustainable Catalysis

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Issue 14/2024

Dai, Peng-Fei; Li, Qiang-Qiang; Qu, Jian-Ping; Kang, Yan-Biao: Recent Developments on the Earth-Abundant-Metal-Catalyzed α,β-Dehydrogenation of Carbonyl Compounds

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Healy, Alan R.: Stereodivergent Carbon–Carbon Bond-Forming Reactions

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Issue 13/2024

Li, Xin; Song, Qiuling: Recent Progress on the Zweifel Olefination: An Update

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Issue 12/2024

Croll, Elizabeth A.; Kwon, Ohyun: Mechanism of the Mitsunobu Reaction: An Ongoing Mystery

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Harusawa, Shinya; Yoneyama, Hiroki; Usami, Yoshihide: Generation of Alkylidene Carbenes through Tetrazole Fragmentation: Recent Advances and Applications in Organic Synthesis

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Zou, Jia-Yu; Xu, Wan-Yi; Wang, Jie; Liu, Qi; He, Ying: Atroposelective Construction of Tetrasubstituted Axially Chiral Alkene Frameworks

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Issue 11/2024

Xu, Wei; Kumagai, Naoya: Recent Advances in Quinoline-Based Macrocycles: Synthesis, Properties, and Applications in Catalytic Reactions

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Hussain, Waseem A.; Parasram, Marvin: Recent Advances in Photoinduced Oxidative Cleavage of Alkenes

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Issue 10/2024

Vystavkin, Nikita; Barday, Manuel; Teskey, Christopher J.: Discovery of Divergent, Light-Controlled Catalysis Triggered by Ligand Photodissociation from Cobalt Complexes

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Kang, Eunsu; Joo, Jung Min: Pyrazolopyridine Ligands in Transition-Metal-Catalyzed C–C and C–Heteroatom Bond-Forming Reactions

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Issue 09/2024

Li, Mengran; Chen, Peng; Liu, Haoqi; Huang, Jian; Chen, Yang: Review of the Total Synthesis of the Aromatic Abietane Diterpenoid Ferruginol

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Bellemin-Laponnaz, Stéphane; Achard, Thierry: Recent Progress in Developing Thioether-Containing Ligands for Catalysis Applications

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Issue 08/2024

Zhao, Xian; Liu, Wei: Recent Advances in Transition-Metal-Catalyzed Sonogashira Cross-Coupling Reactions of Alkyl Electrophiles

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Wang, Zi-Lu; Xu, Yun-He: Progress on the Enantioselective Synthesis of Axially Chiral Cycloalkylidenes

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Issue 07/2024

Das, Ramanand; Das, Malati; Mukherjee, Debaraj; Kundu, Taraknath: Recent Advances on the Synthesis of C-Glycosides from 1,2-Glycals

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Kumar, Sumit; Khan, Yousuf; Arora, Aditi; Kumar, Manish; Rungta, Pallavi; Singh, Brajendra K.; Sharma, Vivek K.; Singh, Sunil K.: Advances in the Synthesis of Spirocyclic Nucleosides

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Issue 05/2024

Van Hoof, Max; Force, Guillaume; Lebœuf, David: Modern Macrolactonization Techniques

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Li, Tao; Chan, Albert S. C.; Meng, Shan-Shui: Direct Reductive Coupling of Nitro Compounds for the Synthesis of Advanced Amines

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Issue 03/2024

Singh, Sanjay; Hazra, Chinmoy K.: Recent Advancements in Typical Friedel–Crafts Alkylation Reactions Focused on Targeting Arene Nucleophiles

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Yang, Liangliang; Wang, Haiyang; Lang, Ming; Peng, Shiyong: Recent Advances on High-Order Dipolar Annulations of Donor–Acceptor Cyclopropanes/Cyclobutanes

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Issue 02/2024

Saito, Fumito: Recent Developments on the Synthesis of Sulfoxides via Sulfenate Anions

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Morrison, Kathleen M.; Stradiotto, Mark: Advances in Nickel-Catalyzed O-Arylation of Aliphatic Alcohols and Phenols with (Hetero)aryl Electrophiles

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Issue 01/2024

Takebe, Hiyori; Matsubara, Seijiro: Decoration on Cubane with an Awareness of Chirality: Development of Substituted Cubane Syntheses

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Bera, Satabdi; Jana, Subhenira; Samanta, Rajarshi: Recent Progress on Copper-Catalyzed C–C Bond Formation via C(sp²)–H Insertions Using Diazo and Related Compounds

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Issue 24/2023

Jiang, Binyang; Shi, Shi-Liang: C–H Functionalization of Arenes via NHC-Supported Ni/Al Bimetallic Catalysis

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Chen, Xia; Guo, Hong-Yu; Zhou, Xiao-Yu; Bao, Ming: Palladium-Catalyzed Homo-Dimerization of Terminal Alkynes

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Issue 23/2023

Shi, Chong-Yang; Zhou, Bo; Teng, Ming-Yu; Ye, Long-Wu: Recent Advances in the Asymmetric Doyle–Kirmse Reaction

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Pramanik, Milan; Melen, Rebecca L.: Activation of Diazo Compounds by Fluorinated Triarylborane Catalysts

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Issue 22/2023

Aquilina, Jake M.; Smith, Myles W.: Synthetic Studies toward the Myrioneuron Alkaloids

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Gualandi, Andrea; Calogero, Francesco; Pinosa, Emanuele; Corbisiero, Dario; Cozzi, Pier Giorgio: Developing Organometallic Nucleophilic Reagents Via Photoredox Catalysis

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Issue 20/2023

Tibbetts, Joshua D.; Askey, Hannah E.; Cao, Qiao; Grayson, James D.; Hobson, Sophie L.; Johnson, George D.; Turner-Dore, Jacob C.; Cresswell, Alexander J.: Decarboxylative, Radical C–C Bond Formation with Alkyl or Aryl Carboxylic Acids: Recent Advances

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Issue 19/2023

Xie, Dezheng; Chen, Ziyi; Wang, Chun-Jiang; Dong, Xiu-Qin: Recent Advances in the Asymmetric Catalytic Synthesis of Phosphonates with an α-Chiral Center

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Tummatorn, Jumreang; Ruchirawat, Somsak; Thongsornkleeb, Charnsak: Halogenative Annulation Reactions of Alkyne-Tethered N- and O-Containing Arenes: Methods for Accessing Aryl-Fused Halogenated N- and O-Heterocycles

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Issue 18/2023

Chen, Huijie; Mo, Yiming: Accelerated Electrosynthesis Development Enabled by High-Throughput Experimentation

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Chen, Xiaohui; Wang, Neng-Zhong; Cheng, Ya-Min; Kong, Xianqiang; Cao, Zhong-Yan: Recent Advances in Electro- or Photochemical Driven Transformations via Cleavage of the C–N Bond of Quaternary Ammonium Salts

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Qin, Jing-Hao; Nan, Ning; Li, Jin-Heng: Electrochemical Difunctionalization of Alkenes

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Wang, Yuying; Liu, Siyuan; Han, Jiangsheng; Wang, Ling; Chen, Jianbin: Photoelectrochemical Cerium Catalysis via Ligand-to-Metal Charge Transfer: A Rising Frontier in Sustainable Organic Synthesis

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Wang, Qian; Liu, Han-Fu; Ren, Sai-Yan; He, Mu-Xue; Pan, Ying-Ming: Research Advances in Electrochemical Synthesis of Spirocyclic Skeleton Compounds

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Zheng, Weipeng; Tao, Yongsheng; Ma, Wan; Lu, Qingquan: Asymmetric Organic Electrochemistry Catalyzed by Transition Metals

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Zhang, Cai; Chen, Demao; Wan, Jie-Ping; Liu, Yunyun: Recent Advances in Electrochemical Cascade Cyclization Reactions

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Faisca Phillips, Ana Maria; Pombeiro, Armando J. L.: Catalytic Enantioselective Synthesis Enabled by Electrochemistry

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Issue 17/2023

Barker, Timothy J.; Bogatkevich, Andrew; Crowder, Dallas W.; Gierszal, Sophia G.; Hayes, Jacob C.; Hollerbach, Michael R.; Russell, Richard W.: Reactions of Benzylboronate Nucleophiles

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Issue 16/2023

Campbell, Aaron D. G.; Armstrong, Roly J.: Synthetic Strategies to Control C–N Atropisomerism in Acyclic Amines and Amides

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Juaristi, Eusebio; Avila-Ortiz, C. Gabriela: Salient Achievements in Synthetic Organic Chemistry Enabled by Mechanochemical Activation

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Issue 15/2023

Liu, Yudong; Woerpel, K. A.: Uncatalyzed Carbometallation Involving Group 13 Elements: Carboboration and Carboalumination of Alkenes and Alkynes

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Rizzacasa, Mark; Ricca, Michael: Chemistry and Biology of Acyloin Natural Products

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Marchese, Austin D.; Mirabi, Bijan; Lautens, Mark: Recent Developments of Palladium- and Rhodium-Catalyzed β-Carbon Elimination Strategies

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Issue 14/2023

Marco-Contelles, José: The Synthesis of 3-Nitrooxypropanol, a Methane Mitigant for Sustainable Farming with Environmental Impact: A Review

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Shi, Chong-Yang; Zhou, Bo; Teng, Ming-Yu; Ye, Long-Wu: Recent Advances in Asymmetric [1,2]-Stevens-Type Rearrangement via Metal Carbenes

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Issue 13/2023

Cala, Lara; Gaviria, Mario A.; Kim, Scott L.; Vogel, Trenton R.; Schindler, Corinna S.: Recognition of Symmetry as a Powerful Tool in Natural Product Synthesis

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Issue 12/2023

Wessig, Pablo; Lehmann, Max: [1,3]-Dioxolo[4,5-f]benzodioxole (DBD) Fluorescent Dyes; Synthesis, Properties, and Applications

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Aradi, Klára; Kiss, Loránd: Recent Advances in the Trifluoromethylation Reactions of Isonitriles To Construct CF₃-Substituted N-Heterocycles

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Issue 11/2023

Ahmed, Jasimuddin; Haug, Graham C.; Nguyen, Viet D.; Porey, Arka; Trevino, Ramon; Larionov, Oleg V.: Catalytic Dienylation: An Emergent Strategy for the Stereoselective Construction of Conjugated Dienes and Polyenes

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Simonet-Davin, Raphaël; Waser, Jerome: Azidation with Hypervalent Iodine Reagents

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Chamness, Stephen A.; Traficante, Emily F.; Vogel, Trenton R.; Schindler, Corinna S.: Synthetic Strategies Towards the Meroterpenoids Cochlearols A and B from Ganoderma cochlear

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Issue 10/2023

Ortiz, Eliezer; Saludares, Connor; Wu, Jessica; Cho, Yoon; Santana, Catherine G.; Krische, Michael J.: Carbonyl Allylation and Crotylation: Historical Perspective, Relevance to Polyketide Synthesis, and Evolution of Enantioselective Ruthenium-Catalyzed Hydrogen Auto-Transfer Processes

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Kranidiotis-Hisatomi, Nektarios; Oestreich, Martin: Advances in Enantioconvergent Transition-Metal-Catalyzed Cross-Coupling Reactions of Racemic α-Silyl and α-Boryl Reagents

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Issue 09/2023

Yan, Xiaoqiang; Wang, Jun: Advances in Exploring Cyclopentadienyl (Cp) Rhodium Catalysts Featuring Diastereotopic or Enantiotopic Cp Faces for Asymmetric C–H Activation

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Issue 08/2023

Wang, Zhan-Yong; Li, Jiarong; Wang, Nan; Liu, Hong; Ding, Wanli; Wang, Kai-Kai: A Decade of Advances of CS₂/Amines in Three-Component Reactions

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Gan, You F.; Li, Yuan Y.; Chen, Xiao Q.; Guo, Yu Y.; Wang, Rui: Recent Advances in Quinone Methide Chemistry for Protein-Proximity Capturing

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Issue 07/2023

Lu, Peng; Lu, Zhan: Earth-Abundant Transition Metal Catalyzed Asymmetric Hydrogenation of Minimally Functionalized Alkenes

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Shi, Yongjie; Rong, Nianxin; Zhang, Xumu; Yin, Qin: Synthesis of Chiral Primary Amines via Enantioselective Reductive Amination: From Academia to Industry

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Issue 06/2023

Doi, Ryohei; Zhou, Yuyang; Ogoshi, Sensuke: Transformation of Tetrafluoroethylene Using Transition-Metal Complexes

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Yang, Ying-Hui; Pang, Xiaobo; Shu, Xing-Zhong: Transition-Metal-Catalyzed Cross-Coupling of Chlorosilanes

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Issue 05/2023

Koide, Kazunori: Mechanistic and Synthetic Studies of Biaryl Birch Reductions

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Wen, Wei; Guo, Qi-Xiang: Recent Advances in Chiral Aldehyde Catalysis for Asymmetric Functionalization of Amines

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Issue 04/2023

Zhou, Min-Jie; Liu, Guixia; Xu, Chen; Huang, Zheng: Acceptorless Dehydrogenation of Aliphatics, Amines, and Alcohols with Homogeneous Catalytic Systems

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Hilt, Gerhard: The Synthetic Approaches to 1,2-Chlorohydrins

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Issue 03/2023

Mahanty, Kingshuk; Halder, Atreyee; Maiti, Debabrata; De Sarkar, Suman: Recent Developments in the Electroreductive Functionalization of Carbon–Halogen Bonds

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Kobayashi, Shoji: Total Synthesis of Geranyl-Resorcinols Isolated from Mushrooms of Genus Hericium

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Issue 02/2023

Didier, Dorian: Forging C–C Bonds through Intramolecular Oxidative Coupling of Organoborates – An Overview

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Dupeux, Aurélien; Michelet, Veronique: Chiral 1,4-Oxazino[4,3-a]indoles as a Challenging Scaffold: Syntheses and Properties

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Chen, Wenzhang; Vincent, Stéphane P.: Copillar[5]arene Chemistry: Synthesis and Applications

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To, Hoang-Minh; Malets, Oleksii; Mazur, Maryna; Mykhailenko, Olha; Kompaniiets, Olena; Ollevier, Thierry: Halodiazirines as Valuable Reagents for the Synthesis of Halocyclo­propanes

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Issue 01/2023

Feray, Laurence; Bertrand, Michèle P.; Galibert-Guijarro, Aurélien: α-Haloenamides: Synthesis and Subsequent Transformations

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Lenarda, Anna; Wirtanen, Tom; Helaja, Juho: Carbon Materials as Catalytic Tools for Oxidative Dehydrogenations and Couplings in Liquid Phase

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Bage, Andrew D.; Nicholson, Kieran; Hunt, Thomas A.; Langer, Thomas; Thomas, Stephen P.: Transborylation-Enabled Boron Catalysis

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Issue 24/2022

Tayama, Eiji: Recent Advances in the Generation of Onium Ylides for Sommelet–Hauser Rearrangements

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Huang, Wei-Sheng; Wang, Qing; Yang, Hua; Xu, Li-Wen: State-of-the-Art Advances in Enantioselective Transition-Metal-Mediated Reactions of Silacyclobutanes

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Paul, Biprajit; Paul, Hrishikesh; Chatterjee, Indranil: Photoredox-Mediated Desulfonylative Radical Reactions: An Excellent Approach Towards C–C and C–Heteroatom Bond Formation

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Issue 23/2022

Yang, Meng-Meng; Wang, Si; Dong, Zhi-Bing: Recent Advances for Chiral Sulfoxides in Asymmetric Catalysis

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Morofuji, Tatsuya; Kano, Naokazu: Recent Progress in C(sp²)–C(sp²) Bond Formation Using Ligand Coupling on Sulfur(IV)

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Issue 22/2022

Yin, Changzhen; Wang, Miao; Cai, Zhenxi; Yuan, Bojun; Hu, Peng: Visible-Light-Induced Iron Group Metal Catalysis: Recent Developments in Organic Synthesis

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Rombach, David; Wagenknecht, Hans-Achim: Photochemical Activation of Sulfur Hexafluoride: A Tool for Fluorination and Pentafluorosulfanylation Reactions

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Su, Hang; Pedersen, Christian Marcus: Ring-System-Based Conformational Switches and their Applications in Sensing and Liposomal Drug Delivery

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Issue 21/2022

Xi, Yang; Chen, Yifeng: Recent Advances in Transition-Metal-Catalyzed Asymmetric Functionalization of Enamides

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Jamshidi, Mahdi; Fastie, Cornelius; Hilt, Gerhard: Applications of Alternating Current/Alternating Potential Electro­lysis in Organic Synthesis

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Issue 20/2022

Cheng, Li; Lin, Quan; Chen, Yunrong; Gong, Hegui: Recent Progress on Transition-Metal-Mediated Reductive C(sp³)–O Bond Radical Addition and Coupling Reactions

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Bensberg, Kathrin; Kirsch, Stefan F.: Reactions with Geminal Diazides: Long Known, Full of Surprises, and New Opportunities

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Issue 19/2022

Reyes, Efraim; Prieto, Liher; Carrillo, Luisa; Uria, Uxue; Vicario, Jose L.: Recent Developments in Transannular Reactions

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Sani, Monica; Zanda, Matteo: Recent Advances in the Synthesis and Medicinal Chemistry of SF₅ and SF₄Cl Compounds

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Issue 18/2022

Chen, Xiao-Yue; Wu, Yichen; Wang, Peng: Recent Advances in Thianthrenation/Phenoxathiination Enabled Site-Selective Functionalization of Arenes

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Vaishya, V.; Singhal, R.; Kriplani, T.; Pilania, M.: Recent Advances in Transition-Metal-Catalyzed Reactions of N-Tosylhydrazones

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Issue 17/2022

Shintani, Ryo: Rhodium-Catalyzed Stitching Reactions for the Facile Synthesis of Extended π-Conjugated Compounds

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Hirano, Koji: Catalytic Asymmetric Construction of CF₃-Substituted Chiral sp³ Carbon Centers

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Issue 15/2022

Wan, Dan-Hong; Yang, Hai-Bin: Research Progress on N-Heterocyclic Carbene Catalyzed Reactions for Synthesizing Ketones through Radical Mechanism

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Zhao, Hongyi; Pan, Huanhuan; Yao, Yi; Huang, Jian; Chen, Yang: Recent Advances in the Total Synthesis of Cephalotane-Type Norditerpenoids from Cephalotaxus sinensis

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Hoque, Md Emdadul; Hassan, Mirja Md Mahamudul; Haldar, Chabush; Dey, Sayan; Guria, Saikat; Chaturvedi, Jagriti; Chattopadhyay, Buddhadeb: Catalyst Engineering through Heterobidentate (N–X-Type) Ligand Design for Iridium-Catalyzed Borylation

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Issue 14/2022

Zhu, Haoran; Driver, Tom G.: Recent Advances to Mediate Reductive Processes of Nitroarenes Using Single-Electron Transfer, Organomagnesium, or Organozinc Reagents

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Ferreira de Paiva, Walysson; de Freitas Rego, Yuri; de Fátima, Ângelo; Fernandes, Sergio Antonio: The Povarov Reaction: A Versatile Method to Synthesize Tetrahydroquinolines, Quinolines and Julolidines

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Issue 13/2022

Borys, Andryj M.; Hevia, Eva: Mechanisms of the Nickel-Catalysed Hydrogenolysis and Cross-Coupling of Aryl Ethers

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Depa, Wojciech; Bisek, Bartosz; Górecki, Marcin; Michalak, Michał: Epoxydibenzo[b,f][1,5]diazocines: From a Hidden Structural Motif to an Efficient Solvent-Free Synthetic Protocol

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Issue 12/2022

Wang, Wanshu; Gao, Lu; Song, Zhenlei: Synthetic Approaches for the Construction of Five- and Six-Membered Silaazacycles

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Nishimoto, Yoshihiro; Sugihara, Naoki; Yasuda, Makoto: C(sp³)–F Bond Transformation of Perfluoroalkyl Compounds Mediated by Visible-Light Photocatalysis: Spin-Center Shifts and Radical/Polar Crossover Processes via Anionic Intermediates

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Beller, Marc Paul; Koert, Ulrich: Synthetic Studies on Chromone Natural Products: The Preusso­chromones

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Issue 11/2022

Hassan, Diandra Safira; Kariapper, F. Safia; Lynch, Ciarán C.; Wolf, Christian: Accelerated Asymmetric Reaction Screening with Optical Assays

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Kawamoto, Takuji; Kamimura, Akio: Recent Advances in Radical Reactions of Vinyl Triflates and Their Derivatives

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Zheng, Yue; Tian, Lifang; Ramadoss, Velayudham; Zhang, Hui; Zhu, Li-Li; Wang, Yahui: Recent Developments in N²-Selective Functionalizations of 1,2,3-Triazoles

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Liu, Ying-Ying; Sun, Shao-Han; Min, Xiang-Ting; Wan, Boshun; Chen, Qing-An: Transition-Metal-Catalyzed Decarbonylative Functionalization of Phthalimides

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Issue 10/2022

Shiozuka, Akira; Sekine, Kohei; Kuninobu, Yoichiro: Photoinduced Organic Reactions by Employing Pyrene Catalysts

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Tsuchiya, Naoki; Sheppard, Tom D.; Nishikata, Takashi: Tertiary Alkylative Suzuki–Miyaura Couplings

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Issue 09/2022

Sun, Xin; Li, Bi-Jie: Acyclic Quaternary Carbon Stereocenters through Transition-Metal-Catalyzed Enantioselective Functionalization of Unsaturated Hydrocarbons

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Sweet, Jamie S.; Knipe, Peter C.: Catalytic Enantioselective Synthesis of C–N Atropisomeric Heterobiaryls

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Ye, Zhi-Shi; Li, Jin-Chen; Wang, Gang: Transition-Metal-Catalyzed Enantioselective Synthesis of Indoles from 2-Alkynylanilines

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Issue 08/2022

Whalley, David M.; Greaney, Michael F.: Recent Advances in the Smiles Rearrangement: New Opportunities for Arylation

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Liu, Ting; Liu, Jian; He, Jin; Hong, Yu; Zhou, Han; Liu, Yin-Ling; Tang, Shi: Recent Advances in Photoinduced Perfluoroalkylation Using Perfluoroalkyl Halides as the Radical Precursors

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Yuan, Wei; He, Chuan: Enantioselective C–H Functionalization toward Silicon-Stereogenic Silanes

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Diesendorf, Nina; Heinrich, Markus R.: Current Advances in Meerwein-type Radical Alkene Functionalizations

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Yan, Biwei; Guo, Wusheng: Recent Advances in Decarboxylative Conversions of Cyclic Carbonates and Beyond

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Issue 07/2022

Katayama, Yuri; Mitsunuma, Harunobu; Kanai, Motomu: Recent Progress in Chromium-Mediated Carbonyl Addition Reactions

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Andrews, Jonathan A.; Willis, Michael C.: DABSO – A Reagent to Revolutionize Organosulfur Chemistry

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Qin, Xu-Long; Xu, Li-Jun; Han, Fu-She: Recent Advances in Organocatalyzed Asymmetric Reduction of Prochiral Ketones: An Update

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Ding, Bo; Xue, Qilin; Jia, Shihu; Cheng, Hong-Gang; Zhou, Qianghui: Recent Advances in Catalytic Nonenzymatic Kinetic Resolution of Tertiary Alcohols

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Issue 06/2022

Tian, Ze-Yu; Ma, Yu; Zhang, Cheng-Pan: Alkylation Reactions with Alkylsulfonium Salts

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Ahsanullah, Ahsanullah; Hassan, Abbas; Ansari, Farzana L.; Rademann, Jörg: Integration of C-Acylation in the Solid-Phase Synthesis of Peptides and Peptidomimetics Employing Meldrum’s Acid, Phosphorus, and Sulfur Ylides

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Hamdane, Yousra; Poupart, Julien; Lubell, William D.: N-Amino-imidazol-2-one (Nai) Residues as Tools for Peptide Mimicry: Synthesis, Conformational Analysis and Biomedical Applications

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Yang, Zhao-Ying; Zhang, Ming; Wang, Xiao-Chen: Synthesis and Applications of Chiral Bicyclic Bisborane Catalysts

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Paris, Timothy J.; Willand-Charnley, Rachel: Modern Synthesis and Chemistry of Stabilized Ketene N,O-Acetals

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Xu, Houchao; Dickschat, Jeroen S.: Mechanistic Investigations on Microbial Type I Terpene Synthases through Site-Directed Mutagenesis

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Issue 05/2022

Ma, Xiao-Yan; Shao, Fu-Qiang; Hu, Xinjun; Liu, Xingyong: Progress in the Synthesis of N-Acyl-N,O-acetals

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Miller, Eric R.; Scheidt, Karl A.: Enantioselective Syntheses of Yohimbine Alkaloids: Proving Grounds for New Catalytic Transformations

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Lu, Zheng; Shang, Mingzhou; Lu, Hongjian: Organic Sulfinic Acids and Salts in Visible Light-Induced Reactions

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Lamberth, Clemens: Organic Isocyanates and Isothiocyanates: Versatile Intermediates in Agrochemistry

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Winterson, Bethan; Patra, Tuhin; Wirth, Thomas: Hypervalent Bromine(III) Compounds: Synthesis, Applications, Prospects

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Issue 03/2022

Wang, Yongtao; Yao, Jia; Li, Haoran: Aerobic Oxidations via Organocatalysis: A Mechanistic Perspective

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Su, Yong-Liang; Doyle, Michael P.: Application of α-Aminoalkyl Radicals as Reaction Activators

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Lee, Kyu Ree; Lee, Yu Lim; Choi, Kyu In; Lee, Sang-gi: Cooperative Rh(II)/Pd(0) Dual Catalysis for the Synthesis of Carbo- and Heterocyclic Compounds

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Goebel, Jonas F.; Zeng, Zhongyi; Gooßen, Lukas J.: Biaryl Synthesis via Electrooxidative Transition-Metal-Catalyzed C–H Activation

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Shin, Inji; Lim, Hee Nam; Hong, Wan Pyo: 1,4-Azaborines: Origin, Modern Synthesis, and Applications as Optoelectronic Materials

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Zhong, Sishi; Xu, Lei; Cai, Yunfei: Recent Advances on Piancatelli Reactions and Related Cascade Processes

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Issue 02/2022

Wei, Baosheng; Knochel, Paul: Recent Advances in Cross-Couplings of Functionalized Organozinc Reagents

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Oroz, Paula; Avenoza, Alberto; Busto, Jesús H.; Corzana, Francisco; Zurbano, María M.; Peregrina, Jesús M.: Strategies for the Synthesis of Selenocysteine Derivatives

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Glueck, David S.: Asymmetric Synthesis of P-Stereogenic Secondary Phosphine ­Oxides (SPOs)

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Zhang, Yong; Sun, Wenxuan; Li, Chao: Nickel-Catalyzed Paired Electrochemical Cross-Coupling of Aryl Halides with Nucleophiles

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Fokin, Igor; Kuessner, Kai-Thorben; Siewert, Inke: Transition Metal Complex Catalyzed Photo- and Electrochemical (De)hydrogenations Involving C=O and C=N Bonds

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Feng, Yanping; Ye, Xiajuan; Huang, Dayun; Guo, Sheng-rong: α-Csp³–H Bond Functionalization of Simple Ethers in Radical Reactions

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Issue 01/2022

Cui, Shu-Qiang; Liao, Wei-Wei: Recent Advances in Transition-Metal-Catalyzed C–H Addition to Nitriles

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He, Peng; Hu, Meng-Yang; Zhang, Xin-Yu; Zhu, Shou-Fei: Transition-Metal-Catalyzed Stereo- and Regioselective Hydrosilylation of Unsymmetrical Alkynes

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Li, Qing-Zhu; Zou, Wen-Lin; Jia, Zhi-Qiang; Li, Jun-Long: Recent Advances on Annulation Reactions with Allyl and Propargyl Sulfonium Salts

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Williams, Dean; Jamshidi, Mohammad P.; Sauvageau, Janelle: Pathogen-Associated Molecular Patterns: The Synthesis of Heptose Phosphates and Derivatives

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Jia, Jie; Hu, Fangdong; Xia, Ying: Transition-Metal-Catalyzed Nucleophilic Dearomatization of Electron-Deficient Heteroarenes

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Ghorai, Sourav; Lee, Daesung: Strain-Induced Transformations of Bicyclo[3.1.0]hex-1-enes

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Issue 24/2021

Melngaile, Renate; Veliks, Janis: Synthetic Applications of Monofluoromethylsulfonium Salts

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Orlandi, Manuel; Escudero-Casao, Margarita; Licini, Giulia: Transition-Metal-Catalyzed Enantioselective α-Arylation of Carbonyl Compounds to Give Tertiary Stereocenters

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Empel, Claire; Jana, Sripati; Koenigs, Rene M.: Advances in [1,2]-Sigmatropic Rearrangements of Onium Ylides via Carbene Transfer Reactions

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Qin, Yu-Nan; Zhang, Chen; Li, Quan; Du, Guang-Yan: Development of Synthetic Strategies to Access Optically Pure ­Feringa’s Motors

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Fontaine, Frédéric-Georges; Desrosiers, Vincent: Boron Lewis Pair Mediated C–H Activation and Borylation

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Issue 23/2021

Varga, Bálint; Csenki, János T.; Tóth, Balázs L.; Béke, Ferenc; Novák, Zoltán; Kotschy, András: Application of Industrially Relevant HydroFluoroOlefin (HFO) Gases in Organic Syntheses

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Xiong, Yang; Li, Sijia; Xiao, Haijing; Zhang, Guozhu: Recent Advances in Visible-Light-Promoted Copper Catalysis in Organic Reactions

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Yu, Xinhui; Zhang, Ting; Liu, Jitian; Li, Xiaoxun: Recent Advances in the Construction of Quaternary Stereocenters via Palladium-Catalyzed Decarboxylative Asymmetric Allylic Alkylation

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Uçar, Sefa; Daştan, Arif: Recent Advances in the Transition-Metal-Free Arylation of Hetero­arenes

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Liu, Le; Duan, Xin-Hua; Guo, Li-Na: Recent Advance in Iminyl Radical Triggered C–H and C–C Bond Functionalization of Oxime Esters via 1,5-HAT and β-Carbon Scission

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Liao, Jin-Xi; Hu, Zhen-Ni; Liu, Hui; Sun, Jian-Song: Advances in the Semi-Synthesis of Triterpenoids

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Issue 21/2021

Sorrentino, Jacob P.; Altman, Ryan A.: Fluorine-Retentive Strategies for the Functionalization of gem-Difluoroalkenes

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Tao, Zhong-Lin; Denmark, Scott E.: Catalytic, Enantioselective Diamination of Alkenes

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Baumann, Marcus; Moody, Thomas S.; Smyth, Megan; Wharry, Scott: Evaluating the Green Credentials of Flow Chemistry towards Industrial Applications

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Liu, Weilong; Winssinger, Nicolas: Synthesis of α-exo-Methylene-γ-butyrolactones: Recent Developments and Applications in Natural Product Synthesis

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Armengol-Relats, Helena; Mato, Mauro; Escofet, Imma; Echavarren, Antonio M.: Assembling Complex Structures through Cascade and Cycloaddition Processes via Non-Acceptor Gold or Rhodium Carbenes

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Issue 20/2021

Fershtat, Leonid L.; Teslenko, Fedor E.: Five-Membered Hetarene N-Oxides: Recent Advances in Synthesis and Reactivity

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Wang, Zhan-Yong; Guo, Qi; Xu, Shaohong; Wang, Kai-Kai: Nucleophilic H-Phosphites, H-Phosphinates, and H-Phosphine Oxides in Organic Reactions

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Ju, Guodong; Tu, Guanglian; Zhao, Yingsheng: Recent Advances in Transition-Metal-Catalyzed Selective C–H Alkoxycarbonyldifluoromethylation Reactions of Aromatic Substrates

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Li, Shen-Huan; Long, Cheng-Yu; Yang, Xin-Ge; Wang, Xue-Qiang: Recent Progress in Amination Enabled by Transition-Metal-Free C(sp²)–O/C(sp²)–S Bond Cleavage Strategy

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Issue 19/2021

Kieslich, David; Christoffers, Jens: Cyanide Anions as Nucleophilic Catalysts in Organic Synthesis

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Slivka, Mikhailo; Onysko, Mikhailo: The Use of Electrophilic Cyclization for the Preparation of Condensed Heterocycles

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Sako, Makoto; Arisawa, Mitsuhiro: Recent Advances in Metal-Nanoparticle-Catalyzed Coupling Reactions Assisted by Microwave Irradiation

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Gao, Biwen; Deng, Danfeng; Huang, Dayun; Sun, Xiangyu: Recent Advances in the Tandem Difunctionalization of Alkynes: Mechanism-Based Classification

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Issue 16/2021

Roche, Stéphane P.: In the Pursuit of (Ald)Imine Surrogates for the Direct Asymmetric Synthesis of Non-Proteinogenic α-Amino Acids

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Majdecki, Maciej; Niedbała, Patryk; Tyszka-Gumkowska, Agata; Jurczak, Janusz: Assisted by Hydrogen-Bond Donors: Cinchona Quaternary Salts as Privileged Chiral Catalysts for Phase-Transfer Reactions

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Zhang, Sheng; Findlater, Michael: Cobalt-Catalyzed Isomerization of Alkenes

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Youssef-Saliba, Sparta; Vallée, Yannick: Sulfur Amino Acids: From Prebiotic Chemistry to Biology and Vice Versa

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Issue 15/2021

Jurinic, Carla K.; Belladona, Andrei L.; Schumacher, Ricardo F.; Godoi, Benhur: Diorganyl Dichalcogenides and Copper/Iron Salts: Versatile Cyclization System To Achieve Carbo- and Heterocycles from Alkynes

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Rubtsov, Aleksandr E.; Malkov, Andrei V.: Recent Advances in the Synthesis of 2,2′-Bipyridines and Their Derivatives

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Zhang, Qiaoling; Xi, Jufang; Ze, He; Qingle, Zeng: Syntheses and Transformations of Sulfinamides

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Rehpenn, Andreas; Walter, Alexandra; Storch, Golo: Molecular Editing of Flavins for Catalysis

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Issue 14/2021

Pedrood, Keyvan; Montazer, Mohammad Nazari; Larijani, Bagher; Mahdavi, Mohammad: Recent Advances in the Synthesis of Heterocycles by the Aza-Wittig Reaction

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Li, Qingjiang; Guo, Zhongwu: Enzymatic Synthesis of Glycosphingolipids: A Review

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Kahlert, Lukas; Schotte, Carsten; Cox, Russell J.: Total Mycosynthesis: Rational Bioconstruction and Bioengineering of Fungal Natural Products

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Livingstone, Keith; Little, Gemma; Jamieson, Craig: Recent Advances in the Generation of Nitrilium Betaine 1,3-Dipoles

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Issue 13/2021

Liu, Jiaming; Chen, Ming: 1,3-Bifunctional Nucleophilic Allylation Reagents: Preparative Methods and Synthetic Applications

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Inoa, Joan; Dominici, Grecia; Eldabagh, Reem; Foley, Jonathan J.; Xing, Yalan: Synthetic Applications and Computational Perspectives on Eosin Y Induced Direct HAT Process

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Issue 12/2021

Neri, Raul; Bossmann, Stefan H.: Isoselenocyanates: Synthesis and Their Use for Preparing Selenium-Based Heterocycles

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Zu, Bing; Guo, Yonghong; Ke, Jie; He, Chuan: Transient- and Native-Directing-Group-Enabled Enantioselective C–H Functionalization

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Issue 11/2021

Ashikari, Yosuke; Nagaki, Aiichiro: Homogeneous Catalyzed Aryl–Aryl Cross-Couplings in Flow

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Issue 10/2021

Zhao, Jia-Jia; Zhang, Hong-Hao; Yu, Shouyun: Enantioselective Radical Functionalization of Imines and Iminium Intermediates via Visible-Light Photoredox Catalysis

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Zheng, Songlin; Hu, Yuanyuan; Yuan, Weiming: Recent Advances in C(sp³)–C(sp³) Cross-Coupling via Metalla­photoredox Strategies

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Mazumdar, Wrickban; Driver, Tom G.: Recent Advances in the Development of Catalytic Methods that Construct Medium-Ring Lactams, Partially Saturated Benzazepines and Their Derivatives

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Issue 09/2021

Singh, Pushpinder; Batra, Aanchal; Singh, Kamal Nain; Mritunjay, Mritunjay: Transition-Metal-Free Strategies for the Synthesis of C-1 Aryl-Substituted Tetrahydroisoquinolines

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Li, Yanjun; Ye, Ziqi; Cai, Jiaxin; Gong, Lei: Visible-Light-Promoted Asymmetric Catalysis by Chiral Complexes of First-Row Transition Metals

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Issue 08/2021

Bartoccini, Francesca; Piersanti, Giovanni: Synthesis and Reactivity of Uhle’s Ketone and Its Derivatives

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Yu, Hsien-Cheng; Mankad, Neal P.: Catalytic Reactions by Heterobimetallic Carbonyl Complexes with Polar Metal–Metal Interactions

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Yu, Jingxun; Luan, Xinjun: Hydroxylamines as One-Atom Nitrogen Sources for Metal-Catalyzed Cycloadditions

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Issue 07/2021

Zhao, Xuchen; Rainier, Jon D.: The Synthesis of Conjugated Bis-Aryl Vinyl Substrates and Their Photoelectrocyclization Reactions towards Phenanthrene Derivatives

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Walther, Melanie; Kipke, Waldemar; Schultzke, Sven; Ghosh, Souvik; Staubitz, Anne: Modification of Azobenzenes by Cross-Coupling Reactions

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Su, Shixia; Wang, Chuan: Catalytic Asymmetric Osmium-Free Dihydroxylation of Alkenes

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Issue 06/2021

Cherepakhin, Valeriy; Williams, Travis J.: Direct Oxidation of Primary Alcohols to Carboxylic Acids

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Jovanovic, Milos D.; Petkovic, Milos R.; Savic, Vladimir M.: Polycyclic Compounds from Allenes via Palladium-Mediated Intramolecular Carbopalladation/Nucleophilic Substitution Cascade Processes

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Nejrotti, Stefano; Prandi, Cristina: Gold Catalysis and Furans: A Powerful Match for Synthetic Connections

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Yang, Chao; Jiang, Chao; Qi, Xiangbing: Alkylzirconocenes in Organic Synthesis: An Overview

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Issue 05/2021

Ura, Yasuyuki: Palladium-Catalyzed Anti-Markovnikov Oxidation of Aromatic and Aliphatic Alkenes to Terminal Acetals and Aldehydes

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Gao, Shuangqiu; Shi, Lili; Chang, Le; Wang, Binglin; Fu, Junkai: Recent Developments in Heck-Type Reaction of Unactivated Alkenes and Alkyl Electrophiles

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Gale-Day, Zachary J.: Recent Advances in Metal-Catalyzed, Electrochemical Coupling Reactions of sp² Halides/Boronic Acids and sp³ Centers

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Wang, Yang; Yang, Bing; Wu, Xin-Xing; Wu, Zheng-Guang: Recent Application of Chiral Aryliodine Based on the 2-Iodo­resorcinol Core in Asymmetric Catalysis

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Issue 04/2021

Chen, Nuan; He, Min; Zhou, Ting; Zhu, Yuqi; Zhang, Hong; Peng, Shiyong: Recent Advances in the Tandem Cyclization/Cycloaddition of Allene Intermediates from Copper-Catalyzed Cross-Coupling of Diazo Compounds with Terminal Alkynes

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Wang, Lili; Ma, Juan; Si, Erbing; Duan, Zheng: Recent Advances in Luminescent Annulated Borepins, Silepins, and Phosphepins

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Xu, Ke; Wang, Ziyuan; Zhu, Tingshun: Recent Progress towards Organocatalyzed Asymmetric (Hetero)Arene Formation

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Gonay, Marie; Batisse, Chloé; Paquin, Jean-François: Recent Advances in the Synthesis of Acyl Fluorides

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Issue 03/2021

Némethová, Ivana; Šebesta, Radovan: Are Organozirconium Reagents Applicable in Current Organic Synthesis?

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Clapham, Margaret L.; Murphy, Emma C.; Douglas, Christopher J.: Synthesis and Crystal Engineering of Rubrene and Its Derivatives

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Jeon, Hongjun; Winkler, Jeffrey D.: Synthesis of Cyclohexane-Angularly-Fused Triquinanes

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Saway, Jason; Salem, Zena M.; Badillo, Joseph J.: Recent Advances in Photoacid Catalysis for Organic Synthesis

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Issue 02/2021

Zhang, Fulin; Xin, Luoting; Yu, Yinghua; Liao, Saihu; Huang, Xueliang: Recent Advances in Palladium-Catalyzed Bridging C–H Activation by Using Alkenes, Alkynes or Diazo Compounds as Bridging Reagents

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Edlová, Tereza; Čubiňák, Marek; Tobrman, Tomáš: Cross-Coupling Reactions of Double or Triple Electrophilic Templates for Alkene Synthesis

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Bandari, Chandrasekhar; Nicholas, Kenneth M.: Deoxygenative Transition-Metal-Promoted Reductive Coupling and Cross-Coupling of Alcohols and Epoxides

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Magyar, Ágnes; Juhász, Kinga; Hell, Zoltán: The Application of 4Å Molecular Sieves in Organic Chemical Syntheses: An Overview

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Issue 01/2021

Muñoz-Molina, José María; Belderrain, Tomás R.; Pérez, Pedro J.: Recent Advances in Copper-Catalyzed Radical C–H Bond Activation Using N–F Reagents

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Shoemaker, Aaron H.; Griffith, Daniel R.: Synthetic Approaches to Non-Tropane, Bridged, Azapolycyclic Ring Systems Containing Seven-Membered Carbocycles

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Carreras, Virginie; Tanbouza, Nour; Ollevier, Thierry: The Power of Iron Catalysis in Diazo Chemistry

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Chen, Tieqiao; Tan, Qihang; Liu, Xue; Liu, Long; Huang, Tianzeng; Han, Li-Biao: Phosphorylation of Carboxylic Acids and Their Derivatives with P(O)–H Compounds Forming P(O)–C Bonds

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Macchia, Antonio; Eitzinger, Andreas; Brière, Jean-François; Waser, Mario; Massa, Antonio: Asymmetric Synthesis of Isoxazol-5-ones and Isoxazolidin-5-ones

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Issue 24/2020

Chen, Jin-Quan; Dong, Zhi-Bing: Recent Progress in Utilization of Functionalized Organometallic Reagents in Cross Coupling Reactions and Nucleophilic Additions

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Al Bujuq, Nader: Methods of Synthesis of Remdesivir, Favipiravir, Hydroxychloroquine, and Chloroquine: Four Small Molecules Repurposed for Clinical Trials during the Covid-19 Pandemic

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Pang, Xiaobo; Peng, Xuejing; Shu, Xing-Zhong: Reductive Cross-Coupling of Vinyl Electrophiles

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Talukdar, Ranadeep: Synthetically Important Ring-Opening Acylations of Alkoxybenzenes

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Yu, Jie; Singh, Anoop S.; Yan, Guobing; Yu, Jian; Tiwari, Vinod K.: Recent Developments on Denitrogenative Functionalization of Benzotriazoles

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Issue 23/2020

Gan, Fuqiang; Luo, Puying; Lin, Junyue; Ding, Qiuping: Recent Advances in the Synthesis and Applications of 2-Arylbenzothiazoles

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Gao, Weiwei; Ding, Shengtao: Progress on Iridium-Catalyzed Hydrosilylation of Alkenes and Alkynes

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Filippov, Ilya P.; Titov, Gleb D.; Rostovskii, Nikolai V.: Recent Advances in Denitrogenative Reactions of Pyridotriazoles

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Khandelwal, Manisha; Ray, Sumit Kumar; Khangarot, Rama Kanwar: Syntheses and Applications of Singh’s Catalyst

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Issue 22/2020

Yorimitsu, Hideki; Yoshimura, Aya; Misaki, Yohji: Catalytic C–H Arylation of Tetrathiafulvalenes for the Synthesis of Functional Materials

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Li, Dan; Chen, Xiaochao; Gao, Wei: Asymmetric Synthesis of C₁-Chiral THIQs with Imines in Isoquinoline Rings

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Issue 21/2020

Mateus-Ruiz, Jeferson B.; Cordero-Vargas, Alejandro: Visible-Light-Mediated Photoredox Reactions in the Total Synthesis of Natural Products

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Moberg, Christina: Silylboranes as Powerful Tools in Organic Synthesis: Stereo- and Regioselective Reactions with 1,n-Enynes

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Issue 20/2020

Calcatelli, Alessio; Cherubini-Celli, Alessio; Carletti, Edoardo; Companyó, Xavier: Unconventional Transformations of Morita–Baylis–Hillman Adducts

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Weißbarth, Hendrik; Mühlhaus, Felix; Gansäuer, Andreas: Titanocene-Catalyzed Regiodivergent Epoxide Opening – From Desymmetrizing meso-Epoxides to Regiodivergent Arylation of Epoxides

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Zhao, Fei; Masci, Domiziana; Tomarelli, Elena; Castagnolo, Daniele: Biocatalytic and Chemo-Enzymatic Approaches for the Synthesis of Heterocycles

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Issue 19/2020

Grygorenko, Oleksandr O.; Moskvina, Viktoriia S.; Hryshchuk, Oleksandr V.; Tymtsunik, Andriy V.: Cycloadditions of Alkenylboronic Derivatives

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Geske, Leander; Sato, Eisuke; Opatz, Till: Anodic Oxidation as an Enabling Tool for the Synthesis of Natural Products

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Arisawa, Mieko: Transition-Metal-Catalyzed Synthesis of Organophosphorus Compounds Involving P–P Bond Cleavage

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Bottcher, Sydney E.; Hutchinson, Lauren E.; Wilger, Dale J.: Nickel-Catalyzed anti-Selective Alkyne Functionalization Reactions

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Issue 18/2020

Large, Benjamin; Prim, Damien: C–H Functionalization Strategies in the Naphthalene Series: Site Selections and Functional Diversity

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Almasalma, Ahmad A.; Mejía, Esteban: Recent Advances on Copper-Catalyzed C–C Bond Formation via C–H Functionalization

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Agrawal, Toolika; Sieber, Joshua D.: Recent Developments in C–C Bond Formation Using Catalytic Reductive Coupling Strategies

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Álvarez-Pérez, Andrea; Saá, Carlos; Varela, Jesús A.: Oxidation of Alkynes via Catalytic Metal-Vinylidenes

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Issue 17/2020

Corti, Vasco; Bertuzzi, Giulio: Organocatalytic Asymmetric Methodologies towards the Synthesis of Atropisomeric N-Heterocycles

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Liang, Dong; Xiao, Wen-Jing; Chen, Jia-Rong: Recent Advances of 1,3,5-Triazinanes in Aminomethylation and Cycloaddition Reactions

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Brechmann, Lea T.; Teichert, Johannes F.: Catch It If You Can: Copper-Catalyzed (Transfer) Hydrogenation Reactions and Coupling Reactions by Intercepting Reactive Intermediates Thereof

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Beltran, Frédéric; Miesch, Laurence: Tertiary Enamides as Versatile and Valuable Substrates to Reach Chemical Diversity

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Issue 16/2020

Yoshimura, Akira; Saito, Akio; Yusubov, Mekhman S.; Zhdankin, Viktor V.: Synthesis of Oxazoline and Oxazole Derivatives by Hypervalent-Iodine-Mediated Oxidative Cycloaddition Reactions

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Liu, Xue; Wu, Xiangmei; Zhang, Ling; Lin, Xiaoyan; Huang, Dayun: Recent Advances in Triarylmethane Synthesis

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Issue 15/2020

Beļaunieks, Rūdolfs; Puriņš, Mikus; Turks, Māris: Manifestation of the β-Silicon Effect in the Reactions of Unsaturated Systems Involving a 1,2-Silyl Shift

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Smolobochkin, Andrey V.; Gazizov, Almir S.; Turmanov, Rakhymzhan A.; Abdullaeva, Dinara S.; Burilov, Alexander R.; Pudovik, Michail A.: N-Phosphorylated Pyrrolidines: An Overview of Synthetic Approaches

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Issue 14/2020

Mittersteiner, Mateus; Bonacorso, Helio G.; Martins, Marcos A. P.; Zanatta, Nilo: Brominated β-Alkoxyvinyl Trihalomethyl Ketones as Promising Synthons in Heterocyclic Synthesis

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Kramer, Søren: Homogeneous Gold-Catalyzed Aryl–Aryl Coupling Reactions

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Issue 13/2020

Danilkina, Natalia A.; Govdi, Anastasia I.; Balova, Irina A.: 5-Iodo-1H-1,2,3-triazoles as Versatile Building Blocks

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Issue 12/2020

Chai, Zhuo: Catalytic Asymmetric Transformations of Racemic Aziridines

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Issue 11/2020

Khan, Muhammad Kamran; Wang, Dandan; Moloney, Mark G.: Functionalised Nitrogen Heterocycles and the Search for New Antibacterials and Bioactives

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Fischer, Jérôme; Nun, Pierrick; Coeffard, Vincent: Visible-Light-Driven Transformations of Phenols via Energy Transfer Catalysis

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Issue 10/2020

Woltornist, Ryan A.; Ma, Yun; Algera, Russell F.; Zhou, Yuhui; Zhang, Zirong; Collum, David B.: Structure, Reactivity, and Synthetic Applications of Sodium Diisopropylamide

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Issue 09/2020

Tu, Hai-Yong; Zhu, Shengqing; Qing, Feng-Ling; Chu, Lingling: Recent Advances in Nickel-Catalyzed Three-Component Difunctionalization of Unactivated Alkenes

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Zheng, Yue; Shao, Xiaoqing; Ramadoss, Velayudham; Tian, Lifang; Wang, Yahui: Recent Developments in Photochemical and Electrochemical Decarboxylative C(sp³)–N Bond Formation

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Issue 08/2020

Zhu, Yannan; Huang, You: Organocatalyzed [3+3] Annulations for the Construction of Heterocycles

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Issue 07/2020

Salom-Roig, Xavier; Bauder, Claude: Recent Applications in the Use of Sulfoxides as Chiral Auxiliaries for the Asymmetric Synthesis of Natural and Biologically Active Products

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Ping, Yuanyuan; Kong, Wangqing: Ni-Catalyzed Reductive Difunctionalization of Alkenes

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Kuang, Guanghua; Liu, Guangyuan; Zhang, Xingxing; Lu, Naihao; Peng, Yiyuan; Xiao, Qiang; Zhou, Yirong: Directing-Group-Assisted Transition-Metal-Catalyzed Direct C–H Oxidative Annulation of Arenes with Alkynes for Facile Construction of Various Oxygen Heterocycles

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Issue 06/2020

Song, Si-Zhe; Dong, Youren; Ge, Guo-Ping; Li, Qiang; Wei, Wen-Ting: Recent Advances in Radical Nitration Using tert-Butyl Nitrite

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Youn, So Won: Transition-Metal-Catalyzed Annulative Coupling Cascade for the Synthesis of 3-Methyleneisoindolin-1-ones

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Hsieh, Jen-Chieh; Su, Haw-Lih: Synthesis of N-Heterocycles via Transition-Metal-Catalyzed Tandem Addition/Cyclization of a Nitrile

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Issue 05/2020

Akkarasamiyo, Sunisa; Ruchirawat, Somsak; Ploypradith, Poonsaksi; Samec, Joseph S. M.: Transition-Metal-Catalyzed Suzuki–Miyaura-Type Cross-Coupling Reactions of π-Activated Alcohols

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Fatykhov, Ramil F.; Chupakhin, Oleg N.; Inyutina, Anna K.; Khalymbadzha, Igor A.: Synthetic Approaches to Unsymmetrically Substituted 5,7-Dihydroxycoumarins

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Meng, Yan-Ping; Wang, Shi-Meng; Fang, Wan-Yin; Xie, Zhi-Zhong; Leng, Jing; Alsulami, Hamed; Qin, Hua-Li: Ethenesulfonyl Fluoride (ESF) and Its Derivatives in SuFEx Click Chemistry and More

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Issue 04/2020

Uttry, Alexander; van Gemmeren, Manuel: Direct C(sp³)–H Activation of Carboxylic Acids

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Pang, Yue; Moser, Daniel; Cornella, Josep: Pyrylium Salts: Selective Reagents for the Activation of Primary Amino Groups in Organic Synthesis

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Baráth, Eszter: Selective Reduction of Carbonyl Compounds via (Asymmetric) Transfer Hydrogenation on Heterogeneous Catalysts

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Issue 03/2020

Nocera, Giuseppe; Murphy, John A.: Ground State Cross-Coupling of Haloarenes with Arenes Initiated by Organic Electron Donors, Formed in situ: An Overview

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Smyshliaeva, Lidiia A.; Varaksin, Mikhail V.; Charushin, Valery N.; Chupakhin, Oleg N.: Azaheterocyclic Derivatives of ortho-Carborane: Synthetic Strategies and Application Opportunities

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De Luca, Lorena; Mezzetti, Antonio: Catalytic Strategies to Enantiopure Benzoins: Past and Future

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Daley, Ryan A.; Topczewski, Joseph J.: Aryl-Decarboxylation Reactions Catalyzed by Palladium: Scope and Mechanism

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Issue 02/2020

Skotnitzki, Juri; Kremsmair, Alexander; Knochel, Paul: Stereoselective Preparation and Reactions of Chiral Secondary Alkyllithiums

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Xiao, Xuan; Zheng, Zi-Tong; Li, Ting; Zheng, Jing-Lin; Tao, Ting; Chen, Li-Mei; Gu, Jin-Ying; Yao, Xu; Lin, Jin-Hong; Xiao, Ji-Chang: Recent Advances in Difluoromethylthiolation

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Issue 01/2020

Baidilov, Daler: On the Mechanism of the Stevens Rearrangement

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Craig, Alexander J.; Hawkins, Bill C.: The Bonding and Reactivity of α-Carbonyl Cyclopropanes

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Issue 24/2019

Zhang, Tong; Wu, Yue-Hua; Wang, Nai-Xing; Xing, Yalan: Advances in C(sp³)–H Bond Functionalization via Radical Processes

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Levi, Noam; Amir, Dafna; Gershonov, Eytan; Zafrani, Yossi: Recent Progress on the Synthesis of CF₂H-Containing Derivatives

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Issue 23/2019

Rakitin, Oleg A.: Recent Developments in the Synthesis of 1,2,5-Thiadiazoles and 2,1,3-Benzothiadiazoles

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Issue 22/2019

Zeidan, Nicolas; Lautens, Mark: Migratory Insertion Strategies for Dearomatization

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Issue 21/2019

Allouche, Emmanuelle M. D.; Charette, André B.: Cyclopropanation Reactions of Semi-stabilized and Non-stabilized Diazo Compounds

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Issue 20/2019

Li, Yuyang; Kluger, Ronald: Metal-Catalyzed Site-Selective Monoacylation of Diols in Aqueous Media

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Issue 19/2019

Rossignon, Alexandre; Bonifazi, Davide: O-Annulation Leading to Five-, Six-, and Seven-Membered Cyclic Diaryl Ethers Involving C–H Cleavage

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Issue 18/2019

Gazizov, Almir S.; Smolobochkin, Andrey V.; Turmanov, Rahimjan A.; Pudovik, Michail A.; Burilov, Alexander R.; Sinyashin, Oleg G.: Synthesis of Phosphaproline Derivatives: A Short Overview

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Issue 14/2019

Senatore, Raffaele; Ielo, Laura; Monticelli, Serena; Castoldi, Laura; Pace, Vittorio: Weinreb Amides as Privileged Acylating Agents for Accessing α-Substituted Ketones

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Mudarra, Ángel L.; Martínez de Salinas, Sara; Pérez-Temprano, Mónica H.: Nucleophilic Trifluoromethylation Reactions Involving Copper(I) Species: From Organometallic Insights to Scope

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Herraiz, Ana G.; Suero, Marcos G.: New Alkene Cyclopropanation Reactions Enabled by Photoredox Catalysis via Radical Carbenoids

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Kunfi, Attila; London, Gábor: Polydopamine: An Emerging Material in the Catalysis of Organic Transformations

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Issue 13/2019

Steven, Alan: Micelle-Mediated Chemistry in Water for the Synthesis of Drug Candidates

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Issue 12/2019

Sbei, Najoua; Listratova, Anna V.; Titov, Alexander A.; Voskressensky, Leonid G.: Recent Advances in Electrochemistry for the Synthesis of N-Heterocycles

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Issue 11/2019

Wang, Zhang: The Chemical Syntheses of Nannocystins

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Hollanders, Karlijn; Maes, Bert U. W.; Ballet, Steven: A New Wave of Amide Bond Formations for Peptide Synthesis

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Issue 10/2019

Colomban, Cédric; Châtelet, Bastien; Martinez, Alexandre: Different Strategies for Obtaining Enantiopure Hemicryptophanes

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Li, Jie; Knochel, Paul: Chromium-Catalyzed Cross-Couplings and Related Reactions

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Issue 09/2019

Parisotto, Stefano; Deagostino, Annamaria: π-Allylpalladium Complexes in Synthesis: An Update

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Kotha, Sambasivarao; Meshram, Milind; Panguluri, Nageswara Rao: Advanced Approaches to Post-Assembly Modification of Peptides by Transition-Metal-Catalyzed Reactions

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Rodriguez, Jean; Quintard, Adrien: Acyl Transfer Strategies as Transient Activations for Enantioselective Synthesis

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Issue 08/2019

Eschliman, Kayla; Bossmann, Stefan H.: Synthesis of Isothiocyanates: An Update

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D’Hollander, Agathe C. A.; Peilleron, Laure; Grayfer, Tatyana D.; Cariou, Kevin: Halonium-Induced Polyene Cyclizations

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Issue 07/2019

Vasilenko, Dmitry A.; Sedenkova, Kseniya N.; Kuznetsova, Tamara S.; Averina, Elena B.: Synthetic Approaches to Nitro-Substituted Isoxazoles

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Usman, Muhammad; Zhang, Xiao-Wen; Liu, Wen-Bo: Silicon-Tethered Frameworks as Directing Groups for Carbon–Carbon and Carbon–Heteroatom Bond Formation

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Issue 06/2019

Pellissier, Hélène: Synthesis of Chiral 3-Substituted 3-Amino-2-oxindoles through Enantioselective Catalytic Domino and Tandem Reactions

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Michelotti, Alessia; Roche, Maxime: 40 Years of Hydrogen–Deuterium Exchange Adjacent to Heteroatoms: A Survey

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Issue 05/2019

Zard, Samir Z.: Sulfur Betaines from S-Propargyl Xanthates. Unusual Chemistry from a Simple Functional Group

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Crawford, Jennifer M.; Sigman, Matthew S.: Conformational Dynamics in Asymmetric Catalysis: Is Catalyst Flexibility a Design Element?

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Ferrer, Sofia; Echavarren, Antonio M.: Synthesis of Bullvalenes: Classical Approaches and Recent Developments

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Maraswami, Manikantha; Loh, Teck-Peng: Transition-Metal-Catalyzed Alkenyl sp² C–H Activation: A Short Account

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Sun, Alexandra C.; McAtee, Rory C.; McClain, Edward J.; Stephenson, Corey R. J.: Advancements in Visible-Light-Enabled Radical C(sp)²–H Alkylation of (Hetero)arenes

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Hu, Fan; Ng, Jerome P. L.; Chiu, Pauline: Pyrroles as Dienes in (4+3) Cycloadditions

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Gagosz, Fabien: Gold Vinylidenes as Useful Intermediates in Synthetic Organic Chemistry

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Groso, Emilia J.; Schindler, Corinna S.: Recent Advances in the Application of Ring-Closing Metathesis for the Synthesis of Unsaturated Nitrogen Heterocycles

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Issue 04/2019

Leonardi, Marco; Estévez, Verónica; Villacampa, Mercedes; Menéndez, J. Carlos: The Hantzsch Pyrrole Synthesis: Non-conventional Variations and Applications of a Neglected Classical Reaction

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Palmieri, Alessandro; Petrini, Marino: Recent Advances in the Synthesis of Unsymmetrical Bisindolylmethane Derivatives

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Issue 03/2019

Vaitla, Janakiram; Bayer, Annette: Sulfoxonium Ylide Derived Metal Carbenoids in Organic Synthesis

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Hrdina, Radim: Directed C–H Functionalization of the Adamantane Framework

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Kancherla, Sindhu; Jørgensen, Kåre B.; Fernández-Ibáñez, M. Ángeles: Recent Developments in Palladium-Catalysed Non-Directed C–H Bond Activation in Arenes

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Issue 02/2019

Ghosh, Manoj K.; Rajkiewicz, Adam A.; Kalek, Marcin: Organocatalytic Group Transfer Reactions with Hypervalent Iodine­ Reagents

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Singh, Kuldeep; Kulbir, Kulbir; Gupta, Tarang; Kaur, Rajneesh; Singh, Raman: Applications of Rozen’s Reagent in Oxygen-Transfer and C–H Activation Reactions

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Passador, Kevin; Thorimbert, Serge; Botuha, Candice: ‘Heteroaromatic Rings of the Future’: Exploration of Unconquered Chemical Space

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Issue 01/2019

Murai, Masahito; Takai, Kazuhiko: Unsymmetrical Difunctionalization of Two Different C–H Bonds in One Pot Under Transition-Metal Catalysis

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Karageorgis, George; Waldmann, Herbert: Guided by Evolution: Biology-Oriented Synthesis of Bioactive Compound Classes

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Barrett, Anthony G. M.; Ma, Tsz-Kan; Mies, Thomas: Recent Developments in Polyene Cyclizations and Their Applications in Natural Product Synthesis

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Zhang, Heng; Lei, Aiwen: Electrochemical/Photochemical Aminations Based on Oxidative Cross-Coupling between C–H and N–H

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Piccardi, Riccardo; Turcaud, Serge; Benedetti, Erica; Micouin, Laurent: Synthesis and Reactivity of Mixed Dimethylalkynylaluminum Reagents

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Kiefer, Alexander; Kazmaier, Uli: Syntheses of Cyclomarins – Interesting Marine Natural Products with Distinct Mode of Action towards Malaria and Tuberculosis

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Wu, Xiang; Gong, Liu-Zhu: Palladium(0)-Catalyzed Difunctionalization of 1,3-Dienes: From Racemic to Enantioselective

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Yoshikai, Naohiko: Recent Advances in Enantioselective C–C Bond Formation via Organocobalt Species

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Erb, William; Mongin, Florence: Twofold Ferrocene C–H Lithiations For One-Step Difunctionalizations

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Lübken, Dennis; Saxarra, Marius; Kalesse, Markus: Tris(acetylacetonato) Iron(III): Recent Developments and Synthetic Applications

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Barde, E.; Guérinot, A.; Cossy, J.: α-Arylation of Amides from α-Halo Amides Using Metal-Catalyzed Cross-Coupling Reactions

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Kumagai, Naoya; Shibasaki, Masakatsu: 7-Azaindoline Auxiliary: A Versatile Attachment Facilitating Enantioselective­ C–C Bond-Forming Catalysis

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Issue 24/2018

Soorukram, Darunee; Pohmakotr, Manat; Kuhakarn, Chutima; Reutrakul, Vichai: Stereoselective Synthesis of Tetrahydrofuran Lignans

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Barthelemy, Anne-Laure; Magnier, Emmanuel; Dagousset, Guillaume: Direct Trifluoromethylthiolation Reactions Involving Radical Processes

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Schettini, Rosaria; Sicignano, Marina; De Riccardis, Francesco; Izzo, Irene; Della Sala, Giorgio: Macrocyclic Hosts in Asymmetric Phase-Transfer Catalyzed Reactions

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Issue 23/2018

Martinez de Marigorta, Edorta; de los Santos, Jesús M.; Ochoa de Retana, Ana M.; Vicario, Javier; Palacios, Francisco: Multicomponent Reactions in the Synthesis of γ-Lactams

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Cholewiak, Agnieszka; Stepniak, Pawel; Jurczak, Janusz: Linear Neutral Receptors for Anions: Synthesis, Structure and Applications

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Jin, Tian; Zhao, Lu; Liu, Xiao; Sun, Liang; Lin, Jia-Fu; Zheng, Zhe-Bin: Recent Advances in the Total Synthesis of Clavaminols

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Issue 21/2018

Roulland, Emmanuel: Tiacumicin B: An Antibiotic of Prime Importance and a Natural Product with an Inspiring Complex Structure

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Dimitrov, Ivaylo; Denny, William A.; Jose, Jiney: Syntheses of Ketamine and Related Analogues: A Mini Review

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Yuan, Yu-Chao; Bruneau, Christian; Gramage-Doria, Rafael: Merging Transition-Metal Catalysis with Phthalimides: A New Entry to Useful Building Blocks

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Issue 20/2018

Gamba-Sánchez, Diego; Prunet, Joëlle: Synthesis of 1,3-Diols by O-Nucleophile Additions to Activated Alkenes

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Nielsen, Christian D.-T.; Abas, Hossay; Spivey, Alan C.: Stereoselective Reactions of ortho-Quinone Methide and ortho-Quinone Methide Imines and Their Utility in Natural Product Synthesis

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Hernández-Ruiz, Raquel; Sanz, Roberto: Dichlorodioxomolybdenum(VI) Complexes: Useful and Readily Available Catalysts in Organic Synthesis

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Issue 19/2018

Ručilová, Veronika; Soural, Miroslav: Recent Advances in the Applications of Triethylsilane in Organic Synthesis

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Rivera-Chao, Eva; Fra, Laura; Fañanás-Mastral, Martín: Synergistic Bimetallic Catalysis for Carboboration of Unsaturated Hydrocarbons

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Dimitrov, Vladimir; Woodward, Simon: Capturing Waste Heat Energy with Charge-Transfer Organic Thermoelectrics

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Chen, Jing-Biao; Whiting, Andrew: Recent Advances in Copper-Catalyzed Asymmetric Hydroboration of Electron-Deficient Alkenes: Methodologies and Mechanism

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Issue 18/2018

Guyon, Hélène; Boussonnière, Anne; Castanet, Anne-Sophie: Transition-Metal-Free Enantioselective Reactions of Organo­magnesium Reagents Mediated by Chiral Ligands

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Oulyadi, Hassan: Recent Advances in NMR: Aggregation, Solvation, and Dynamics of Selected Organolithium Compounds

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Brikci-Nigassa, Nahida Mokhtari; Bentabed-Ababsa, Ghenia; Erb, William; Mongin, Florence: In Situ ‘Trans-Metal Trapping’: An Efficient Way to Extend the Scope of Aromatic Deprotometalation

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Smith, Keith; Alshammari, Mohammed B.; El-Hiti, Gamal A.: Unravelling Factors Affecting Directed Lithiation of Acylamino­aromatics

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Plasseraud, Laurent: Organotin(IV) Complexes Containing Sn–O–Se Moieties: A Structural Inventory

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Dagorne, Samuel: Recent Developments on N-Heterocyclic Carbene Supported Zinc Complexes: Synthesis and Use in Catalysis

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Issue 16/2018

Listunov, Dymytrii; Joly, Etienne; Rullière, Pauline; Gaspard, Hafida; Bernardes-Génisson, Vania; Génisson, Yves; Maraval, Valérie; Chauvin, Remi: From Natural to Artificial Antitumor Lipidic Alkynylcarbinols: Asymmetric Synthesis, Enzymatic Resolution, and Refined SARs

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Issue 15/2018

Segundo, Marcos San; Correa, Arkaitz: Cross-Dehydrogenative Coupling Reactions for the Functionalization of α-Amino Acid Derivatives and Peptides

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Dhara, Ayan; Beuerle, Florian: Synthetic Strategies for the Regioselective Functionalization of Tribenzotriquinacenes

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Issue 14/2018

Gomes, Ana T. P. C.; Forezi, Luana da S. M.; Simões, Mário M. Q.; Gonzaga, Daniel T.; Cardoso, Mariana F. C.; Da Silva, Fernando de C.; Neves, Maria G. P. M. S.; Ferreira, Vítor F.; Cavaleiro, José A. S.: Carbene-Type Species in the Functionalization of Porphyrin Derivatives

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Leitch, Jamie A.; Frost, Christopher G.: Regioselective Transition-Metal-Catalyzed C–H Functionalization of Anilines

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Riley, Darren L.; Neyt, Nicole C.: Approaches for Performing Reductions under Continuous-Flow Conditions

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Issue 13/2018

Dalpozzo, Renato; Mancuso, Raffaella: Enantioselective Vinylogous Reactions of 3-Alkylidene Oxindoles

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da Silva, Amanda F.; Fernandes, Alessandra A. G.; Thurow, Samuel; Stivanin, Mateus L.; Jurberg, Igor D.: Isoxazol-5-ones as Strategic Building Blocks in Organic Synthesis

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Issue 12/2018

Kirupakaran, Sujenth; Korth, Hans-Gert; Hirschhäuser, Christoph: A Complementary Toolbox of Iterative Methods for the Stereo­selective Synthesis of Heteroatom-Rich Motives from C₁-Building Blocks

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Bergman, Jan: Comparison of Two Reagents for Thionations

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Issue 11/2018

Murarka, Sandip; Antonchick, Andrey P.: Metal-Catalyzed Oxidative Coupling of Ketones and Ketone Enolates

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Botubol-Ares, José Manuel; Durán-Peña, María Jesús; Hanson, James R.; Hernández-Galán, Rosario; Collado, Isidro G.: Cp₂Ti(III)Cl and Analogues as Sustainable Templates in Organic Synthesis

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Issue 10/2018

Wu, Wei; Weng, Zhiqiang: Synthesis of Aryl Trifluoromethyl Ketones

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Issue 09/2018

Silva, Eduarda M. P.; Rocha, Djenisa H. A.; Silva, Artur M. S.: Diels–Alder Reactions of 1,2-Dihydropyridines: An Efficient Tool for the Synthesis of Isoquinuclidines

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Fasano, Valerio; Ingleson, Michael J.: Recent Advances in Water-Tolerance in Frustrated Lewis Pair Chemistry

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Issue 08/2018

Mousavizadeh, Farnoush; Meyer, Daniel; Giannis, Athanassios: Synthesis of C-Nor-D-homo-steroidal Alkaloids and Their Derivatives

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Bogdanov, Andrei V.; Mironov, Vladimir F.: Advances in the Synthesis of Isatins: A Survey of the Last Decade

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Issue 07/2018

Boyle, Joshua William; Zhao, Yichao; Chan, Philip Wai Hong: Product Divergence in Coinage-Metal-Catalyzed Reactions of π-Rich Compounds

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Méndez, María V.; Bracca, Andrea B. J.; Kaufman, Teodoro S.: Isolation, Synthesis, and Biological Activity of Quindoline, a Valuable­ Indoloquinoline Natural Product and Useful Key Intermediate­

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Issue 06/2018

Bürglová, Kristýna; Hlaváč, Jan: Application of Trimethylsilanolate Alkali Salts in Organic Synthesis

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Albano, Gianluigi; Aronica, Laura Antonella: Cyclization Reactions for the Synthesis of Phthalans and Isoindolines­

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Meanwell, Michael; Britton, Robert: Synthesis of Heterobenzylic Fluorides

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Issue 05/2018

Wang, Pu-Sheng; Shen, Meng-Lan; Gong, Liu-Zhu: Transition-Metal-Catalyzed Asymmetric Allylation of Carbonyl Compounds with Unsaturated Hydrocarbons

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Balasubramaniam, Sivaraman; Sankaran, Ganapathy Subramanian; Badle, Sneh Sanjay: Perspective on FTY720, an Immunosuppressant

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Chardon, Aurélien; Morisset, Eléonore; Rouden, Jacques; Blanchet, Jérôme: Recent Advances in Amide Reductions

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Issue 04/2018

Ohno, Hiroaki; Inuki, Shinsuke: Recent Progress in Palladium-Catalyzed Cascade Cyclizations for Natural Product Synthesis

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Li, Pengfei; Jia, Xiaodong: tert-Butyl Nitrite (TBN) as a Versatile Reagent in Organic Synthesis

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Len, Christophe; Delbecq, Frederic; Cara Corpas, Cristobal; Ruiz Ramos, Encarnacion: Continuous Flow Conversion of Glycerol into Chemicals: An Overview

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Issue 03/2018

Martín-Heras, Víctor; Parra, Alejandro; Tortosa, Mariola: Cyclopropyl- and Cyclobutylboronates and -silanes: A Stereo­selective Approach

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Kiyokawa, Kensuke; Nagata, Takaya; Minakata, Satoshi: Recent Advances in the Synthesis of β-Ketonitriles

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Richmond, Edward; Moran, Joseph: Recent Advances in Nickel Catalysis Enabled by Stoichiometric Metallic Reducing Agents

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Issue 02/2018

Ramesh, Perla; Suman, Devatha; Reddy, Koti Siva Nagi: Asymmetric Synthetic Strategies of (R)-(–)-Baclofen: An Antispastic Drug

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Vorobyeva, Daria V.; Osipov, Sergey N.: Selective Synthesis of 2- and 7-Substituted Indole Derivatives via Chelation-Assisted Metallocarbenoid C–H Bond Functionalization

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Largeron, Martine; Nguyen, Khac Minh Huy: Recent Advances in the Synthesis of Benzimidazole Derivatives from the Oxidative Coupling of Primary Amines

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Issue 01/2018

Ajay, Sama; Shaw, Arun K.: Studies Towards the Synthesis of (+)- and (–)-Anisomycin and Their Analogues

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Chen, Yue-Gang; Xu, Xue-Tao; Zhang, Kun; Li, Yi-Qian; Zhang, Li-Pu; Fang, Ping; Mei, Tian-Sheng: Transition-Metal-Catalyzed Carboxylation of Organic Halides and Their Surrogates with Carbon Dioxide

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Eivgi, Or; Lemcoff, N. Gabriel: Turning the Light On: Recent Developments in Photoinduced Olefin Metathesis

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Issue 24/2017

Castro-Alvarez, Alejandro; Carneros, Héctor; Costa, Anna M; Vilarrasa, Jaume: Computer-Aided Insight into the Relative Stability of Enamines

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Wang, Chuan: Electrophilic Ring Opening of Small Heterocycles

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Issue 23/2017

Pankova, Alena S.; Kuznetsov, Mikhail A.: Recent Advances in the Chemistry of 2-Acylaziridines

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Kimura, Tsutomu: Recent Advances in Magnesium Carbenoid Chemistry

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Issue 22/2017

Hu, Wen-Li; Hu, Xiang-Guo; Hunter, Luke: Recent Developments in the Deoxyfluorination of Alcohols and Phenols: New Reagents, Mechanistic Insights, and Applications

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Pathipati, Stalin R.; van der Werf, Angela; Selander, Nicklas: Indium(III)-Catalyzed Transformations of Alkynes: Recent Advances in Carbo- and Heterocyclization Reactions

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Issue 21/2017

Gusarova, Nina K.; Chernysheva, Nataliya A.; Trofimov, Boris A.: Catalyst- and Solvent-Free Addition of the P–H Species to Alkenes and Alkynes: A Green Methodology for C–P Bond Formation

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Zhao, Qun; Poisson, Thomas; Pannecoucke, Xavier; Besset, Tatiana: The Transient Directing Group Strategy: A New Trend in Transition-Metal-Catalyzed C–H Bond Functionalization

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Issue 20/2017

Aziz, Jessy; Piguel, Sandrine: An Update on Direct C–H Bond Functionalization of Nitrogen-Containing Fused Heterocycles

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Henry, Martyn C.; Mostafa, Mohamed A. B.; Sutherland, Andrew: Recent Advances in Transition-Metal-Catalyzed, Directed Aryl C–H/N–H Cross-Coupling Reactions

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Issue 19/2017

Feng, Minghao; Jiang, Xuefeng: Reactions of Arynes Involving Transition-Metal Catalysis

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Barroso, Raquel; Cabal, María P.; Valdés, Carlos: Pd-catalyzed Auto-Tandem Cascades Based on N-Sulfonylhydrazones: Hetero- and Carbocyclization Processes

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Issue 18/2017

Míguez-Lago, Sandra; Cid, María Magdalena: Axially Chiral Shape-Persistent Encapsulating Agents

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Issue 17/2017

Guo, Qihang; Lu, Zhan: Recent Advances in Nitrogen–Nitrogen Bond Formation

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Pfund, Emmanuel; Lequeux, Thierry: Synthesis of Fluoropyrrolidines and (Fluoroalkyl)pyrrolidines

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Issue 16/2017

Arava, Shlomy; Diesendruck, Charles E.: Strategies for the Synthesis of N-Arylammonium Salts

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Issue 15/2017

Chen, Yi-Hung; Ellwart, Mario; Malakhov, Vladimir; Knochel, Paul: Solid Organozinc Pivalates: A New Class of Zinc Organometallics with Greatly Enhanced Air- and Moisture-Stability

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Breugst, Martin; von der Heiden, Daniel; Schmauck, Julie: Novel Noncovalent Interactions in Catalysis: A Focus on Halogen, Chalcogen, and Anion-π Bonding

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Bartolo, Nicole D.; Read, Jacquelyne A.; Valentín, Elizabeth M.; Woerpel, K. A.: Reactions of Allylmagnesium Halides with Carbonyl Compounds: Reactivity, Structure, and Mechanism

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Mąkosza, Mieczysław: How Does Nucleophilic Aromatic Substitution in Nitroarenes Really Proceed: General Mechanism

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Tabolin, Andrey A.; Sukhorukov, Alexey Yu.; Ioffe, Sema L.; Dilman, Alexander D.: Recent Advances in the Synthesis and Chemistry of Nitronates

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Parchomyk, Tobias; Koszinowski, Konrad: Iron-Catalyzed Cross-Coupling: Mechanistic Insight for Rational Applications in Synthesis

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Dana, Suman; Ramakrishna, Isai; Baidya, Mahiuddin: Ambident Reactivity of Nitroso Compounds for Direct Amination and Hydroxylation of Carbonyls

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Reissig, Hans-Ulrich; Zimmer, Reinhold: Cyclizations of Alkoxyallenes: Mechanisms, Intermediates, ­Products – A Personal Account on Solved and Unsolved Problems with Unique Allene Building Blocks

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Hartley, Will C.; O’Riordan, Timothy J. C.; Smith, Andrew D.: Aryloxide-Promoted Catalyst Turnover in Lewis Base Organo­catalysis

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Fantin, Marco; Lorandi, Francesca; Gennaro, Armando; Isse, Abdirisak A.; Matyjaszewski, Krzysztof: Electron Transfer Reactions in Atom Transfer Radical Polymerization

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Armstrong, Roly J.; Aggarwal, Varinder K.: 50 Years of Zweifel Olefination: A Transition-Metal-Free Coupling

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Abe, Manabu; Chitose, Youhei; Jakkampudi, Satish; Thuy, Pham Thi Thu; Lin, Qianghua; Van, Bui Thi; Yamada, Ayato; Oyama, Ryoko; Sasaki, Miyu; Katan, Claudine: Design and Synthesis of Two-Photon Responsive Chromophores for Near-Infrared Light-Induced Uncaging Reactions

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Micheletti, Gabriele; Boga, Carla: Nucleophile/Electrophile Combinations in Aromatic Substitution: From Wheland to Wheland–Meisenheimer Intermediates Using Strongly Activated Arenes

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Zhao, Rong; Chang, Denghu; Shi, Lei: Recent Advances in Cyclic Diacyl Peroxides: Reactivity and Selectivity Enhancement Brought by the Cyclic Structure

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Asahara, Haruyasu: Recent Advances in the Carbon–Carbon Bond-Forming Reactions of N-Acylketimines

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Maji, Biplab; Barman, Milan K.: Recent Developments of Manganese Complexes for Catalytic Hydrogenation and Dehydrogenation Reactions

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Krishnamoorthy, Sankarganesh; Prakash, G. K. Surya: Silicon-Based Reagents for Difluoromethylation and Difluoromethylenation Reactions

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Gao, Pin; Gu, Yu-Rui; Duan, Xin-Hua: Direct C–H Functionalization of Heteroarenes via Redox-Neutral Radical Process: A Facile Route to C–C Bonds Formation

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Denegri, Bernard; Matić, Mirela; Kronja, Olga: Impact of Electronic Effects on the Nucleofugality of Leaving Groups

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Gualandi, Andrea; Mengozzi, Luca; Cozzi, Pier Giorgio: Stereoselective S_N1-Type Reaction of Enols and Enolates

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Quint, Valentin; Noël-Duchesneau, Ludovik; Lagadic, Elodie; Morlet-Savary, Fabrice; Lalevée, Jacques; Gaumont, Annie- Claude; Lakhdar, Sami: Metal-Free Generation of Phosphorus-Centered Radicals for the Synthesis of Phosphorus-Based Heterocycles: A Personal Account

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Issue 14/2017

Budynina, Ekaterina M.; Ivanov, Konstantin L.; Sorokin, Ivan D.; Melnikov, Mikhail Ya.: Ring Opening of Donor–Acceptor Cyclopropanes with N-Nucleo­philes

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Keglevich, György; Kiss, Nóra Zsuzsa; Grün, Alajos; Bálint, Erika; Kovács, Tamara: Advantages of the Microwave Tool in Organophosphorus Syntheses

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Issue 13/2017

Broggini, Gianluigi; Borelli, Tea; Giofré, Sabrina; Mazza, Alberto: Intramolecular Oxidative Palladium-Catalyzed Amination Involving Double C–H Functionalization of Unactivated Olefins

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Döndas, H. Ali; de Gracia Retamosa, María; Sansano, José M.: Current Trends towards the Synthesis of Bioactive Heterocycles and Natural Products Using 1,3-Dipolar Cycloadditions (1,3-DC) with Azomethine Ylides

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Issue 12/2017

Glinsky-Olivier, Nicolas; Guinchard, Xavier: Enantioselective Catalytic Methods for the Elaboration of Chiral Tetrahydro-β-carbolines and Related Scaffolds

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Naidoo, Shivani; Jeena, Vineet: Synthesis of 2,4-Disubstituted Quinoline Derivatives via A³-Coupling: An EcoScale Evaluation

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Issue 11/2017

Pires, Marina J. D.; Purificação, Sara I.; Santos, A. Sofia; Marques, M. Manuel B.: The Role of PEG on Pd- and Cu-Catalyzed Cross-Coupling Reactions

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Fuse, Shinichiro; Morita, Taiki; Nakamura, Hiroyuki: Step-by-Step Multifunctionalization of Isoxazoles Based On S_EAr Reactions and C–H Direct Arylations

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Mostinski, Yelena; Lankri, David; Tsvelikhovsky, Dmitry: Transition-Metal-Catalyzed Synthesis of Spirolactones

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Issue 10/2017

Annibaletto, Julien; Oudeyer, Sylvain; Levacher, Vincent; Brière, Jean-François: Catalytic Enantioselective Syntheses of Isoxazolidin-5-ones

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Issue 09/2017

Carraro, Massimo; Pisano, Luisa; Azzena, Ugo: Silica Gel Stabilized Na and Na/K Alloys: Highly Effective, Versatile and Environmentally Friendly Reducing Agents

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Merad, Jérémy; Candy, Mathieu; Pons, Jean-Marc; Bressy, Cyril: Catalytic Enantioselective Desymmetrization of Meso Compounds in Total Synthesis of Natural Products: Towards an Economy of Chiral Reagents

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Issue 08/2017

Schröder, Birte; Gaich, Tanja: Methoxatin as a Target in Total Synthesis

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Polák, Peter; Dvořák, Dalimil; Tobrman, Tomáš: Cyanogen: A Versatile Reagent for Diversity-Oriented Synthesis

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Blouin, Sarah; Blond, Gaelle; Donnard, Morgan; Gulea, Mihaela; Suffert, Jean: Cyclocarbopalladation as a Key Step in Cascade Reactions: Recent Developments

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Jackman, Mary M.; Cai, Yu; Castle, Steven L.: Recent Advances in Iminyl Radical Cyclizations

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Issue 07/2017

Fraile, José M.; García, José I.; Herrerías, Clara I.; Pires, Elisabet: Synthetic Transformations for the Valorization of Fatty Acid Derivatives

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Thaima, Thanaphat; Zamani, Farzad; Hyland, Christopher J. T.; Pyne, Stephen G.: Allenylation and Propargylation Reactions of Ketones, Aldehydes, Imines, and Iminium Ions Using Organoboronates and Related Derivatives

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Coussanes, Guilhem; Vila, Xavier; Diaba, Faïza; Bonjoch, Josep: Radical Cyclization of Trichloroacetamides: Synthesis of Lactams

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Lebœuf, David; Gandon, Vincent: Carbon–Carbon and Carbon–Heteroatom Bond-Forming Transformations Catalyzed by Calcium(II) Triflimide

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Issue 06/2017

Zhang, Min; Zhu, Chunyin; Ye, Long-Wu: Recent Advances in Dual Visible Light Photoredox and Gold-Catalyzed­ Reactions

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Lepori, Clément; Hannedouche, Jérôme: First-Row Late Transition Metals for Catalytic (Formal) Hydro­amination of Unactivated Alkenes

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Comas-Barceló, Júlia; Harrity, Joseph P. A.: Metal Acetylides in Cycloaddition Reactions

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Grimaud, Laurence; Jutand, Anny: Role of Fluoride Ions in Palladium-Catalyzed Cross-Coupling Reactions­

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Issue 05/2017

Liu, Jie; Wang, Lei: Recent Advances in Asymmetric Reactions Catalyzed by Proline and Its Derivatives

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Lanari, Daniela; Piermatti, Oriana; Morozzi, Chiara; Santoro, Stefano; Vaccaro, Luigi: Recent Applications of Solid-Supported Ammonium Fluorides in Organic Synthesis

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Mizar, Pushpak; Wirth, Thomas: Iodoaminations of Alkenes

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Ordóñez, Mario; Viveros-Ceballos, José Luis; Sayago, Francisco J.; Cativiela, Carlos: Stereoselective Synthesis of α-Amino-H-phosphinic Acids and Derivatives

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Issue 04/2017

Legnani, Luca; Bhawal, Benjamin N.; Morandi, Bill: Recent Developments in the Direct Synthesis of Unprotected Primary­ Amines

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Adeleke, A. Francis; Brown, Alexander P. N.; Cheng, Li-Jie; Mosleh, Kari A. M.; Cordier, Christopher J.: Recent Advances in Catalytic Transformations Involving Copper Acetylides

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Otero-Fraga, Jorge; Montesinos-Magraner, Marc; Mendoza, Abraham: Perspectives on Intermolecular Azomethine Ylide [3+2] Cycloadditions with Non-Electrophilic Olefins

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Chen, Wenyi; Bakewell, Clare; Crimmin, Mark R.: Functionalisation of Carbon–Fluorine Bonds with Main Group Reagents

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Eisink, Niek N. H. M.; Minnaard, Adriaan J.; Witte, Martin D.: Chemo- and Regioselective Oxidation of Secondary Alcohols in Vicinal Diols

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Mayer, Susanne; Lang, Kathrin: Tetrazines in Inverse-Electron-Demand Diels–Alder Cycloadditions and Their Use in Biology

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Issue 03/2017

Barré, Anaïs; Ţînţaş, Mihaela-Liliana; Levacher, Vincent; Papamicaël, Cyril; Gembus, Vincent: An Overview of the Synthesis of Highly Versatile N-Hydroxysuccinimide Esters

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Aullón, Gabriel; Romea, Pedro; Urpí, Fèlix: Substrate-Controlled Aldol Reactions from Chiral α-Hydroxy Ketones

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Yuan, Ling-Zhi; Hamze, Abdallah; Alami, Mouad; Provot, Olivier: Synthesis of Substituted Benzils from Diarylalkyne Oxidation

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Mangeney, Pierre; Gérard, Hélène; Vrancken, Emmanuel: Li⁺-Controlled Diastereoselectivity of the Addition of Allenyl Cuprate Reagents to Aldehydes

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Issue 02/2017

Moegling, Julian; Hoffmann, Alexander; Herres-Pawlis, Sonja: Insights into Copper-Poly(pyrazolyl)methane-Catalyzed Reactions for Organic Transformations

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Schmid, Fabian; Baro, Angelika; Laschat, Sabine: Strategies for the Synthesis of Deoxypropionates

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Issue 01/2017

Qureshi, Zafar; Toker, Christina; Lautens, Mark: Secondary Alkyl Groups in Palladium-Catalyzed Cross-Coupling Reactions

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Selter, Lars; Zygalski, Lukas; Kerste, Eric; Koert, Ulrich: Vicinal Tricarbonyl Compounds: Versatile Building Blocks for Natural Product Synthesis

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Jalani, Hitesh B.; Karagöz, Aysun Çapcı; Tsogoeva, Svetlana B.: Synthesis of Substituted 1,2,3-Triazoles via Metal-Free Click Cycloaddition Reactions and Alternative Cyclization Methods

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Issue 24/2016

Ganesh, Venkataraman; Chandrasekaran, Srinivasan: Recent Advances in the Synthesis and Reactivity of Vinylcyclopropanes

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Shang, Ming; Sun, Shang-Zheng; Wang, Hong-Li; Wang, Ming-Ming; Dai, Hui-Xiong: Recent Progress on Copper-Mediated Directing-Group-Assisted C(sp²)–H Activation

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Indukuri, Kiran; Cornelissen, Loïc; Riant, Olivier: Recent Developments in the Chemistry of Vinylsiloxanes

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Issue 23/2016

Tian, Qingshan; Zhang, Guozhu: Recent Advances in the Asymmetric Nozaki–Hiyama–Kishi Reaction

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Moni, Lisa; Banfi, Luca; Riva, Renata; Basso, Andrea: External-Oxidant-Based Multicomponent Reactions

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Pons, Amandine; Poisson, Thomas; Pannecoucke, Xavier; Charette, André B.; Jubault, Philippe: Synthesis and Applications of Fluorocyclopropanes

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Issue 22/2016

Rintjema, Jeroen; Kleij, Arjan W.: Substrate-Assisted Carbon Dioxide Activation as a Versatile Approach for Heterocyclic Synthesis

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Besson, Thierry; Fruit, Corinne: Recent Developments in Microwave-Assisted Metal-Catalyzed C–H Functionalization of Heteroarenes for Medicinal Chemistry and Material Applications

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Vargas-Caporali, Jorge; Juaristi, Eusebio: The Diamino Analogues of Privileged Corey–Bakshi–Shibata and Jørgensen–Hayashi Catalysts: A Comparison of Their Performance

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Issue 21/2016

Zani, Lorenzo; Mordini, Alessandro; Calamante, Massimo; Reginato, Gianna: Preparation of Reduced Pyrazino[2,1-a]isoquinoline Derivatives: Important Heterocycles in the Field of Bioactive Compounds

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Renaud, Jean-Luc; Gaillard, Sylvain: Recent Advances in Iron- and Cobalt-Complex-Catalyzed Tandem/Consecutive Processes Involving Hydrogenation

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Fülöpová, Veronika; Soural, Miroslav: Solid-Phase Synthesis of Heterocycles with α-Haloketones as the Key Building Blocks

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Issue 20/2016

Ajitha, Manjaly J.; Huang, Kuo-Wei: Non-Classical C–H···X Hydrogen Bonding and Its Role in Asymmetric Organocatalysis

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Serrano-Molina, David; Martín-Castro, Ana M.: Tandem Sequences Involving Michael Additions and Sigmatropic Rearrangements

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Varela, Jesús A.; Saá, Carlos: Metal-Catalyzed Cyclizations to Pyran and Oxazine Derivatives

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Issue 18/2016

Sloan, Nikki L.; Sutherland, Andrew: Recent Advances in Transition-Metal-Catalyzed Iodination of Arenes

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Wencel-Delord, Joanna; Colobert, Françoise: Stereoselective Metal-Catalyzed C–C Bond Coupling Reactions by Stereoconvergence, Dynamic Kinetic Asymmetric Transformation, or Dynamic Kinetic Resolution

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Alezra, Valérie; Kawabata, Takeo: Recent Progress in Memory Of Chirality (MOC): An Advanced Chiral Pool

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Issue 17/2016

Amat, Mercedes; Llor, Núria; Guignard, Guillaume; Bosch, Joan: Synthesis of Fluvirucins and Their Aglycons, the Fluvirucinins

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Giustiniano, Mariateresa; Novellino, Ettore; Tron, Gian Cesare: Nitrile N-Oxides and Nitrile Imines as New Fuels for the Discovery of Novel Isocyanide-Based Multicomponent Reactions

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Nielsen, Mogens Brøndsted: Sonogashira-Like Coupling Reactions with Phosphine–Gold(I) Alkynyl Complexes

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Issue 16/2016

Echeverria, Pierre-Georges; Ayad, Tahar; Phansavath, Phannarath; Ratovelomanana-Vidal, Virginie: Recent Developments in Asymmetric Hydrogenation and Transfer Hydrogenation of Ketones and Imines through Dynamic Kinetic Resolution

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Yoshida, Hiroto: Stannylation Reactions under Base Metal Catalysis: Some Recent Advances

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Roselló, María Sánchez; del Pozo, Carlos; Fustero, Santos: A Decade of Advance in the Asymmetric Vinylogous Mannich Reaction

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Issue 15/2016

García-Cabeza, Ana Leticia; Moreno-Dorado, F. Javier; Ortega, María J.; Guerra, Francisco M.: Copper-Catalyzed Oxidation of Alkenes and Heterocycles

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Vicente, Rubén: Recent Progresses towards the Strengthening of Cyclopropene Chemistry

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Banert, Klaus: The Chemistry of Unusually Functionalized Azides

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Issue 14/2016

Zeng, Yuwen; Hu, Jinbo: Bridging Fluorine and Aryne Chemistry: Vicinal Difunctionalization of Arynes Involving Nucleophilic Fluorination, Trifluoromethylation, or Trifluoromethylthiolation

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Montesinos-Magraner, Marc; Vila, Carlos; Blay, Gonzalo; Pedro, José R.: Catalytic Enantioselective Friedel–Crafts Reactions of Naphthols and Electron-Rich Phenols

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Sánchez-Sancho, Francisco; Csákÿ, Aurelio G.: C–H Bond Formation with Boronic Acids and Derivatives by Transition-Metal-Free Conjugate Addition Reactions

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Issue 13/2016

Sasaki, I.: Recent Uses of Kröhnke Methodology: A Short Survey

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Florio, Saverio; Salomone, Antonio: Heterocycle-Mediated ortho-Functionalization of Aromatic Compounds: The DoM Methodology and Synthetic Utility

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Tanoury, Gerald J.: Photochemical Synthesis of Azaheterocycles

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Issue 12/2016

Chen, Zhang-Pei; Zhou, Yong-Gui: Asymmetric Hydrogenation of Heteroarenes with Multiple Heteroatoms

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Hoffmann, Norbert: Photochemical Electron and Hydrogen Transfer in Organic Synthesis: The Control of Selectivity

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Issue 11/2016

Kindt, Stephanie; Heinrich, Markus R.: Recent Advances in Meerwein Arylation Chemistry

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Heinrich, Clément F.; Peter, Clovis; Miesch, Laurence; Geoffroy, Philippe; Miesch, Michel: Diastereo- and Enantioselective Synthesis of Polyfunctionalized Diquinanes, Hydrindanes, and Decalins Bearing a Hydroxyl Group at the Ring Junction

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Issue 10/2016

Erhardt, Hellmuth; Kirsch, Stefan F.: Geminal Bis- and Tristriazoles: Long-known but still Uncommon Heterocyclic Entities

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Collins, Súil; Bartlett, Sean; Nie, Feilin; Sore, Hannah F.; Spring, David R.: Diversity-Oriented Synthesis of Macrocycle Libraries for Drug Discovery and Chemical Biology

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Issue 09/2016

Das, Sudarshan; Santra, Sougata; Mondal, Pallab; Majee, Adinath; Hajra, Alakananda: Zwitterionic Imidazolium Salt: Recent Advances in Organocatalysis

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Nishiwaki, Nagatoshi: Development of a Pseudo-Intramolecular Process

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Issue 08/2016

Benischke, Andreas D.; Ellwart, Mario; Becker, Matthias R.; Knochel, Paul: Polyfunctional Zinc and Magnesium Organometallics for Organic Synthesis: Some Perspectives

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Issue 07/2016

Meazza, Marta; Rios, Ramon: Merging Transition-Metal Activation and Aminocatalysis

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Issue 06/2016

Bag, Sukdev; Maiti, Debabrata: Palladium-Catalyzed Olefination of Aryl C–H Bonds by Using Directing­ Scaffolds

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Issue 05/2016

Lundberg, Helena; Adolfsson, Hans: Catalytic α-Alkylation/Reduction of Ketones with Primary Alcohols To Furnish Secondary Alcohols

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Merino, Pedro; Tejero, Tomás; Delso, Ignacio; Matute, Rosa: Recent Advances on Asymmetric Nitroso Aldol Reaction

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Issue 04/2016

Pullarkat, Sumod A.: Recent Progress in Palladium-Catalyzed Asymmetric Hydrophos­phination

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Issue 03/2016

Dai, Qiang; Jiang, Yan; Yu, Jin-Tao; Cheng, Jiang: Peroxide: A Novel Methylating Reagent

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Issue 02/2016

Tilly, David; Chevallier, Floris; Mongin, Florence: Synthesis of Heterobiaryls Featuring 1,4 N···S Inter-Ring Interactions

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Issue 01/2016

Jia, Xiaodong: Radical Cation Salts: From Single-Electron Oxidation to C–H Activation­

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Issue 23/2015

Xu, Zheng; Huang, Wei-Sheng; Zhang, Jin; Xu, Li-Wen: Recent Advances in Transition-Metal-Catalyzed Silylations of Arenes with Hydrosilanes: C–X Bond Cleavage or C–H Bond Activation­ Synchronized with Si–H Bond Activation

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Issue 22/2015

Gu, Jing; Du, Wei; Chen, Ying-Chun: Combined Asymmetric Aminocatalysis and Carbene Catalysis

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Issue 17/2015

Chatalova-Sazepin, Claire; Hemelaere, Rémy; Paquin, Jean-François; Sammis, Glenn M.: Recent Advances in Radical Fluorination

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Issue 16/2015

Sharma, Ritika; Kumar, Rakesh; Kumar, Inder; Singh, Bikram; Sharma, Upendra: Selective C–Si Bond Formation through C–H Functionalization

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Issue 14/2015

Wu, Hua; He, Yu-Ping; Shi, Feng: Recent Advances in Chiral Phosphoric Acid Catalyzed Asymmetric Reactions for the Synthesis of Enantiopure Indole Derivatives

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Issue 13/2015

Praveen, P. J.; Parameswaran, P. S.; Majik, M. S.: Bis(indolyl)methane Alkaloids: Isolation, Bioactivity, and Syntheses

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Issue 12/2015

Kuzmina, Olesya M.; Steib, Andreas K.; Moyeux, Alban; Cahiez, Gérard; Knochel, Paul: Recent Advances in Iron-Catalyzed Csp²–Csp² Cross-Couplings

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Shang, Xiaojie; Liu, Zhong-Quan: Iron-Catalyzed Alkylation of Alkenes and Alkynes Using Alcohols as the Alkylating Reagent

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Issue 11/2015

Pfund, Emmanuel; Lequeux, Thierry; Gueyrard, David: Synthesis of Fluorinated and Trifluoromethyl-Substituted Alkenes through the Modified Julia Olefination: An Update

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Issue 10/2015

Sarkar, Anirban; Santra, Sougata; Kundu, Shrishnu Kumar; Ghosal, Nirnita Chakraborty; Hajra, Alakananda; Majee, Adinath: Zinc Tetrafluoroborate: A Versatile and Robust Catalyst for Various­ Organic Reactions and Transformations

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Issue 09/2015

Liu, Yun-Lin; Zhou, Jian: Catalytic Asymmetric Strecker Reaction: Bifunctional Chiral Tertiary Amine/Hydrogen-Bond Donor Catalysis Joins the Field

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Issue 08/2015

Saeidian, Hamid; Abdoli, Morteza; Mirjafary, Zohreh: Synthesis of Acyclic and Cyclic Sulfamates: A Review

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Issue 07/2015

Hu, Xin-Hu; Liu, Zhen-Ting; Shao, Long; Hu, Xiang-Ping: Recent Advances in Catalytic Stereocontrolled Cycloaddition with Terminal Propargylic Compounds

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Issue 06/2015

Ager, David J.: Popular Synthetic Approaches To Pharmaceuticals

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Issue 05/2015

Chen, Jia-Rong; Yu, Xiao-Ye; Xiao, Wen-Jing: Tandem Radical Cyclization of N-Arylacrylamides: An Emerging Platform for the Construction of 3,3-Disubstituted Oxindoles

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Issue 04/2015

Xie, Jian-Hua; Bao, Deng-Hui; Zhou, Qi-Lin: Recent Advances in the Development of Chiral Metal Catalysts for the Asymmetric Hydrogenation of Ketones

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Issue 03/2015

Champagne, Pier Alexandre; Desroches, Justine; Paquin, Jean-François: Organic Fluorine as a Hydrogen-Bond Acceptor: Recent Examples and Applications

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Issue 02/2015

Li, Yan; Zhang, Qian: N-Fluorobenzenesulfonimide: An Efficient Nitrogen Source for C–N Bond Formation

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Issue 01/2015

Li, Hui; Wu, Jimmy: (3+2)-Cycloaddition Reactions of Oxyallyl Cations

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Issue 22/2014

Anbarasan, Pazhamalai; Yadagiri, Dongari; Rajasekar, Shanmugam: Recent Advances in Transition-Metal-Catalyzed Denitrogenative Transformations­ of 1,2,3-Triazoles and Related Compounds

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Issue 21/2014

Chong, Eugene; Garcia, Pierre; Schafer, Laurel L.: Hydroaminoalkylation: Early-Transition-Metal-Catalyzed α-Alkylation of Amines

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Issue 20/2014

Deeming, Alex S.; Emmett, Edward J.; Richards-Taylor, Charlotte S.; Willis, Michael C.: Rediscovering the Chemistry of Sulfur Dioxide: New Developments in Synthesis and Catalysis

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Issue 19/2014

Bhat, Chinmay; Bugde, Sandesh T.; Tilve, Santosh G.: Conhydrine: An Account of Isolation, Biological Perspectives and Synthesis

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Issue 18/2014

Lahm, Günther; Orejarena Pacheco, Julio Cesar; Opatz, Till: Rearrangements of Nitrile-Stabilized Ammonium Ylides

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Issue 17/2014

Corpet, Martin; Gosmini, Corinne: Recent Advances in Electrophilic Amination Reactions

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Issue 16/2014

Mahoney, Kevin P. P.; Smith, Duncan R. M.; Bogosyan, Emma J. A.; Goss, Rebecca J. M.: Access to High Value Natural and Unnatural Products through Hyphenating Chemical Synthesis and Biosynthesis

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Issue 15/2014

Li, Jingjie; Shi, Li-Li; Chen, Jiahua; Gong, Jianxian; Yang, Zhen: Thioureas as Ligands in Organometallic Reactions

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Issue 14/2014

Fernandes, Rodney A.; Mulay, Sandip V.: Chiral Cups (Calixarenes) via Dötz Benzannulation

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Issue 13/2014

Abdel-Wahab, Bakr F.; Shaaban, Saad: Thiazolothiadiazoles and Thiazolooxadiazoles: Synthesis and Biological Applications

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Issue 12/2014

Maertens, Gaëtan; Ménard, Marc-André; Canesi, Sylvain: Catalytic Enantioselective Desymmetrizations of Prochiral Dienone Systems

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Issue 11/2014

Hafner, Andreas; Jung, Nicole; Bräse, Stefan: Silver-Mediated Perfluoroalkylation Reactions

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Issue 08/2014

Sun, Jiansong; Laval, Stéphane; Yu, Biao: Glycosylation Reactions in the Synthesis of Flavonoid Glycosides

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Issue 06/2014

O’Reilly, Steven; Guiry, Patrick J.: Recent Applications of C₁-Symmetric Bis(oxazoline)-Containing Ligands in Asymmetric Catalysis

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Issue 05/2014

Chen, Jie; Zhou, Ling: Recent Progress in the Asymmetric Intermolecular Halogenation of Alkenes

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Issue 04/2014

Sidduri, Achyutharao; Tilley, Jefferson W.; Fotouhi, Nader: Functionalized Organozinc Reagents in Medicinal Chemistry: Discovery of Novel Drug Candidates

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Issue 03/2014

Deore, Prashant S.; Argade, Narshinha P.: Metal-Catalyzed Cross-Coupling Reactions of Halomaleic Anhydrides and Halomaleimides: Synthesis of Structurally Interesting and Biologically ­Important Natural and Unnatural Products

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Issue 01/2014

Baeza, Alejandro; Nájera, Carmen: Recent Advances in the Direct Nucleophilic Substitution of Allylic Alcohols through S_N1-Type Reactions

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Issue 24/2013

Chakraborty, Indrajit; Jana, Samaresh: Synthetic Developments on the Indolizidine Alkaloid, Harmicine

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Issue 23/2013

Nithiy, Nisha; Rosa, David; Orellana, Arturo: Carbon–Carbon Bond Formation through Palladium Homoenolates

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Issue 22/2013

Li, Huan; Zhang, Yan; Wang, Jianbo: Reaction of Diazo Compounds with Organoboron Compounds

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Issue 21/2013

Vitale, Paola; Scilimati, Antonio: Functional 3-Arylisoxazoles and 3-Aryl-2-isoxazolines from Reaction of Aryl Nitrile Oxides and Enolates: Synthesis and Reactivity

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Issue 20/2013

Eckermann, Ruben; Gaich, Tanja: The Akuammiline Alkaloids; Origin and Synthesis

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Issue 18/2013

Singh, Fateh V.; Wirth, Thomas: Oxidative Rearrangements with Hypervalent Iodine Reagents

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Issue 14/2013

Baidya, Mahiuddin; Yamamoto, Hisashi: Advancements in the Nascent Nitroso-Ene Reaction

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Issue 12/2013

García Mancheño, Olga; Stopka, Tobias: TEMPO Derivatives as Alternative Mild Oxidants in Carbon–Carbon Coupling Reactions

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Issue 08/2013

Korneev, Sergei M.: Hydrocinnamic Acids: Application and Strategy of Synthesis

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Issue 05/2013

Ferraccioli, Raffaella: Palladium-Catalyzed Synthesis of Carbo- and Heterocycles through Norbornene-Mediated ortho C–H Functionalization

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Issue 01/2013

Evano, Gwilherm; Jouvin, Kévin; Coste, Alexis: General Amination Reactions for the Synthesis of Ynamides

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Issue 22/2012

Lee, Doris; Taylor, Mark S.: Catalyst-Controlled Regioselective Reactions of Carbohydrate Derivatives

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Issue 17/2012

Majik, Mahesh S.; Tilve, Santosh G.: Pyrrolizidine Alkaloids Pyrrolams A–D: A Survey of Synthetic Efforts, Biological Activity, and Studies on Their Stability

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Issue 16/2012

Miao, Zhenyuan; Chen, Fener: Asymmetric Aldol Reactions of Heterocyclic Dienolsilanes and α,β-Unsaturated Carbonyl Derived Dienolsilanes

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Issue 15/2012

Ralston, Kevin J.; Hulme, Alison N.: The Evans–Tishchenko Reaction: Scope and Applications

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Issue 13/2012

Kiss, Loránd; Nonn, Melinda; Fülöp, Ferenc: Syntheses of Isoxazoline-Based Amino Acids by Cycloaddition of Nitrile Oxides and Their Conversion into Highly Functionalized Bioactive Amino Acid Derivatives

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Issue 12/2012

Mei, Tian-Sheng; Kou, Lei; Ma, Sandy; Engle, Keary M.; Yu, Jin-Quan: Heterocycle Formation via Palladium-Catalyzed C–H Functionalization

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Issue 10/2012

Bisai, Vishnumaya: Organocatalytic Asymmetric Vinylogous Aldol Reactions

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