Synthesis

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Issue eFirst

Takahashi, Hiroto; Honjo, Yusaku; Shibata, Yu; Nagashima, Yuki; Tanaka, Ken: Dienylation of Unfunctionalized Arenes with 1,6-Diynes via Rhodium-Catalyzed Directing-Group-Free C–H Bond Activation
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0585_ga_10-1055_a-1328-6436.gif
Gu, Zheng-Yang; Wu, Yang; Jin, Feng; Bao, Xiaoguang; Xia, Ji-Bao: Intermolecular C–H Amidation of Alkenes with Carbon Monoxide and Azides via Tandem Palladium Catalysis
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0053_ga_10-1055_a-1401-4486.gif
Khatana, Anil Kumar; Singh, Vikram; Gupta, Manoj Kumar; Tiwari, Bhoopendra: A Highly Efficient NHC-Catalyzed Aerobic Oxidation of Aldehydes to Carboxylic Acids
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0219_ga_10-1055_s-0037-1610069.gif
Ryan, Jonathon S.; Schindler, Corinna S.: Total Synthesis of Mycocyclosin and the Herqulines
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0034_ga_10-1055_a-1403-4312.gif
Ishida, Naoyoshi; Iwamoto, Hiroaki; Sunagawa, Denise Eimi; Ohashi, Masato; Ogoshi, Sensuke: CsF-Catalyzed Fluoroacylation of Tetrafluoroethylene Using Acyl Fluorides for the Synthesis of Pentafluoroethyl Ketones
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0481_ga_10-1055_s-0040-1705962.gif
Nocera, Giuseppe; Murphy, John A.: Ground State Cross-Coupling of Haloarenes with Arenes Initiated by Organic Electron Donors, Formed in situ: An Overview
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0401_ga_10-1055_s-0039-1690614.gif
Sperger, Theresa; Schoenebeck, Franziska: α-Arylation of Esters and Ketones Enabled by a Bench-Stable Pd(I) Dimer Catalyst
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0285_ga_10-1055_s-0037-1610087.gif
Wan, Bin; Zhang, Yanghui: Synthesis of Unsymmetrically Substituted Tetraphenylenes through Palladium-Catalyzed C(sp2)–H Activation
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0016_ga_10-1055_a-1416-9737.gif
Cole, Charles J. F.; Chi, Hyung Min; DeBacker, Kenneth C.; Snyder, Scott A.: Synthesis of Enhanced, Isolable Disulfanium Salts and their Application to Thiiranium-Promoted Polyene Cyclizations
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0184_ga_10-1055_s-0037-1609754.gif
Wang, Zheng; Ji, Hongtao; He, Wei-Min; Xiong, Yang; Zhang, Guozhu: Chromium-Catalyzed Asymmetric Dearomatization–Addition Reactions of Halomethyloxazoles and Indoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0070_ga_10-1055_s-0037-1609753.gif
Xu, Wengang; Wu, Mingbo; Yoshikai, Naohiko: Iron-Catalyzed Remote C–H Alkylation of 8-Amidoquinolines with Cycloalkanes
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0595_ga_10-1055_a-1337-5416.gif
Lindner, Marcin; Krasiński, Antoni; Jurczak, Janusz: Facile, Stereocontrolled Synthetic Route towards Bis-functionalised Pyrrolizidines
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0359_ga_10-1055_s-0037-1609582.gif
Watanabe, Hikaru; Nakajima, Kazuki; Ekuni, Kento; Edagawa, Ryota; Akagi, Yuta; Okuda, Yasuhiro; Wakamatsu, Kan; Orita, Akihiro: Custom-Made Pyrene Photocatalyst-Promoted Desulfonylation of Arylethenyl Sulfones Using Green-Light-Emitting Diodes
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0005_ga_10-1055_s-0040-1706025.gif
Lam, Heather; Abel-Snape, Xavier; Köllen, Martin F.; Lautens, Mark: Recent Advances in Transition-Metal-Free (4+3)-Annulations
https://www.thieme-connect.de/media/synthesis/EFirst/i_z0520_ga_10-1055_s-0040-1706023.gif
Oberg, Kevin M.; Cochran, Brian M.; Cook, Matthew J.; Rovis, Tomislav: The Catalytic Alkylative Desymmetrization of Anhydrides in a Formal Synthesis of Ionomycin
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0160_ga_10-1055_s-0037-1610108.gif
Pang, Jia Hao; Ong, Derek Yiren; Watanabe, Kohei; Takita, Ryo; Chiba, Shunsuke: Leaving Group Ability in Nucleophilic Aromatic Amination by Sodium Hydride–Lithium Iodide Composite
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0368_ga_10-1055_s-0039-1690010.gif
Akahori, Shuhei; Fujihara, Tetsuaki; Tsuji, Yasushi; Shinokubo, Hiroshi; Miyake, Yoshihiro: Synthesis of Tetrasilatetrathia[8]circulenes through C–I and C–H Silylation
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0107_ga_10-1055_a-1437-9917.gif
Zhang, Yongda; Lao, Kendricks S.; Sieber, Joshua D.; Xu, Yibo; Wu, Linglin; Wang, Xiao-Jun; Desrosiers, Jean-Nicolas; Lee, Heewon; Haddad, Nizar; Han, Zhengxu S.; Yee, Nathan K.; Song, Jinhua J.; Howell, Amy R.; Senanayake, Chris H.: Modular Dihydrobenzoazaphosphole Ligands for Suzuki–Miyaura Cross-Coupling
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0181_ga_10-1055_s-0037-1610158.gif
Liddon, John T. R.; Rossi-Ashton, James A.; Clarke, Aimee K.; Lynam, Jason M.; Taylor, Richard J. K.; Unsworth, William P.: Divergent Reactivity of Indole-Tethered Ynones with Silver(I) and Gold(I) Catalysts: A Combined Synthetic and Computational Study
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0211_ga_10-1055_s-0037-1610181.gif
Joshi, Madhur S.; Pigge, F. Christopher: Sequential Pyridine Dearomatization–Mizoroki–Heck Cyclization for the Construction of Fused (Dihydropyrido)isoindolinone Ring Systems
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0093_ga_10-1055_s-0037-1610133.gif
Inai, Yasuhito; Usuki, Yoshinosuke; Satoh, Tetsuya: Synthesis of Benzo-Fused Cyclic Compounds via Rhodium-Catalyzed Decarboxylative Coupling of Aromatic Carboxylic Acids with Alkynes
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0071_ga_10-1055_a-1416-6997.gif
Wertjes, William; Ayers, Sloan; Gao, Qi; Simmons, Eric M.; Beutner, Gregory L.: A Divergent Nickel-Catalyzed Synthesis of Quinazolinediones and Benzoxazinone Imines
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0192_ga_10-1055_s-0037-1610140.gif
Tang, Zhi; Tong, Zhou; Qiu, Renhua; Yin, Shuang-Feng; Kambe, Nobuaki: Recent Advances on Benzofuranones: Synthesis and Transformation via C–H Functionalization
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0039_ga_10-1055_a-1405-5761.gif
Denizot, Natacha; Guillot, Régis; Kouklovsky, Cyrille; Vincent, Guillaume: N-Iodosuccinimide-Mediated Oxidative Coupling of Indoles and Phenols: A Synthetic Study toward the Benzofuroindoline Moiety of Bipleiophylline
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0092_ga_10-1055_s-0036-1592002.gif
Kawakami, Haruka; Nohira, Itsuki; Chatani, Naoto: Nickel-Catalyzed C–F/N–H Annulation of 2-(2-Fluoroaryl) N-Heteroaromatic Compounds with Alkynes: Activation of C–F Bonds
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0614_ga_10-1055_a-1337-5504.gif
Ziegler, Dorothée S.; Klier, Lydia; Müller, Nicolas; Karaghiosoff, Konstantin; Knochel, Paul: Directed Zincation or Magnesiation of 2- and 4-Pyrones and Their Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0411_ga_10-1055_s-0037-1610215.gif
Garlets, Zachary J.; Wolfe, John P.: Asymmetric Synthesis of Six-Membered Cyclic Sulfamides via Palladium-Catalyzed Alkene Carboamination Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0078_ga_10-1055_s-0036-1591574.gif
Fukumoto, Yoshiya; Shiratani, Motohiro; Noguchi, Hikaru; Chatani, Naoto: Iridium-Catalyzed Direct Amidation of Imidazoles at the C-2 Position with Isocyanates in the Presence of Hydrosilanes Leading to Imidazole-2-Carboxamides
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0637_ga_10-1055_a-1375-5283.gif
Yamamoto, Sonoka; Shibuya, Yushin; Suzuki, Toyoko; Okano, Kentaro; Horie, Masaki; Mori, Atsunori: One-Shot Deprotonative Metalation/Transmetalation/Polymerization of Halothiophenes Catalyzed by Nickel Complex for Polythiophene Synthesis
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0653_ga_10-1055_a-1368-7072.jpg

Issue Accepted Manuscripts

Kiyosu, Yuuki; Tanaka, Shino; Okumura, Sota; Kiyokawa, Kensuke; Minakata, Satoshi: Synthesis of Fused Diaziridine Derivatives from Cyclic Secondary Amines Utilizing N-Bromosulfonamides as an Aminating Reagent
Kanyiva, Kyalo Stephen; Nigel Tang, King Hung; Wang, Jiarui; Shibata, Takanori: Palladium-Catalyzed sp3 C–H Benzoxylation of Alanine Derivatives Using Aldehydes under Ambient Conditions
Ishida, Tamao; Zhang, Zhenzhong; Murayama, Haruno; Yamamoto, Eiji; Tokunaga, Makoto: C-H bond functionalization using Pd and Au supported catalysts with mechanistic insights of the active species
Dalal, Arup; Arulananda Babu, Srinivasarao: Pd(II)-catalyzed directing group-aided C-H arylation and alkylation of pyrene core. Synthesis of C1,C2- and C1,C10-disubstituted pyrene motifs
Oonishi, Yoshihiro; Sakamoto, Shunki; Agata, Shuya; Sato, Yoshihiro: Rh(I)-Catalyzed Enantioselective Cyclization of Enyne through Site-Selective C(sp3)-H Bond Activation Triggered by Formation of Rhodacycle
Pan, Feng-Feng; Guo, Peng; huang, Xiaochuang; Shu, Xing-Zhong: Dibenzyls synthesis by nickel-catalyzed homocoupling of benzyl alcohols
De, Pinaki Bhusan; Asako, Sobi; Ilies, Laurean: Recent Advances in Use of Sodium Dispersion for Organic Synthesis
Kona, Chandrababu Naidu; Oku, Rikuto; Nishii, Yuji; Miura, Masahiro: Peri-Selective Direct Acylmethylation and Amidation of Naphthalene Derivatives Using Iridium and Rhodium Catalysts
Shimazumi, Ryoma; Morita, Kosuke; Yoshida, Tomoki; Yasui, Kousuke; Tobisu, Mamoru: Late-stage Derivatization of Buflavine by Nickel-catalyzed Direct Substitution of a Methoxy Group via C-O Bond Activation
Morimoto, Tsumoru; Wang, Chuang; Tanimoto, Hiroki; Artok, Levent; Kakiuchi, Kiyomi: Rhodium(I)-Catalyzed CO Gas-Free Arylative Dual-Carbonylation of Alkynes with Arylboronic Acids via the Formyl C-H Activation of Formaldehyde
Yabe, Ryota; Ebe, Yusuke; Nishimura, Takahiro: Iridium-Catalyzed Direct C–H Allylation of Ketimines
Wienhold, Sebastian; Fritz, Lukas; Judt, Tatjana; Hackl, Sabrina; Neubauer, Thomas; Sauerer, Bastian; Bach, Thorsten: Studies towards the Synthesis of (-)-Pulvomycin: Construction of the C12-C40 Segment by a Stereoselective Aldol Reaction

Issue 02/2021

Arjona-Esteban, Alhama; Rausch, Anja; Vysotsky, Myroslav O.; Würthner, Frank: Merocyanine Dyes with Extended Polymethine Chains by Simple Two-Step Condensation Sequence
https://www.thieme-connect.de/media/synthesis/202102/i_c0240_ga_10-1055_s-0040-1707896.gif
Yoshimura, Aya; Henmi, Keisuke; Kimura, Hitoshi; Sakakibara, Ryo; Ochi, Rika; Shirahata, Takashi; Yorimitsu, Hideki; Misaki, Yohji: Synthesis of Peripherally Arylated Tetrathiafulvalenes Extended with an Anthraquinoid Spacer via Pd-Catalyzed C–H Arylation and Construction of a Double-Helical Cobalt-Based Metal-Organic Framework
https://www.thieme-connect.de/media/synthesis/202102/i_c0266_ga_10-1055_s-0040-1707177.gif
Widner, Florian J.; Kieninger, Christoph; Wurst, Klaus; Deery, Evelyne; Lawrence, Andrew D.; Warren, Martin J.; Kräutler, Bernhard: Synthesis, Spectral Characterization and Crystal Structure of Chlororhodibalamin: A Synthesis Platform for Rhodium Analogues of Vitamin B12 and for Rh-Based Antivitamins B12
https://www.thieme-connect.de/media/synthesis/202102/i_c0397_ga_10-1055_s-0040-1707288.gif
Yan, Feng-Zhi; Shao, Yuan-Guang; Zhang, Zibin; Shen, Yan-Feng; Huang, Xue-Chun; Zhang, Pei-Ling; Li, Shijun: Synthesis of Catenanes from a BMP32C10-Based Cryptand Tuned by the Linkage Length of Paraquat Salts
https://www.thieme-connect.de/media/synthesis/202102/i_c0428_ga_10-1055_s-0040-1707290.gif
Mei, Peifeng; Kurosaki, Ryo; Matsumoto, Akinobu; Yamada, Hiroko; Aratani, Naoki: One-Pot Synthesis of a Cyclic Pyrene Octamer from Two Bifunctionalized Pyrene Monomers
https://www.thieme-connect.de/media/synthesis/202102/i_c0439_ga_10-1055_s-0040-1705950.gif

Issue 24/2020

Qin, Jing-Hao; Li, Jin-Heng; An, De-Lie: Recent Advances in Cycloaddition Reactions with Alkynes to Construct Heterocycles
https://www.thieme-connect.de/media/synthesis/202024/i_c0230_ga_10-1055_s-0040-1707355.gif
Pellissier, Hélène: The Use of Domino Reactions for the Synthesis of Chiral Rings
https://www.thieme-connect.de/media/synthesis/202024/i_c0191_ga_10-1055_s-0040-1707905.gif
Wei, Bin; Li, Ke-Wei; Wu, Yan-Chen; Tong, Shi-Qi; Song, Ren-Jie: Radical Strategy for the Transition-Metal-Catalyzed Synthesis of γ-Lactones: A Review
https://www.thieme-connect.de/media/synthesis/202024/i_c0226_ga_10-1055_s-0040-1707835.jpg
Huang, Min-Hua; Hao, Wen-Juan; Jiang, Bo: Iridium(III)-Catalyzed Difluoroalkylation–Bicyclization of 1,7-Enynes toward Benzo[a]fluoren-5-ones under Visible-Light Photoredox Conditions
https://www.thieme-connect.de/media/synthesis/202024/i_c0182_ga_10-1055_s-0040-1707863.gif

Issue 22/2020

Maligres, Peter E.; Song, Zhiguo Jake; Strotman, Neil A.; Yin, Jinquin; Pei, Tao; Strotman, Hallena R.; Itoh, Tetsuji; Sherer, Edward C.; Humphrey, Guy R.: Synthesis of Fused Oxepane HIV Integrase Inhibitor MK-1376
https://www.thieme-connect.de/media/synthesis/202022/i_c0045_ga_10-1055_s-0040-1707994.gif
Toussaint, Frédéric C.; Defrance, Thierry; Decouvreur, Serge; Carly, Nicolas; Merschaert, Alain: Intensification of Free-Radical Racemization for a Non-activated Amine in a Continuous Flow Reactor
https://www.thieme-connect.de/media/synthesis/202022/i_c0232_ga_10-1055_s-0040-1707339.jpg
Wächtler, Andreas; Bremer, Matthias; Maillard, David; Mohr, Thomas: Controlling the All-trans Stereochemistry in Liquid Crystalline 4,4′-Dialkyl-[1,1′-bicyclohexyl] Compounds
https://www.thieme-connect.de/media/synthesis/202022/i_c0256_ga_10-1055_s-0040-1707349.gif
Stumpf, Andreas; St-Jean, Frédéric; Lao, David; Cheng, Zhigang Ken; Angelaud, Remy; Gosselin, Francis: Practical Early Development Synthesis of Nav1.7 Inhibitor GDC-0310
https://www.thieme-connect.de/media/synthesis/202022/i_c0207_ga_10-1055_s-0040-1707859.gif
Chen, Chengsheng; Wu, Ling; Wang, Yuwen; Wu, Linglin; Zhang, Yongda: Copper-Catalyzed Asymmetric Hydroamination of Styrenes with pivZPhos as Ligand
https://www.thieme-connect.de/media/synthesis/202022/i_c0264_ga_10-1055_s-0040-1707346.gif
Crawford, James J.; Liao, Daohong; Kolesnikov, Aleksandr; Lee, Wendy; Landry, Matthew L.: Synthesis of an Azabicyclo[3.1.0]hexanone-Containing Inhibitor of NF-κΒ Inducing Kinase via Catalytic C–H Activation
https://www.thieme-connect.de/media/synthesis/202022/i_c0401_ga_10-1055_s-0040-1707279.gif

Issue 21/2020

Shiri, Morteza; Farajinia-Lehi, Noushin; Salehi, Parvin; Tanbakouchian, Zahra: Transition Metal and Inner Transition Metal Catalyzed Amide Derivatives Formation through Isocyanide Chemistry
https://www.thieme-connect.de/media/synthesis/202021/i_c0308_ga_10-1055_s-0040-1707357.jpg
Manne, Srinivasa Rao; de la Torre, Beatriz G.; El-Faham, Ayman; Albericio, Fernando: OxymaPure Coupling Reagents: Beyond Solid-Phase Peptide Synthesis
https://www.thieme-connect.de/media/synthesis/202021/i_c0384_ga_10-1055_s-0040-1706296.jpg
Zhao, Baoli; Liu, Yunyun: Step-Economical C–H Activation Reactions Directed by In Situ Amidation
https://www.thieme-connect.de/media/synthesis/202021/i_c0172_ga_10-1055_s-0040-1707124.gif
Spiliopoulou, Nikoleta; Constantinou, Constantinos T.; Triandafillidi, Ierasia; Kokotos, Christoforos G.: Synthetic Approaches to Acyl Hydrazides and Their Use as Synthons in Organic Synthesis
https://www.thieme-connect.de/media/synthesis/202021/i_c0186_ga_10-1055_s-0040-1707394.gif
Kolympadi Marković, Maria; Marković, Dean; Laclef, Sylvain: Amide Synthesis by Transamidation of Primary Carboxamides
https://www.thieme-connect.de/media/synthesis/202021/i_c0202_ga_10-1055_s-0040-1707133.gif
Shiri, Morteza; Gholami-Koupaei, Zahra; Bandehali-Naeini, Farzaneh; Tonekaboni, Maryam-Sadat; Soheil-Moghaddam, Saeedeh; Ebrahimi, Delaram; Karami, Sima; Notash, Behrouz: Highly Selective Synthesis of α-Hydroxy, α-Oxy, and α-Oxo Amides by a Post-Passerini Condensation Transformation
https://www.thieme-connect.de/media/synthesis/202021/i_c0210_ga_10-1055_s-0040-1707132.gif
Movahed, Farzaneh Soleymani; Sawant, Dinesh N.; Bagal, Dattatraya B.; Saito, Susumu: Tris(o-phenylenedioxy)cyclotriphosphazene as a Promoter for the Formation of Amide Bonds Between Aromatic Acids and Amines
https://www.thieme-connect.de/media/synthesis/202021/i_c0222_ga_10-1055_s-0040-1707174.gif
Smolobochkin, Andrey V.; Gazizov, Almir S.; Otegen, Nazerke K.; Voronina, Julia K.; Strelnik, Anna G.; Samigullina, Aida I.; Burilov, Alexander R.; Pudovik, Michail A.: Nucleophilic Cyclization/Electrophilic Substitution of (2,2-Dialkoxyethyl)ureas: Highly Regioselective Access to Novel 4-(Het)arylimidazolidinones and Benzo[d][1,3]diazepinones
https://www.thieme-connect.de/media/synthesis/202021/i_c0158_ga_10-1055_s-0040-1707864.gif
Verma, Saumya; Kumar, Puneet; Khatana, Anil K.; Chandra, Dinesh; Yadav, Ajay K.; Tiwari, Bhoopendra; Jat, Jawahar L.: Zinc(II)-Catalyzed Synthesis of Secondary Amides from Ketones via Beckmann Rearrangement Using Hydroxylamine-O-sulfonic Acid in Aqueous Media
https://www.thieme-connect.de/media/synthesis/202021/i_c0225_ga_10-1055_s-0040-1707809.gif
Kabes, Connor Q.; Gunn, Jack H.; Selbst, Maximilian A.; Lucas, Reagan F.; Gladysz, John A.: Syntheses of Enantiopure 1,2-Ethylenediamines with Tethered Secondary Amines of the Formula H2NCH2CH[(CH2)nNHMe]NH2 (n = 1–4) from α-Amino Acids: New Agents for Asymmetric Catalysis
https://www.thieme-connect.de/media/synthesis/202021/i_c0235_ga_10-1055_s-0040-1707146.jpg
Zhang, Rui; Zhang, Jun-Chao; Zhang, Wei-Yi; He, Yu-Qing; Cheng, Hua; Chen, Cheng; Gu, Yu-Cheng: A Practical Approach for the Transamidation of N,N-Dimethyl Amides with Primary Amines Promoted by Sodium tert-Butoxide under Solvent-Free Conditions
https://www.thieme-connect.de/media/synthesis/202021/i_c0297_ga_10-1055_s-0040-1705892.gif

Issue 08/2020

Connon, Robert; Carroll, Laura; Guiry, Patrick J.: A Base-Promoted One-Pot Asymmetric Friedel–Crafts Alkylation/Michael Addition of 4-Substituted Indoles
https://www.thieme-connect.de/media/synthesis/202008/i_c0474_ga_10-1055_s-0039-1690241.gif
Yang, Yuzhong; Zhou, Liwei; Yang, Xiumei; Luo, Xiai; Deng, Guobo; Yang, Yuan; Liang, Yun: Synthesis of Phenanthrenes via Palladium-Catalyzed Three-Component Domino Reaction of Aryl Iodides, Internal Alkynes, and o-Bromobenzoic Acids
https://www.thieme-connect.de/media/synthesis/202008/i_c0487_ga_10-1055_s-0039-1690737.gif
Henkel, Michael; Bach, Thorsten: Annulation of Indoles with 1,n-Dibromoalkanes by a Pd(II)-Catalyzed and Norbornene-Mediated Reaction Cascade
https://www.thieme-connect.de/media/synthesis/202008/i_c0495_ga_10-1055_s-0039-1690693.gif
Shen, Zican; Li, Chen; Mercado, Brandon Q.; Ellman, Jonathan A.: Cobalt(III)-Catalyzed Diastereoselective Three-Component C–H Bond Addition to Butadiene and Activated Ketones
https://www.thieme-connect.de/media/synthesis/202008/i_c0566_ga_10-1055_s-0039-1690741.gif
Lee, Sumin; Jang, Young Jin; Phipps, Erik J. T.; Lei, Honghui; Rovis, Tomislav: Rhodium(III)-Catalyzed Three-Component 1,2-Diamination of Unactivated Terminal Alkenes
https://www.thieme-connect.de/media/synthesis/202008/i_c0606_ga_10-1055_s-0039-1690756.gif
Sun, Manman; Li, Jinshan; Chen, Weida; Wu, Haijian; Yang, Jianguo; Wang, Zhiming: Palladium-Catalyzed [4+2] Annulation of Aryl and Alkenyl Carboxamides with 1,3-Dienes via C–H Functionalization: Synthesis of 3,4-Dihydroisoquinolones and 5,6-Dihydropyridinones
https://www.thieme-connect.de/media/synthesis/202008/i_t0490_ga_10-1055_s-0039-1690219.gif

Issue 23/2019

Special Topic Cover Page
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Sutherland, Andrew: Radiohalogenation of Organic Compounds: Practical Considerations and Challenges for Molecular Imaging
https://www.thieme-connect.de/media/synthesis/201923/i_s0302_ga_10-1055_s-0037-1611885.jpg
Milicevic Sephton, Selena; Zhou, Xiaoyun; Thompson, Stephen; Aigbirhio, Franklin I.: Preparation of the Serotonin Transporter PET Radiotracer 2-({2-[(Dimethylamino)methyl]phenyl}thio)-5-[18F]fluoroaniline (4-[18F]ADAM): Probing Synthetic and Radiosynthetic Methods
https://www.thieme-connect.de/media/synthesis/201923/i_c0355_ga_10-1055_s-0039-1690522.gif
Kitahara, Kazumasa; Mizutani, Haruna; Iwasa, Seiji; Shibatomi, Kazutaka: Asymmetric Synthesis of α-Chloro-α-halo Ketones by Decarboxylative Chlorination of α-Halo-β-ketocarboxylic Acids
https://www.thieme-connect.de/media/synthesis/201923/i_c0320_ga_10-1055_s-0039-1690009.gif
Dubost, Emmanuelle; Babin, Victor; Benoist, Florian; Hébert, Alexandra; Pigrée, Gilbert; Bouillon, Jean-Philippe; Fabis, Frédéric; Cailly, Thomas: Improvements of C–H Radio-Iodination of N-Acylsulfonamides toward Implementation in Clinics
https://www.thieme-connect.de/media/synthesis/201923/i_s0301_ga_10-1055_s-0037-1611884.gif
Thompson, Stephen; Lee, So Jeong; Jackson, Isaac M.; Ichiishi, Naoko; Brooks, Allen F.; Sanford, Melanie S.; Scott, Peter J. H.: Synthesis of [18F]-γ-Fluoro-α,β-unsaturated Esters and Ketones via Vinylogous 18F-Fluorination of α-Diazoacetates with [18F]AgF
https://www.thieme-connect.de/media/synthesis/201923/i_c0373_ga_10-1055_s-0039-1690012.jpg
Sarie, Jérôme C.; Neufeld, Jessica; Daniliuc, Constantin G.; Gilmour, Ryan: Willgerodt-Type Dichloro(aryl)-λ3-Iodanes: A Structural Study
https://www.thieme-connect.de/media/synthesis/201923/i_s0315_ga_10-1055_s-0037-1611886.gif

Issue 13/2019

Special Topic Cover Page
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Podyacheva, Evgeniya; Afanasyev, Oleg I.; Tsygankov, Alexey A.; Makarova, Maria; Chusov, Denis: Hitchhiker’s Guide to Reductive Amination
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Lai, Wing In; Leung, Man Pan; Choy, Pui Ying; Kwong, Fuk Yee: Sterically Hindered Amination of Aryl Chlorides Catalyzed by a New Carbazolyl-Derived P,N-Ligand-Composed Palladium Complex
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Purkait, Anisha; Jana, Chandan K.: N-Aminations of Benzylamines and Alicyclic Amines with Nitrosoarenes to Hydrazones and Hydrazides
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Li, Quan-Zhe; Wang, Xun-Hui; Hou, Si-Hua; Ma, Yan-Yan; Zhao, Deng-Gao; Zhang, Shu-Yu; Bai, He-Yuan; Ding, Tong-Mei: Silver-Catalyzed para-Selective C–H Amination of 1-Naphthyl­amides with Azodicarboxylates at Room Temperature
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Pratap, Ramendra; Yorimitsu, Hideki: Palladium-Catalyzed Amination of Aryl Sulfides and Sulfoxides with Azaarylamines of Poor Nucleophilicity
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Zhou, Huan; Zhao, Wenlei; Zhang, Tao; Guo, Haodong; Huang, Haizhou; Chang, Mingxin: Enantioselective Synthesis of 2-Substituted Pyrrolidines via Intramolecular­ Reductive Amination
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Issue 12/2019

Special Topic Cover Page
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Zhou, Yongyun; Khan, Ruhima; Fan, Baomin; Xu, Lijin: Ruthenium-Catalyzed Selective Reduction of Carboxylic Esters and Carboxamides
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Deshmukh, Dewal S.; Bhanage, Bhalchandra M.: Ruthenium-Catalyzed Annulation of N-Cbz Hydrazones via C–H/N–N Bond Activation for the Rapid Synthesis of Isoquinolines
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Das, Riki; Khot, Nandkishor Prakash; Deshpande, Akanksha Santosh; Kapur, Manmohan: Ruthenium-Catalyzed Directed C(3)–H Olefination of N-Acetyl-1,2-dihydroisoquinolines: A Method to Achieve C3-Olefinated Isoquinolines
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Bairy, Gurupada; Nandi, Arijit; Manna, Kartic; Jana, Ranjan: Ruthenium(II)-Catalyzed Migratory C–H Allylation/Hydroamination Cascade for the Synthesis of Rutaecarpine Analogues
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Tran, Christine; Haddad, Mansour; Ratovelomanana-Vidal, Virginie: Ruthenium-Catalyzed [2+2+2] Cycloaddition of α,ω-Diynes and Selenocyanates: An Entry to Selenopyridine Derivatives
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Kawano, Teruhiro; Watari, Ryo; Kayaki, Yoshihito; Ikariya, Takao: Catalytic Hydrogenation of Carboxamides with a Bifunctional Cp*Ru Catalyst Bearing an Imidazol-2-ylidene with a Protic Aminoethyl Side Chain
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Issue 17/2018

Special Topic Cover Page
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Oh, Eun Hye; Kim, Hyun Jin; Han, Soo Bong: Recent Developments in Visible-Light-Catalyzed Multicomponent Trifluoromethylation of Unsaturated Carbon–Carbon Bonds
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Zhou, Wen-Jun; Zhang, Yi-Han; Gui, Yong-Yuan; Sun, Liang; Yu, Da-Gang: Merging Transition-Metal Catalysis with Photoredox Catalysis: An Environmentally Friendly Strategy for C–H Functionalization
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Du, Yuliu; Wei, Zheng; Wang, Ting: Visible-Light-Mediated Synthesis of Oxidized Amides via Organic Photoredox Catalysis
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An, Xiao-De; Yu, Shouyun: Photoredox-Catalyzed Radical Relay Reaction Toward Functionalized Vicinal Diamines
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Voutyritsa, Errika; Nikitas, Nikolaos F.; Apostolopoulou, Mary K.; Gerogiannopoulou, Anna Dimitra D.; Kokotos, Christoforos G.: Photoorganocatalytic Atom Transfer Radical Addition of Bromoacetonitrile to Aliphatic Olefins
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Otomura, Nobutaka; Okugawa, Yuto; Hirano, Koji; Miura, Masahiro: Bromine Cation Initiated vic-Diphosphination of Styrenes with Diphosphines under Photoredox Catalysis
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Issue 16/2018

Special Topic Cover Page
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Baumann, Andreas N.; Eisold, Michael; Music, Arif; Didier, Dorian: One-Pot Preparation of Stable Organoboronate Reagents for the Functionalization of Unsaturated Four- and Five-Membered Carbo­- and Heterocycles
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Yamaguchi, Eiji; Kamito, Yuji; Matsuo, Kazuki; Ishihara, Jun; Itoh, Akichika: Photooxidative Keto-Trifluoromethylation of Styrenes by Means of an Anthraquinone-Based Organocatalyst
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Chen, Yizhou; Wang, Shanlu; Zhao, Li; Rong, Chenyan; Liu, Tong; Sun, Han; Wang, Yuping; Zhang, Jian; Zhong, Guofu: A Metal-Free Synthesis of 3-Phenoxyimidazo Heterocycles by Catalytic Oxidative Cyclization of 2-Amino-azaarenes with Lignin Models
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Suen, Linda M.; Wang, Cheng; Hunter, David N.; Mitchell, Helen J.; Converso, Antonella; ElMarrouni, Abdellatif: Synthesis of HIV NNRTI Doravirine Analogues via Visible-Light Photoredox Decarboxylative Cross-Coupling
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Liu, Yang; Daka, Mario; Bandini, Marco: Regio- and Stereoselective Nickel-Catalyzed Coupling of Boronic Acids with Allenoates
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Park, Jaerim; Song, Kwang Ho; Lee, Sunwoo: Palladium-Catalyzed Decarboxylative Coupling Reactions of Propiolic Acid Derivatives and Arylsulfonyl Hydrazide
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Torregrosa, Robert R. P.; Mendis, Shehani N.; Davies, Alex; Tunge, Jon A.: Palladium-Catalyzed Decarboxylative Benzylation of Acetylides and Enolates
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Li, Jing; Wang, Zhong-Xia: Nickel-Catalyzed Transformation of Aryl 2-Pyridyl Ethers via Cleavage of the Carbon–Oxygen Bond: Synthesis of Mono-α-arylated­ Ketones
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De, Pinaki Bhusan; Pradhan, Sourav; Shah, Tariq A.; Punniyamurthy, Tharmalingam: Iodine-Mediated Intramolecular C–H Amination of Benzimidazoles: A Metal-Free Route to Dihydroimidazobenzimidazoles
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Guan, Weiye; Liao, Jennie; Watson, Mary P.: Vinylation of Benzylic Amines via C–N Bond Functionalization of Benzylic Pyridinium Salts
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Yin, Zhiping; Power, Dennis J.; Wang, Zechao; Stewart, Scott G.; Wu, Xiao-Feng: Synthesis of 1,3,4-Oxadiazoles via Annulation of Hydrazides and Benzene-1,3,5-triyl Triformate under Metal-Free Conditions
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Issue 15/2018

Special Topic Cover Page
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Zhang, Qi; Raveendra Babu, Kaki; Huang, Zhouliang; Song, Jinna; Bi, Xihe: Visible-Light-Induced Radical Polynitration of Arylboronic Acids: Synthesis of Polynitrophenols
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Wu, Kui; Fang, Cheng; Kaur, Sarbjeet; Liu, Peng; Wang, Ting: Methylene Blue-Catalyzed Oxidative Cleavage of N-Carbonylated Indoles
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Wang, Guang-Zu; Shang, Rui; Fu, Yao: Irradiation-Induced Palladium-Catalyzed Direct C–H Alkylation of Heteroarenes with Tertiary and Secondary Alkyl Bromides
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Hamsath, Akil; Galloway, Jordan D.; Baxter, Ryan D.: Quinone C–H Alkylations via Oxidative Radical Processes
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Li, Longji; Yang, Qi; Jia, Zongbin; Luo, Sanzhong: Organocatalytic Electrochemical C–H Lactonization of Aromatic Carboxylic Acids
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Levin, Vitalij V.; Agababyan, Daniil P.; Struchkova, Marina I.; Dilman, Alexander D.: Dimerization of Benzyl and Allyl Halides via Photoredox-Mediated Disproportionation of Organozinc Reagents
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Manick, Anne-Doriane; Tanaka, Hirotaka; Oisaki, Kounosuke; Kanai, Motomu: Organophotoredox/Copper Hybrid Catalysis for Regioselective Allylic­ Aminodecarboxylation of β,γ-Unsaturated Carboxylic Acids
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Egami, Hiromichi; Ito, Yuta; Ide, Takafumi; Masuda, Shuya; Hamashima, Yoshitaka: Simple Photo-Induced Trifluoromethylation of Aromatic Rings
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Gharpure, Santosh J.; Niranjana, P.; Porwal, Suheel K.: Cascade Radical Cyclization to Vinylogous Carbonates/Carbamates for the Synthesis of Oxa- and Aza-Angular Triquinanes: Diastereoselectivity Depends on the Ring Size of Radical Precursor
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Li, Cheng-Kun; Zhang, Dong-Liang; Olamiji, Ogundipe Olukayode; Zhang, Pei-Zhi; Shoberu, Adedamola; Zou, Jian-Ping; Zhang, Wei: Mn(OAc)3-Mediated Regioselective Radical Alkoxycarbonylation of Indoles, Pyrimidinones, and Pyridinones
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Deng, Weili; Li, Yajun; Li, You-Gui; Bao, Hongli: Iron-Catalyzed Carboiodination of Alkynes
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Zhao, Xinxin; Chen, Ming; Huang, Binbin; Yang, Chao; Gao, Yuan; Xia, Wujiong: Photoinduced Cross-Coupling of Amines with 1,2-Diiodobenzene and Its Application in the Synthesis of Carbazoles
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Luo, Kai; Zhang, Ling; Wei, Kai; Yang, Wen-Chao; Wu, Lei: Latent Radical Cleavage of α-Allenylic C–O Bonds: Potassium Persulfate Mediated Thiolation of Allenylphosphine Oxides
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Mei, Chong; Hu, Yixin; Lu, Wenjun: Visible-Light-Driven Oxidation of N-Alkylamides to Imides Using Oxone/H2O and Catalytic KBr
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Das, Dipendu; Khan, Hina P. A.; Chakraborty, Tushar Kanti: Ti(III)-Mediated Radical-Induced Approach to a Bicyclic δ-Lactone with a Bridgehead β-Hydroxy Group
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Fukuyama, Takahide; Bando, Takanobu; Ryu, Ilhyong: Electron-Transfer-Induced Intramolecular Heck Carbonylation Reactions Leading to Benzolactones and Benzolactams
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Baguia, Hajar; Deldaele, Christopher; Romero, Eugénie; Michelet, Bastien; Evano, Gwilherm: Copper-Catalyzed Photoinduced Radical Domino Cyclization of Ynamides and Cyanamides: A Unified Entry to Rosettacin, Luotonin A, and Deoxyvasicinone
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Issue 21/2017

Special Topic Cover Page
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Takenouchi, Yuta; Ito, Hajime: Copper(I)-Catalyzed Boryl Substitution of Allyl Aminals: Selective Synthesis of Linear γ-Aminoallylboronates
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Miura, Wataru; Hirano, Koji; Miura, Masahiro: Iridium-Catalyzed Site-Selective C–H Borylation of 2-Pyridones
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Jang, Won Jun; Han, Jung Tae; Yun, Jaesook: NHC-Copper-Catalyzed Tandem Hydrocupration and Allylation of Alkenyl Boronates
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Pinet, Sandra; Liautard, Virginie; Debiais, Mégane; Pucheault, Mathieu: Radical Metal-Free Borylation of Aryl Iodides
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Saito, Hayate; Nogi, Keisuke; Yorimitsu, Hideki: Palladium-Catalyzed Double Borylation of Diaryl Sulfoxides with Diboron
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Farre, Albert; Briggs, Rachel; Pubill-Ulldemolins, Cristina; Bonet, Amadeu: Developing a Bench-Scale Green Diboration Reaction toward Industrial Application
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Issue 20/2017

Special Topic Cover Page
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Couly, Florence; Dubouilh-Benard, Carole; Besson, Thierry; Fruit, Corinne: Late-Stage C–H Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one Backbone: Synthesis of an Array of Potential Kinase Inhibitors
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Sabat, Nazarii; Smoleń, Sabina; Nauš, Petr; Perlíková, Pavla; Cebová, Magdaléna; Poštová Slavětínská, Lenka; Hocek, Michal: Synthesis of 2,6-Substituted 7-(Het)aryl-7-deazapurine Nucleobases (2,4-Disubstituted 5-(Het)aryl-pyrrolo[2,3-d]pyrimidines)
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Skonieczny, Kamil; Jaźwiński, Jarosław; Gryko, Daniel T.: The Synthesis of Imidazo[1,2-f]phenanthridines, Phenanthro-[9,10-d]imidazoles, and Phenanthro[9′,10′:4,5]imidazo[1,2-f]-phenanthridines via Intramolecular Oxidative Aromatic Coupling
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Yu, Zhao; Bo, Tang; Aiying, Guan; Weiwei, Wang; Zhenhua, Zhang; Mingan, Wang: Synthesis and Fungicidal Activity of (E)-5-[1-(4-Phenyl-2-oxo-1-oxaspiro[4.5]dec-3-en-3-yl)ethylidene]-2-aminoimidazolin-4-one Derivatives
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Tokumaru, Kazuyuki; Bera, Kalisankar; Johnston, Jeffrey N.: 1,3,4-Oxadiazole and Heteroaromatic-Fused 1,2,4-Triazole Synthesis­ Using Diverted Umpolung Amide Synthesis
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Lessi, Marco; Panzetta, Gianmarco; Marianetti, Giulia; Bellina, Fabio: Improved Synthesis of Symmetrical 2,5-Diarylimidazoles by One-Pot Palladium-Catalyzed Direct Arylation Tailored on the Electronic Features of the Aryl Halide
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Zhang, Xiaojuan; Han, Xiuling; Hu, Zhiyong; Lu, Xiyan: Synthesis of Substituted Piperidines via Cationic Palladium(II)-Catalyzed Reductive Coupling of N-Tosyl-Tethered Alkynones
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Shang, Xiao-Jie; Liu, Zhong-Quan: A Catalyzed Aerobic Intramolecular C–O Bond Formation: Facile Access to Ring-Fused Dihydrobenzoxazine Derivatives
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Issue 18/2017

Special Topic Cover Page
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Abe, Takumi; Haruyama, Tomohiro; Yamada, Koji: C4 Pictet–Spengler Reactions for the Synthesis of Core Structures in Hyrtiazepine Alkaloids
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Pertschi, Romain; Miaskiewicz, Solène; Weibel, Jean-Marc; Pale, Patrick; Blanc, Aurélien: Gold(I)-Catalyzed Cascade: Synthesis of 2,5-Disubstituted Pyrroles from N-Sulfonyl-2-(1-ethoxypropargyl)azetidines through Cyclization/Nucleophilic Substitution/Elimination
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Cacchi, Sandro; Fabrizi, Giancarlo; Goggiamani, Antonella; Iazzetti, Antonia; Verdiglione, Rosanna: 2-(Aminomethyl)-3-arylindoles from 3-(o-Trifluoroacetamidoaryl)-1-propargylic Alcohols, Aryl Halides, and Amines: A Domino Palladium-Catalyzed Three-Component Approach
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Zheng, Min; Chen, Kai; Zhu, Shifa: One-Pot Synthesis of Indole Derivatives from the Reaction of Nitroalkynes and Alkynes via a Mercury-Carbene Intermediate
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Shimizu, Maki; Hayama, Noboru; Kimachi, Tetsutaro; Inamoto, Kiyofumi: Copper-Catalyzed Intramolecular C–H Amination: A New Entry to Substituted Xanthine Derivatives
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Opsomer, Tomas; Thomas, Joice; Dehaen, Wim: Chemoselectivity in the Synthesis of 1,2,3-Triazoles from Enolizable Ketones, Primary Alkylamines, and 4-Nitrophenyl Azide
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Fujita, Shoji; Shibuya, Masatoshi; Yamamoto, Yoshihiko: Intramolecular Hydroalkoxylation/Reduction and Hydroamination/Reduction of Unactivated Alkynes Using a Silane–Iodine Catalytic System
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Paul, Kartick; Jalal, Swapnadeep; Kundal, Sandip; Chakraborty, Baitan; Jana, Umasish: Iron-Catalyzed Intramolecular Alkyne–Carbonyl Metathesis: A New Cyclization Strategy for the Synthesis of Benzocarbazole and Azepino[1,2-a]indole Derivatives
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Li, Xue-Fei; Lin, Jin-Shun; Liu, Xin-Yuan: Catalytic Radical Intramolecular Aminoperfluoroalkylation and Aminodifluoromethylation of Unactivated Alkenes with Fluoro­alkylsulfonyl Chlorides
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Mullapudi, Venkannababu; Bhogade, Ravindra B.; Deshpande, Mukund V.; Ramana, Chepuri V.: Phenol Oxidative Dearomatization of Modified Nucleoside Templates: A Simple Access to the C7-Spiroannulated Octosyl Acid Framework
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Ghosh, Arun K.; Tomaine, Anthony J.; Cantwell, Kelsey E.: Lewis Acid Mediated Cyclizations: Diastereoselective Synthesis of Six- to Eight-Membered Substituted Cyclic Ethers
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Lee, Sang Eun; Lee, Seong Jong; Cheon, Cheol-Hong: Concise Total Syntheses of Paullone and Kenpaullone via Cyanide-Catalyzed Intramolecular Imino-Stetter Reaction
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Triandafillidi, Ierasia; Sideri, Ioanna K.; Tzaras, Dimitrios Ioannis; Spiliopoulou, Nikoleta; Kokotos, Christoforos G.: Green Organocatalytic Synthesis of Dihydrobenzofurans by Oxidation–Cyclization of Allylphenols
https://www.thieme-connect.de/media/synthesis/201718/i_c0154_ga_10-1055_s-0036-1588998.gif
Nayak, Sanatan; Prabagar, B.; Ghosh, Nayan; Mallick, Rajendra K.; Sahoo, Akhila K.: Ag(I)-Catalyzed Cycloisomerization and Cyclization of Ketene Aminals: Construction of Azepine and 1,2-Dihydropyridine Derivatives
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Nagamoto, Midori; Nishimura, Takahiro; Yorimitsu, Hideki: Iridium-Catalyzed Intramolecular Oxidative Cyclization of Alkenyl Amides and Alkenoic Acids
https://www.thieme-connect.de/media/synthesis/201718/i_c0211_ga_10-1055_s-0036-1588435.gif
Li, Dianjun; Li, Ying; Yu, Wei: tert-Butyl Hypochlorite Induced Cyclization of Ethyl 2-(N-Aryl­carbamoyl)-2-iminoacetates
https://www.thieme-connect.de/media/synthesis/201718/i_c0243_ga_10-1055_s-0036-1588462.gif
Li, Jie; Xiao, Jun-An; Zhao, Shu-Juan; Xiang, Hao-Yue; Yang, Hua: Facile Construction of Pyrrolo[1,2-a]indolenine Scaffold via Dia­stereoselective [3+2] Annulation of Donor–Acceptor Cyclopropane with Indolenine
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Issue 17/2017

Special Topic Cover Page
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Hammann, Jeffrey M.; Hofmayer, Maximilian S.; Lutter, Ferdinand H.; Thomas, Lucie; Knochel, Paul: Recent Advances in Cobalt-Catalyzed Csp2 and Csp3 Cross-Couplings
https://www.thieme-connect.de/media/synthesis/201717/i_c0069_ga_10-1055_s-0036-1588430.gif
Ferrand, Laura; Lyu, Ye; Rivera-Hernández, Alejandro; Fallon, Brendan J.; Amatore, Muriel; Aubert, Corinne; Petit, Marc: Hydroboration and Diboration of Internal Alkynes Catalyzed by a Well-Defined Low-Valent Cobalt Catalyst
https://www.thieme-connect.de/media/synthesis/201717/i_c0089_ga_10-1055_s-0036-1588996.gif
Joshi, Hemant; Ghosh, Subrata K.; Gladysz, John A.: Enantioselective Additions of Stabilized Carbanions to Imines Generated from α-Amido Sulfones By Using Lipophilic Salts of Chiral Tris(1,2-diphenylethylenediamine) Cobalt(III) Trications as Hydrogen Bond Donor Catalysts
https://www.thieme-connect.de/media/synthesis/201717/i_c0236_ga_10-1055_s-0036-1590502.gif
Suo, Jian-Feng; Zhao, Xue-Mei; Zhang, Kai-Xin; Zhou, Sheng-Li; Niu, Jun-Long; Song, Mao-Ping: Cobalt-Catalyzed Perfluoroalkylation of Quinoline Amides at the C5 Position
https://www.thieme-connect.de/media/synthesis/201717/i_c0033_ga_10-1055_s-0036-1588160.gif
Hofmayer, Maximilian S.; Hammann, Jeffrey M.; Lutter, Ferdinand H.; Knochel, Paul: Large-Scale Cobalt-Catalyzed Cross-Couplings of Functionalized Bench-Stable Arylzinc Pivalates with (Hetero)Aryl and Alkenyl Halides­
https://www.thieme-connect.de/media/synthesis/201717/i_c0090_ga_10-1055_s-0036-1588986.gif
Xu, Kun; Tan, Zhoumei; Zhang, Haonan; Zhang, Sheng: Cobalt-Catalyzed Monoselective ortho-C–H Ethylation of Carboxamides with Triethylaluminum
https://www.thieme-connect.de/media/synthesis/201717/i_c0095_ga_10-1055_s-0036-1589010.gif
Kalsi, Deepti; Barsu, Nagaraju; Dahiya, Pardeep; Sundararaju, Basker: C–H and N–H Bond Annulation of Benzamides with Isonitriles Catalyzed by Cobalt(III)
https://www.thieme-connect.de/media/synthesis/201717/i_c0137_ga_10-1055_s-0036-1589011.gif
Cabré, Albert; Verdaguer, Xavier; Riera, Antoni: Ethylene Glycol Assisted Intermolecular Pauson–Khand Reaction
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Jamieson, Megan L.; Brant, Nicola Z.; Brimble, Margaret A.; Furkert, Daniel P.: Remarkable Influence of Cobalt Catalysis on Epoxide Ring-Opening with Sulfoxonium Ylides
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Midya, Siba P.; Mondal, Akash; Begum, Ayesha; Balaraman, Ekambaram: A Simple Cobalt(II) Chloride Catalyzed N-Alkylation of Amines with Alcohols
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Issue 16/2017

Special Topic Cover Page
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Watabe, Yota; Kanazawa, Kohei; Fujita, Takeshi; Ichikawa, Junji: Nickel-Catalyzed Hydroalkenylation of Alkynes through C–F Bond Activation: Synthesis of 2-Fluoro-1,3-dienes
https://www.thieme-connect.de/media/synthesis/201716/i_c0187_ga_10-1055_s-0036-1588842.gif
Xiao, Jian; Wang, Ya-Wen; Peng, Yu: Nickel-Promoted Reductive Cyclization Cascade: A Short Synthesis of a New Aromatic Strigolactone Analogue
https://www.thieme-connect.de/media/synthesis/201716/i_c0156_ga_10-1055_s-0036-1588804.gif
Barday, Manuel; Janot, Christopher; Clare, Daniel; Carr-Knox, Caitlin; Higginson, Bradley; Ho, Kelvin Y. T.; Aïssa, Christophe: On the Regioselectivity of the Nickel-Catalyzed Insertion of Alkynes into the Carbon–Carbon Bond of Oxetan-3-one
https://www.thieme-connect.de/media/synthesis/201716/i_c0213_ga_10-1055_s-0036-1589052.gif
Sumida, Yuto; Sumida, Tomoe; Hosoya, Takamitsu: Nickel-Catalyzed Reductive Cross-Coupling of Aryl Triflates and Nonaflates with Alkyl Iodides
https://www.thieme-connect.de/media/synthesis/201716/i_c0215_ga_10-1055_s-0036-1588464.gif
Shi, Shicheng; Szostak, Michal: Nickel-Catalyzed Negishi Cross-Coupling of N-Acylsuccinimides: Stable, Amide-Based, Twist-Controlled Acyl-Transfer Reagents via N–C Activation
https://www.thieme-connect.de/media/synthesis/201716/i_c0192_ga_10-1055_s-0036-1588845.jpg

Issue 13/2017

Special Topic Cover Page
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Parmeggiani, Camilla; Matassini, Camilla; Cardona, Francesca; Goti, Andrea: On the Oxidation of Hydroxylamines with o-Iodoxybenzoic Acid (IBX)
https://www.thieme-connect.de/media/synthesis/201713/i_c0240_ga_10-1055_s-0036-1588457.gif
Muñiz, Kilian; Fra, Laura: Enantioselective 4-Hydroxylation of Phenols under Chiral Organoiodine(I/III) Catalysis
https://www.thieme-connect.de/media/synthesis/201713/i_c0133_ga_10-1055_s-0036-1588808.gif
Kiyokawa, Kensuke; Takemoto, Kenta; Yahata, Shunsuke; Kojima, Takumi; Minakata, Satoshi: Oxidative Cyclization of β,γ-Unsaturated Carboxylic Acids Using Hypervalent Iodine Reagents: An Efficient Synthesis of 4-Substituted Furan-2-ones
https://www.thieme-connect.de/media/synthesis/201713/i_c0096_ga_10-1055_s-0036-1588987.gif
Fujita, Morifumi; Lee, Hee Jin; Ichihara, Chisaki; Sugimura, Takashi: E/Z-Selectivity Controlled by Participation of Internal Oxy Group During Electrophilic Substitution of Alk-1-enylboronate with Bis(2,4,6-trimethylpyridine)iodonium Salt
https://www.thieme-connect.de/media/synthesis/201713/i_c0884_ga_10-1055_s-0036-1558967.gif
Li, Guangchen; Zhang-Negrerie, Daisy; Du, Yunfei: Synthesis of N-Substituted 2-Amino-3,4-diiodofurans from Allenes via NIS-Mediated Intramolecular Electrophilic Iodocyclization
https://www.thieme-connect.de/media/synthesis/201713/i_c0126_ga_10-1055_s-0036-1588792.gif
Dagenais, Robin; Lauriers, Antoine Jobin-Des; Legault, Claude Y.: Iodine(III)-Mediated Oxidative Hydrolysis of Haloalkenes: Investigation of the Effect of Iodine(III) Reagents
https://www.thieme-connect.de/media/synthesis/201713/i_c0216_ga_10-1055_s-0036-1588439.gif

Issue 17/2016

Shaw, Subrata; White, James D.: Asymmetric Catalysis with Iron–Salen Complexes
https://www.thieme-connect.de/media/synthesis/201617/i_c0181_ga_10-1055_s-0035-1562103.gif
Liu, Cheng-Yuan; Chen, Ying-Ho; Chen, Chih-Hao; Yu, Ming-Shiuan; Tsai, Fu-Yu; Ong, Tiow-Gan: Selective C(8)–H Activation of Imidazopyridines Mediated by Cooperative Nickel–Aluminum Catalysis
https://www.thieme-connect.de/media/synthesis/201617/i_c0130_ga_10-1055_s-0035-15661438.gif
Kumar, Ravindra; Tamai, Eri; Ohnishi, Akira; Nishimura, Akira; Hoshimoto, Yoichi; Ohashi, Masato; Ogoshi, Sensuke: Nickel-Catalyzed Enantioselective Synthesis of Cyclobutenes via [2+2] Cycloaddition of α,β-Unsaturated Carbonyls with 1,3-Enynes
https://www.thieme-connect.de/media/synthesis/201617/i_c0174_ga_10-1055_s-0035-1561669.gif
Malineni, Jagadeesh; Jezorek, Ryan L.; Zhang, Na; Percec, Virgil: An Indefinitely Air-Stable σ-NiII Precatalyst for Quantitative Cross-Coupling of Unreactive Aryl Halides and Mesylates with Aryl Neopentylglycolboronates
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Malineni, Jagadeesh; Jezorek, Ryan L.; Zhang, Na; Percec, Virgil: NiIICl(1-Naphthyl)(PCy3)2, An Air-Stable σ-NiII Precatalyst for Quantitative Cross-Coupling of Aryl C–O Electrophiles with Aryl Neopentylglycolboronates
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Moragas, Toni; Martin, Ruben: Nickel-Catalyzed Reductive Carboxylation of Cyclopropyl Motifs with Carbon Dioxide
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Sugiyama, Yu-ki; Heigozono, Shiori; Tamura, Kazuhiro; Okamoto, Sentaro: Iron-Catalyzed Reductive Metalation–Allylation and Metalative Cyclization of 2,3-Disubstituted Oxetanes and Their Stereoselectivity
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Zhang, Qingchen; Wang, Xuan; Qian, Qun; Gong, Hegui: Nickel-Catalyzed Reductive Cross-Coupling of Benzyl Halides with Aryl Halides
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Xi, Tuo; Chen, Xu; Zhang, Heyi; Lu, Zhan: Reductive Cyclization of 1,6- and 1,7-Enynes Catalyzed by Iron Complexes
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Issue 16/2016

Cai, Pin-Wen; You, Zhi-Hao; Xie, Liang-Hui; Tan, Rui; Tong, Zhi-Ping; Liu, Yan-Kai: The Attractive Application of Lactol Chemistry: From Racemic Lactol to Natural Product Skeleton
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Su, Lin; Xu, Ming-Hua: Asymmetric Reformatsky-Type Reaction of Isatin-Derived N-Sulfinyl Ketimines: Efficient and Practical Synthesis of Enantiopure Chiral 2-Oxoindolinyl-β3,3-Amino Esters
https://www.thieme-connect.de/media/synthesis/201616/i_c0034_ga_10-1055_s-0035-1561426.gif
Gao, Xing; Han, Jianwei; Wang, Limin: Chiral Iminophosphorane Organocatalyzed Asymmetric Sulfenyl­ation of 3-Substituted Oxindoles: Substrate-Interrelated Enantio­selectivities
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Nishimura, Takahiro; Nagai, Tomotaka; Takechi, Ryosuke; Ebe, Yusuke: Rhodium-Catalyzed Enantioselective Addition of Tricyclopropylboroxin to N-Sulfonylimines
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Chen, Shi; Mondal, Mukulesh; Ibrahim, Ahmad A.; Wheeler, Kraig A.; Kerrigan, Nessan J.: Asymmetric Synthesis of Dipropionate Derivatives through Catalytic Hydrogenation of Enantioenriched E-Ketene Heterodimers
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Sun, Shutao; Liu, Lei: Catalytic Enantioselective Alkynylation of Tetrahydroisoquinoline-Based N-Acyl Hemiaminals
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Feng, Yangyang; Huang, Ruofeng; Hu, Liangzhen; Xiong, Yan; Coeffard, Vincent: Chiral C2-Symmetric Iodoarene-Catalyzed Asymmetric α-Oxidation of β-Keto Esters
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Berti, Francesco; Favero, Lucilla; Pineschi, Mauro: Asymmetric Synthesis of Methylphenidate and Quinolizidinones by Addition of Aldehydes to Piperidine-Based Conjugated N-Acyl­iminium Ions
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Dai, Wen; Mi, Yuan; Lv, Ying; Shang, Sensen; Li, Guosong; Chen, Guangwen; Gao, Shuang: Development of a Continuous-Flow Microreactor for Asymmetric Epoxidation of Electron-Deficient Olefins
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Salomó, Ernest; Orgué, Sílvia; Riera, Antoni; Verdaguer, Xavier: Efficient Preparation of (S)- and (R)-tert-Butylmethylphosphine–Borane: A Novel Entry to Important P-Stereogenic Ligands
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Shibata, Takanori; Fukai, Miku; Sekine, Ryosuke; Hazra, Madhurima; Kanyiva, Kyalo Stephen: Enantioselective Synthesis of Planar-Chiral 1,n-Dioxa[n]paracyclophane-Based Phosphites and Their Application as Chiral Ligands
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Vishwanath, Manjunatha; Prakash, Muthuraj; Vinayagam, Poopathy; Kesavan, Venkitasamy: Construction of Polycyclic Fused Pyrrolidines with Three Contiguous Stereocenters via Michael Addition of Vinylmalononitriles to Nitrostyrenes­ Using l-Proline-Derived Thiourea
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Issue 12/2016

Wildermuth, Raphael; Speck, Klaus; Magauer, Thomas: Gold(I)-Catalyzed Enyne Cyclizations: Studies Toward the Total Synthesis of (+)-Aureol
https://www.thieme-connect.de/media/synthesis/201612/i_c0046_ga_10-1055_s-0035-1561589.gif
Shi, Shicheng; Lalancette, Roger; Szostak, Michal: Cyclization of Imides to 2-Azabicycles via Aminoketyl Radicals by Using Samarium(II) Iodide–Water: Reaction Development, Synthetic Scope, and Mechanistic Studies
https://www.thieme-connect.de/media/synthesis/201612/i_c0066_ga_10-1055_s-0035-1560437.gif
Sugimoto, Kenji; Hoshiba, Yuya; Tsuge, Kiyoshi; Matsuya, Yuji: Synthesis of Substituted Pyrrolo[2,1-a]isoquinolines by Gold-Catalyzed Domino Cyclization of Alkynyl Iminoesters
https://www.thieme-connect.de/media/synthesis/201612/i_c0072_ga_10-1055_s-0035-1561423.gif
Shirke, Rajendra P.; Reddy, Virsinha; Anand, R. Vijaya; Ramasastry, S. S. V.: Furans to Benzofurans: Intramolecular Cross-Benzoin Reactions Catalysed by N-Heterocyclic Carbenes
https://www.thieme-connect.de/media/synthesis/201612/i_c0133_ga_10-1055_s-0035-1560432.gif
Gandeepan, Parthasarathy; Rajamalli, Pachaiyappan; Cheng, Chien-Hong: Palladium-Catalyzed C–H Activation and Cyclization of Anilides with 2-Iodoacetates and 2-Iodobenzoates: An Efficient Method toward Oxindoles and Phenanthridones
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Malkina, Anastasiya G.; Stepanov, Anton V.; Sobenina, Lyubov N.; Shemyakina, Olesya A.; Ushakov, Igor A.; Smirnov, Vladimir I.; Trofimov, Boris A.: Organocatalyzed Microwave-Assisted Competing Cyclization of Cyanopropargylic Alcohols with Carboxylic Acids: 4-Cyano-3(2H)-furanones versus 4-Cyano-[(Z)-3-cyanomethylene]-2,3-dihydro­furans
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Nambu, Hisanori; Ono, Naoki; Yakura, Takayuki: Acid-Catalyzed Ring-Opening Cyclization of Spirocyclopropanes for the Construction of a 2-Arylbenzofuran Skeleton: Total Synthesis of Cuspidan B
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Parker, Patrick D.; Pierce, Joshua G.: Synthesis of 1,2,4-Oxadiazoles via DDQ-Mediated Oxidative Cyclization of Amidoximes
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Cavitt, Marchello A.; France, Stefan: Aluminum(III)-Catalyzed, Formal Homo-Nazarov-Type Ring-Opening Cyclizations toward the Synthesis of Functionalized Tetrahydroindolizines
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Ren, Zhi-Hui; Zhao, Mi-Na; Yi, Yukun; Wang, Yao-Yu; Guan, Zheng-Hui: Copper-Catalyzed Aerobic Oxidative Cyclization of Ketoxime Acetates with Pyridines for the Synthesis of Imidazo[1,2-a]pyridines
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Morita, Nobuyoshi; Mashiko, Rie; Hakuta, Dai; Eguchi, Daisuke; Ban, Shintaro; Hashimoto, Yoshimitsu; Okamoto, Iwao; Tamura, Osamu: Gold-Catalyzed Dimeric Cyclization of Isoeugenol and Related 1-Phenylpropenes in Ionic Liquid: Environmentally Friendly and Stereoselective Synthesis of 1,2,3-Trisubstituted 2,3-Dihydro-1H-indenes
https://www.thieme-connect.de/media/synthesis/201612/i_c0078_ga_10-1055_s-0035-1561604.gif
Yu, Mangfei; Zhang, Qian; Wang, Jia; Huang, Peng; Yan, Pengfei; Zhang, Rui; Dong, Dewen: Triflic Anhydride Mediated Ring-Opening/Recyclization Reaction of α-Carbamoyl α-Oximyl Cyclopropanes with DMF: Synthetic Route to 5-Aminoisoxazoles
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Issue 11/2016

Li, Zhilong; Tong, Rongbiao: Asymmetric Total Syntheses of the trans-2-Aryl-6-alkyltetrahydropyrans Diospongin B and Parvistones D and E from a Common Precursor
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Kousara, Mohammad; Bideau, Franck Le; Ibrahim, Rama; Ferry, Angélique; Venot, Pierre-Etienne; Dejean, Camille; Raingeaud, Joël; Dubois, Joëlle; Retailleau, Pascal; Dumas, Françoise: Suberosanes as Potential Antitumor Agents: First Enantioselective Total Synthesis of (1S)-Suberosanone and Configurational Assignment of Suberosenol A
https://www.thieme-connect.de/media/synthesis/201611/i_c0040_ga_10-1055_s-0035-1561430.jpg
Nakayama, Yasuaki; Maeda, Yuichiro; Hama, Naoto; Sato, Takaaki; Chida, Noritaka: Total Synthesis of (–)-Stemoamide by Sequential Overman/Claisen Rearrangement
https://www.thieme-connect.de/media/synthesis/201611/i_c0050_ga_10-1055_s-0035-1561948.gif
García-Ruiz, Cristina; Cheng-Sánchez, Iván; Sarabia, Francisco: Synthesis of (–)- and (+)-Gummiferol via Asymmetric Synthesis of Glycidic Amides
https://www.thieme-connect.de/media/synthesis/201611/i_c0102_ga_10-1055_s-0035-1561606.gif
Konda, Saidulu; Khatravath, Mahender; Mallurwar, Naveen Kumar; Rao, Pallavi; Sripelly, Shivashankar; Iqbal, Javed; Arya, Prabhat: Stereoselective Synthesis of the C27–C35 Eribulin Fragment and Its Utilization in Building Structurally Diverse Macrocycles
https://www.thieme-connect.de/media/synthesis/201611/i_c0084_ga_10-1055_s-0035-1561431.gif
Ye, Jian-Liang; Liu, Yang; Zhang, Yu-Feng; Yang, Zhi-Ping; Huang, Pei-Qiang: Studies on the Second-Generation Approach to Loline Alkaloids: Synthesis of N-Bus-norloline through N-tert-Butanesulfinyl Imine Based Asymmetric Vinylogous Mannich Reaction
https://www.thieme-connect.de/media/synthesis/201611/i_c0116_ga_10-1055_s-0035-1561432.gif
Yang, Xiaoyu; Yu, Biao: Synthesis of Landomycin D: Studies on the Saccharide Assembly
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Hunter, Thomas J.; Wang, Yanping; Zheng, Jiamin; O’Doherty, George A.: Asymmetric Iterative Hydration of Polyene Strategy to Cryptocaryols A and B
https://www.thieme-connect.de/media/synthesis/201611/i_c0125_ga_10-1055_s-0035-1561607.gif

Issue 19/2015

Liu, Le; Zhang-Negrerie, Daisy; Du, Yunfei; Zhao, Kang: Hypervalent Iodine Mediated C–C Double Bond Activation: A Cascade Access to α-Keto Diacetates from Readily Available Cinnamic Acids
https://www.thieme-connect.de/media/synthesis/201519/i_c0218_ga_10-1055_s-0034-1378718.gif
Sun, Gui-Jun; Wang, Yong; Kang, Qiang: Palladium-Catalyzed Allylic Amination of Homoallylic Alcohols with Amines via Carbon–Carbon Bond Cleavage
https://www.thieme-connect.de/media/synthesis/201519/i_c0189_ga_10-1055_s-0034-1380418.gif
Okuma, Kentaro; Horigami, Kenta; Nagahora, Noriyoshi; Shioji, Kosei: Enantioselective Synthesis of 4,4′-Biaryl-BINOLs from Arynes and β-Diketones
https://www.thieme-connect.de/media/synthesis/201519/i_c0278_ga_10-1055_s-0034-1380452.gif
Aoyama, Tadashi; Hayakawa, Mamiko; Kubota, Sho; Ogawa, Sumire; Nakajima, Erika; Mitsuyama, Emi; Iwabuchi, Taku; Kaneko, Haruki; Obara, Rina; Takido, Toshio; Kodomari, Mitsuo; Ouchi, Akihiko: Simple Method for sp2–sp3 and sp3–sp3 Carbon–Carbon Bond Activation in 2-Substituted 1,3-Diketones
https://www.thieme-connect.de/media/synthesis/201519/i_c0277_ga_10-1055_s-0034-1378862.gif
Choi, Jeongae; Jung, Hyunuk; Yeo, Jeong-Eun; Koo, Sangho: Synthesis of Tribenzotropone by Ring Expansion of Phenanthrene-9,10-dione
https://www.thieme-connect.de/media/synthesis/201519/i_c0244_ga_10-1055_s-0034-1381045.gif
Shadrin, Ivan A.; Rzhevskii, Sergey A.; Rybakov, Victor B.; Babaev, Eugene V.: Sonogashira Reaction of the Indolizine Ring
https://www.thieme-connect.de/media/synthesis/201519/i_c0259_ga_10-1055_s-0034-1378861.gif
Parida, Amarchand; Sharique, Mohd.; Kakde, Badrinath N.; Ghosh, Santanu; Bisai, Alakesh: Efficient Synthesis of 3-Alkynyl-2-(hydroxymethyl)cyclohex-2-en-1-ones by a Stork–Danheiser Sequence from Vinylogous Esters and Terminal Alkynes
https://www.thieme-connect.de/media/synthesis/201519/i_c0264_ga_10-1055_s-0034-1380451.gif
Ou, Yang; Qin, Chong; Song, Song; Jiao, Ning: An Iron-Catalyzed Direct Approach to Amides from Benzyl Azides via C–C Bond Cleavage
https://www.thieme-connect.de/media/synthesis/201519/i_c0307_ga_10-1055_s-0034-1380222.gif

Issue 18/2015

Luo, Guo-Ying; Wu, Hao; Tang, Yu; Li, Hui; Yeom, Hyun-Suk; Yang, Ka; Hsung, Richard P.: A Total Synthesis of (±)-Rhododaurichromanic Acid A via an Oxa-[3+3] Annulation of Resorcinols
https://www.thieme-connect.de/media/synthesis/201518/i_c0219_ga_10-1055_s-0034-1380429.gif
Kumar, Raju Suresh; Almansour, Abdulrahman I.; Arumugam, Natarajan; Menéndez, J. Carlos; Osman, Hasnah; Kumar, Raju Ranjith: Dipolar Cycloaddition-Based Multicomponent Reactions in Ionic Liquids: A Green, Fully Stereoselective Synthesis of Novel Polycyclic Cage Systems with the Generation of Two New Azaheterocyclic Rings
https://www.thieme-connect.de/media/synthesis/201518/i_c0234_ga_10-1055_s-0034-1379931.gif
Zhao, Yating; Huang, Binbin; Yang, Chao; Li, Bing; Xia, Wujiong: Metal-Free [3+2] Oxidative Coupling of Phenols with Alkenes: Synthesis of Dihydrobenzofurans
https://www.thieme-connect.de/media/synthesis/201518/i_c0155_ga_10-1055_s-0034-1380419.gif
Cserép, Gergely B.; Demeter, Orsolya; Bätzner, Effi; Kállay, Mihály; Wagenknecht, Hans-Achim; Kele, Péter: Synthesis and Evaluation of Nicotinic Acid Derived Tetrazines for Bioorthogonal Labeling
https://www.thieme-connect.de/media/synthesis/201518/i_c0157_ga_10-1055_s-0034-1380721.gif
Islam, Kobirul; Das, Deb K.; Akram, Ejaz; Khan, Abu T.: Exploration of C5–C6-Unsubstituted 1,4-Dihydropyridines for the Construction of exo-Hexahydro-1H-chromeno[3,4-h][1,6]naphthyridine-3-carboxylates Using a Stereoselective Povarov Reaction
https://www.thieme-connect.de/media/synthesis/201518/i_c0223_ga_10-1055_s-0034-1380431.gif
Olson, Christopher A.; Shaner, Courtnay E.; Roche, Sydney C.; Ferrence, Gregory M.; Mitchell, T. Andrew: Hexahydro-1H-Isoindolinone-Like Scaffolds from Electronically Deactivated and Sterically Hindered Dienes: Synthesis in the Context­ of Muironolide A
https://www.thieme-connect.de/media/synthesis/201518/i_c0283_ga_10-1055_s-0034-1380221.gif
Högermeier, Jens; Trawny, Daniel; Zimmer, Reinhold; Reissig, Hans-Ulrich: Diels–Alder Reactions of 1,3-Dienes Incorporated into 8-Oxa- and 8-Thiabicyclo[3.2.1]octane Skeletons: A Convenient Access to Complex Tri- and Tetracyclic Compounds
https://www.thieme-connect.de/media/synthesis/201518/i_c0299_ga_10-1055_s-0034-1381037.gif
Lopchuk, Justin M.; Song, Mia; Butler, Blythe; Gribble, Gordon W.: Synthesis of Heteroaryl-Substituted Pyrroles via the 1,3-Dipolar Cycloaddition of Unsymmetrical Münchnones and Nitrovinylheterocycles
https://www.thieme-connect.de/media/synthesis/201518/i_c0162_ga_10-1055_s-0034-1380720.gif
Ribeiro Laia, Fernanda M.; Pinho e Melo, Teresa M. V. D.: Synthesis and Reactivity of Aziridines with Internal Dipolarophiles: An Approach to 1,4-Dihydrochromeno[4,3-b]pyrroles and 3-Methylenechromano[4,3-b]pyrroles
https://www.thieme-connect.de/media/synthesis/201518/i_c0235_ga_10-1055_s-0034-1378717.jpg
Miller, Daniel K.; Bailey, Christopher A.; Sammelson, Robert E.: Synthesis of Isoxazolines and Isoxazoles Inspired by Fipronil
https://www.thieme-connect.de/media/synthesis/201518/i_c0263_ga_10-1055_s-0034-1378737.gif
Pop, Lidia; Golban, Mirabela Ligia; Hădade, Niculina D.; Socaci, Crina; Grosu, Ion: CuAAC Synthesis of Tetragonal Building Blocks Decorated with Nucleobases
https://www.thieme-connect.de/media/synthesis/201518/i_c0288_ga_10-1055_s-0034-1378782.gif
Kratzer, Philipp; Gerster, Holger; Maas, Gerhard: Cycloaddition Reactions of Propyne Iminium Salts and Enol Ethers
https://www.thieme-connect.de/media/synthesis/201518/i_c0319_ga_10-1055_s-0034-1380223.gif
Yamaoka, Yousuke; Taniguchi, Marie; Yamada, Ken-ichi; Takasu, Kiyosei: Asymmetric Total Synthesis of Tylophorine through a Formal [2+2] Cycloaddition Followed by Migrative Ring Opening of a Cyclobutane
https://www.thieme-connect.de/media/synthesis/201518/i_c0267_ga_10-1055_s-0034-1380430.gif
Seck, Insa; Fall, Alioune; Lago, Carmen; Sène, Massène; Gaye, Mohamed; Seck, Matar; Gómez, Generosa; Fall, Yagamare: Synthesis of a Cholesterol Side-Chain Triazole Analogue via ‘Click’ Chemistry
https://www.thieme-connect.de/media/synthesis/201518/i_c0282_ga_10-1055_s-0034-1381053.gif

Issue 17/2015

Dobrydnev, Alexey V.; Popova, Maria V.; Saffon-Merceron, Nathalie; Listunov, Dymytrii; Volovenko, Yulian M.: Synthesis of the First Representatives of Spiro-1λ6-isothiazolidine-1,1,4-triones
https://www.thieme-connect.de/media/synthesis/201517/i_t0209_ga_10-1055_s-0034-1380434.gif
Zhang, Shuang; Hu, Xiu-Qin; Wang, Zhu-Yin; Xu, Peng-Fei: Reactions of Sulfonium Salts with 2,3-Dioxopyrrolidine Derivatives: A Concise Synthesis of Spirocyclopropane
https://www.thieme-connect.de/media/synthesis/201517/i_c0093_ga_10-1055_s-0034-1380522.gif
Peng, Jing; Ran, Guang-Yao; Du, Wei; Chen, Ying-Chun: Tertiary-Amine-Catalyzed Asymmetric [3+2] Annulations of Morita–Baylis–Hillman Carbonates of Isatins with Nitroolefins to Construct Spirooxindoles
https://www.thieme-connect.de/media/synthesis/201517/i_c0186_ga_10-1055_s-0034-1378716.gif
Xiao, Fenfen; Zhang, Qing; Wang, Yunxia; Hu, Xiangdong: Synthetic Studies toward Bi-linderone Lead To Unexpected 6π-Electrocyclization Reactions: A Facile Construction of Highly Congested Spiro Compounds
https://www.thieme-connect.de/media/synthesis/201517/i_f0346_ga_10-1055_s-0034-1381054.gif
Cormier, Morgan; Chardon, Aurélien; Blanchet, Jérôme; Rouden, Jacques; Maddaluno, Jacques; De Paolis, Michaël: An Organocatalytic Access to Spiro[4.5]decanes and Spiro[4.6]undecanes Containing Aminolactones and 3-Aminopyrrolidines
https://www.thieme-connect.de/media/synthesis/201517/i_c0767_ga_10-1055_s-0034-1380146.gif

Issue 16/2015

Philipps, Arne R.; Fritze, Lars; Erdmann, Nico; Enders, Dieter: An Asymmetric Organocatalytic Quadruple Domino Reaction Employing a Vinylogous Friedel–Crafts/Michael/Michael/Aldol Condensation Sequence
https://www.thieme-connect.de/media/synthesis/201516/i_c0127_ga_10-1055_s-0034-1380197.jpg
Garbarino, Silvia; Protti, Stefano; Basso, Andrea: Toward a Green Atom Economy: Development of a Sustainable Multicomponent Reaction
https://www.thieme-connect.de/media/synthesis/201516/i_c0183_ga_10-1055_s-0034-1380719.jpg
Firth, James D.; Zhang, Rong; Morgentin, Rémy; Guilleux, Rachel; Kalliokoski, Tuomo; Warriner, Stuart; Foster, Richard; Marsden, Stephen P.; Nelson, Adam: Exploitation of the Ugi–Joullié Reaction in the Synthesis of Libraries of Drug-Like Bicyclic Hydantoins
https://www.thieme-connect.de/media/synthesis/201516/i_c0208_ga_10-1055_s-0034-1378704.gif
Neochoritis, Constantinos G.; Zhang, Ji; Dömling, Alexander: Leuckart–Wallach Approach to Sugar Isocyanides and Its IMCRs
https://www.thieme-connect.de/media/synthesis/201516/i_c0249_ga_10-1055_s-0034-1381046.jpg
Xu, Shibo; Su, Shikuan; Zhang, Huiting; Tian, Lumin; Liang, Pengcheng; Chen, Jiawen; Zhang, Yuan; Li, Chunju; Jia, Xueshun; Li, Jian: Isocyanide-Based Multicomponent Reactions: Rapid Synthesis of a 5,5-Fused Bicyclic Skeleton from α,β-Unsaturated Ketones and Allenoates
https://www.thieme-connect.de/media/synthesis/201516/i_c0250_ga_10-1055_s-0034-1378736.gif
Neo, Ana G.; Castellano, Teresa G.; Marcos, Carlos F.: Enol-Ugi Reaction of Hydroxycoumarins: Straightforward Synthesis of Amino Acid Derived Coumarin Enamines
https://www.thieme-connect.de/media/synthesis/201516/i_c0258_ga_10-1055_s-0034-1380436.gif
Carboni, Aude; Dagousset, Guillaume; Magnier, Emmanuel; Masson, Géraldine: Three-Component Photoredox-Mediated Chloro-, Bromo-, or Iodotrifluoromethylation of Alkenes
https://www.thieme-connect.de/media/synthesis/201516/i_c0200_ga_10-1055_s-0034-1378715.gif
Qureshi, Zafar; Schlundt, Waldemar; Lautens, Mark: Introduction of Hindered Electrophiles via C–H Functionalization in a Palladium-Catalyzed Multicomponent Domino Reaction
https://www.thieme-connect.de/media/synthesis/201516/i_z0123_ga_10-1055_s-0034-1380198.gif

Issue 15/2015

Du, Haiying; Rodriguez, Jean; Bugaut, Xavier; Constantieux, Thierry: Michael Addition Initiated Substrate- or Catalyst-Controlled Chemodivergent Three-Component Construction of Fused and Bridged Polycyclic Heterocycles
https://www.thieme-connect.de/media/synthesis/201515/i_z0663_ga_10-1055_s-0034-1380229.gif
Vízcaíno-Milla, Pascuala; Sansano, José M.; Nájera, Carmen; Fiser, Béla; Gómez-Bengoa, Enrique: Primary Amine–2-Aminopyrimidine Chiral Organocatalysts for the Enantioselective Conjugate Addition of Branched Aldehydes to Maleimides
https://www.thieme-connect.de/media/synthesis/201515/i_c0196_ga_10-1055_s-0034-1380718.gif
Fu, Niankai; Guo, Yinliang; Zhang, Long; Luo, Sanzhong: Chiral Primary Amine Catalyzed Asymmetric Tandem Reduction–Michael Addition–Protonation Reaction between Alkylidene Meldrum’s Acid and α-Substituted Vinyl Ketones
https://www.thieme-connect.de/media/synthesis/201515/i_c0142_ga_10-1055_s-0034-1380717.gif
Rideau, Emeline; Mäsing, Florian; Fletcher, Stephen P.: Asymmetric Conjugate Addition of Alkylzirconocenes to Cyclopent-4-ene-1,3-dione Monoacetals
https://www.thieme-connect.de/media/synthesis/201515/i_c0203_ga_10-1055_s-0034-1379928.gif
Tai, Hung-Che; Chavan, Arjun S.; Chuang, Shih-Ching: Nucleophilic Conjugate 1,5-Addition of Gilman Reagents to (E)-Hex-2-en-4-ynedioates: An Access to β(γ′)-Substituted Muconates
https://www.thieme-connect.de/media/synthesis/201515/i_c0211_ga_10-1055_s-0034-1378856.gif
Roscales, Silvia; Sancho, Ainhoa; Csákÿ, Aurelio G.: Metal-Free Conjugate Addition of Alkenylboronic Acids to Enedicarbonyl Compounds towards the Synthesis of Pyridazine Derivatives
https://www.thieme-connect.de/media/synthesis/201515/i_c0139_ga_10-1055_s-0034-1380525.gif
Peck, Cheryl L.; Calderone, Joseph A.; Santos, Webster L.: Copper(II)-Catalyzed β-Borylation of Acetylenic Esters in Water
https://www.thieme-connect.de/media/synthesis/201515/i_c0153_ga_10-1055_s-0034-1380524.gif
Witte, Swjatoslaw N. R.; Voigt, Benjamin; Mahrwald, Rainer: Amine-Catalyzed Cascade Reactions of Unprotected and Unactivated­ Carbohydrates: Direct Access to C-Glycosides
https://www.thieme-connect.de/media/synthesis/201515/i_c0159_ga_10-1055_s-0034-1380416.gif
Nishimura, Katsumi; Fukuyama, Naoshi; Yamashita, Mitsuaki; Sumiyoshi, Takaaki; Yamamoto, Yasutomo; Yamada, Ken-ichi; Tomioka, Kiyoshi: Cyclic Model for the Asymmetric Conjugate Addition of Organolithiums with Enoates
https://www.thieme-connect.de/media/synthesis/201515/i_c0169_ga_10-1055_s-0034-1380702.gif
Sugiura, Masaharu; Ishikawa, Wakoto; Kuboyama, Yukinobu; Nakajima, Makoto: Conjugate Addition of Diboron Catalyzed by O-Monoacyltartaric Acids
https://www.thieme-connect.de/media/synthesis/201515/i_c0172_ga_10-1055_s-0034-1378835.gif

Issue 17/2014

Mori, Yasuyuki; Mori, Takamichi; Onodera, Gen; Kimura, Masanari: Nickel-Catalyzed Multicomponent Coupling of Alkyne, Buta-1,3-diene, and Dimethylzinc under Carbon Dioxide
https://www.thieme-connect.de/media/synthesis/201417/i_c0134_ga_10-1055_s-0033-1339024.gif
Strack, Martin; Metzler-Nolte, Nils; Albada, H. Bauke: Copper-Free Cleavage-Sonogashira Conjugation of Silylacetylene Immobilized Peptides
https://www.thieme-connect.de/media/synthesis/201417/i_c0144_ga_10-1055_s-0034-1378207.gif
Ma, Wenbo; Ackermann, Lutz: Silver-Mediated Alkyne Annulations by C–H/P–H Functionalizations: Step-Economical Access to Benzophospholes
https://www.thieme-connect.de/media/synthesis/201417/i_c0151_ga_10-1055_s-0033-1338630.gif
Park, Youngchul; Kang, Dongjin; Jeon, Woo Hyung; Ryu, Taekyu; Lee, Phil Ho: Synthesis of Ethyl Arylpropiolates through Palladium-Catalyzed Cross-Coupling­ Reactions of Aryl Iodides with In Situ Generated Lithium Tetrakis(ethoxycarbonylethynyl)indates
https://www.thieme-connect.de/media/synthesis/201417/i_c0123_ga_10-1055_s-0033-1339110.gif

Issue 16/2014

Guo, Wei; Xia, Yuanzhi: THF Solvent as a Proton Shuttle in the AuCl3-Catalyzed Cycloisomerization of a Bromoallenyl Ketone: A Mechanistic DFT Study
https://www.thieme-connect.de/media/synthesis/201416/i_c0272_ga_10-1055_s-0034-1378281.gif
Lee, Ji Hyung; Jeong, Wook; Rhee, Young Ho: Unique Divergent Reactivity of Boc-Protected Homopropargylic Alkoxyalkylamines in the Gold(I)-Catalyzed Domino Catalytic Reactions: Application to the Formal Synthesis of (–)-Pseudodistomin B
https://www.thieme-connect.de/media/synthesis/201416/i_c0191_ga_10-1055_s-0033-1338639.gif
Liu, Meng-Qi; Zhou, Ai-Hua; Jiang, Shuang; Wang, Jia-Qi; Ye, Long-Wu: Highly Diastereoselective Synthesis of Cyclopentenones via a One-Pot Gold Catalysis, Nazarov Cyclization and Alkylation Cascade
https://www.thieme-connect.de/media/synthesis/201416/i_c0114_ga_10-1055_s-0033-1341204.gif
Wei, Fang; Wang, Xianghua; Peng, Shasha; Jia, Qiuhui; Jiang, Chao; Liu, Shili; Xu, Zhenghu: Direct Gold-Catalyzed Regioselective Tetrafunctionalization of Nonactivated Alkynes
https://www.thieme-connect.de/media/synthesis/201416/i_c0133_ga_10-1055_s-0033-1341271.gif

Issue 14/2014

Zhou, Mingxin; Song, Qiuling: Synthesis of α-Ketoamides from Aryl Methyl Ketones and N,N-Dimethylformamide via Copper-Catalyzed Aerobic Oxidative Coupling
https://www.thieme-connect.de/media/synthesis/201414/i_c0127_ga_10-1055_s-0033-1339109.gif
Belhomme, Marie-Charlotte; Dru, Delphine; Xiong, Heng-Ying; Cahard, Dominique; Besset, Tatiana; Poisson, Thomas; Pannecoucke, Xavier: Copper-Mediated Direct Functionalization of Unsaturated C–C Bonds with Ethyl Bromo(difluoro)acetate: A Straightforward Access to Highly Valuable Difluoromethylated Alkenes
https://www.thieme-connect.de/media/synthesis/201414/i_c0137_ga_10-1055_s-0033-1338637.gif
Székely, Anna; Sinai, Ádám; Tóth, Edina B.; Novák, Zoltán: Utilization of a Copper on Iron Catalyst for the Synthesis of Biaryl Systems and Benzoxazines via Oxidative Arylation of Anilide Derivatives
https://www.thieme-connect.de/media/synthesis/201414/i_c0145_ga_10-1055_s-0033-1338642.gif
Duong, Hung A.; Nguyen, Tuan Minh; Rosman, Nurul Zubaidah Binte; Tan, Lionel Jia Liang: Carboxylation of Organoboronic Esters with Potassium Methyl Carbonate under Copper Catalysis
https://www.thieme-connect.de/media/synthesis/201414/i_c0122_ga_10-1055_s-0033-1339119.gif
Sahoo, Santosh K.; Jena, Himanshu Sekhar; Majji, Ganesh; Patel, Bhisma K.: Formation of Imidazolidine-benzothiazole–Copper(II) Complexes via a Copper-Mediated Room-Temperature C–H Activation of Imidazolidinecarbothioamides
https://www.thieme-connect.de/media/synthesis/201414/i_c0238_ga_10-1055_s-0033-1339127.gif
Zhao, Chenglong; Tan, Zhuozhen; Liang, Zhuye; Deng, Wei; Gong, Hegui: Nickel-Catalyzed Reductive Allylation of Ketones with Allylic Carbonates
https://www.thieme-connect.de/media/synthesis/201414/i_c0174_ga_10-1055_s-0033-1339111.gif
Luo, Long; Zhang, Jian-Jian; Ling, Wei-Jian; Shao, Yong-Liang; Wang, Ya-Wen; Peng, Yu: Unified Synthesis of (–)-Folicanthine and (–)-Ditryptophenaline Enabled by a Room Temperature Nickel-Mediated Reductive Dimerization
https://www.thieme-connect.de/media/synthesis/201414/i_c0189_ga_10-1055_s-0033-1339126.gif
Liu, Jiangguang; Yan, Jiajie; Qin, Dongguang; Cai, Qian: An Unexpected Inversion of Enantioselectivity in a Copper-Catalyzed Intramolecular­ Desymmetric Aryl C–N Coupling Reaction
https://www.thieme-connect.de/media/synthesis/201414/i_c0121_ga_10-1055_s-0033-1338638.gif
Kageyuki, Ikuo; Yoshida, Hiroto; Takaki, Ken: Three-Component Carboboration of Alkenes under Copper Catalysis
https://www.thieme-connect.de/media/synthesis/201414/i_c0143_ga_10-1055_s-0033-1341267.gif
Gurung, Santosh K.; Thapa, Surendra; Shrestha, Bijay; Giri, Ramesh: Copper-Catalyzed Cross-Coupling of Aryl- and Heteroaryltriethoxysilanes with Aryl and Heteroaryl Iodides and Bromides
https://www.thieme-connect.de/media/synthesis/201414/i_c0146_ga_10-1055_s-0033-1339108.gif
Ambler, Brett R.; Peddi, Santosh; Altman, Ryan A.: Copper-Catalyzed Decarboxylative Trifluoromethylation of Propargyl Bromodifluoroacetates
https://www.thieme-connect.de/media/synthesis/201414/i_c0147_ga_10-1055_s-0033-1339128.gif

Issue 10/2014

Tang, Weijun; Xiao, Jianliang: Asymmetric Hydrogenation of Imines via Metal–Organo Cooperative Catalysis
https://www.thieme-connect.de/media/synthesis/201410/i_c0049_ga_10-1055_s-0033-1338603.gif
Deiana, Luca; Ghisu, Lorenza; Córdova, Oscar; Afewerki, Samson; Zhang, Renyun; Córdova, Armando: Efficient and Highly Enantioselective Aerobic Oxidation–Michael–Carbocyclization Cascade Transformations by Integrated Pd(0)-CPG Nanoparticle/Chiral Amine Relay Catalysis
https://www.thieme-connect.de/media/synthesis/201410/i_c0014_ga_10-1055_s-0033-1340883.gif
Diezel, Sonja; Breit, Bernhard: Tandem Regioselective Rhodium-Catalyzed Hydroformylation–Enantioselective Aminocatalytic anti-Mannich Reaction
https://www.thieme-connect.de/media/synthesis/201410/i_c0025_ga_10-1055_s-0033-1338602.gif
Gualandi, Andrea; Mengozzi, Luca; Wilson, Claire Margaret; Cozzi, Pier Giorgio: Synergistic Stereoselective Organocatalysis with Indium(III) Salts
https://www.thieme-connect.de/media/synthesis/201410/i_c0033_ga_10-1055_s-0033-1341022.gif
Lee, Hwa-Jung; Shyam, Pranab Kumar; Yoon, Woojin; Yun, Hoseop; Jang, Hye-Young: Diastereo- and Enantioselective Synthesis of Hexasubstituted Cyclohexanes via a Metal–Organocatalytic Quadruple Cascade Sequence
https://www.thieme-connect.de/media/synthesis/201410/i_c0009_ga_10-1055_s-0033-1341103.gif
Praveen, Chandrasekaran; Levêque, Sabine; Vitale, Maxime R.; Michelet, Véronique; Ratovelomanana-Vidal, Virginie: Synergistic Iron-and-Amine Catalysis in Carbocyclizations
https://www.thieme-connect.de/media/synthesis/201410/i_c0018_ga_10-1055_s-0033-1338612.gif
Liu, Lu; Daka, Philias; Sarkisian, Ryan; Deng, Yongming; Wheeler, Kraig; Wang, Hong: Oxa-Diels–Alder Reaction of Isatins and Acyclic α,β-Unsaturated Methyl Ketones through Cooperative Dienamine and Metal Lewis Acid Catalysis
https://www.thieme-connect.de/media/synthesis/201410/i_c0028_ga_10-1055_s-0033-1338613.gif
Jing, Changcheng; Xing, Dong; Qian, Yu; Hu, Wenhao: Rh2(OAc)4 and Chiral Phosphoric Acid Cocatalyzed Highly Diastereo- and Enantioselective Four-Component Reactions: Facile Synthesis of Chiral α,β-Diamino Acid Derivatives
https://www.thieme-connect.de/media/synthesis/201410/i_c0085_ga_10-1055_s-0033-1341051.gif
Li, Nan; Chen, Dian-Feng; Wang, Pu-Sheng; Han, Zhi-Yong; Gong, Liu-Zhu: Relay Catalytic Cascade Hydrosiloxylation and Asymmetric Hetero-Diels–Alder Reaction
https://www.thieme-connect.de/media/synthesis/201410/i_c0068_ga_10-1055_s-0033-1340905.gif
Yang, Jinming; Yu, Xingxin; Wu, Jie: A Facile Route to H-Pyrazolo[5,1-a]isoquinolines through a Multicomponent Reaction of 2-Alkynylbenzaldehyde, Sulfonylhydrazine, and Benzyne
https://www.thieme-connect.de/media/synthesis/201410/i_c0162_ga_10-1055_s-0033-1341102.gif
Yoshida, Masanori; Masaki, Erika; Terumine, Tatsuaki; Hara, Shoji: Asymmetric α-Allylation of α-Branched Aldehydes with Allyl Alcohols by Synergistic Catalysis Using an Achiral Palladium Complex and a Chiral Primary Amino Acid
https://www.thieme-connect.de/media/synthesis/201410/i_c0838_ga_10-1055_s-0033-1340901.gif

Issue 19/2013

Reboredo, Silvia; Vicario, Jose L.; Carrillo, Luisa; Reyes, Efraím; Uria, Uxue: A Simple Synthesis of Polysubstituted Pyrrolidines by an Organocatalytic Three-Component Approach Featuring a One-Pot Condensation and [3+2]-Cycloaddition Reaction in Aqueous Medium
https://www.thieme-connect.de/media/synthesis/201319/i_c0127_ga_10-1055_s-0033-1338922.gif
Reitel, Kärt; Lippur, Kristin; Järving, Ivar; Kudrjašova, Marina; Lopp, Margus; Kanger, Tõnis: Asymmetric Aminocatalytic Michael Addition of Cyclopropane-Containing Aldehydes to Nitroalkenes
https://www.thieme-connect.de/media/synthesis/201319/i_c0131_ga_10-1055_s-0033-1338704.gif
Shimada, Yoshiko; Hattori, Kasumi; Tada, Norihiro; Miura, Tsuyoshi; Itoh, Akichika: Facile Aerobic Photooxidation of Alcohols Using 2-Chloroanthraquinone under Visible Light Irradiation
https://www.thieme-connect.de/media/synthesis/201319/i_c0164_ga_10-1055_s-0033-1338420.gif
Paria, Suva; Pirtsch, Michael; Kais, Viktor; Reiser, Oliver: Visible-Light-Induced Intermolecular Atom-Transfer Radical Addition of Benzyl Halides to Olefins: Facile Synthesis of Tetrahydroquinolines
https://www.thieme-connect.de/media/synthesis/201319/i_c0169_ga_10-1055_s-0033-1338910.gif
Cismesia, Megan A.; Ischay, Michael A.; Yoon, Tehshik P.: Reductive Cyclizations of Nitroarenes to Hydroxamic Acids by Visible Light Photoredox Catalysis
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Issue 15/2013

Mochizuki, Katsufumi; Sakai, Kazunori; Kochi, Takuya; Kakiuchi, Fumitoshi: Rhodium-Catalyzed Dimerization of Arylacetylenes and Addition of Malonates­ to 1,3-Enynes
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Yamada, Yoichi M. A.; Ohta, Hidetoshi; Yuyama, Yoshinari; Uozumi, Yasuhiro: Polymeric Bimetallic Catalyst-Promoted In-Water Dehydrative Alkylation of Ammonia and Amines with Alcohols
https://www.thieme-connect.de/media/synthesis/201315/i_c0144_ga_10-1055_s-0033-1338797.gif
Arnold, Jeffrey S.; Nguyen, Hien M.: Rhodium-Catalyzed Asymmetric Amination of Allylic Trichloroacetimidates
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Ye, Ke-Yin; Zhao, Zhuo-An; Lai, Zeng-Wei; Dai, Li-Xin; You, Shu-Li: Highly Regioselective Allylic Substitution Reactions Catalyzed by an Air-Stable (π-Allyl)iridium Complex Derived from Dinaphthocyclooctatetraene and a Phosphoramidite Ligand
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Obora, Yasushi; Sawaguchi, Takuya; Tsubakimoto, Keiko; Yoshida, Hiroshi; Ogawa, Shinji; Hatanaka, Shintaro: Iridium-Catalyzed Synthesis of ω-Hydroxy Homoallylic Alcohols
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Apsunde, Tushar Dattu; Trudell, Mark L.: Microwave-Assisted Iridium-Catalyzed Synthesis of Nicotine and Anabasine Derivatives
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Wang, Hui; Xu, Ming-Hua: Rhodium-Catalyzed Highly Enantioselective Addition of Arylboronic Acids to Cyclic Aldimines: Practical Asymmetric Synthesis of Cyclic Sulfamidates
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Suzuki, Takeyuki; Ishizaka, Yuka; Ghozati, Kazem; Zhou, Da-Yang; Asano, Kaori; Sasai, Hiroaki: Enantioselective Multicatalytic Synthesis of α-Benzyl-β-hydroxyindan-1-ones
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Liu, Wenting; Hong, Xiaohu; Xu, Bin: Rhodium-Catalyzed Oxidative Coupling of Aryl Hydrazones with Internal Alkynes: Efficient Synthesis of Multisubstituted Isoquinolines
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Issue 12/2013

Fukata, Yukihiro; Miyaji, Ryota; Okamura, Takaaki; Asano, Keisuke; Matsubara, Seijiro: Asymmetric Cycloetherifications by Bifunctional Aminothiourea Catalysts: The Importance of Hydrogen Bonding
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Jakab, Gergely; Hosseini, Abolfazl; Hausmann, Heike; Schreiner, Peter R.: Mild and Selective Organocatalytic Iodination of Activated Aromatic Compounds
https://www.thieme-connect.de/media/synthesis/201312/i_c0157_ga_10-1055_s-0033-1338468.gif
Kumar, Vikas; Ray, Bidisha; Rathi, Preeti; Mukherjee, Santanu: Catalytic Asymmetric Direct Vinylogous Michael Addition of γ-Aryl-Substituted Deconjugated Butenolides to Nitroolefins and N-Phenylmaleimide
https://www.thieme-connect.de/media/synthesis/201312/i_c0191_ga_10-1055_s-0033-1338705.gif
Duan, Shu-Wen; Liu, Yi-Yin; Ding, Wei; Li, Tian-Ren; Shi, De-Qing; Chen, Jia-Rong; Xiao, Wen-Jing: Chiral Squaramide Catalyzed Asymmetric Conjugate Additions of 3-Substituted Oxindoles to Vinylphosphonates
https://www.thieme-connect.de/media/synthesis/201312/i_c0080_ga_10-1055_s-0032-1316919.gif
Chen, Guo-Ying; Lu, Yixin: Highly Enantioselective Michael Addition of α-Substituted Nitrophosphonates to a Vinyl Sulfone
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Raimondi, Wilfried; Sanchez Duque, Maria del Mar; Goudedranche, Sébastien; Quintard, Adrien; Constantieux, Thierry; Bugaut, Xavier; Bonne, Damien; Rodriguez, Jean: Activation of 1,2- and 1,3-Ketoamides with Thiourea Organocatalyst for the Enantioselective Domino Synthesis of Functionalized Cyclohexanes
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Issue 18/2012

Hassink, Matthew D.; Fox, Joseph M.: Functionalized Cyclopropenes and Methylenecyclopropenes from Dianions of 3-Hydroxymethylcyclopropenes
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Rotstein, Benjamin H.; Yudin, Andrei K.: Aziridine-2-carboxaldehyde Dimers Undergo Homo-Ugi 4-Component-5-center Reactions
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Walker, Daniel P.; Eklov, Brian M.; Bedore, Matthew W.: Practical Synthesis of 3-Oxa-6-azabicyclo[3.1.1]heptane Hydrotosylate; A Novel Morpholine-Based Building Block
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Di Bussolo, Valeria; Frau, Ileana; Pineschi, Mauro; Crotti, Paolo: d-Allal- and d-Galactal-Derived Vinyl N-Mesylaziridines: Regio- and Stereoselectivity in Addition Reactions of O-, C-, N-, and S-Nucleophiles
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Florio, Saverio: Unraveling the Synthetic Utility of the Regio- and Stereoselective Lithiation of Aziridines
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Issue 16/2012

Lei, Ming; Tian, Wan; Hu, Ruijun; Li, Wei; Zhang, Hong: An Efficient Synthesis of 2-(Trifluoromethyl)-2H-[1,3]oxazino[2,3-a]isoquinolines via a Three-Component Cascade Approach Using a Continuous-Flow Microreactor
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Rodriguez, Antonio M.; Juan, Alberto; Gómez, M. Victoria; Moreno, Andres; de la Hoz, Antonio: Continuous-Flow Microliter Microwave Irradiation in the Synthesis of Isoxazole Derivatives: An Optimization Procedure
https://www.thieme-connect.de/media/synthesis/201216/c0216_ga.jpg
Slocum, D. W.; Reinscheld, Thomas K.; Austin, Nick D.; Kusmic, Damir; Whitley, Paul E.: Near-Ambient Temperature Halogen–Lithium Exchange of p-Bromoanisole and Related Substrates: Flow/Batch Studies
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Pagano, Nicholas; Heil, Marintha L.; Cosford, Nicholas D. P.: Automated Multistep Continuous Flow Synthesis of 2-(1H-Indol-3-yl)thiazole Derivatives
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Ullah, Farman; Zang, Qin; Javed, Salim; Porubsky, Patrick; Neuenswander, Benjamin; Lushington, Gerald H.; Hanson, Paul R.; Organ, Michael G.: Synthesis of an Isoindoline-Annulated, Tricyclic Sultam Library via Microwave-Assisted, Continuous-Flow Organic Synthesis (MACOS)
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Fukuyama, Takahide; Kajihara, Yoshito; Ryu, Ilhyong; Studer, Armido: Nitroxide-Mediated Polymerization of Styrene, Butyl Acrylate, or Methyl Methacrylate by Microflow Reactor Technology
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Issue 14/2012

Wu, Xingxing; Zhang, Junliang: Y(OTf)3-Catalyzed Diastereoselective [3+2] Cycloaddition of N-Tosyl­aziridines and Imines; Efficient Synthesis of Multisubstituted Imidazolidines
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Yamazaki, Shoko; Fukushima, Yugo; Ukai, Tetsuma; Tatsumi, Kohei; Ogawa, Akiya: Lewis Acid Promoted Reactions of 1,1-Diarylallenes and Ketone Derivatives: Synthesis of Indenes by an Addition/Cyclization Reaction
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Beckendorf, Stephan; Mancheño, Olga García: 'Click'-BINOLs: A New Class of Tunable Ligands for Asymmetric Catalysis
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Auvil, Tyler J.; Mattson, Anita E.: Internal Lewis Acid Assisted Benzoic Acid Catalysis
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Lanari, Daniela; Piermatti, Oriana; Pizzo, Ferdinando; Vaccaro, Luigi: Copper(II) Triflate–Sodium Dodecyl Sulfate Catalyzed Preparation of 1,2-Diphenyl-2,3-dihydro-4-pyridones in Aqueous Acidic Medium
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Komai, Hirotomo; Yoshino, Tatsuhiko; Matsunaga, Shigeki; Kanai, Motomu: Lewis Acid Catalyzed Benzylic C–H Bond Functionalization of Azaarenes; Addition to Imines and Enones
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Schweighauser, Luca; Bodoky, Ina; Kessler, Simon N.; Häussinger, Daniel; Wegner, Hermann A.: Bidentate Lewis Acid Catalyzed Inverse-Electron-Demand Diels–Alder Reaction for the Selective Functionalization of Aldehydes
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Issue 12/2012

Shao, Jun; Huang, Xiaomei; Hong, Xiaohu;