Synthesis

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Issue eFirst

See, Nicholas W.; Pierens, Gregory K.; Krenske, Elizabeth H.; Ferro, Vito: C-5 Epimerisation of d-Mannopyranosyl Fluorides: The Influence of Anomeric Configuration on Radical Reactivity
https://www.thieme-connect.de/media/synthesis/EFirst/i_b0292_ga_10-1055_a-2149-4586.gif
Khatana, Anil Kumar; Singh, Vikram; Gupta, Manoj Kumar; Tiwari, Bhoopendra: A Highly Efficient NHC-Catalyzed Aerobic Oxidation of Aldehydes to Carboxylic Acids
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0219_ga_10-1055_s-0037-1610069.gif
Sperger, Theresa; Schoenebeck, Franziska: α-Arylation of Esters and Ketones Enabled by a Bench-Stable Pd(I) Dimer Catalyst
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0285_ga_10-1055_s-0037-1610087.gif
Lindner, Marcin; Krasiński, Antoni; Jurczak, Janusz: Facile, Stereocontrolled Synthetic Route towards Bis-functionalised Pyrrolizidines
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0359_ga_10-1055_s-0037-1609582.gif
Oberg, Kevin M.; Cochran, Brian M.; Cook, Matthew J.; Rovis, Tomislav: The Catalytic Alkylative Desymmetrization of Anhydrides in a Formal Synthesis of Ionomycin
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0160_ga_10-1055_s-0037-1610108.gif
Pang, Jia Hao; Ong, Derek Yiren; Watanabe, Kohei; Takita, Ryo; Chiba, Shunsuke: Leaving Group Ability in Nucleophilic Aromatic Amination by Sodium Hydride–Lithium Iodide Composite
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0368_ga_10-1055_s-0039-1690010.gif
Zhang, Yongda; Lao, Kendricks S.; Sieber, Joshua D.; Xu, Yibo; Wu, Linglin; Wang, Xiao-Jun; Desrosiers, Jean-Nicolas; Lee, Heewon; Haddad, Nizar; Han, Zhengxu S.; Yee, Nathan K.; Song, Jinhua J.; Howell, Amy R.; Senanayake, Chris H.: Modular Dihydrobenzoazaphosphole Ligands for Suzuki–Miyaura Cross-Coupling
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0181_ga_10-1055_s-0037-1610158.gif
Liddon, John T. R.; Rossi-Ashton, James A.; Clarke, Aimee K.; Lynam, Jason M.; Taylor, Richard J. K.; Unsworth, William P.: Divergent Reactivity of Indole-Tethered Ynones with Silver(I) and Gold(I) Catalysts: A Combined Synthetic and Computational Study
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0211_ga_10-1055_s-0037-1610181.gif
Joshi, Madhur S.; Pigge, F. Christopher: Sequential Pyridine Dearomatization–Mizoroki–Heck Cyclization for the Construction of Fused (Dihydropyrido)isoindolinone Ring Systems
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0093_ga_10-1055_s-0037-1610133.gif
Wertjes, William; Ayers, Sloan; Gao, Qi; Simmons, Eric M.; Beutner, Gregory L.: A Divergent Nickel-Catalyzed Synthesis of Quinazolinediones and Benzoxazinone Imines
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0192_ga_10-1055_s-0037-1610140.gif
Kaieda, Yuya; Yamamoto, Kosuke; Toguchi, Hiroyuki; Hanazawa, Natsumi; Kuriyama, Masami; Onomura, Osamu: Oxidative C–N Bond Cleavage of Cyclic Amines with Ammonium Hypochlorite
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0043_ga_10-1055_a-2062-8680.gif
Denizot, Natacha; Guillot, Régis; Kouklovsky, Cyrille; Vincent, Guillaume: N-Iodosuccinimide-Mediated Oxidative Coupling of Indoles and Phenols: A Synthetic Study toward the Benzofuroindoline Moiety of Bipleiophylline
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0092_ga_10-1055_s-0036-1592002.gif
Ziegler, Dorothée S.; Klier, Lydia; Müller, Nicolas; Karaghiosoff, Konstantin; Knochel, Paul: Directed Zincation or Magnesiation of 2- and 4-Pyrones and Their Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0411_ga_10-1055_s-0037-1610215.gif
Garlets, Zachary J.; Wolfe, John P.: Asymmetric Synthesis of Six-Membered Cyclic Sulfamides via Palladium-Catalyzed Alkene Carboamination Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0078_ga_10-1055_s-0036-1591574.gif
Nocera, Giuseppe; Murphy, John A.: Ground State Cross-Coupling of Haloarenes with Arenes Initiated by Organic Electron Donors, Formed in situ: An Overview
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0401_ga_10-1055_s-0039-1690614.gif
Cole, Charles J. F.; Chi, Hyung Min; DeBacker, Kenneth C.; Snyder, Scott A.: Synthesis of Enhanced, Isolable Disulfanium Salts and their Application to Thiiranium-Promoted Polyene Cyclizations
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0184_ga_10-1055_s-0037-1609754.gif
Wang, Zheng; Ji, Hongtao; He, Wei-Min; Xiong, Yang; Zhang, Guozhu: Chromium-Catalyzed Asymmetric Dearomatization–Addition Reactions of Halomethyloxazoles and Indoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0070_ga_10-1055_s-0037-1609753.gif
Seki, Katsunori; Makikawa, Takumi; Toshima, Kazunobu; Takahashi, Daisuke: Synthesis and Immunological Evaluation of Escherichia coli O1- Derived Oligosaccharide–Protein Conjugates toward Avian Pathogenic Escherichia coli O1 Vaccine Development
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0324_ga_10-1055_a-2152-0255.gif

Issue 04/2024

Qin, Yang; Liu, Sheng; Shi, Shi-Liang: Transition-Metal-Free Cross-Coupling of Acetals and Grignard Reagents To Form Diarylmethyl Alkyl Ethers and Triarylmethanes
https://www.thieme-connect.de/media/synthesis/202404/i_b0141_ga_10-1055_a-2088-5000.gif
Khan, Farooq-Ahmad; Yaqoob, Sana; Qasim, Muhammad Wasim; Ali, Shujaat; Wang, Yan; Jiang, Zi-Hua: A Robust, Gram-Scale and High-Yield Synthesis of MDP Congeners for Activation of the NOD2 Receptor and Vaccine Adjuvantation
https://www.thieme-connect.de/media/synthesis/202404/i_b0528_ga_10-1055_a-2004-5883.gif
Chaskar, Sudhir P.; Honparkhe, Ramchandra; Aghao, Arvind K.; Thorat, Rakesh G.; Pramanik, Chinmoy: An Alternative Formal Synthesis of (S)-(+)-Vigabatrin
https://www.thieme-connect.de/media/synthesis/202404/i_c0128_ga_10-1055_s-0042-1751470.gif
Chen, Yang; Li, Qiao-Yue; Xie, Xiao-Yan; Wang, Wei; Li, Dashan; Wang, Wen-Jing; Shao, Li-Dong: Construction of an Epoxy-lactone Moiety on the C/D Ring of Highly Oxygenated Triterpenes through a Modified SeO2-Promoted Oxidative Cyclization
https://www.thieme-connect.de/media/synthesis/202404/i_c0152_ga_10-1055_a-2122-4021.gif
Varga, Petra Regina; Belovics, Alexandra; Karaghiosoff, Konstantin; Szabó, Rita; Bősze, Szilvia; Drahos, László; Keglevich, György: Efficient Synthesis of Diethyl, Dialkyl α-Hydroxy-propylenebisphosphonates and Related 5-Phosphonoyl-1,2-oxaphospholane 2-Oxides
https://www.thieme-connect.de/media/synthesis/202404/i_c0184_ga_10-1055_a-2122-4178.gif
Cui, Hai-Bo; Ma, Ting; Zhang, Ru-Yue; Shan, Jing; Wang, Zhong-Qiang; Bai, Mei; Chen, Yong-Zheng: Biocatalytic Synthesis of Chiral Benzylic Alcohols via Enantioselective Hydroxylation by a Self-Sufficient Cytochrome P450 from Deinococcus gobiensis
https://www.thieme-connect.de/media/synthesis/202404/i_g0096_ga_10-1055_a-2076-9792.gif
Kumar, Kankanala Naveen; Mhate, Mouzma; Ravichandiran, Velayutham; Swain, Sharada Prasanna: Bis(pinacoloto)diboron/4-Phenylpyridine System for One-Pot Photocatalyzed Borylation and Reduction of Aldehyde: Synthesis of Tavaborole in a Flow Reactor
https://www.thieme-connect.de/media/synthesis/202404/i_g0318_ga_10-1055_a-2169-6200.gif
Tintori, Guillaume; Jacob, Clément; Delsarte, Christine; Potié, François; Grimaud, Laurence; Vitale, Maxime; Echeverria, Pierre-Georges: Efficient and Scalable Synthesis of 6,6-Dimethyl-3-oxabicyclo [3.1.0]hexan-2-one through Organocatalyzed Desymmetrization and Chemoselective Reduction
https://www.thieme-connect.de/media/synthesis/202404/i_j0435_ga_10-1055_a-2217-0996.gif
Bera, Shyamal Kanti; Bhanja, Rosalin; Sahu, Chandan Chittapriya; Mal, Prasenjit: An Intramolecular Radical C–N Coupling by N-Iodosuccinimide
https://www.thieme-connect.de/media/synthesis/202404/i_m0068_ga_10-1055_a-2063-0221.gif
Nakahara, Yuichi; Endo, Yuta; Takahashi, Kazutoshi; Kawaguchi, Tomoko; Kato, Keisuke; Matsuda, Yutaka; Nagaki, Aiichiro: A Manufacturing Strategy Utilizing a Continuous-Mode Reactor toward Homogeneous PEGylated Bioconjugate Production
https://www.thieme-connect.de/media/synthesis/202404/i_m0093_ga_10-1055_a-2077-6187.gif
Ramu, Chennam; Kumaraguru, T.; Reddy, M. Sridhar; Rode, Haridas B.; Ghosh, Subhash; Reddy, Ch. Raji; Sudhakar, Gangarajula: Synthesis of Ledipasvir through a Late-Stage Cyclopropanation and Fluorination Process
https://www.thieme-connect.de/media/synthesis/202404/i_m0494_ga_10-1055_s-0042-1751437.gif
Sunny, Steeva; Maingle, Mohit; Sheeba, Loddipalle; Pathan, Firojkhan Rajekhan; J., Gowri Sankar; Juloori, Harika; Gadewar, Sainath Ganesh; Seth, Kapileswar: Pd-Nanoparticles-Catalyzed C(sp2)–H Arylation for the Synthesis of Functionalized Heterocycles: Recent Progress and Prospects
https://www.thieme-connect.de/media/synthesis/202404/i_r0041_ga_10-1055_a-2060-3488.gif
Zhang, Fei; Zhou, Yong; Wang, Shuangqiang; Zhao, Yao; Wu, Xiaojin; Chen, Rizhi: Palladium-Loading Ceramic Catalytic Membrane Reactors for Mizoroki–Heck Reaction
https://www.thieme-connect.de/media/synthesis/202404/i_b0222_ga_10-1055_a-2119-5236.gif
Ohashi, Eisaku; Sahara, Naoto; Hirano, Yoichi; Hosoya, Masahiro; Takahashi, Yusaku; Tsuno, Naoki: An Effective Additive for Introducing the Triazole Unit of Ensitrelvir: Combination of LiCl and Et3N to Easily Generate Lithium Triazinolate
https://www.thieme-connect.de/media/synthesis/202404/i_c0088_ga_10-1055_a-2085-6342.gif
Mahajan, Bhushan; Aand, Dnyaneshwar; Purwa, Mandeep; Mujawar, Taufiqueahmed; Ghosh, Subhash; Pabbaraja, Srihari; Singh, Ajay K.: Elements-Continuous-Flow Platform for Coupling Reactions and Anti-viral Daclatasvir API Synthesis
https://www.thieme-connect.de/media/synthesis/202404/i_c0518_ga_10-1055_a-2022-2063.gif
Adaoudi, Omaïma; Le Bescont, Julie; Bruneau-Voisine, Antoine; Evano, Gwilherm: Copper-Catalyzed Carbonylative Cross-Coupling of Alkyl Iodides with Alcohols and Sodium Hydroxide: Synthesis of Esters and Carboxylic Acids
https://www.thieme-connect.de/media/synthesis/202404/i_m0029_ga_10-1055_a-2042-3417.gif
Dash, Rupashri; Hota, Sudhir Kumar; Murarka, Sandip: Base-Promoted 1,6-Aza-Michael Addition of Azauracils to para-Quinone Methides
https://www.thieme-connect.de/media/synthesis/202404/i_m0215_ga_10-1055_a-2104-5943.gif
Algera, Russell F.; Davidson, Andrew; Herbert, David K.; Lian, Yajing; Liu, Fangfang; Liu, Yiyang; Nematalla, Asaad; Piper, Jared L.; Magano, Javier; Monfette, Sebastien; Nguyen, Bao; Raggon, Jeffrey W.; Rainville, Joseph P.; Rane, Anil; Tao, Yong; Wang, Ke; Yayla, Hatice G.: Exploratory Process Development of a Pulmonary Arterial Hypertension Clinical Compound via a Late-Stage Pd-Catalyzed Buchwald–Hartwig C–N Coupling
https://www.thieme-connect.de/media/synthesis/202404/i_m0254_ga_10-1055_s-0040-1720087.gif
Das, Soumyadip; Chanda, Kaushik: One-Pot Telescopic Approach to Synthesize Disubstituted Benz­imidazoles in Deep Eutectic Solvent
https://www.thieme-connect.de/media/synthesis/202404/i_t0135_ga_10-1055_a-2102-1192.jpg

Issue 01/2024

Zhang, Pengke; Hua, Lin; Takahashi, Tamotsu; Jin, Shengnan; Wang, Qilin: Recent Advances in the Dearomative Skeletal Editing of Mono-azaarenes
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Dehnert, Brady W.; Dworkin, Jeremy H.; Kwon, Ohyun: Dealkenylative Functionalizations: Conversion of Alkene C(sp3)–C(sp2) Bonds into C(sp3)–X Bonds via Redox-Based Radical Processes
https://www.thieme-connect.de/media/synthesis/202401/i_r0006_ga_10-1055_a-2044-4571.gif
Schwartz, Zachary; Valiton, Chelsea; Lovasz, Myles; Roberts, Andrew G.: Recent Applications of Ammonium Ylide Based [2,3]-Sigmatropic and [1,2]-Stevens Rearrangements To Transform Amines into Natural Products
https://www.thieme-connect.de/media/synthesis/202401/i_r0053_ga_10-1055_s-0042-1751446.gif
Martin, Brandon S.; Ma, Donghui; Saito, Takeru; Gallagher, Katelyn S.; Dai, Mingji: Concise Total Synthesis of Complanadine A Enabled by Pyrrole-to-Pyridine Molecular Editing
https://www.thieme-connect.de/media/synthesis/202401/i_c0073_ga_10-1055_a-2107-5159.gif
Gillard, Rachel M.; Zhang, Jiajun; Steel, Richard; Wang, Jocelyn; Strull, Jessica L.; Cai, Bin; Chakraborty, Nilanjana; Boger, Dale L.: Aryl Annulation: A Powerful Simplifying Retrosynthetic Disconnection
https://www.thieme-connect.de/media/synthesis/202401/i_c0449_ga_10-1055_a-1959-2088.gif
Shimazumi, Ryoma; Kodama, Takuya; Tobisu, Mamoru: Palladium-Catalyzed Unimolecular Fragment Coupling of N-Allylamides Bearing a Tethered Nucleophile with the Translocation of an Amide Group
https://www.thieme-connect.de/media/synthesis/202401/i_c0559_ga_10-1055_a-2022-1905.gif

Issue 21/2023

Taskesenligil, Yunus; Saracoglu, Nurullah: C6–H Bond Functionalization of Indoles: A New Gate
https://www.thieme-connect.de/media/synthesis/202321/i_r0049_ga_10-1055_a-2050-4897.gif
Khatua, Hillol; Das, Subrata; Patra, Sima; Chattopadhyay, Buddhadeb: C–H Bond Silylation of Heteroarenes
https://www.thieme-connect.de/media/synthesis/202321/i_r0099_ga_10-1055_a-2110-4581.gif
Basak, Shubhajit; Paul, Tripti; Mandal, Santu; Karjee, Pallab; Nanjegowda, Maniya Vadakanamala; Punniyamurthy, Tharmalingam: Transition-Metal-Catalyzed Directed C8–H Carbon–Carbon Bond Formation in Quinolines and 1,2,3,4-Tetrahydroquinolines
https://www.thieme-connect.de/media/synthesis/202321/i_r0104_ga_10-1055_a-2058-0695.gif
Gramage-Doria, Rafael; Bruneau, Christian: Carbon–Carbon Bond Forming Reactions in Diazines via Transition-Metal-Catalyzed C–H Bond Activation
https://www.thieme-connect.de/media/synthesis/202321/i_r0223_ga_10-1055_a-2134-0307.gif
Wanic, Daria K.; Melvin, Rebecca; Barker, Graeme: Zinc-Mediated C–H Metalations in Modern Organic Synthesis
https://www.thieme-connect.de/media/synthesis/202321/i_r0294_ga_10-1055_a-2155-3423.gif
Liu, Linhao; Doucet, Henri: Scope and Limitations of the Palladium-Catalyzed Direct 1,2-Diheteroarylation of 1,2-Dihalobenzene Derivatives
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Naharwal, Sushma; Kharat, Narendra Dinkar; Mahesha, Chikkagundagal K.; Bajaj, Kiran; Sakhuja, Rajeev: Palladium-Catalyzed Regioselective C-Arylation and C,N-Diarylation of N-Aryl-2,3-dihydrophthalazine-1,4-diones Using Diaryliodonium Salts
https://www.thieme-connect.de/media/synthesis/202321/i_m0036_ga_10-1055_a-2048-8030.gif
Nguyen, Thanh V. Q.; Levoin, Armand; Poli, Lorenzo: Palladium-Catalyzed C7–H (Hetero)arylation of Pyrazolo[1,5-a]pyrazines with Heteroarenes and Aryl Iodides with the Assistance of Silver Salts
https://www.thieme-connect.de/media/synthesis/202321/i_c0606_ga_10-1055_s-0041-1738433.gif
Kaur, Ramandeep; Singh, Harcharan; Babu, Srinivasarao Arulananda: Pd(II)-Catalyzed Directing-Group-Aided C–H Arylation, Alkylation, Benzylation, and Methoxylation of Carbazole-3-carboxamides toward C2,C3,C4-Functionalized Carbazoles
https://www.thieme-connect.de/media/synthesis/202321/i_f0651_ga_10-1055_a-2056-2363.gif
Intelli, Andrew John; Pal, Mohan; Selvaraju, Manikandan; Altman, Ryan A.: Palladium-Catalyzed Dearomatization of Benzothiophenes: Isolation and Functionalization of a Discrete Dearomatized Intermediate
https://www.thieme-connect.de/media/synthesis/202321/i_v0046_ga_10-1055_a-2092-9012.gif
Kumar, Saurabh; Prabhakar, Neha Sharma; Kishor, Kaushal; Singh, Krishna Nand: Decarboxylative Alkenylation of Imidazo[1,2-a]pyridines Using α,β-Unsaturated Carboxylic Acids via Pd-Catalyzed C–H Functionalization
https://www.thieme-connect.de/media/synthesis/202321/i_t0035_ga_10-1055_a-2067-4041.gif
Hayashi, Mikishiro; Michikita, Ryudai; Usuki, Yoshinosuke; Satoh, Tetsuya: Construction of Thienopyrroles through Rhodium-Catalyzed Direct Annulation of (Acetylamino)thiophenes with Alkynes
https://www.thieme-connect.de/media/synthesis/202321/i_f0645_ga_10-1055_a-2015-4466.gif
Roger, Julien; Sire, Charline; Tsivery, Anthonia; Cattey, Hélène; Hierso, Jean-Cyrille: Aryl Triflates in Phosphorus-Directed Rhodium(III)-Catalyzed C–H Activation
https://www.thieme-connect.de/media/synthesis/202321/i_t0501_ga_10-1055_a-2018-0965.gif
Kalshetti, Rupali G.; Halnor, Swapnil V.; Ramana, Chepuri V.: Rh-Catalyzed C–H Functionalization of the (Pyrazol-5-yl)pyridine Core of GBT-440
https://www.thieme-connect.de/media/synthesis/202321/i_t0167_ga_10-1055_a-2116-6734.gif
Ramkumar, Alagumalai; Gandhi, Thirumanavelan: Sustainable Ru(II)-Catalyzed ortho-C(sp2)–H Hydroxyalkylation of Phthalazinones Using Ethyl Glyoxalate: Access to α,α′-Arylcarboxy sec-Alcohols
https://www.thieme-connect.de/media/synthesis/202321/i_j0151_ga_10-1055_a-2114-5426.gif
Zhang, Zhou; Yi, Jun-Jie; Aslam, Muhammad; Wan, Jie-Ping; Sun, Meng: Rh(III)-Catalyzed Stereoselective C–H Homoallylation of Indolines with 4-Vinyl-1,3-dioxan-2-ones
https://www.thieme-connect.de/media/synthesis/202321/i_b0555_ga_10-1055_a-2002-5931.gif
Ferro, Rita; Viduedo, Nuno; Santos, A. Sofia; Silva, Artur M. S.; Royo, Beatriz; Marques, M. Manuel B.: Bimetallic Catalyzed Synthesis of 2-Arylindoles
https://www.thieme-connect.de/media/synthesis/202321/i_t0631_ga_10-1055_a-2035-6420.gif
Shinde, Vikki N.; Bhawani, Bhawani; Nipate, Dhanajay S.; Sonam, Sonam; Meena, Neha; Rangan, Krishnan; Kumar, Dalip; Kumar, Anil: Manganese-Catalyzed ortho-Hydroalkylation of Aryl-Substituted N-Heteroaromatic Compounds with Maleimides
https://www.thieme-connect.de/media/synthesis/202321/i_j0083_ga_10-1055_a-2066-1131.gif
Owens, Philippa K.; Smith, Blair I. P.; Campos, Sebastien; Lindsay, David M.; Kerr, William J.: Selective Deuteration of Heterocycle N-Oxides via Iridium-Catalysed Hydrogen Isotope Exchange
https://www.thieme-connect.de/media/synthesis/202321/i_m0108_ga_10-1055_a-2088-4302.gif
Jeon, Ju Eun; Jeong, Siyeon; Kwak, Hayeon; Joo, Jung Min: Gold-Catalyzed Cyclization of Alkynyl Heteroarenes with a Norbornene Bridge
https://www.thieme-connect.de/media/synthesis/202321/i_f0040_ga_10-1055_a-2039-5521.gif
Romero-Ibañez, Julio; Sandoval-Lira, Jacinto; Cruz-Gregorio, Silvano; Hernández-Pérez, Julio M.; Quintero, Leticia; Sartillo-Piscil, Fernando: On the Reaction Mechanism of the Selective C(sp3)–H Functionalization of N-Benzylpiperidines Mediated by TEMPO Oxoammonium Cation
https://www.thieme-connect.de/media/synthesis/202321/i_m0058_ga_10-1055_a-2053-9558.gif
Delouche, Thomas; Gadiry-Diallo, Abdoul; Besson, Thierry; Ogoshi, Sensuke; Fruit, Corinne: Photocatalyst-Free, Visible-Light-Mediated C–H Perfluoroalkylation of Quinazolin-4(3H)-ones with perfluoroalkyl Iodides
https://www.thieme-connect.de/media/synthesis/202321/i_c0044_ga_10-1055_a-2054-0482.gif
Singh, Shashank; Naskar, Kalyan S.; Kundu, Arindam; Singh, Ravi P.: Visible-Light-Induced Metal-Free Selenation of Tryptamines/3-Substituted Indoles
https://www.thieme-connect.de/media/synthesis/202321/i_f0169_ga_10-1055_a-2112-2353.gif
Sikdar, Papiya; Choudhuri, Tathagata; Paul, Suvam; Das, Sourav; Kumar, Anil; Bagdi, Avik Kumar: Photocatalyst-Free Visible-Light-Promoted C–H Selenylation of Pyrazolo[1,5-a]pyrimidines
https://www.thieme-connect.de/media/synthesis/202321/i_c0168_ga_10-1055_a-2124-5485.gif

Issue 09/2023

Schäfer, Gabriel; Reber, Stefan; Ahmetovic, Muhamed; Fleischer, Tony; Leuenberger, Daniel; Blumer, Nicole; Udry, Megan; Abele, Stefan: Robust and Scalable Reductive Amination Protocol for Electron-Poor Heterocyclic Amines Using Et3SiH/TFA as Reducing Agent
https://www.thieme-connect.de/media/synthesis/202309/i_c0441_ga_10-1055_a-1981-2727.gif
Huang, Jhih-Yi; Delbianco, Martina: Recent Developments in Solid-Phase Glycan Synthesis
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Kręcijasz, Remigiusz B.; Malinčík, Juraj; Šolomek, Tomáš: Exploring Silyl Protecting Groups for the Synthesis of Carbon Nanohoops
https://www.thieme-connect.de/media/synthesis/202309/i_c0520_ga_10-1055_a-2008-9505.gif
Murakami, Sho; Brudy, Cosima; Bachmann, Moritz; Takemoto, Yoshiji; Pieber, Bartholomäus: Photocatalytic Cleavage of Trityl Protected Thiols and Alcohols
https://www.thieme-connect.de/media/synthesis/202309/i_m0491_ga_10-1055_a-1979-5933.gif
Röckl, Johannes L.; Lundberg, Helena: Samarium and Ytterbium in Organic Electrosynthesis
https://www.thieme-connect.de/media/synthesis/202309/i_r0579_ga_10-1055_a-1997-0939.gif
Zeisel, Lukas; Maier, Martin S.; Thorn-Seshold, Oliver: Efficient and Scalable Syntheses of 1,2-Thiaselenane-4-amine and 1,2-Thiaselenane-5-amine
https://www.thieme-connect.de/media/synthesis/202309/i_c0496_ga_10-1055_a-2022-1398.gif
La Torre, Mathéo; Maton, William; Cleator, Ed; Jouffroy, Matthieu: Pd/C Catalyzed Dehalogenation of (Hetero)aryls Using Triethyl­silane as Hydrogen Donor
https://www.thieme-connect.de/media/synthesis/202309/i_c0534_ga_10-1055_s-0042-1753402.gif
Liu, Can; Shen, Ni; Shang, Rui: Photocatalytic Defluoroalkylation of Trifluoroacetates with Alkenes using 4-(Acetamido)thiophenol
https://www.thieme-connect.de/media/synthesis/202309/i_m0487_ga_10-1055_a-2019-1532.gif

Issue 06/2023

Fujimoto, Hayato; Yamamura, Shisato; Takenaka, Namiki; Tobisu, Mamoru: Phosphine-Catalyzed Z-Selective Carbofluorination of Alkynoates Bearing an N-Heteroarene Unit
https://www.thieme-connect.de/media/synthesis/202306/i_c0369_ga_10-1055_a-1948-3234.gif
Zhang, Li; Shi, Jianxun; Fang, Yewen: An Alternative to the Arbuzov Reaction: Generation and Transformation of α-Dialkyl-Substituted Methylphosphonate Carbanions via an SET Reduction Process
https://www.thieme-connect.de/media/synthesis/202306/i_c0379_ga_10-1055_a-1959-2742.gif
Picthall, Daniel; Surgenor, Brian A.; Kilian, Petr: Convenient and Scalable Synthesis of Aryldichlorophosphines and Primary Arylphosphines via Perthiophosphonic Anhydrides
https://www.thieme-connect.de/media/synthesis/202306/i_c0422_ga_10-1055_a-1994-2301.gif
Woof, Callum R.; Linford-Wood, Thomas G.; Mahon, Mary F.; Webster, Ruth L.: Catalytic Hydrophosphination of Allenes Using an Iron(II) β-Diketiminate Complex
https://www.thieme-connect.de/media/synthesis/202306/i_c0290_ga_10-1055_a-1902-5592.gif
Endo, Chikako; Inoue, Yurika; Maruyama, Toshifumi; Minoura, Mao; Murai, Toshiaki: Two-Step Transesterification of Phosphates, Phosphorothioates, and Phosphonates with a Binaphthyl Group for the Synthesis of P-Chirogenic Phosphates and Phosphonates
https://www.thieme-connect.de/media/synthesis/202306/i_c0357_ga_10-1055_a-1948-3003.gif

Issue 22/2022

Sarmah, Manashi; Hazarika, Hemanta; Gogoi, Pranjal: Aryne Annulations for the Synthesis of Carbocycles and Heterocycles: An Updated Review
https://www.thieme-connect.de/media/synthesis/202222/i_r0146_ga_10-1055_a-1863-8622.gif
Kabuki, Akira; Yamaguchi, Junichiro: Formal Syntheses of Dictyodendrins B, C, and E by a Multi-Substituted Indole Synthesis
https://www.thieme-connect.de/media/synthesis/202222/i_f0070_ga_10-1055_a-1786-9881.jpg
Iwata, Takayuki; Hyodo, Mizuki; Fujiwara, Takumi; Kawano, Ryusei; Kuhn, Leah; Alabugin, Igor V.; Shindo, Mitsuru: 3-Trifluoromethylbenzyne: Precise Orientation in Cycloaddition Reaction Enabled Regioselective Synthesis of Trifluoromethylated Triptycenes
https://www.thieme-connect.de/media/synthesis/202222/i_f0130_ga_10-1055_a-1818-0576.gif
Tawatari, Tsukasa; Kato, Ritsuki; Takasu, Kiyosei; Takikawa, Hiroshi: Intramolecular Propargylic Ene Reaction of Benzyne En Route to Highly Functionalized Allenes and Allenamides
https://www.thieme-connect.de/media/synthesis/202222/i_f0135_ga_10-1055_a-1826-2545.gif
Metze, Bryan E.; Bhattacharjee, Avik; McCormick, Theresa M.; Stuart, David R.: Parameterization of Arynophiles: Experimental Investigations towards a Quantitative Understanding of Aryne Trapping Reactions
https://www.thieme-connect.de/media/synthesis/202222/i_f0166_ga_10-1055_a-1845-3066.gif
Artigas, Albert; Hagebaum-Reignier, Denis; Carissan, Yannick; Coquerel, Yoann: Multidimensional Isotropic Magnetic Shielding Contour Maps for the Visualization of Aromaticity in ortho-Arynes and Their Reactions
https://www.thieme-connect.de/media/synthesis/202222/i_f0169_ga_10-1055_a-1867-0674.jpg
Miyabe, Hideto: Regiocontrol by Halogen Substituent on Arynes: Generation of 3-Haloarynes and Their Synthetic Reactions
https://www.thieme-connect.de/media/synthesis/202222/i_r0136_ga_10-1055_a-1814-9853.gif
Nagai, Akira; Kobayashi, Akihiro; Sakata, Yuki; Minami, Yasunori; Uchida, Keisuke; Hosoya, Takamitsu; Yoshida, Suguru: Synthesis of Multisubstituted Benzenes from Phenols via Multisubstituted Benzynes
https://www.thieme-connect.de/media/synthesis/202222/i_f0139_ga_10-1055_a-1834-2927.gif
Rai, Shweta; Samatha, Polasani; Addipilli, Ramunaidu; Mainkar, Prathama S.; Sripadi, Prabhakar; Adepu, Raju; Chandrasekhar, Srivari: Poly(ethylene glycol) Dimethyl Ethers (PEGDME): Efficient and Recyclable Solvents for Aryne-Involved Reactions
https://www.thieme-connect.de/media/synthesis/202222/i_f0147_ga_10-1055_a-1846-5598.gif
Agudelo, Brian Castro; Rigoulet, Florian; Giorgi, Michel; Sayah, Babak; Rodriguez, Jean; Coquerel, Yoann: Synthesis of Axially Chiral Cationic Benzo[c]phenanthridinium Derivatives
https://www.thieme-connect.de/media/synthesis/202222/i_f0170_ga_10-1055_a-1845-3128.gif
Yang, Yun; Jones, Christopher R.: The Aryne Ene Reaction
https://www.thieme-connect.de/media/synthesis/202222/i_f0171_ga_10-1055_a-1827-2987.gif
Heinz, Benjamin; Djukanovic, Dimitrije; Siemens, Fiona; Idriess, Mohamed; Martin, Benjamin; Knochel, Paul: Regioselective Amination or Alkoxylation of Halogenated Amino-, Thio- or Alkoxypyridines via Pyridyne Intermediates
https://www.thieme-connect.de/media/synthesis/202222/i_f0548_ga_10-1055_s-0037-1610786.gif
Zhang, Ruirui; Peng, Xia; Tan, Jiajing: Recent Advances in Construction of C(sp2)–O Bonds via Aryne Participated Multicomponent Coupling Reactions
https://www.thieme-connect.de/media/synthesis/202222/i_f0770_ga_10-1055_a-1748-7448.gif

Issue 21/2022

Yang, Zhenjie; Cheng, Hong-Gang; Chen, Ruiming; Cao, Liming; Wei, Qiang; Wang, Qingqing; Zhou, Qianghui: Eight-Step Asymmetric Synthesis of (–)-Berkelic Acid
https://www.thieme-connect.de/media/synthesis/202221/i_g0085_ga_10-1055_a-1799-0459.gif
Huang, Long-Tao; Hirata, Yuki; Kato, Yoshimi; Lin, Luqing; Kojima, Masahiro; Yoshino, Tatsuhiko; Matsunaga, Shigeki: Ruthenium(II)/Chiral Carboxylic Acid Catalyzed Enantioselective C–H Functionalization of Sulfoximines
https://www.thieme-connect.de/media/synthesis/202221/i_g0414_ga_10-1055_a-1588-0072.gif
Huang, Xiao-Ling; Li, Chong; Wang, Juan; Yang, Shang-Dong: Direct Copper-Catalyzed C-3 Arylation of Diphenylphosphine Oxide Indoles
https://www.thieme-connect.de/media/synthesis/202221/i_g0472_ga_10-1055_a-1633-8792.gif
Pototskiy, Roman A.; Boym, Mikhail A.; Nelyubina, Yulia V.; Perekalin, Dmitry S.: Synthesis of Ruthenium Catalysts with a Chiral Arene Ligand Derived from Natural Camphor
https://www.thieme-connect.de/media/synthesis/202221/i_g0590_ga_10-1055_a-1668-2075.gif
Wang, Huiying; Wang, Mengmeng; Ma, Biao; Dai, Hui-Xiong: Rhodium-Catalyzed C–H Activation of Indoles for the Construction of Spiroindole Scaffolds
https://www.thieme-connect.de/media/synthesis/202221/i_g0035_ga_10-1055_a-1791-7218.gif
Li, Mingliang; Wang, Jun: Recent Advances on Transition-Metal-Catalyzed Asymmetric C–H Arylation Reactions
https://www.thieme-connect.de/media/synthesis/202221/i_g0577_ga_10-1055_a-1677-5870.gif
Murakami, Kotone; Sakamoto, Kana; Nishimura, Takahiro: Enantioselective C–H Alkylation of N-Arylbenzamides with Vinyl Ethers Catalyzed by an Iridium/Chiral Phosphoramidite–Olefin Complex
https://www.thieme-connect.de/media/synthesis/202221/i_g0582_ga_10-1055_a-1672-6284.gif
Shirai, Tomohiko; Yamamoto, Yasunori: Cationic Iridium/Chiral Bidentate Phosphoramidite Catalyzed Asymmetric Hydroarylation
https://www.thieme-connect.de/media/synthesis/202221/i_g0594_ga_10-1055_a-1683-9455.gif
Xu, Weiwei; Ye, Mengchun: Enantioselective Cobalt-Catalyzed C–H Functionalization
https://www.thieme-connect.de/media/synthesis/202221/i_r0078_ga_10-1055_a-1801-2595.gif
Qian, Pu-Fan; Li, Jun-Yi; Zhou, Tao; Shi, Bing-Feng: Synthesis of P- and S-Stereogenic Compounds via Enantioselective C–H Functionalization
https://www.thieme-connect.de/media/synthesis/202221/i_r0088_ga_10-1055_a-1802-6793.gif
Wang, Pu-Sheng; Gong, Liu-Zhu: Asymmetric C–H Functionalization Enabled by Pd/Chiral Phosphoric Acid Combined Catalysis
https://www.thieme-connect.de/media/synthesis/202221/i_r0530_ga_10-1055_a-1662-7096.gif

Issue 19/2022

Brandão, Pedro; Pineiro, Marta; Burke, Anthony J.: Tryptanthrin and Its Derivatives in Drug Discovery: Synthetic Insights
https://www.thieme-connect.de/media/synthesis/202219/i_r0723_ga_10-1055_s-0040-1719901.jpg
Nori, Valeria; Sinibaldi, Arianna; Pesciaioli, Fabio; Carlone, Armando: Impact of Design of Experiments in the Optimisation of Catalytic Reactions in Academia
https://www.thieme-connect.de/media/synthesis/202219/i_r0735_ga_10-1055_a-1736-6703.gif
Federsel, Hans-Jürgen: Taking the Green Road Towards Pharmaceutical Manufacturing
https://www.thieme-connect.de/media/synthesis/202219/i_r0774_ga_10-1055_a-1752-5471.jpg
Carreiro, Elisabete P.; Gastalho, Carlos M.; Ernesto, Sofia; Costa, Ana R.; Antunes, Célia M.; Burke, Anthony J.: Synthesis and Antiproliferative Activity of Novel Quercetin-1,2,3-Triazole Hybrids using the 1,3-Dipolar Cycloaddition (Click) Reaction
https://www.thieme-connect.de/media/synthesis/202219/i_t0074_ga_10-1055_s-0040-1719928.gif
Sebald, Michael A.; Gebauer, Julian; Koch, Matthias: Concise Syntheses of Alternariol, Alternariol-9-monomethyl Ether and Their D3-Isotopologues
https://www.thieme-connect.de/media/synthesis/202219/i_f0536_ga_10-1055_a-1698-8328.gif
Kachkovskyi, Georgii; Cieślak, Marcin; Graczyk, Piotr; Zawadzki, Przemysław; Kalinowska-Tłuścik, Justyna; Werłos, Mateusz: Photocatalytic Approach to α,α-Difluoroalkyl Alcohols
https://www.thieme-connect.de/media/synthesis/202219/i_f0729_ga_10-1055_s-0041-1737546.gif
Marques, Carolina S.; López, Óscar; Leitzbach, Luisa; Fernández-Bolaños, José G.; Stark, Holger; Burke, Anthony J.: Survey of New, Small-Molecule Isatin-Based Oxindole Hybrids as Multi-Targeted Drugs for the Treatment of Alzheimer’s Disease
https://www.thieme-connect.de/media/synthesis/202219/i_m0728_ga_10-1055_s-0041-1737343.gif

Issue 17/2022

Remete, Attila M.; Nonn, Melinda; Volk, Balázs; Kiss, Loránd: Developments in the Alkynyltrifluoromethylations of Alkenes and Alkynes
https://www.thieme-connect.de/media/synthesis/202217/i_r0123_ga_10-1055_a-1811-8679.gif
Fichez, Jeanne; Dupommier, Dorian; Besset, Tatiana: Direct Synthesis of Disubstituted Trifluoromethylthiolated Alkenes
https://www.thieme-connect.de/media/synthesis/202217/i_r0707_ga_10-1055_s-0040-1719891.gif
Gonda, Zsombor; Földesi, Tamás; Nagy, Bálint; Novák, Zoltán: Modular Synthesis of Carbazole-Substituted Phthalimides as Potential Photocatalysts
https://www.thieme-connect.de/media/synthesis/202217/i_z0437_ga_10-1055_a-1647-7292.jpg
Salamon-Krokosz, Katarzyna; Gołdyn, Mateusz; Siodła, Tomasz; Bartoszak-Adamska, Elżbieta; Koroniak, Henryk; Koroniak-Szejn, Katarzyna: Fluorinated Olefinic Lactams: The Case of Amino Acids – Preparation and Mechanistic Studies
https://www.thieme-connect.de/media/synthesis/202217/i_c0658_ga_10-1055_s-0041-1737346.jpg
Uchikura, Tatsuhiro; Yokohama, Sosuke; Murakami, Mona; Akiyama, Takahiko: Chiral Calcium Phosphate Catalyzed Enantioselective Synthesis of All-Carbon Quaternary Center by Friedel–Crafts Alkylation Reaction of Pyrroles and Trifluoromethylated Nitrostyrenes
https://www.thieme-connect.de/media/synthesis/202217/i_f0701_ga_10-1055_s-0040-1719879.gif
Cruz-Hernández, Carlos; Juaristi, Eusebio: On the Synthesis of a Novel Chiral Phosphorodiamidic Acid Containing­ the α-Phenylethyl Moiety: Insights on its Conformation and Reactivity
https://www.thieme-connect.de/media/synthesis/202217/i_t0561_ga_10-1055_a-1689-3626.gif
El Haimer, Mohamed; Faragó, Tünde; Schelz, Zsuzsanna; Zupkó, István; Palkó, Márta: Synthesis of Alicyclic 2-Methylenethiazolo[2,3-b]quinazolinone Derivatives via Base-Promoted Cascade Reactions
https://www.thieme-connect.de/media/synthesis/202217/i_t0623_ga_10-1055_s-0040-1720028.gif
Garnes-Portolés, Francisco; Miguélez, Rubén; Grayson, Matthew N.; Barrio, Pablo: Heteroatom-Tethered ω-Alkenylallylboronates: Stereoselective Synthesis of Heterocyclic Derived Alcohols
https://www.thieme-connect.de/media/synthesis/202217/i_t0690_ga_10-1055_s-0040-1719890.gif
Dargó, Gyula; Nagy, Sándor; Kis, Dávid; Bagi, Péter; Mátravölgyi, Béla; Tóth, Blanka; Huszthy, Péter; Drahos, László; Kupai, József: Application of Proline-Derived (Thio)squaramide Organocatalysts in Asymmetric Diels–Alder and Conjugate Addition Reactions
https://www.thieme-connect.de/media/synthesis/202217/i_z0619_ga_10-1055_s-0040-1719886.gif
Raji, Mounir; Le, Tam Minh; Csámpai, Antal; Nagy, Viktória; Zupkó, István; Szakonyi, Zsolt: Stereoselective Synthesis and Applications of Pinane-Based Chiral 1,4-Amino Alcohol Derivatives
https://www.thieme-connect.de/media/synthesis/202217/i_z0668_ga_10-1055_s-0040-1719887.gif
Molnár, István G.; Mucsi, Zoltán; Kovács, Ervin; Nyerges, Miklós: Electrocyclization and Unexpected Reactions of Non-Stabilized α,β:γ,δ-Unsaturated Azomethine Ylides: Experimental and Theoretical Studies
https://www.thieme-connect.de/media/synthesis/202217/i_m0713_ga_10-1055_a-1742-2005.gif
Cserép, Gergely B.; Németh, Krisztina; Szatmári, Ágnes; Horváth, Flóra; Imre, Tímea; Németh, Krisztina; Kele, Péter: Beyond the Bioorthogonal Inverse-Electron-Demand Diels–Alder Reactions of Tetrazines: 2-Pyrone-Functionalized Fluorogenic Probes
https://www.thieme-connect.de/media/synthesis/202217/i_t0622_ga_10-1055_a-1761-4672.jpg
Szabó, Tímea; Görür, Funda Lidya; Horváth, Simon; Volk, Balázs; Milen, Mátyás: Synthesis of Racemic and Enantiopure Forms of β-Carboline Alkaloid Brevicolline
https://www.thieme-connect.de/media/synthesis/202217/i_t0720_ga_10-1055_s-0041-1737830.gif
Berecz, Gábor; Dancsó, András; Németh, Dóra R.; Kiss, Loránd; Simig, Gyula; Volk, Balázs: Towards Tianeptine Analogues: Synthesis of New Ring Systems Containing a Dibenzo[c,f][1,2]thiazepine S,S-Dioxide Core
https://www.thieme-connect.de/media/synthesis/202217/i_t0733_ga_10-1055_s-0040-1719885.gif
Takao, Go; Hakozaki, Tomohiro; Miura, Keisuke; Urushibara, Yusuke; Fuchibe, Kohei; Ichikawa, Junji: Construction of Substituted [4]Acene Frameworks Based on Double Cationic Cyclizations of Fluoroalkenes
https://www.thieme-connect.de/media/synthesis/202217/i_f0693_ga_10-1055_s-0037-1610791.gif
Harsági, Nikoletta; Kiss, Nóra Zsuzsa; Drahos, László; Keglevich, György: Synthesis of Cyclic Phosphinates by Microwave-Assisted Ionic-Liquid-Promoted Alcoholysis
https://www.thieme-connect.de/media/synthesis/202217/i_t0208_ga_10-1055_a-1504-8924.gif

Issue 15/2022

Amaya-García, Fabián; Unterlass, Miriam M.: Synthesis of 2,3-Diarylquinoxaline Carboxylic Acids in High-Temperature Water
https://www.thieme-connect.de/media/synthesis/202215/i_t0120_ga_10-1055_s-0040-1719922.gif
Vanderghinste, Jaro; Das, Shoubhik: Applications of Photoredox Catalysis for the Radical-Induced Cleavage of C–C Bonds
https://www.thieme-connect.de/media/synthesis/202215/i_t0633_ga_10-1055_a-1702-6193.gif
Swan, Charlie; Maggi, Lorenzo; Park, Mahri; Taylor, Sophie; Shepherd, William; Ball, Liam T.: Generation of Thiyl Radicals from Air-Stable, Odorless Thiophenol Surrogates: Application to Visible-Light-Promoted C–S Cross-Coupling
https://www.thieme-connect.de/media/synthesis/202215/i_z0611_ga_10-1055_s-0041-1737816.gif
Bortolato, Tommaso; Dyguda, Mateusz; Vega-Peñaloza, Alberto; Dell’Amico, Luca: Properties and Synthetic Performances of Phenylamino Cyanoarenes under One-Photon Excitation Manifolds
https://www.thieme-connect.de/media/synthesis/202215/i_c0750_ga_10-1055_a-1776-0929.gif
Monasson, Olivier; Malinowski, Maciej; Lubin-Germain, Nadège; Ferry, Angélique: Hirao Cross-Coupling Reaction as an Efficient Tool to Build Non-natural C2-Phosphonylated Sugars
https://www.thieme-connect.de/media/synthesis/202215/i_m0624_ga_10-1055_a-1709-3305.gif
Wech, Felix; Gellrich, Urs: Hydrogenation of Olefins, Alkynes, Allenes, and Arenes by Borane-Based Frustrated Lewis Pairs
https://www.thieme-connect.de/media/synthesis/202215/i_r0616_ga_10-1055_a-1684-5552.gif
Patra, Subrata; Mosiagin, Ivan; Giri, Rahul; Katayev, Dmitry: Organic Nitrating Reagents
https://www.thieme-connect.de/media/synthesis/202215/i_r0727_ga_10-1055_s-0040-1719905.gif
Abuhafez, Naba; Perennes, Antoine; Gramage-Doria, Rafael: Mimicking Enzymes: Taking Advantage of the Substrate-Recognition Properties of Metalloporphyrins in Supramolecular Catalysis
https://www.thieme-connect.de/media/synthesis/202215/i_r0743_ga_10-1055_a-1729-9223.gif
Veth, Lukas; Grab, Hanusch A.; Dydio, Paweł: Recent Trends in Group 9 Catalyzed C–H Borylation Reactions: Different Strategies To Control Site-, Regio-, and Stereoselectivity
https://www.thieme-connect.de/media/synthesis/202215/i_z0615_ga_10-1055_a-1711-5889.gif

Issue 04/2022

Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.: IntraMolecular Diels–Alder Reactions of Vinylarenes and Alkynyl Arenes (the IMDAV Reaction)
https://www.thieme-connect.de/media/synthesis/202204/i_z0484_ga_10-1055_s-0040-1705983.gif
Hopf, Henning; Sherburn, Michael S.: Allenes in Diels–Alder Cycloadditions
https://www.thieme-connect.de/media/synthesis/202204/i_m0291_ga_10-1055_s-0040-1706052.gif
Biswas, Anup; Kundu, Samrat; Pal, Dhananjoy; Pal, Amit; Maji, Modhu Sudan: Organocatalyzed Oxa-Diels–Alder Reactions: Recent Progress
https://www.thieme-connect.de/media/synthesis/202204/i_r0218_ga_10-1055_a-1514-1049.gif
Pookkandam Parambil, Shandev; Pulikkal Veettil, Santhini; Dehaen, Wim: The Synthesis of Five-Membered N-Heterocycles by Cycloaddition of Nitroalkenes with (In)Organic Azides and Other 1,3-Dipoles
https://www.thieme-connect.de/media/synthesis/202204/i_t0322_ga_10-1055_a-1547-0196.gif
He, Jian; Liu, Qiang: Highly Efficient Visible-Light-Driven [2+2] Cycloaddition of Maleimides to Alkenes and Alkynes for the Synthesis of 3-Aza­bicyclo[3.2.0]heptane-Fused Scaffolds
https://www.thieme-connect.de/media/synthesis/202204/i_g0154_ga_10-1055_a-1480-3215.gif
Kumar, Ketan; Vivekanand, T.; Singh, Bara; Ramasastry, S. S. V.: C(sp3)–H Activation Enabled by (η3-Indolylmethyl)palladium Complexes: Synthesis of Monosubstituted Tetrahydrocarbazoles
https://www.thieme-connect.de/media/synthesis/202204/i_m0241_ga_10-1055_a-1516-7960.gif
He, Xiao-Yu; Ma, Yu-Hong; Yang, Qing-Qing; Xiao, Wen-Jing: [4+n] Annulation Reactions Using ortho-Chloromethyl Anilines as Aza-ortho-Quinone Methide Precursors
https://www.thieme-connect.de/media/synthesis/202204/i_m0311_ga_10-1055_a-1529-7739.gif
Qureshi, Asif Ali; Sanjeeva Kumar, Arpula; Chauhan, Sachin; Kumara Swamy, K. C.: Stereo- and Regioselective [3+2] Cycloaddition of Acetoxy Allenoates with Azides: Metal-Free Synthesis of Multisubstituted Triazoles
https://www.thieme-connect.de/media/synthesis/202204/i_m0423_ga_10-1055_s-0040-1719838.gif
Sara, Alexandru A.; Um-e-Farwa, Um-e-Farwa; Saeed, Aamer; Kalesse, Markus: Recent Applications of the Diels–Alder Reaction in the Synthesis of Natural Products (2017–2020)
https://www.thieme-connect.de/media/synthesis/202204/i_r0249_ga_10-1055_a-1532-4763.gif
Ledovskaya, Maria S.; Voronin, Vladimir V.; Rodygin, Konstantin S.; Ananikov, Valentine P.: Acetylene and Ethylene: Universal C2 Molecular Units in Cycloaddition Reactions
https://www.thieme-connect.de/media/synthesis/202204/i_r0524_ga_10-1055_a-1654-2318.gif
Ghosh, Prasanjit; Mondal, Swati Lekha; Baidya, Mahiuddin: Ascending of Cycloaddition Strategy for N–O Heterocycles
https://www.thieme-connect.de/media/synthesis/202204/i_r0636_ga_10-1055_a-1703-6448.gif
Hofmann, Fabian; Gärtner, Cornelius; Kretzschmar, Martin; Schneider, Christoph: Asymmetric Synthesis of Fused Tetrahydroquinolines via Intra­molecular Aza-Diels–Alder Reaction of ortho-Quinone Methide Imines
https://www.thieme-connect.de/media/synthesis/202204/i_t0233_ga_10-1055_a-1517-7515.gif
Barday, Manuel; Nicolas, Eva; Higginson, Bradley; Delmotte, François; Appelmans, Martin; Aïssa, Christophe: Tandem Nickel-Catalyzed Dimerization/(4+2) Cycloaddition of Terminal Alkynes with Four-Membered Ring Ketones
https://www.thieme-connect.de/media/synthesis/202204/i_t0564_ga_10-1055_a-1671-8497.gif
Chuyko, Alexey; Dolgonos, Grygoriy; Shivanyuk, Alexander; Fetyukhin, Volodymyr; Lukin, Oleg: Simple Synthesis of Complex Amines from the Diels–Alder Adducts of (–)-Cytisine
https://www.thieme-connect.de/media/synthesis/202204/i_z0205_ga_10-1055_s-0040-1706282.gif
Ugarriza, Iratxe; Reyes, Efraím; Prieto, Liher; Uria, Uxue; Carrillo, Luisa; Vicario, Jose L.: An Approach to the Synthesis of a Hepatitis C Virus Inhibitor through a Proline-Catalyzed 1,3-Dipolar Cycloaddition Using Acrolein
https://www.thieme-connect.de/media/synthesis/202204/i_f0626_ga_10-1055_s-0040-1719858.gif

Issue 22/2021

Lam, Heather; Abel-Snape, Xavier; Köllen, Martin F.; Lautens, Mark: Recent Advances in Transition-Metal-Free (4+3)-Annulations
https://www.thieme-connect.de/media/synthesis/202122/i_z0520_ga_10-1055_s-0040-1706023.gif
Ryan, Jonathon S.; Schindler, Corinna S.: Total Synthesis of Mycocyclosin and the Herqulines
https://www.thieme-connect.de/media/synthesis/202122/i_m0034_ga_10-1055_a-1403-4312.gif
Sokol, Kevin Rafael; Magauer, Thomas: Total Synthesis of Oxepin and Dihydrooxepin Containing Natural Products
https://www.thieme-connect.de/media/synthesis/202122/i_r0210_ga_10-1055_s-0037-1610776.gif
Martín-Heras, Víctor; Daniliuc, Constantin G.; Gilmour, Ryan: An I(I)/I(III) Catalysis Route to the Heptafluoroisopropyl Group: A Privileged Module in Contemporary Agrochemistry
https://www.thieme-connect.de/media/synthesis/202122/i_m0189_ga_10-1055_a-1485-4916.gif
Wood, Devin P.; Guan, Weiyang; Lin, Song: Titanium and Cobalt Bimetallic Radical Redox Relay for the Isomerization of N-Bz Aziridines to Allylic Amides
https://www.thieme-connect.de/media/synthesis/202122/i_m0275_ga_10-1055_s-0037-1610779.gif
Garry, Olivia L.; Mansfield, Steven J.; Anderson, Edward A.: Regio- and Stereoselective Addition of Brønsted Acids to Yndiamides: Synthesis of N,O,N- and N,S,N-Trisubstituted Ketene Acetals
https://www.thieme-connect.de/media/synthesis/202122/i_m0496_ga_10-1055_a-1638-5783.gif
Tien, Chieh-Hung; Trofimova, Alina; Shao, Wenjie; Yudin, Andrei K.: Synthesis of Borylated Hydrazino Acid Derivatives
https://www.thieme-connect.de/media/synthesis/202122/i_t0192_ga_10-1055_s-0040-1706046.gif
Kasim, Johanes K.; Kavianinia, Iman; Bull, Matthew; Harris, Paul W. R.; Smaill, Jeff B.; Patterson, Adam V.; Brimble, Margaret A.: Fourth-Generation Analogues of the Anticancer Peptaibol Culicinin D: Probing the Effects of Hydrophobicity and Halogenation on Cytotoxicity
https://www.thieme-connect.de/media/synthesis/202122/i_m0124_ga_10-1055_s-0040-1706264.gif
Wienhold, Sebastian; Fritz, Lukas; Judt, Tatjana; Hackl, Sabrina; Neubauer, Thomas; Sauerer, Bastian; Bach, Thorsten: Studies towards the Synthesis of (–)-Pulvomycin: Construction of the C12–C40 Segment by a Stereoselective Aldol Reaction
https://www.thieme-connect.de/media/synthesis/202122/i_m0156_ga_10-1055_a-1464-2576.gif
El Khoury, Anton; Seidler, Paul M.; Eisenberg, David S.; Harran, Patrick G.: Catalytic Synthesis of PEGylated EGCG Conjugates that Disaggregate Alzheimer’s Tau
https://www.thieme-connect.de/media/synthesis/202122/i_m0212_ga_10-1055_a-1509-5904.gif
Caldora, Henry P.; Govaerts, Sebastian; Dighe, Shashikant U.; Turner, Oliver J.; Leonori, Daniele: A de novo Synthesis of Oxindoles from Cyclohexanone-Derived γ-Keto-Ester Acceptors Using a Desaturative Amination–Cyclization Approach
https://www.thieme-connect.de/media/synthesis/202122/i_m0336_ga_10-1055_a-1538-8429.gif
Wong, Jonathan J.; Chen, Xiangyang; Houk, Kendall N.; Vollhardt, K. Peter C.: The Trajectory of the (η5-Cyclopentadienyl)cobalt-Mediated Cycloisomerization of Ene-Yne-Ene-Type Allyl Propargylic Ethers to Furans: A DFT Appraisal
https://www.thieme-connect.de/media/synthesis/202122/i_m0475_ga_10-1055_a-1645-2632.gif
Davis, Christopher W.; Bingham, Tanner W.; Okumura, Mikiko; Sarlah, David: Dearomative syn-1,2-Diamination of Benzene and Naphthalene
https://www.thieme-connect.de/media/synthesis/202122/i_m0523_ga_10-1055_s-0040-1719842.gif
Jaye, Joseph A.; Sletten, Ellen M.: Simple Synthesis of Fluorinated Ene-Ynes via In Situ Generation of Allenes
https://www.thieme-connect.de/media/synthesis/202122/i_t0155_ga_10-1055_s-0037-1610774.gif
Wang, Lin; Ni, Shengyang; Cornella, Josep: Validation of Arylphosphorothiolates as Convergent Substrates for Ar-SF4Cl and Ar-SF5 Synthesis
https://www.thieme-connect.de/media/synthesis/202122/i_t0216_ga_10-1055_s-0040-1706039.gif

Issue 18/2021

Basak, Sumon; Biswas, Jyoti Prasad; Maiti, Debabrata: Transition-Metal-Catalyzed C–H Arylation Using Organoboron Reagents
https://www.thieme-connect.de/media/synthesis/202118/i_f0145_ga_10-1055_a-1485-4666.gif
De, Pinaki Bhusan; Asako, Sobi; Ilies, Laurean: Recent Advances in the Use of Sodium Dispersion for Organic Synthesis
https://www.thieme-connect.de/media/synthesis/202118/i_f0182_ga_10-1055_a-1478-7061.gif
Tang, Zhi; Tong, Zhou; Qiu, Renhua; Yin, Shuang-Feng; Kambe, Nobuaki: Recent Advances on Benzofuranones: Synthesis and Transformation via C–H Functionalization
https://www.thieme-connect.de/media/synthesis/202118/i_f0039_ga_10-1055_a-1405-5761.gif
Misal Castro, Luis C.; Sultan, Ibrahim; Tsurugi, Hayato; Mashima, Kazushi: Pyridine-Mediated B–B Bond Activation of (RO)2B–B(OR)2 for Generating Borylpyridine Anions and Pyridine-Stabilized Boryl Radicals as Useful Boryl Reagents in Organic Synthesis
https://www.thieme-connect.de/media/synthesis/202118/i_f0104_ga_10-1055_a-1486-8169.gif
Maeda, Kyogo; Motokura, Ken: Recent Advances in Heterogeneous Ir Complex Catalysts for Aromatic C–H Borylation
https://www.thieme-connect.de/media/synthesis/202118/i_f0142_ga_10-1055_a-1478-6118.gif
Doiuchi, Daiki; Uchida, Tatsuya: Recent Strategies in Non-Heme-Type Metal Complex-Catalyzed Site-, Chemo-, and Enantioselective C–H Oxygenations
https://www.thieme-connect.de/media/synthesis/202118/i_f0253_ga_10-1055_a-1525-4335.gif
Sihag, Pinki; Jeganmohan, Masilamani: Recent Advances in Transition-Metal-Catalyzed C–H Functionalization Reactions Involving Aza/Oxabicyclic Alkenes
https://www.thieme-connect.de/media/synthesis/202118/i_f0263_ga_10-1055_a-1528-1711.gif
Jung, Jieun; Saito, Susumu: Recent Advances in Light-Driven Carbon–Carbon Bond Formation via Carbon Dioxide Activation
https://www.thieme-connect.de/media/synthesis/202118/i_f0295_ga_10-1055_a-1577-5947.jpg
Ishida, Tamao; Zhang, Zhenzhong; Murayama, Haruno; Yamamoto, Eiji; Tokunaga, Makoto: C–H Bond Functionalization Using Pd- and Au-Supported Catalysts with Mechanistic Insights of the Active Species
https://www.thieme-connect.de/media/synthesis/202118/i_f0140_ga_10-1055_a-1468-1455.jpg
Zhang, Zhuo-Zhuo; Zhou, Gang; Huang, Fan-Rui; Shi, Bing-Feng: Cobalt-Catalyzed Oxidative [4+2] Annulation of Benzamides with Dihydrofuran: A Facile Route to Tetrahydrofuro[2,3-c]isoquinolinones
https://www.thieme-connect.de/media/synthesis/202118/i_f0268_ga_10-1055_a-1521-5800.gif
Wan, Bin; Zhang, Yanghui: Synthesis of Unsymmetrically Substituted Tetraphenylenes through Palladium-Catalyzed C(sp2)–H Activation
https://www.thieme-connect.de/media/synthesis/202118/i_f0016_ga_10-1055_a-1416-9737.gif
Dalal, Arup; Babu, Srinivasarao Arulananda: Pd(II)-Catalyzed Directing-Group-Aided C–H Arylation and Alkylation of Pyrene Core: Synthesis of C1,C2- and C1,C10-Disubstituted Pyrene Motifs
https://www.thieme-connect.de/media/synthesis/202118/i_f0113_ga_10-1055_a-1472-0881.gif
Wei, Yunlong; Chen, Zhiqi; Wu, Zhen; Xu, Yaohui; Wu, Xinxin; Zhu, Chen: Radical Carbosulfonylation of Propellane: Synthesis of Sulfonyl β-Keto-bicyclo[1,1,1]pentanes
https://www.thieme-connect.de/media/synthesis/202118/i_f0143_ga_10-1055_a-1484-1028.gif
Hassan, Mirja Md Mahamudul; Hoque, Md Emdadul; Dey, Sayan; Guria, Saikat; Roy, Brindaban; Chattopadhyay, Buddhadeb: Iridium-Catalyzed Site-Selective Borylation of 8-Arylquinolines
https://www.thieme-connect.de/media/synthesis/202118/i_f0179_ga_10-1055_a-1506-3884.gif
Yuan, Shuqing; Ling, Liang; Tang, Jinghua; Luo, Meiming; Zeng, Xiaoming: Chromium-Catalyzed Reductive Cleavage of Unactivated Aromatic and Benzylic C–O Bonds
https://www.thieme-connect.de/media/synthesis/202118/i_f0232_ga_10-1055_a-1507-6419.gif
Minami, Yasunori; Matsuyama, Nao; Matsuo, Yasuaki; Tamura, Masanori; Sato, Kazuhiko; Nakajima, Yumiko: Catalytic Reductive Cleavage of Poly(phenylene sulfide) Using a Hydrosilane
https://www.thieme-connect.de/media/synthesis/202118/i_f0259_ga_10-1055_a-1518-9010.gif
Xu, Wei; Kohei, Miki; Shibasaki, Masakatsu; Kumagai, Naoya: Strategic Synthesis of Asymmetrically Substituted C4N4 Fluorophores
https://www.thieme-connect.de/media/synthesis/202118/i_f0270_ga_10-1055_a-1516-9399.jpg
Gu, Zheng-Yang; Wu, Yang; Jin, Feng; Bao, Xiaoguang; Xia, Ji-Bao: Intermolecular C–H Amidation of Alkenes with Carbon Monoxide and Azides via Tandem Palladium Catalysis
https://www.thieme-connect.de/media/synthesis/202118/i_f0053_ga_10-1055_a-1401-4486.gif
Morimoto, Tsumoru; Wang, Chuang; Tanimoto, Hiroki; Artok, Levent; Kakiuchi, Kiyomi: Rhodium(I)-Catalyzed CO-Gas-Free Arylative Dual-Carbonylation of Alkynes with Arylboronic Acids via the Formyl C–H Activation of Formaldehyde
https://www.thieme-connect.de/media/synthesis/202118/i_f0130_ga_10-1055_a-1468-8377.gif
Kimura, Naoki; Katta, Shiori; Kitazawa, Yoichi; Kochi, Takuya; Kakiuchi, Fumitoshi: Deuterium-Labeling Studies on the C–H/Olefin Coupling of Aromatic Ketones Catalyzed by Fe(PMe3)4
https://www.thieme-connect.de/media/synthesis/202118/i_f0186_ga_10-1055_s-0040-1706040.gif
Jinnai, Seihou; Oi, Ayumi; Seo, Takuji; Moriyama, Taichi; Minami, Ryunosuke; Higashida, Suguru; Ie, Yutaka: Electron-Accepting π-Conjugated Compound Containing Cyano-Substituted Naphthobisthiadiazole as Nonfullerene Acceptor in Organic Solar Cells
https://www.thieme-connect.de/media/synthesis/202118/i_f0214_ga_10-1055_a-1528-1632.gif
Rawat, Vishal Kumar; Higashida, Kosuke; Sawamura, Masaya: Nickel-Catalyzed Homocoupling of Aryl Ethers with Magnesium Anthracene Reductant
https://www.thieme-connect.de/media/synthesis/202118/i_f0235_ga_10-1055_a-1509-5954.gif
Fukuyama, Takahide; Hamada, Yuki; Ryu, Ilhyong: A New Protocol for Catalytic Reduction of Alkyl Chlorides Using an Iridium/Bis(benzimidazol-2′-yl)pyridine Catalyst and Triethylsilane
https://www.thieme-connect.de/media/synthesis/202118/i_f0258_ga_10-1055_a-1527-4526.gif

Issue 17/2021

Korvorapun, Korkit; Samanta, Ramesh C.; Rogge, Torben; Ackermann, Lutz: Remote C–H Functionalizations by Ruthenium Catalysis
https://www.thieme-connect.de/media/synthesis/202117/i_f0171_ga_10-1055_a-1485-5156.gif
Vijaykumar, Muniyappa; Punji, Benudhar: Advances in Transition-Metal-Catalyzed C–H Bond Oxygenation of Amides
https://www.thieme-connect.de/media/synthesis/202117/i_f0146_ga_10-1055_a-1481-2584.gif
Ohno, Shohei; Miyoshi, Makoto; Murai, Kenichi; Arisawa, Mitsuhiro: Non-Directed β- or γ-C(sp3)–H Functionalization of Saturated Nitrogen-Containing Heterocycles
https://www.thieme-connect.de/media/synthesis/202117/i_f0110_ga_10-1055_a-1483-4575.gif
Aldhous, Timothy P.; Chung, Raymond W. M.; Dalling, Andrew G.; Bower, John F.: Enantioselective Intermolecular Murai-Type Alkene Hydroarylation Reactions
https://www.thieme-connect.de/media/synthesis/202117/i_f0144_ga_10-1055_s-0040-1720406.gif
Oonishi, Yoshihiro; Sakamoto, Shunki; Agata, Shuya; Sato, Yoshihiro: Rhodium(I)-Catalyzed Enantioselective Cyclization of Enynes through Site-Selective C(sp3)–H Bond Activation Triggered by Formation of Rhodacycle
https://www.thieme-connect.de/media/synthesis/202117/i_f0125_ga_10-1055_a-1469-7408.gif
Watanabe, Hikaru; Nakajima, Kazuki; Ekuni, Kento; Edagawa, Ryota; Akagi, Yuta; Okuda, Yasuhiro; Wakamatsu, Kan; Orita, Akihiro: Custom-Made Pyrene Photocatalyst-Promoted Desulfonylation of Arylethenyl Sulfones Using Green-Light-Emitting Diodes
https://www.thieme-connect.de/media/synthesis/202117/i_f0005_ga_10-1055_s-0040-1706025.gif
Akahori, Shuhei; Fujihara, Tetsuaki; Tsuji, Yasushi; Shinokubo, Hiroshi; Miyake, Yoshihiro: Synthesis of Tetrasilatetrathia[8]circulenes through C–I and C–H Silylation
https://www.thieme-connect.de/media/synthesis/202117/i_f0107_ga_10-1055_a-1437-9917.gif
Seo, Jia; Chen, Che-Wei; Lee, Woohyeong; Jeon, Ju Eun; Chen, Pei-Ling; Chuang, Shih-Ching; Joo, Jung Min: Palladium-Catalyzed C–H Benzannulation of Functionalized Furans and Pyrroles with Alkynes
https://www.thieme-connect.de/media/synthesis/202117/i_f0134_ga_10-1055_a-1502-3641.gif
Fukumoto, Yoshiya; Shiratani, Motohiro; Noguchi, Hikaru; Chatani, Naoto: Iridium-Catalyzed Direct Amidation of Imidazoles at the C-2 Position with Isocyanates in the Presence of Hydrosilanes Leading to Imidazole-2-Carboxamides
https://www.thieme-connect.de/media/synthesis/202117/i_f0637_ga_10-1055_a-1375-5283.gif
Ozaki, Tomoya; Kaga, Atsushi; Saito, Hayate; Yorimitsu, Hideki: Generation of Aryllithium Reagents from N-Arylpyrroles Using Lithium
https://www.thieme-connect.de/media/synthesis/202117/i_z0120_ga_10-1055_a-1482-2567.gif
Inai, Yasuhito; Usuki, Yoshinosuke; Satoh, Tetsuya: Synthesis of Benzo-Fused Cyclic Compounds via Rhodium-Catalyzed Decarboxylative Coupling of Aromatic Carboxylic Acids with Alkynes
https://www.thieme-connect.de/media/synthesis/202117/i_f0071_ga_10-1055_a-1416-6997.gif
Shimazumi, Ryoma; Morita, Kosuke; Yoshida, Tomoki; Yasui, Kosuke; Tobisu, Mamoru: Late-Stage Derivatization of Buflavine by Nickel-Catalyzed Direct Substitution of a Methoxy Group via C–O Bond Activation
https://www.thieme-connect.de/media/synthesis/202117/i_f0122_ga_10-1055_a-1467-2494.gif
You, Jingwen; Chen, Qiang; Nishihara, Yasushi: Nickel-Catalyzed Decarbonylative Thioetherification of Acyl Fluorides via C–F Bond Activation
https://www.thieme-connect.de/media/synthesis/202117/i_f0133_ga_10-1055_a-1484-6216.gif
Yabe, Ryota; Ebe, Yusuke; Nishimura, Takahiro: Iridium-Catalyzed Direct C–H Allylation of Ketimines
https://www.thieme-connect.de/media/synthesis/202117/i_f0137_ga_10-1055_a-1477-7059.gif
Ohmura, Toshimichi; Yagi, Kaito; Torigoe, Takeru; Suginome, Michinori: Intramolecular Addition of a Dimethylamino C(sp3)–H Bond across C–C Triple Bonds Using IrCl(DTBM-SEGPHOS)(ethylene) Catalyst: Synthesis of Indoles from 2-Alkynyl-N-methylanilines
https://www.thieme-connect.de/media/synthesis/202117/i_f0252_ga_10-1055_a-1511-1025.gif
Takahashi, Hiroto; Honjo, Yusaku; Shibata, Yu; Nagashima, Yuki; Tanaka, Ken: Dienylation of Unfunctionalized Arenes with 1,6-Diynes via Rhodium-Catalyzed Directing-Group-Free C–H Bond Activation
https://www.thieme-connect.de/media/synthesis/202117/i_f0585_ga_10-1055_a-1328-6436.gif
Kawakami, Haruka; Nohira, Itsuki; Chatani, Naoto: Nickel-Catalyzed C–F/N–H Annulation of 2-(2-Fluoroaryl) N-Heteroaromatic Compounds with Alkynes: Activation of C–F Bonds
https://www.thieme-connect.de/media/synthesis/202117/i_f0614_ga_10-1055_a-1337-5504.gif
Yamamoto, Sonoka; Shibuya, Yushin; Suzuki, Toyoko; Okano, Kentaro; Horie, Masaki; Mori, Atsunori: One-Shot Deprotonative Metalation/Transmetalation/Polymerization of Halothiophenes Catalyzed by Nickel Complex for Polythiophene Synthesis
https://www.thieme-connect.de/media/synthesis/202117/i_f0653_ga_10-1055_a-1368-7072.jpg
Kanyiva, Kyalo Stephen; Tang, King Hung Nigel; Wang, Jiarui; Shibata, Takanori: Palladium-Catalyzed sp3 C–H Benzoxylation of Alanine Derivatives Using Aldehydes under Ambient Conditions
https://www.thieme-connect.de/media/synthesis/202117/i_f0024_ga_10-1055_a-1422-9632.gif
Pan, Feng-Feng; Guo, Peng; Huang, Xiaochuang; Shu, Xing-Zhong: Synthesis of Dibenzyls by Nickel-Catalyzed Homocoupling of Benzyl Alcohols
https://www.thieme-connect.de/media/synthesis/202117/i_f0108_ga_10-1055_a-1467-2432.gif
Kiyosu, Yuuki; Tanaka, Shino; Okumura, Sota; Kiyokawa, Kensuke; Minakata, Satoshi: Synthesis of Fused Diaziridine Derivatives from Cyclic Secondary Amines by Utilizing N-Bromosulfonamides as an Aminating Reagent
https://www.thieme-connect.de/media/synthesis/202117/i_f0129_ga_10-1055_a-1468-8275.gif
Ninokata, Ryo; Korogi, Riho; Nakao, Junya; Fukuda, Tsutomu; Onodera, Gen; Kimura, Masanari: Reconstruction of Carbon Bond Frameworks via Oxapalladacycles Promoted by the Synergistic Effect of Palladium Catalyst and Triethylborane
https://www.thieme-connect.de/media/synthesis/202117/i_f0132_ga_10-1055_a-1485-5781.gif
Tanaka, Shinji; Iwase, Shoutaro; Kanda, Sena; Kato, Marie; Kiriyama, Yutaro; Kitamura, Masato: Ruthenium-Catalyzed Asymmetric Dehydrative Allylic Cyclization of Five-Membered Chalcogen Heteroaromatics
https://www.thieme-connect.de/media/synthesis/202117/i_f0141_ga_10-1055_a-1523-6826.gif
Kona, Chandrababu Naidu; Oku, Rikuto; Nishii, Yuji; Miura, Masahiro: Peri-Selective Direct Acylmethylation and Amidation of Naphthalene Derivatives Using Iridium and Rhodium Catalysts
https://www.thieme-connect.de/media/synthesis/202117/i_f0150_ga_10-1055_a-1472-1059.gif
Ishida, Naoyoshi; Iwamoto, Hiroaki; Sunagawa, Denise Eimi; Ohashi, Masato; Ogoshi, Sensuke: CsF-Catalyzed Fluoroacylation of Tetrafluoroethylene Using Acyl Fluorides for the Synthesis of Pentafluoroethyl Ketones
https://www.thieme-connect.de/media/synthesis/202117/i_f0481_ga_10-1055_s-0040-1705962.gif
Xu, Wengang; Wu, Mingbo; Yoshikai, Naohiko: Iron-Catalyzed Remote C–H Alkylation of 8-Amidoquinolines with Cycloalkanes
https://www.thieme-connect.de/media/synthesis/202117/i_f0595_ga_10-1055_a-1337-5416.gif

Issue 02/2021

Arjona-Esteban, Alhama; Rausch, Anja; Vysotsky, Myroslav O.; Würthner, Frank: Merocyanine Dyes with Extended Polymethine Chains by Simple Two-Step Condensation Sequence
https://www.thieme-connect.de/media/synthesis/202102/i_c0240_ga_10-1055_s-0040-1707896.gif
Yoshimura, Aya; Henmi, Keisuke; Kimura, Hitoshi; Sakakibara, Ryo; Ochi, Rika; Shirahata, Takashi; Yorimitsu, Hideki; Misaki, Yohji: Synthesis of Peripherally Arylated Tetrathiafulvalenes Extended with an Anthraquinoid Spacer via Pd-Catalyzed C–H Arylation and Construction of a Double-Helical Cobalt-Based Metal-Organic Framework
https://www.thieme-connect.de/media/synthesis/202102/i_c0266_ga_10-1055_s-0040-1707177.gif
Widner, Florian J.; Kieninger, Christoph; Wurst, Klaus; Deery, Evelyne; Lawrence, Andrew D.; Warren, Martin J.; Kräutler, Bernhard: Synthesis, Spectral Characterization and Crystal Structure of Chlororhodibalamin: A Synthesis Platform for Rhodium Analogues of Vitamin B12 and for Rh-Based Antivitamins B12
https://www.thieme-connect.de/media/synthesis/202102/i_c0397_ga_10-1055_s-0040-1707288.gif
Yan, Feng-Zhi; Shao, Yuan-Guang; Zhang, Zibin; Shen, Yan-Feng; Huang, Xue-Chun; Zhang, Pei-Ling; Li, Shijun: Synthesis of Catenanes from a BMP32C10-Based Cryptand Tuned by the Linkage Length of Paraquat Salts
https://www.thieme-connect.de/media/synthesis/202102/i_c0428_ga_10-1055_s-0040-1707290.gif
Mei, Peifeng; Kurosaki, Ryo; Matsumoto, Akinobu; Yamada, Hiroko; Aratani, Naoki: One-Pot Synthesis of a Cyclic Pyrene Octamer from Two Bifunctionalized Pyrene Monomers
https://www.thieme-connect.de/media/synthesis/202102/i_c0439_ga_10-1055_s-0040-1705950.gif

Issue 24/2020

Qin, Jing-Hao; Li, Jin-Heng; An, De-Lie: Recent Advances in Cycloaddition Reactions with Alkynes to Construct Heterocycles
https://www.thieme-connect.de/media/synthesis/202024/i_c0230_ga_10-1055_s-0040-1707355.gif
Pellissier, Hélène: The Use of Domino Reactions for the Synthesis of Chiral Rings
https://www.thieme-connect.de/media/synthesis/202024/i_c0191_ga_10-1055_s-0040-1707905.gif
Wei, Bin; Li, Ke-Wei; Wu, Yan-Chen; Tong, Shi-Qi; Song, Ren-Jie: Radical Strategy for the Transition-Metal-Catalyzed Synthesis of γ-Lactones: A Review
https://www.thieme-connect.de/media/synthesis/202024/i_c0226_ga_10-1055_s-0040-1707835.jpg
Huang, Min-Hua; Hao, Wen-Juan; Jiang, Bo: Iridium(III)-Catalyzed Difluoroalkylation–Bicyclization of 1,7-Enynes toward Benzo[a]fluoren-5-ones under Visible-Light Photoredox Conditions
https://www.thieme-connect.de/media/synthesis/202024/i_c0182_ga_10-1055_s-0040-1707863.gif

Issue 22/2020

Maligres, Peter E.; Song, Zhiguo Jake; Strotman, Neil A.; Yin, Jinquin; Pei, Tao; Strotman, Hallena R.; Itoh, Tetsuji; Sherer, Edward C.; Humphrey, Guy R.: Synthesis of Fused Oxepane HIV Integrase Inhibitor MK-1376
https://www.thieme-connect.de/media/synthesis/202022/i_c0045_ga_10-1055_s-0040-1707994.gif
Toussaint, Frédéric C.; Defrance, Thierry; Decouvreur, Serge; Carly, Nicolas; Merschaert, Alain: Intensification of Free-Radical Racemization for a Non-activated Amine in a Continuous Flow Reactor
https://www.thieme-connect.de/media/synthesis/202022/i_c0232_ga_10-1055_s-0040-1707339.jpg
Wächtler, Andreas; Bremer, Matthias; Maillard, David; Mohr, Thomas: Controlling the All-trans Stereochemistry in Liquid Crystalline 4,4′-Dialkyl-[1,1′-bicyclohexyl] Compounds
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Stumpf, Andreas; St-Jean, Frédéric; Lao, David; Cheng, Zhigang Ken; Angelaud, Remy; Gosselin, Francis: Practical Early Development Synthesis of Nav1.7 Inhibitor GDC-0310
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Chen, Chengsheng; Wu, Ling; Wang, Yuwen; Wu, Linglin; Zhang, Yongda: Copper-Catalyzed Asymmetric Hydroamination of Styrenes with pivZPhos as Ligand
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Crawford, James J.; Liao, Daohong; Kolesnikov, Aleksandr; Lee, Wendy; Landry, Matthew L.: Synthesis of an Azabicyclo[3.1.0]hexanone-Containing Inhibitor of NF-κΒ Inducing Kinase via Catalytic C–H Activation
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Issue 21/2020

Shiri, Morteza; Farajinia-Lehi, Noushin; Salehi, Parvin; Tanbakouchian, Zahra: Transition Metal and Inner Transition Metal Catalyzed Amide Derivatives Formation through Isocyanide Chemistry
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Manne, Srinivasa Rao; de la Torre, Beatriz G.; El-Faham, Ayman; Albericio, Fernando: OxymaPure Coupling Reagents: Beyond Solid-Phase Peptide Synthesis
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Zhao, Baoli; Liu, Yunyun: Step-Economical C–H Activation Reactions Directed by In Situ Amidation
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Spiliopoulou, Nikoleta; Constantinou, Constantinos T.; Triandafillidi, Ierasia; Kokotos, Christoforos G.: Synthetic Approaches to Acyl Hydrazides and Their Use as Synthons in Organic Synthesis
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Kolympadi Marković, Maria; Marković, Dean; Laclef, Sylvain: Amide Synthesis by Transamidation of Primary Carboxamides
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Shiri, Morteza; Gholami-Koupaei, Zahra; Bandehali-Naeini, Farzaneh; Tonekaboni, Maryam-Sadat; Soheil-Moghaddam, Saeedeh; Ebrahimi, Delaram; Karami, Sima; Notash, Behrouz: Highly Selective Synthesis of α-Hydroxy, α-Oxy, and α-Oxo Amides by a Post-Passerini Condensation Transformation
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Movahed, Farzaneh Soleymani; Sawant, Dinesh N.; Bagal, Dattatraya B.; Saito, Susumu: Tris(o-phenylenedioxy)cyclotriphosphazene as a Promoter for the Formation of Amide Bonds Between Aromatic Acids and Amines
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Smolobochkin, Andrey V.; Gazizov, Almir S.; Otegen, Nazerke K.; Voronina, Julia K.; Strelnik, Anna G.; Samigullina, Aida I.; Burilov, Alexander R.; Pudovik, Michail A.: Nucleophilic Cyclization/Electrophilic Substitution of (2,2-Dialkoxyethyl)ureas: Highly Regioselective Access to Novel 4-(Het)arylimidazolidinones and Benzo[d][1,3]diazepinones
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Verma, Saumya; Kumar, Puneet; Khatana, Anil K.; Chandra, Dinesh; Yadav, Ajay K.; Tiwari, Bhoopendra; Jat, Jawahar L.: Zinc(II)-Catalyzed Synthesis of Secondary Amides from Ketones via Beckmann Rearrangement Using Hydroxylamine-O-sulfonic Acid in Aqueous Media
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Kabes, Connor Q.; Gunn, Jack H.; Selbst, Maximilian A.; Lucas, Reagan F.; Gladysz, John A.: Syntheses of Enantiopure 1,2-Ethylenediamines with Tethered Secondary Amines of the Formula H2NCH2CH[(CH2)nNHMe]NH2 (n = 1–4) from α-Amino Acids: New Agents for Asymmetric Catalysis
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Zhang, Rui; Zhang, Jun-Chao; Zhang, Wei-Yi; He, Yu-Qing; Cheng, Hua; Chen, Cheng; Gu, Yu-Cheng: A Practical Approach for the Transamidation of N,N-Dimethyl Amides with Primary Amines Promoted by Sodium tert-Butoxide under Solvent-Free Conditions
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Issue 08/2020

Connon, Robert; Carroll, Laura; Guiry, Patrick J.: A Base-Promoted One-Pot Asymmetric Friedel–Crafts Alkylation/Michael Addition of 4-Substituted Indoles
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Yang, Yuzhong; Zhou, Liwei; Yang, Xiumei; Luo, Xiai; Deng, Guobo; Yang, Yuan; Liang, Yun: Synthesis of Phenanthrenes via Palladium-Catalyzed Three-Component Domino Reaction of Aryl Iodides, Internal Alkynes, and o-Bromobenzoic Acids
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Henkel, Michael; Bach, Thorsten: Annulation of Indoles with 1,n-Dibromoalkanes by a Pd(II)-Catalyzed and Norbornene-Mediated Reaction Cascade
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Shen, Zican; Li, Chen; Mercado, Brandon Q.; Ellman, Jonathan A.: Cobalt(III)-Catalyzed Diastereoselective Three-Component C–H Bond Addition to Butadiene and Activated Ketones
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Lee, Sumin; Jang, Young Jin; Phipps, Erik J. T.; Lei, Honghui; Rovis, Tomislav: Rhodium(III)-Catalyzed Three-Component 1,2-Diamination of Unactivated Terminal Alkenes
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Sun, Manman; Li, Jinshan; Chen, Weida; Wu, Haijian; Yang, Jianguo; Wang, Zhiming: Palladium-Catalyzed [4+2] Annulation of Aryl and Alkenyl Carboxamides with 1,3-Dienes via C–H Functionalization: Synthesis of 3,4-Dihydroisoquinolones and 5,6-Dihydropyridinones
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Issue 23/2019

Special Topic Cover Page
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Sutherland, Andrew: Radiohalogenation of Organic Compounds: Practical Considerations and Challenges for Molecular Imaging
https://www.thieme-connect.de/media/synthesis/201923/i_s0302_ga_10-1055_s-0037-1611885.jpg
Milicevic Sephton, Selena; Zhou, Xiaoyun; Thompson, Stephen; Aigbirhio, Franklin I.: Preparation of the Serotonin Transporter PET Radiotracer 2-({2-[(Dimethylamino)methyl]phenyl}thio)-5-[18F]fluoroaniline (4-[18F]ADAM): Probing Synthetic and Radiosynthetic Methods
https://www.thieme-connect.de/media/synthesis/201923/i_c0355_ga_10-1055_s-0039-1690522.gif
Kitahara, Kazumasa; Mizutani, Haruna; Iwasa, Seiji; Shibatomi, Kazutaka: Asymmetric Synthesis of α-Chloro-α-halo Ketones by Decarboxylative Chlorination of α-Halo-β-ketocarboxylic Acids
https://www.thieme-connect.de/media/synthesis/201923/i_c0320_ga_10-1055_s-0039-1690009.gif
Dubost, Emmanuelle; Babin, Victor; Benoist, Florian; Hébert, Alexandra; Pigrée, Gilbert; Bouillon, Jean-Philippe; Fabis, Frédéric; Cailly, Thomas: Improvements of C–H Radio-Iodination of N-Acylsulfonamides toward Implementation in Clinics
https://www.thieme-connect.de/media/synthesis/201923/i_s0301_ga_10-1055_s-0037-1611884.gif
Thompson, Stephen; Lee, So Jeong; Jackson, Isaac M.; Ichiishi, Naoko; Brooks, Allen F.; Sanford, Melanie S.; Scott, Peter J. H.: Synthesis of [18F]-γ-Fluoro-α,β-unsaturated Esters and Ketones via Vinylogous 18F-Fluorination of α-Diazoacetates with [18F]AgF
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Sarie, Jérôme C.; Neufeld, Jessica; Daniliuc, Constantin G.; Gilmour, Ryan: Willgerodt-Type Dichloro(aryl)-λ3-Iodanes: A Structural Study
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Issue 13/2019

Special Topic Cover Page
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Podyacheva, Evgeniya; Afanasyev, Oleg I.; Tsygankov, Alexey A.; Makarova, Maria; Chusov, Denis: Hitchhiker’s Guide to Reductive Amination
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Lai, Wing In; Leung, Man Pan; Choy, Pui Ying; Kwong, Fuk Yee: Sterically Hindered Amination of Aryl Chlorides Catalyzed by a New Carbazolyl-Derived P,N-Ligand-Composed Palladium Complex
https://www.thieme-connect.de/media/synthesis/201913/i_h0168_ga_10-1055_s-0037-1611534.gif
Purkait, Anisha; Jana, Chandan K.: N-Aminations of Benzylamines and Alicyclic Amines with Nitrosoarenes to Hydrazones and Hydrazides
https://www.thieme-connect.de/media/synthesis/201913/i_c0091_ga_10-1055_s-0037-1610701.gif
Li, Quan-Zhe; Wang, Xun-Hui; Hou, Si-Hua; Ma, Yan-Yan; Zhao, Deng-Gao; Zhang, Shu-Yu; Bai, He-Yuan; Ding, Tong-Mei: Silver-Catalyzed para-Selective C–H Amination of 1-Naphthyl­amides with Azodicarboxylates at Room Temperature
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Pratap, Ramendra; Yorimitsu, Hideki: Palladium-Catalyzed Amination of Aryl Sulfides and Sulfoxides with Azaarylamines of Poor Nucleophilicity
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Zhou, Huan; Zhao, Wenlei; Zhang, Tao; Guo, Haodong; Huang, Haizhou; Chang, Mingxin: Enantioselective Synthesis of 2-Substituted Pyrrolidines via Intramolecular­ Reductive Amination
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Issue 12/2019

Special Topic Cover Page
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Zhou, Yongyun; Khan, Ruhima; Fan, Baomin; Xu, Lijin: Ruthenium-Catalyzed Selective Reduction of Carboxylic Esters and Carboxamides
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Deshmukh, Dewal S.; Bhanage, Bhalchandra M.: Ruthenium-Catalyzed Annulation of N-Cbz Hydrazones via C–H/N–N Bond Activation for the Rapid Synthesis of Isoquinolines
https://www.thieme-connect.de/media/synthesis/201912/i_c0127_ga_10-1055_s-0037-1611795.gif
Das, Riki; Khot, Nandkishor Prakash; Deshpande, Akanksha Santosh; Kapur, Manmohan: Ruthenium-Catalyzed Directed C(3)–H Olefination of N-Acetyl-1,2-dihydroisoquinolines: A Method to Achieve C3-Olefinated Isoquinolines
https://www.thieme-connect.de/media/synthesis/201912/i_c0102_ga_10-1055_s-0037-1611807.gif
Bairy, Gurupada; Nandi, Arijit; Manna, Kartic; Jana, Ranjan: Ruthenium(II)-Catalyzed Migratory C–H Allylation/Hydroamination Cascade for the Synthesis of Rutaecarpine Analogues
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Tran, Christine; Haddad, Mansour; Ratovelomanana-Vidal, Virginie: Ruthenium-Catalyzed [2+2+2] Cycloaddition of α,ω-Diynes and Selenocyanates: An Entry to Selenopyridine Derivatives
https://www.thieme-connect.de/media/synthesis/201912/i_c0078_ga_10-1055_s-0037-1610704.gif
Kawano, Teruhiro; Watari, Ryo; Kayaki, Yoshihito; Ikariya, Takao: Catalytic Hydrogenation of Carboxamides with a Bifunctional Cp*Ru Catalyst Bearing an Imidazol-2-ylidene with a Protic Aminoethyl Side Chain
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Issue 17/2018

Special Topic Cover Page
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Oh, Eun Hye; Kim, Hyun Jin; Han, Soo Bong: Recent Developments in Visible-Light-Catalyzed Multicomponent Trifluoromethylation of Unsaturated Carbon–Carbon Bonds
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Zhou, Wen-Jun; Zhang, Yi-Han; Gui, Yong-Yuan; Sun, Liang; Yu, Da-Gang: Merging Transition-Metal Catalysis with Photoredox Catalysis: An Environmentally Friendly Strategy for C–H Functionalization
https://www.thieme-connect.de/media/synthesis/201817/i_c0386_ga_10-1055_s-0037-1610222.gif
Du, Yuliu; Wei, Zheng; Wang, Ting: Visible-Light-Mediated Synthesis of Oxidized Amides via Organic Photoredox Catalysis
https://www.thieme-connect.de/media/synthesis/201817/i_c0144_ga_10-1055_s-0036-1591988.gif
An, Xiao-De; Yu, Shouyun: Photoredox-Catalyzed Radical Relay Reaction Toward Functionalized Vicinal Diamines
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Voutyritsa, Errika; Nikitas, Nikolaos F.; Apostolopoulou, Mary K.; Gerogiannopoulou, Anna Dimitra D.; Kokotos, Christoforos G.: Photoorganocatalytic Atom Transfer Radical Addition of Bromoacetonitrile to Aliphatic Olefins
https://www.thieme-connect.de/media/synthesis/201817/i_c0112_ga_10-1055_s-0037-1610138.gif
Otomura, Nobutaka; Okugawa, Yuto; Hirano, Koji; Miura, Masahiro: Bromine Cation Initiated vic-Diphosphination of Styrenes with Diphosphines under Photoredox Catalysis
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Issue 16/2018

Special Topic Cover Page
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Baumann, Andreas N.; Eisold, Michael; Music, Arif; Didier, Dorian: One-Pot Preparation of Stable Organoboronate Reagents for the Functionalization of Unsaturated Four- and Five-Membered Carbo­- and Heterocycles
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Yamaguchi, Eiji; Kamito, Yuji; Matsuo, Kazuki; Ishihara, Jun; Itoh, Akichika: Photooxidative Keto-Trifluoromethylation of Styrenes by Means of an Anthraquinone-Based Organocatalyst
https://www.thieme-connect.de/media/synthesis/201816/i_c0116_ga_10-1055_s-0036-1592003.gif
Chen, Yizhou; Wang, Shanlu; Zhao, Li; Rong, Chenyan; Liu, Tong; Sun, Han; Wang, Yuping; Zhang, Jian; Zhong, Guofu: A Metal-Free Synthesis of 3-Phenoxyimidazo Heterocycles by Catalytic Oxidative Cyclization of 2-Amino-azaarenes with Lignin Models
https://www.thieme-connect.de/media/synthesis/201816/i_c0133_ga_10-1055_s-0037-1610139.gif
Suen, Linda M.; Wang, Cheng; Hunter, David N.; Mitchell, Helen J.; Converso, Antonella; ElMarrouni, Abdellatif: Synthesis of HIV NNRTI Doravirine Analogues via Visible-Light Photoredox Decarboxylative Cross-Coupling
https://www.thieme-connect.de/media/synthesis/201816/i_c0175_ga_10-1055_s-0037-1610155.gif
Liu, Yang; Daka, Mario; Bandini, Marco: Regio- and Stereoselective Nickel-Catalyzed Coupling of Boronic Acids with Allenoates
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Park, Jaerim; Song, Kwang Ho; Lee, Sunwoo: Palladium-Catalyzed Decarboxylative Coupling Reactions of Propiolic Acid Derivatives and Arylsulfonyl Hydrazide
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Torregrosa, Robert R. P.; Mendis, Shehani N.; Davies, Alex; Tunge, Jon A.: Palladium-Catalyzed Decarboxylative Benzylation of Acetylides and Enolates
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Li, Jing; Wang, Zhong-Xia: Nickel-Catalyzed Transformation of Aryl 2-Pyridyl Ethers via Cleavage of the Carbon–Oxygen Bond: Synthesis of Mono-α-arylated­ Ketones
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De, Pinaki Bhusan; Pradhan, Sourav; Shah, Tariq A.; Punniyamurthy, Tharmalingam: Iodine-Mediated Intramolecular C–H Amination of Benzimidazoles: A Metal-Free Route to Dihydroimidazobenzimidazoles
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Guan, Weiye; Liao, Jennie; Watson, Mary P.: Vinylation of Benzylic Amines via C–N Bond Functionalization of Benzylic Pyridinium Salts
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Yin, Zhiping; Power, Dennis J.; Wang, Zechao; Stewart, Scott G.; Wu, Xiao-Feng: Synthesis of 1,3,4-Oxadiazoles via Annulation of Hydrazides and Benzene-1,3,5-triyl Triformate under Metal-Free Conditions
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Issue 15/2018

Special Topic Cover Page
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Zhang, Qi; Raveendra Babu, Kaki; Huang, Zhouliang; Song, Jinna; Bi, Xihe: Visible-Light-Induced Radical Polynitration of Arylboronic Acids: Synthesis of Polynitrophenols
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Wu, Kui; Fang, Cheng; Kaur, Sarbjeet; Liu, Peng; Wang, Ting: Methylene Blue-Catalyzed Oxidative Cleavage of N-Carbonylated Indoles
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Wang, Guang-Zu; Shang, Rui; Fu, Yao: Irradiation-Induced Palladium-Catalyzed Direct C–H Alkylation of Heteroarenes with Tertiary and Secondary Alkyl Bromides
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Hamsath, Akil; Galloway, Jordan D.; Baxter, Ryan D.: Quinone C–H Alkylations via Oxidative Radical Processes
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Li, Longji; Yang, Qi; Jia, Zongbin; Luo, Sanzhong: Organocatalytic Electrochemical C–H Lactonization of Aromatic Carboxylic Acids
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Levin, Vitalij V.; Agababyan, Daniil P.; Struchkova, Marina I.; Dilman, Alexander D.: Dimerization of Benzyl and Allyl Halides via Photoredox-Mediated Disproportionation of Organozinc Reagents
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Manick, Anne-Doriane; Tanaka, Hirotaka; Oisaki, Kounosuke; Kanai, Motomu: Organophotoredox/Copper Hybrid Catalysis for Regioselective Allylic­ Aminodecarboxylation of β,γ-Unsaturated Carboxylic Acids
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Egami, Hiromichi; Ito, Yuta; Ide, Takafumi; Masuda, Shuya; Hamashima, Yoshitaka: Simple Photo-Induced Trifluoromethylation of Aromatic Rings
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Gharpure, Santosh J.; Niranjana, P.; Porwal, Suheel K.: Cascade Radical Cyclization to Vinylogous Carbonates/Carbamates for the Synthesis of Oxa- and Aza-Angular Triquinanes: Diastereoselectivity Depends on the Ring Size of Radical Precursor
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Li, Cheng-Kun; Zhang, Dong-Liang; Olamiji, Ogundipe Olukayode; Zhang, Pei-Zhi; Shoberu, Adedamola; Zou, Jian-Ping; Zhang, Wei: Mn(OAc)3-Mediated Regioselective Radical Alkoxycarbonylation of Indoles, Pyrimidinones, and Pyridinones
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Deng, Weili; Li, Yajun; Li, You-Gui; Bao, Hongli: Iron-Catalyzed Carboiodination of Alkynes
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Zhao, Xinxin; Chen, Ming; Huang, Binbin; Yang, Chao; Gao, Yuan; Xia, Wujiong: Photoinduced Cross-Coupling of Amines with 1,2-Diiodobenzene and Its Application in the Synthesis of Carbazoles
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Luo, Kai; Zhang, Ling; Wei, Kai; Yang, Wen-Chao; Wu, Lei: Latent Radical Cleavage of α-Allenylic C–O Bonds: Potassium Persulfate Mediated Thiolation of Allenylphosphine Oxides
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Mei, Chong; Hu, Yixin; Lu, Wenjun: Visible-Light-Driven Oxidation of N-Alkylamides to Imides Using Oxone/H2O and Catalytic KBr
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Das, Dipendu; Khan, Hina P. A.; Chakraborty, Tushar Kanti: Ti(III)-Mediated Radical-Induced Approach to a Bicyclic δ-Lactone with a Bridgehead β-Hydroxy Group
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Fukuyama, Takahide; Bando, Takanobu; Ryu, Ilhyong: Electron-Transfer-Induced Intramolecular Heck Carbonylation Reactions Leading to Benzolactones and Benzolactams
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Baguia, Hajar; Deldaele, Christopher; Romero, Eugénie; Michelet, Bastien; Evano, Gwilherm: Copper-Catalyzed Photoinduced Radical Domino Cyclization of Ynamides and Cyanamides: A Unified Entry to Rosettacin, Luotonin A, and Deoxyvasicinone
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Issue 21/2017

Special Topic Cover Page
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Takenouchi, Yuta; Ito, Hajime: Copper(I)-Catalyzed Boryl Substitution of Allyl Aminals: Selective Synthesis of Linear γ-Aminoallylboronates
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Miura, Wataru; Hirano, Koji; Miura, Masahiro: Iridium-Catalyzed Site-Selective C–H Borylation of 2-Pyridones
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Jang, Won Jun; Han, Jung Tae; Yun, Jaesook: NHC-Copper-Catalyzed Tandem Hydrocupration and Allylation of Alkenyl Boronates
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Pinet, Sandra; Liautard, Virginie; Debiais, Mégane; Pucheault, Mathieu: Radical Metal-Free Borylation of Aryl Iodides
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Saito, Hayate; Nogi, Keisuke; Yorimitsu, Hideki: Palladium-Catalyzed Double Borylation of Diaryl Sulfoxides with Diboron
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Farre, Albert; Briggs, Rachel; Pubill-Ulldemolins, Cristina; Bonet, Amadeu: Developing a Bench-Scale Green Diboration Reaction toward Industrial Application
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Issue 20/2017

Special Topic Cover Page
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Couly, Florence; Dubouilh-Benard, Carole; Besson, Thierry; Fruit, Corinne: Late-Stage C–H Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one Backbone: Synthesis of an Array of Potential Kinase Inhibitors
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Sabat, Nazarii; Smoleń, Sabina; Nauš, Petr; Perlíková, Pavla; Cebová, Magdaléna; Poštová Slavětínská, Lenka; Hocek, Michal: Synthesis of 2,6-Substituted 7-(Het)aryl-7-deazapurine Nucleobases (2,4-Disubstituted 5-(Het)aryl-pyrrolo[2,3-d]pyrimidines)
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Skonieczny, Kamil; Jaźwiński, Jarosław; Gryko, Daniel T.: The Synthesis of Imidazo[1,2-f]phenanthridines, Phenanthro-[9,10-d]imidazoles, and Phenanthro[9′,10′:4,5]imidazo[1,2-f]-phenanthridines via Intramolecular Oxidative Aromatic Coupling
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Yu, Zhao; Bo, Tang; Aiying, Guan; Weiwei, Wang; Zhenhua, Zhang; Mingan, Wang: Synthesis and Fungicidal Activity of (E)-5-[1-(4-Phenyl-2-oxo-1-oxaspiro[4.5]dec-3-en-3-yl)ethylidene]-2-aminoimidazolin-4-one Derivatives
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Tokumaru, Kazuyuki; Bera, Kalisankar; Johnston, Jeffrey N.: 1,3,4-Oxadiazole and Heteroaromatic-Fused 1,2,4-Triazole Synthesis­ Using Diverted Umpolung Amide Synthesis
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Lessi, Marco; Panzetta, Gianmarco; Marianetti, Giulia; Bellina, Fabio: Improved Synthesis of Symmetrical 2,5-Diarylimidazoles by One-Pot Palladium-Catalyzed Direct Arylation Tailored on the Electronic Features of the Aryl Halide
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Zhang, Xiaojuan; Han, Xiuling; Hu, Zhiyong; Lu, Xiyan: Synthesis of Substituted Piperidines via Cationic Palladium(II)-Catalyzed Reductive Coupling of N-Tosyl-Tethered Alkynones
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Shang, Xiao-Jie; Liu, Zhong-Quan: A Catalyzed Aerobic Intramolecular C–O Bond Formation: Facile Access to Ring-Fused Dihydrobenzoxazine Derivatives
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Issue 18/2017

Special Topic Cover Page
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Abe, Takumi; Haruyama, Tomohiro; Yamada, Koji: C4 Pictet–Spengler Reactions for the Synthesis of Core Structures in Hyrtiazepine Alkaloids
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Pertschi, Romain; Miaskiewicz, Solène; Weibel, Jean-Marc; Pale, Patrick; Blanc, Aurélien: Gold(I)-Catalyzed Cascade: Synthesis of 2,5-Disubstituted Pyrroles from N-Sulfonyl-2-(1-ethoxypropargyl)azetidines through Cyclization/Nucleophilic Substitution/Elimination
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Cacchi, Sandro; Fabrizi, Giancarlo; Goggiamani, Antonella; Iazzetti, Antonia; Verdiglione, Rosanna: 2-(Aminomethyl)-3-arylindoles from 3-(o-Trifluoroacetamidoaryl)-1-propargylic Alcohols, Aryl Halides, and Amines: A Domino Palladium-Catalyzed Three-Component Approach
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Zheng, Min; Chen, Kai; Zhu, Shifa: One-Pot Synthesis of Indole Derivatives from the Reaction of Nitroalkynes and Alkynes via a Mercury-Carbene Intermediate
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Shimizu, Maki; Hayama, Noboru; Kimachi, Tetsutaro; Inamoto, Kiyofumi: Copper-Catalyzed Intramolecular C–H Amination: A New Entry to Substituted Xanthine Derivatives
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Opsomer, Tomas; Thomas, Joice; Dehaen, Wim: Chemoselectivity in the Synthesis of 1,2,3-Triazoles from Enolizable Ketones, Primary Alkylamines, and 4-Nitrophenyl Azide
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Fujita, Shoji; Shibuya, Masatoshi; Yamamoto, Yoshihiko: Intramolecular Hydroalkoxylation/Reduction and Hydroamination/Reduction of Unactivated Alkynes Using a Silane–Iodine Catalytic System
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Paul, Kartick; Jalal, Swapnadeep; Kundal, Sandip; Chakraborty, Baitan; Jana, Umasish: Iron-Catalyzed Intramolecular Alkyne–Carbonyl Metathesis: A New Cyclization Strategy for the Synthesis of Benzocarbazole and Azepino[1,2-a]indole Derivatives
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Li, Xue-Fei; Lin, Jin-Shun; Liu, Xin-Yuan: Catalytic Radical Intramolecular Aminoperfluoroalkylation and Aminodifluoromethylation of Unactivated Alkenes with Fluoro­alkylsulfonyl Chlorides
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Mullapudi, Venkannababu; Bhogade, Ravindra B.; Deshpande, Mukund V.; Ramana, Chepuri V.: Phenol Oxidative Dearomatization of Modified Nucleoside Templates: A Simple Access to the C7-Spiroannulated Octosyl Acid Framework
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Ghosh, Arun K.; Tomaine, Anthony J.; Cantwell, Kelsey E.: Lewis Acid Mediated Cyclizations: Diastereoselective Synthesis of Six- to Eight-Membered Substituted Cyclic Ethers
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Lee, Sang Eun; Lee, Seong Jong; Cheon, Cheol-Hong: Concise Total Syntheses of Paullone and Kenpaullone via Cyanide-Catalyzed Intramolecular Imino-Stetter Reaction
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Triandafillidi, Ierasia; Sideri, Ioanna K.; Tzaras, Dimitrios Ioannis; Spiliopoulou, Nikoleta; Kokotos, Christoforos G.: Green Organocatalytic Synthesis of Dihydrobenzofurans by Oxidation–Cyclization of Allylphenols
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Nayak, Sanatan; Prabagar, B.; Ghosh, Nayan; Mallick, Rajendra K.; Sahoo, Akhila K.: Ag(I)-Catalyzed Cycloisomerization and Cyclization of Ketene Aminals: Construction of Azepine and 1,2-Dihydropyridine Derivatives
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Nagamoto, Midori; Nishimura, Takahiro; Yorimitsu, Hideki: Iridium-Catalyzed Intramolecular Oxidative Cyclization of Alkenyl Amides and Alkenoic Acids
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Li, Dianjun; Li, Ying; Yu, Wei: tert-Butyl Hypochlorite Induced Cyclization of Ethyl 2-(N-Aryl­carbamoyl)-2-iminoacetates
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Li, Jie; Xiao, Jun-An; Zhao, Shu-Juan; Xiang, Hao-Yue; Yang, Hua: Facile Construction of Pyrrolo[1,2-a]indolenine Scaffold via Dia­stereoselective [3+2] Annulation of Donor–Acceptor Cyclopropane with Indolenine
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Issue 17/2017

Special Topic Cover Page
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Hammann, Jeffrey M.; Hofmayer, Maximilian S.; Lutter, Ferdinand H.; Thomas, Lucie; Knochel, Paul: Recent Advances in Cobalt-Catalyzed Csp2 and Csp3 Cross-Couplings
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Ferrand, Laura; Lyu, Ye; Rivera-Hernández, Alejandro; Fallon, Brendan J.; Amatore, Muriel; Aubert, Corinne; Petit, Marc: Hydroboration and Diboration of Internal Alkynes Catalyzed by a Well-Defined Low-Valent Cobalt Catalyst
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Joshi, Hemant; Ghosh, Subrata K.; Gladysz, John A.: Enantioselective Additions of Stabilized Carbanions to Imines Generated from α-Amido Sulfones By Using Lipophilic Salts of Chiral Tris(1,2-diphenylethylenediamine) Cobalt(III) Trications as Hydrogen Bond Donor Catalysts
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Suo, Jian-Feng; Zhao, Xue-Mei; Zhang, Kai-Xin; Zhou, Sheng-Li; Niu, Jun-Long; Song, Mao-Ping: Cobalt-Catalyzed Perfluoroalkylation of Quinoline Amides at the C5 Position
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Hofmayer, Maximilian S.; Hammann, Jeffrey M.; Lutter, Ferdinand H.; Knochel, Paul: Large-Scale Cobalt-Catalyzed Cross-Couplings of Functionalized Bench-Stable Arylzinc Pivalates with (Hetero)Aryl and Alkenyl Halides­
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Xu, Kun; Tan, Zhoumei; Zhang, Haonan; Zhang, Sheng: Cobalt-Catalyzed Monoselective ortho-C–H Ethylation of Carboxamides with Triethylaluminum
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Kalsi, Deepti; Barsu, Nagaraju; Dahiya, Pardeep; Sundararaju, Basker: C–H and N–H Bond Annulation of Benzamides with Isonitriles Catalyzed by Cobalt(III)
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Cabré, Albert; Verdaguer, Xavier; Riera, Antoni: Ethylene Glycol Assisted Intermolecular Pauson–Khand Reaction
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Jamieson, Megan L.; Brant, Nicola Z.; Brimble, Margaret A.; Furkert, Daniel P.: Remarkable Influence of Cobalt Catalysis on Epoxide Ring-Opening with Sulfoxonium Ylides
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Midya, Siba P.; Mondal, Akash; Begum, Ayesha; Balaraman, Ekambaram: A Simple Cobalt(II) Chloride Catalyzed N-Alkylation of Amines with Alcohols
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Issue 16/2017

Special Topic Cover Page
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Watabe, Yota; Kanazawa, Kohei; Fujita, Takeshi; Ichikawa, Junji: Nickel-Catalyzed Hydroalkenylation of Alkynes through C–F Bond Activation: Synthesis of 2-Fluoro-1,3-dienes
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Xiao, Jian; Wang, Ya-Wen; Peng, Yu: Nickel-Promoted Reductive Cyclization Cascade: A Short Synthesis of a New Aromatic Strigolactone Analogue
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Barday, Manuel; Janot, Christopher; Clare, Daniel; Carr-Knox, Caitlin; Higginson, Bradley; Ho, Kelvin Y. T.; Aïssa, Christophe: On the Regioselectivity of the Nickel-Catalyzed Insertion of Alkynes into the Carbon–Carbon Bond of Oxetan-3-one
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Sumida, Yuto; Sumida, Tomoe; Hosoya, Takamitsu: Nickel-Catalyzed Reductive Cross-Coupling of Aryl Triflates and Nonaflates with Alkyl Iodides
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Shi, Shicheng; Szostak, Michal: Nickel-Catalyzed Negishi Cross-Coupling of N-Acylsuccinimides: Stable, Amide-Based, Twist-Controlled Acyl-Transfer Reagents via N–C Activation
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Issue 13/2017

Special Topic Cover Page
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Parmeggiani, Camilla; Matassini, Camilla; Cardona, Francesca; Goti, Andrea: On the Oxidation of Hydroxylamines with o-Iodoxybenzoic Acid (IBX)
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Muñiz, Kilian; Fra, Laura: Enantioselective 4-Hydroxylation of Phenols under Chiral Organoiodine(I/III) Catalysis
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