Synthesis

Current Issue eFirst

Khatana, Anil Kumar; Singh, Vikram; Gupta, Manoj Kumar; Tiwari, Bhoopendra: A Highly Efficient NHC-Catalyzed Aerobic Oxidation of Aldehydes to Carboxylic Acids

• Full Text
• HTML
• PDF (192 kb)

Nocera, Giuseppe; Murphy, John A.: Ground State Cross-Coupling of Haloarenes with Arenes Initiated by Organic Electron Donors, Formed in situ: An Overview

• Full Text
• HTML
• PDF (247 kb)

Sperger, Theresa; Schoenebeck, Franziska: α-Arylation of Esters and Ketones Enabled by a Bench-Stable Pd(I) Dimer Catalyst

• Full Text
• HTML
• PDF (209 kb)

Maligres, Peter E.; Song, Zhiguo Jake; Strotman, Neil A.; Yin, Jinquin; Pei, Tao; Strotman, Hallena R.; Itoh, Tetsuji; Sherer, Edward C.; Humphrey, Guy R.: Synthesis of Fused Oxepane HIV Integrase Inhibitor MK-1376

• Full Text
• HTML
• PDF (296 kb)

Cole, Charles J. F.; Chi, Hyung Min; DeBacker, Kenneth C.; Snyder, Scott A.: Synthesis of Enhanced, Isolable Disulfanium Salts and their Application to Thiiranium-Promoted Polyene Cyclizations

• Full Text
• HTML
• PDF (212 kb)

Wang, Zheng; Ji, Hongtao; He, Wei-Min; Xiong, Yang; Zhang, Guozhu: Chromium-Catalyzed Asymmetric Dearomatization–Addition Reactions of Halomethyloxazoles and Indoles

• Full Text
• HTML
• PDF (195 kb)

Lindner, Marcin; Krasiński, Antoni; Jurczak, Janusz: Facile, Stereocontrolled Synthetic Route towards Bis-functionalised Pyrrolizidines

• Full Text
• HTML
• PDF (418 kb)

Oberg, Kevin M.; Cochran, Brian M.; Cook, Matthew J.; Rovis, Tomislav: The Catalytic Alkylative Desymmetrization of Anhydrides in a Formal Synthesis of Ionomycin

• Full Text
• HTML
• PDF (228 kb)

Pang, Jia Hao; Ong, Derek Yiren; Watanabe, Kohei; Takita, Ryo; Chiba, Shunsuke: Leaving Group Ability in Nucleophilic Aromatic Amination by Sodium Hydride–Lithium Iodide Composite

• Full Text
• HTML
• PDF (180 kb)

Zhang, Yongda; Lao, Kendricks S.; Sieber, Joshua D.; Xu, Yibo; Wu, Linglin; Wang, Xiao-Jun; Desrosiers, Jean-Nicolas; Lee, Heewon; Haddad, Nizar; Han, Zhengxu S.; Yee, Nathan K.; Song, Jinhua J.; Howell, Amy R.; Senanayake, Chris H.: Modular Dihydrobenzoazaphosphole Ligands for Suzuki–Miyaura Cross-Coupling

• Full Text
• HTML
• PDF (376 kb)

Liddon, John T. R.; Rossi-Ashton, James A.; Clarke, Aimee K.; Lynam, Jason M.; Taylor, Richard J. K.; Unsworth, William P.: Divergent Reactivity of Indole-Tethered Ynones with Silver(I) and Gold(I) Catalysts: A Combined Synthetic and Computational Study

• Full Text
• HTML
• PDF (229 kb)

Joshi, Madhur S.; Pigge, F. Christopher: Sequential Pyridine Dearomatization–Mizoroki–Heck Cyclization for the Construction of Fused (Dihydropyrido)isoindolinone Ring Systems

• Full Text
• HTML
• PDF (269 kb)

Spiliopoulou, Nikoleta; Constantinou, Constantinos T.; Triandafillidi, Ierasia; Kokotos, Christoforos G.: Synthetic Approaches to Acyl Hydrazides and Their Use as Synthons in Organic Synthesis

• Full Text
• HTML
• PDF (915 kb)

Wertjes, William; Ayers, Sloan; Gao, Qi; Simmons, Eric M.; Beutner, Gregory L.: A Divergent Nickel-Catalyzed Synthesis of Quinazolinediones and Benzoxazinone Imines

• Full Text
• HTML
• PDF (531 kb)

Verma, Saumya; Kumar, Puneet; Khatana, Anil K.; Chandra, Dinesh; Yadav, Ajay K.; Tiwari, Bhoopendra; Jat, Jawahar L.: Zinc(II)-Catalyzed Synthesis of Secondary Amides from Ketones via Beckmann Rearrangement Using Hydroxylamine-O-sulfonic Acid in Aqueous Media

• Full Text
• HTML
• PDF (186 kb)

Denizot, Natacha; Guillot, Régis; Kouklovsky, Cyrille; Vincent, Guillaume: N-Iodosuccinimide-Mediated Oxidative Coupling of Indoles and Phenols: A Synthetic Study toward the Benzofuroindoline Moiety of Bipleiophylline

• Full Text
• HTML
• PDF (376 kb)

Ziegler, Dorothée S.; Klier, Lydia; Müller, Nicolas; Karaghiosoff, Konstantin; Knochel, Paul: Directed Zincation or Magnesiation of 2- and 4-Pyrones and Their Derivatives

• Full Text
• HTML
• PDF (273 kb)

Garlets, Zachary J.; Wolfe, John P.: Asymmetric Synthesis of Six-Membered Cyclic Sulfamides via Palladium-Catalyzed Alkene Carboamination Reactions

• Full Text
• HTML
• PDF (222 kb)

Current Issue 08/2020

Connon, Robert; Carroll, Laura; Guiry, Patrick J.: A Base-Promoted One-Pot Asymmetric Friedel–Crafts Alkylation/Michael Addition of 4-Substituted Indoles

• Full Text
• HTML
• PDF (927 kb)

Yang, Yuzhong; Zhou, Liwei; Yang, Xiumei; Luo, Xiai; Deng, Guobo; Yang, Yuan; Liang, Yun: Synthesis of Phenanthrenes via Palladium-Catalyzed Three-Component Domino Reaction of Aryl Iodides, Internal Alkynes, and o-Bromobenzoic Acids

• Full Text
• HTML
• PDF (227 kb)

Henkel, Michael; Bach, Thorsten: Annulation of Indoles with 1,n-Dibromoalkanes by a Pd(II)-Catalyzed and Norbornene-Mediated Reaction Cascade

• Full Text
• HTML
• PDF (200 kb)

Shen, Zican; Li, Chen; Mercado, Brandon Q.; Ellman, Jonathan A.: Cobalt(III)-Catalyzed Diastereoselective Three-Component C–H Bond Addition to Butadiene and Activated Ketones

• Full Text
• HTML
• PDF (267 kb)

Lee, Sumin; Jang, Young Jin; Phipps, Erik J. T.; Lei, Honghui; Rovis, Tomislav: Rhodium(III)-Catalyzed Three-Component 1,2-Diamination of Unactivated Terminal Alkenes

• Full Text
• HTML
• PDF (662 kb)

Sun, Manman; Li, Jinshan; Chen, Weida; Wu, Haijian; Yang, Jianguo; Wang, Zhiming: Palladium-Catalyzed [4+2] Annulation of Aryl and Alkenyl Carboxamides with 1,3-Dienes via C–H Functionalization: Synthesis of 3,4-Dihydroisoquinolones and 5,6-Dihydropyridinones

• Full Text
• HTML
• PDF (339 kb)

Current Issue 23/2019

Special Topic Cover Page

• Full Text
• PDF (2080 kb)

Sutherland, Andrew: Radiohalogenation of Organic Compounds: Practical Considerations and Challenges for Molecular Imaging

• Full Text
• HTML
• PDF (330 kb)

Milicevic Sephton, Selena; Zhou, Xiaoyun; Thompson, Stephen; Aigbirhio, Franklin I.: Preparation of the Serotonin Transporter PET Radiotracer 2-({2-[(Dimethylamino)methyl]phenyl}thio)-5-[¹⁸F]fluoroaniline (4-[¹⁸F]ADAM): Probing Synthetic and Radiosynthetic Methods

• Full Text
• HTML
• PDF (219 kb)

Kitahara, Kazumasa; Mizutani, Haruna; Iwasa, Seiji; Shibatomi, Kazutaka: Asymmetric Synthesis of α-Chloro-α-halo Ketones by Decarboxylative Chlorination of α-Halo-β-ketocarboxylic Acids

• Full Text
• HTML
• PDF (226 kb)

Dubost, Emmanuelle; Babin, Victor; Benoist, Florian; Hébert, Alexandra; Pigrée, Gilbert; Bouillon, Jean-Philippe; Fabis, Frédéric; Cailly, Thomas: Improvements of C–H Radio-Iodination of N-Acylsulfonamides toward Implementation in Clinics

• Full Text
• HTML
• PDF (684 kb)

Thompson, Stephen; Lee, So Jeong; Jackson, Isaac M.; Ichiishi, Naoko; Brooks, Allen F.; Sanford, Melanie S.; Scott, Peter J. H.: Synthesis of [¹⁸F]-γ-Fluoro-α,β-unsaturated Esters and Ketones via Vinylogous ¹⁸F-Fluorination of α-Diazoacetates with [¹⁸F]AgF

• Full Text
• HTML
• PDF (449 kb)

Sarie, Jérôme C.; Neufeld, Jessica; Daniliuc, Constantin G.; Gilmour, Ryan: Willgerodt-Type Dichloro(aryl)-λ³-Iodanes: A Structural Study

• Full Text
• HTML
• PDF (3071 kb)

Current Issue 13/2019

Special Topic Cover Page

• Full Text
• PDF (1732 kb)

Podyacheva, Evgeniya; Afanasyev, Oleg I.; Tsygankov, Alexey A.; Makarova, Maria; Chusov, Denis: Hitchhiker’s Guide to Reductive Amination

• Full Text
• HTML
• PDF (1329 kb)

Lai, Wing In; Leung, Man Pan; Choy, Pui Ying; Kwong, Fuk Yee: Sterically Hindered Amination of Aryl Chlorides Catalyzed by a New Carbazolyl-Derived P,N-Ligand-Composed Palladium Complex

• Full Text
• HTML
• PDF (686 kb)

Purkait, Anisha; Jana, Chandan K.: N-Aminations of Benzylamines and Alicyclic Amines with Nitrosoarenes to Hydrazones and Hydrazides

• Full Text
• HTML
• PDF (339 kb)

Li, Quan-Zhe; Wang, Xun-Hui; Hou, Si-Hua; Ma, Yan-Yan; Zhao, Deng-Gao; Zhang, Shu-Yu; Bai, He-Yuan; Ding, Tong-Mei: Silver-Catalyzed para-Selective C–H Amination of 1-Naphthyl­amides with Azodicarboxylates at Room Temperature

• Full Text
• HTML
• PDF (202 kb)

Pratap, Ramendra; Yorimitsu, Hideki: Palladium-Catalyzed Amination of Aryl Sulfides and Sulfoxides with Azaarylamines of Poor Nucleophilicity

• Full Text
• HTML
• PDF (186 kb)

Zhou, Huan; Zhao, Wenlei; Zhang, Tao; Guo, Haodong; Huang, Haizhou; Chang, Mingxin: Enantioselective Synthesis of 2-Substituted Pyrrolidines via Intramolecular­ Reductive Amination

• Full Text
• HTML
• PDF (188 kb)

Current Issue 12/2019

Special Topic Cover Page

• Full Text
• PDF (1528 kb)

Zhou, Yongyun; Khan, Ruhima; Fan, Baomin; Xu, Lijin: Ruthenium-Catalyzed Selective Reduction of Carboxylic Esters and Carboxamides

• Full Text
• HTML
• PDF (508 kb)

Deshmukh, Dewal S.; Bhanage, Bhalchandra M.: Ruthenium-Catalyzed Annulation of N-Cbz Hydrazones via C–H/N–N Bond Activation for the Rapid Synthesis of Isoquinolines

• Full Text
• HTML
• PDF (445 kb)

Das, Riki; Khot, Nandkishor Prakash; Deshpande, Akanksha Santosh; Kapur, Manmohan: Ruthenium-Catalyzed Directed C(3)–H Olefination of N-Acetyl-1,2-dihydroisoquinolines: A Method to Achieve C3-Olefinated Isoquinolines

• Full Text
• HTML
• PDF (224 kb)

Bairy, Gurupada; Nandi, Arijit; Manna, Kartic; Jana, Ranjan: Ruthenium(II)-Catalyzed Migratory C–H Allylation/Hydroamination Cascade for the Synthesis of Rutaecarpine Analogues

• Full Text
• HTML
• PDF (323 kb)

Tran, Christine; Haddad, Mansour; Ratovelomanana-Vidal, Virginie: Ruthenium-Catalyzed [2+2+2] Cycloaddition of α,ω-Diynes and Selenocyanates: An Entry to Selenopyridine Derivatives

• Full Text
• HTML
• PDF (245 kb)

Kawano, Teruhiro; Watari, Ryo; Kayaki, Yoshihito; Ikariya, Takao: Catalytic Hydrogenation of Carboxamides with a Bifunctional Cp*Ru Catalyst Bearing an Imidazol-2-ylidene with a Protic Aminoethyl Side Chain

• Full Text
• HTML
• PDF (266 kb)

Current Issue 17/2018

Special Topic Cover Page

• Full Text
• PDF (950 kb)

Oh, Eun Hye; Kim, Hyun Jin; Han, Soo Bong: Recent Developments in Visible-Light-Catalyzed Multicomponent Trifluoromethylation of Unsaturated Carbon–Carbon Bonds

• Full Text
• HTML
• PDF (543 kb)

Zhou, Wen-Jun; Zhang, Yi-Han; Gui, Yong-Yuan; Sun, Liang; Yu, Da-Gang: Merging Transition-Metal Catalysis with Photoredox Catalysis: An Environmentally Friendly Strategy for C–H Functionalization

• Full Text
• HTML
• PDF (686 kb)

Du, Yuliu; Wei, Zheng; Wang, Ting: Visible-Light-Mediated Synthesis of Oxidized Amides via Organic Photoredox Catalysis

• Full Text
• HTML
• PDF (1150 kb)

An, Xiao-De; Yu, Shouyun: Photoredox-Catalyzed Radical Relay Reaction Toward Functionalized Vicinal Diamines

• Full Text
• HTML
• PDF (317 kb)

Voutyritsa, Errika; Nikitas, Nikolaos F.; Apostolopoulou, Mary K.; Gerogiannopoulou, Anna Dimitra D.; Kokotos, Christoforos G.: Photoorganocatalytic Atom Transfer Radical Addition of Bromoacetonitrile to Aliphatic Olefins

• Full Text
• HTML
• PDF (185 kb)

Otomura, Nobutaka; Okugawa, Yuto; Hirano, Koji; Miura, Masahiro: Bromine Cation Initiated vic-Diphosphination of Styrenes with Diphosphines under Photoredox Catalysis

• Full Text
• HTML
• PDF (210 kb)

Current Issue 16/2018

Special Topic Cover Page

• Full Text
• PDF (2431 kb)

Baumann, Andreas N.; Eisold, Michael; Music, Arif; Didier, Dorian: One-Pot Preparation of Stable Organoboronate Reagents for the Functionalization of Unsaturated Four- and Five-Membered Carbo­- and Heterocycles

• Full Text
• HTML
• PDF (264 kb)

Yamaguchi, Eiji; Kamito, Yuji; Matsuo, Kazuki; Ishihara, Jun; Itoh, Akichika: Photooxidative Keto-Trifluoromethylation of Styrenes by Means of an Anthraquinone-Based Organocatalyst

• Full Text
• HTML
• PDF (375 kb)

Chen, Yizhou; Wang, Shanlu; Zhao, Li; Rong, Chenyan; Liu, Tong; Sun, Han; Wang, Yuping; Zhang, Jian; Zhong, Guofu: A Metal-Free Synthesis of 3-Phenoxyimidazo Heterocycles by Catalytic Oxidative Cyclization of 2-Amino-azaarenes with Lignin Models

• Full Text
• HTML
• PDF (233 kb)

Suen, Linda M.; Wang, Cheng; Hunter, David N.; Mitchell, Helen J.; Converso, Antonella; ElMarrouni, Abdellatif: Synthesis of HIV NNRTI Doravirine Analogues via Visible-Light Photoredox Decarboxylative Cross-Coupling

• Full Text
• HTML
• PDF (324 kb)

Liu, Yang; Daka, Mario; Bandini, Marco: Regio- and Stereoselective Nickel-Catalyzed Coupling of Boronic Acids with Allenoates

• Full Text
• HTML
• PDF (231 kb)

Park, Jaerim; Song, Kwang Ho; Lee, Sunwoo: Palladium-Catalyzed Decarboxylative Coupling Reactions of Propiolic Acid Derivatives and Arylsulfonyl Hydrazide

• Full Text
• HTML
• PDF (201 kb)

Torregrosa, Robert R. P.; Mendis, Shehani N.; Davies, Alex; Tunge, Jon A.: Palladium-Catalyzed Decarboxylative Benzylation of Acetylides and Enolates

• Full Text
• HTML
• PDF (238 kb)

Li, Jing; Wang, Zhong-Xia: Nickel-Catalyzed Transformation of Aryl 2-Pyridyl Ethers via Cleavage of the Carbon–Oxygen Bond: Synthesis of Mono-α-arylated­ Ketones

• Full Text
• HTML
• PDF (213 kb)

De, Pinaki Bhusan; Pradhan, Sourav; Shah, Tariq A.; Punniyamurthy, Tharmalingam: Iodine-Mediated Intramolecular C–H Amination of Benzimidazoles: A Metal-Free Route to Dihydroimidazobenzimidazoles

• Full Text
• HTML
• PDF (216 kb)

Guan, Weiye; Liao, Jennie; Watson, Mary P.: Vinylation of Benzylic Amines via C–N Bond Functionalization of Benzylic Pyridinium Salts

• Full Text
• HTML
• PDF (204 kb)

Yin, Zhiping; Power, Dennis J.; Wang, Zechao; Stewart, Scott G.; Wu, Xiao-Feng: Synthesis of 1,3,4-Oxadiazoles via Annulation of Hydrazides and Benzene-1,3,5-triyl Triformate under Metal-Free Conditions

• Full Text
• HTML
• PDF (186 kb)

Current Issue 15/2018

Special Topic Cover Page

• Full Text
• PDF (2545 kb)

Zhang, Qi; Raveendra Babu, Kaki; Huang, Zhouliang; Song, Jinna; Bi, Xihe: Visible-Light-Induced Radical Polynitration of Arylboronic Acids: Synthesis of Polynitrophenols

• Full Text
• HTML
• PDF (213 kb)

Wu, Kui; Fang, Cheng; Kaur, Sarbjeet; Liu, Peng; Wang, Ting: Methylene Blue-Catalyzed Oxidative Cleavage of N-Carbonylated Indoles

• Full Text
• HTML
• PDF (699 kb)

Wang, Guang-Zu; Shang, Rui; Fu, Yao: Irradiation-Induced Palladium-Catalyzed Direct C–H Alkylation of Heteroarenes with Tertiary and Secondary Alkyl Bromides

• Full Text
• HTML
• PDF (375 kb)

Hamsath, Akil; Galloway, Jordan D.; Baxter, Ryan D.: Quinone C–H Alkylations via Oxidative Radical Processes

• Full Text
• HTML
• PDF (294 kb)

Li, Longji; Yang, Qi; Jia, Zongbin; Luo, Sanzhong: Organocatalytic Electrochemical C–H Lactonization of Aromatic Carboxylic Acids

• Full Text
• HTML
• PDF (187 kb)

Levin, Vitalij V.; Agababyan, Daniil P.; Struchkova, Marina I.; Dilman, Alexander D.: Dimerization of Benzyl and Allyl Halides via Photoredox-Mediated Disproportionation of Organozinc Reagents

• Full Text
• HTML
• PDF (193 kb)

Manick, Anne-Doriane; Tanaka, Hirotaka; Oisaki, Kounosuke; Kanai, Motomu: Organophotoredox/Copper Hybrid Catalysis for Regioselective Allylic­ Aminodecarboxylation of β,γ-Unsaturated Carboxylic Acids

• Full Text
• HTML
• PDF (277 kb)

Egami, Hiromichi; Ito, Yuta; Ide, Takafumi; Masuda, Shuya; Hamashima, Yoshitaka: Simple Photo-Induced Trifluoromethylation of Aromatic Rings

• Full Text
• HTML
• PDF (210 kb)

Gharpure, Santosh J.; Niranjana, P.; Porwal, Suheel K.: Cascade Radical Cyclization to Vinylogous Carbonates/Carbamates for the Synthesis of Oxa- and Aza-Angular Triquinanes: Diastereoselectivity Depends on the Ring Size of Radical Precursor

• Full Text
• HTML
• PDF (426 kb)

Li, Cheng-Kun; Zhang, Dong-Liang; Olamiji, Ogundipe Olukayode; Zhang, Pei-Zhi; Shoberu, Adedamola; Zou, Jian-Ping; Zhang, Wei: Mn(OAc)₃-Mediated Regioselective Radical Alkoxycarbonylation of Indoles, Pyrimidinones, and Pyridinones

• Full Text
• HTML
• PDF (193 kb)

Deng, Weili; Li, Yajun; Li, You-Gui; Bao, Hongli: Iron-Catalyzed Carboiodination of Alkynes

• Full Text
• HTML
• PDF (196 kb)

Zhao, Xinxin; Chen, Ming; Huang, Binbin; Yang, Chao; Gao, Yuan; Xia, Wujiong: Photoinduced Cross-Coupling of Amines with 1,2-Diiodobenzene and Its Application in the Synthesis of Carbazoles

• Full Text
• HTML
• PDF (366 kb)

Luo, Kai; Zhang, Ling; Wei, Kai; Yang, Wen-Chao; Wu, Lei: Latent Radical Cleavage of α-Allenylic C–O Bonds: Potassium Persulfate Mediated Thiolation of Allenylphosphine Oxides

• Full Text
• HTML
• PDF (275 kb)

Mei, Chong; Hu, Yixin; Lu, Wenjun: Visible-Light-Driven Oxidation of N-Alkylamides to Imides Using Oxone/H₂O and Catalytic KBr

• Full Text
• HTML
• PDF (201 kb)

Das, Dipendu; Khan, Hina P. A.; Chakraborty, Tushar Kanti: Ti(III)-Mediated Radical-Induced Approach to a Bicyclic δ-Lactone with a Bridgehead β-Hydroxy Group

• Full Text
• HTML
• PDF (255 kb)

Fukuyama, Takahide; Bando, Takanobu; Ryu, Ilhyong: Electron-Transfer-Induced Intramolecular Heck Carbonylation Reactions Leading to Benzolactones and Benzolactams

• Full Text
• HTML
• PDF (227 kb)

Baguia, Hajar; Deldaele, Christopher; Romero, Eugénie; Michelet, Bastien; Evano, Gwilherm: Copper-Catalyzed Photoinduced Radical Domino Cyclization of Ynamides and Cyanamides: A Unified Entry to Rosettacin, Luotonin A, and Deoxyvasicinone

• Full Text
• HTML
• PDF (278 kb)

Current Issue 21/2017

Special Topic Cover Page

• Full Text
• PDF (1675 kb)

Takenouchi, Yuta; Ito, Hajime: Copper(I)-Catalyzed Boryl Substitution of Allyl Aminals: Selective Synthesis of Linear γ-Aminoallylboronates

• Full Text
• HTML
• PDF (209 kb)

Miura, Wataru; Hirano, Koji; Miura, Masahiro: Iridium-Catalyzed Site-Selective C–H Borylation of 2-Pyridones

• Full Text
• HTML
• PDF (227 kb)

Jang, Won Jun; Han, Jung Tae; Yun, Jaesook: NHC-Copper-Catalyzed Tandem Hydrocupration and Allylation of Alkenyl Boronates

• Full Text
• HTML
• PDF (208 kb)

Pinet, Sandra; Liautard, Virginie; Debiais, Mégane; Pucheault, Mathieu: Radical Metal-Free Borylation of Aryl Iodides

• Full Text
• HTML
• PDF (232 kb)

Saito, Hayate; Nogi, Keisuke; Yorimitsu, Hideki: Palladium-Catalyzed Double Borylation of Diaryl Sulfoxides with Diboron

• Full Text
• HTML
• PDF (210 kb)

Farre, Albert; Briggs, Rachel; Pubill-Ulldemolins, Cristina; Bonet, Amadeu: Developing a Bench-Scale Green Diboration Reaction toward Industrial Application

• Full Text
• HTML
• PDF (825 kb)

Current Issue 20/2017

Special Topic Cover Page

• Full Text
• PDF (1315 kb)

Couly, Florence; Dubouilh-Benard, Carole; Besson, Thierry; Fruit, Corinne: Late-Stage C–H Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one Backbone: Synthesis of an Array of Potential Kinase Inhibitors

• Full Text
• HTML
• PDF (225 kb)

Sabat, Nazarii; Smoleń, Sabina; Nauš, Petr; Perlíková, Pavla; Cebová, Magdaléna; Poštová Slavětínská, Lenka; Hocek, Michal: Synthesis of 2,6-Substituted 7-(Het)aryl-7-deazapurine Nucleobases (2,4-Disubstituted 5-(Het)aryl-pyrrolo[2,3-d]pyrimidines)

• Full Text
• HTML
• PDF (400 kb)

Skonieczny, Kamil; Jaźwiński, Jarosław; Gryko, Daniel T.: The Synthesis of Imidazo[1,2-f]phenanthridines, Phenanthro-[9,10-d]imidazoles, and Phenanthro[9′,10′:4,5]imidazo[1,2-f]-phenanthridines via Intramolecular Oxidative Aromatic Coupling

• Full Text
• HTML
• PDF (561 kb)

Yu, Zhao; Bo, Tang; Aiying, Guan; Weiwei, Wang; Zhenhua, Zhang; Mingan, Wang: Synthesis and Fungicidal Activity of (E)-5-[1-(4-Phenyl-2-oxo-1-oxaspiro[4.5]dec-3-en-3-yl)ethylidene]-2-aminoimidazolin-4-one Derivatives

• Full Text
• HTML
• PDF (205 kb)

Tokumaru, Kazuyuki; Bera, Kalisankar; Johnston, Jeffrey N.: 1,3,4-Oxadiazole and Heteroaromatic-Fused 1,2,4-Triazole Synthesis­ Using Diverted Umpolung Amide Synthesis

• Full Text
• HTML
• PDF (196 kb)

Lessi, Marco; Panzetta, Gianmarco; Marianetti, Giulia; Bellina, Fabio: Improved Synthesis of Symmetrical 2,5-Diarylimidazoles by One-Pot Palladium-Catalyzed Direct Arylation Tailored on the Electronic Features of the Aryl Halide

• Full Text
• HTML
• PDF (342 kb)

Zhang, Xiaojuan; Han, Xiuling; Hu, Zhiyong; Lu, Xiyan: Synthesis of Substituted Piperidines via Cationic Palladium(II)-Catalyzed Reductive Coupling of N-Tosyl-Tethered Alkynones

• Full Text
• HTML
• PDF (185 kb)

Shang, Xiao-Jie; Liu, Zhong-Quan: A Catalyzed Aerobic Intramolecular C–O Bond Formation: Facile Access to Ring-Fused Dihydrobenzoxazine Derivatives

• Full Text
• HTML
• PDF (185 kb)

Current Issue 18/2017

Special Topic Cover Page

• Full Text
• PDF (4349 kb)

Abe, Takumi; Haruyama, Tomohiro; Yamada, Koji: C4 Pictet–Spengler Reactions for the Synthesis of Core Structures in Hyrtiazepine Alkaloids

• Full Text
• HTML
• PDF (273 kb)

Pertschi, Romain; Miaskiewicz, Solène; Weibel, Jean-Marc; Pale, Patrick; Blanc, Aurélien: Gold(I)-Catalyzed Cascade: Synthesis of 2,5-Disubstituted Pyrroles from N-Sulfonyl-2-(1-ethoxypropargyl)azetidines through Cyclization/Nucleophilic Substitution/Elimination

• Full Text
• HTML
• PDF (484 kb)

Cacchi, Sandro; Fabrizi, Giancarlo; Goggiamani, Antonella; Iazzetti, Antonia; Verdiglione, Rosanna: 2-(Aminomethyl)-3-arylindoles from 3-(o-Trifluoroacetamidoaryl)-1-propargylic Alcohols, Aryl Halides, and Amines: A Domino Palladium-Catalyzed Three-Component Approach

• Full Text
• HTML
• PDF (274 kb)

Zheng, Min; Chen, Kai; Zhu, Shifa: One-Pot Synthesis of Indole Derivatives from the Reaction of Nitroalkynes and Alkynes via a Mercury-Carbene Intermediate

• Full Text
• HTML
• PDF (237 kb)

Shimizu, Maki; Hayama, Noboru; Kimachi, Tetsutaro; Inamoto, Kiyofumi: Copper-Catalyzed Intramolecular C–H Amination: A New Entry to Substituted Xanthine Derivatives

• Full Text
• HTML
• PDF (195 kb)

Opsomer, Tomas; Thomas, Joice; Dehaen, Wim: Chemoselectivity in the Synthesis of 1,2,3-Triazoles from Enolizable Ketones, Primary Alkylamines, and 4-Nitrophenyl Azide

• Full Text
• HTML
• PDF (395 kb)

Fujita, Shoji; Shibuya, Masatoshi; Yamamoto, Yoshihiko: Intramolecular Hydroalkoxylation/Reduction and Hydroamination/Reduction of Unactivated Alkynes Using a Silane–Iodine Catalytic System

• Full Text
• HTML
• PDF (235 kb)

Paul, Kartick; Jalal, Swapnadeep; Kundal, Sandip; Chakraborty, Baitan; Jana, Umasish: Iron-Catalyzed Intramolecular Alkyne–Carbonyl Metathesis: A New Cyclization Strategy for the Synthesis of Benzocarbazole and Azepino[1,2-a]indole Derivatives

• Full Text
• HTML
• PDF (224 kb)

Li, Xue-Fei; Lin, Jin-Shun; Liu, Xin-Yuan: Catalytic Radical Intramolecular Aminoperfluoroalkylation and Aminodifluoromethylation of Unactivated Alkenes with Fluoro­alkylsulfonyl Chlorides

• Full Text
• HTML
• PDF (517 kb)

Mullapudi, Venkannababu; Bhogade, Ravindra B.; Deshpande, Mukund V.; Ramana, Chepuri V.: Phenol Oxidative Dearomatization of Modified Nucleoside Templates: A Simple Access to the C7-Spiroannulated Octosyl Acid Framework

• Full Text
• HTML
• PDF (216 kb)

Ghosh, Arun K.; Tomaine, Anthony J.; Cantwell, Kelsey E.: Lewis Acid Mediated Cyclizations: Diastereoselective Synthesis of Six- to Eight-Membered Substituted Cyclic Ethers

• Full Text
• HTML
• PDF (531 kb)

Lee, Sang Eun; Lee, Seong Jong; Cheon, Cheol-Hong: Concise Total Syntheses of Paullone and Kenpaullone via Cyanide-Catalyzed Intramolecular Imino-Stetter Reaction

• Full Text
• HTML
• PDF (220 kb)

Triandafillidi, Ierasia; Sideri, Ioanna K.; Tzaras, Dimitrios Ioannis; Spiliopoulou, Nikoleta; Kokotos, Christoforos G.: Green Organocatalytic Synthesis of Dihydrobenzofurans by Oxidation–Cyclization of Allylphenols

• Full Text
• HTML
• PDF (320 kb)

Nayak, Sanatan; Prabagar, B.; Ghosh, Nayan; Mallick, Rajendra K.; Sahoo, Akhila K.: Ag(I)-Catalyzed Cycloisomerization and Cyclization of Ketene Aminals: Construction of Azepine and 1,2-Dihydropyridine Derivatives

• Full Text
• HTML
• PDF (267 kb)

Nagamoto, Midori; Nishimura, Takahiro; Yorimitsu, Hideki: Iridium-Catalyzed Intramolecular Oxidative Cyclization of Alkenyl Amides and Alkenoic Acids

• Full Text
• HTML
• PDF (248 kb)

Li, Dianjun; Li, Ying; Yu, Wei: tert-Butyl Hypochlorite Induced Cyclization of Ethyl 2-(N-Aryl­carbamoyl)-2-iminoacetates

• Full Text
• HTML
• PDF (226 kb)

Li, Jie; Xiao, Jun-An; Zhao, Shu-Juan; Xiang, Hao-Yue; Yang, Hua: Facile Construction of Pyrrolo[1,2-a]indolenine Scaffold via Dia­stereoselective [3+2] Annulation of Donor–Acceptor Cyclopropane with Indolenine

• Full Text
• HTML
• PDF (358 kb)

Current Issue 17/2017

Special Topic Cover Page

• Full Text
• PDF (1040 kb)

Hammann, Jeffrey M.; Hofmayer, Maximilian S.; Lutter, Ferdinand H.; Thomas, Lucie; Knochel, Paul: Recent Advances in Cobalt-Catalyzed Csp² and Csp³ Cross-Couplings

• Full Text
• HTML
• PDF (447 kb)

Ferrand, Laura; Lyu, Ye; Rivera-Hernández, Alejandro; Fallon, Brendan J.; Amatore, Muriel; Aubert, Corinne; Petit, Marc: Hydroboration and Diboration of Internal Alkynes Catalyzed by a Well-Defined Low-Valent Cobalt Catalyst

• Full Text
• HTML
• PDF (229 kb)

Joshi, Hemant; Ghosh, Subrata K.; Gladysz, John A.: Enantioselective Additions of Stabilized Carbanions to Imines Generated from α-Amido Sulfones By Using Lipophilic Salts of Chiral Tris(1,2-diphenylethylenediamine) Cobalt(III) Trications as Hydrogen Bond Donor Catalysts

• Full Text
• HTML
• PDF (532 kb)

Suo, Jian-Feng; Zhao, Xue-Mei; Zhang, Kai-Xin; Zhou, Sheng-Li; Niu, Jun-Long; Song, Mao-Ping: Cobalt-Catalyzed Perfluoroalkylation of Quinoline Amides at the C5 Position

• Full Text
• HTML
• PDF (381 kb)

Hofmayer, Maximilian S.; Hammann, Jeffrey M.; Lutter, Ferdinand H.; Knochel, Paul: Large-Scale Cobalt-Catalyzed Cross-Couplings of Functionalized Bench-Stable Arylzinc Pivalates with (Hetero)Aryl and Alkenyl Halides­

• Full Text
• HTML
• PDF (202 kb)

Xu, Kun; Tan, Zhoumei; Zhang, Haonan; Zhang, Sheng: Cobalt-Catalyzed Monoselective ortho-C–H Ethylation of Carboxamides with Triethylaluminum

• Full Text
• HTML
• PDF (190 kb)

Kalsi, Deepti; Barsu, Nagaraju; Dahiya, Pardeep; Sundararaju, Basker: C–H and N–H Bond Annulation of Benzamides with Isonitriles Catalyzed by Cobalt(III)

• Full Text
• HTML
• PDF (220 kb)

Cabré, Albert; Verdaguer, Xavier; Riera, Antoni: Ethylene Glycol Assisted Intermolecular Pauson–Khand Reaction

• Full Text
• HTML
• PDF (203 kb)

Jamieson, Megan L.; Brant, Nicola Z.; Brimble, Margaret A.; Furkert, Daniel P.: Remarkable Influence of Cobalt Catalysis on Epoxide Ring-Opening with Sulfoxonium Ylides

• Full Text
• HTML
• PDF (190 kb)

Midya, Siba P.; Mondal, Akash; Begum, Ayesha; Balaraman, Ekambaram: A Simple Cobalt(II) Chloride Catalyzed N-Alkylation of Amines with Alcohols

• Full Text
• HTML
• PDF (185 kb)

Current Issue 16/2017

Special Topic Cover Page

• Full Text
• PDF (508 kb)

Watabe, Yota; Kanazawa, Kohei; Fujita, Takeshi; Ichikawa, Junji: Nickel-Catalyzed Hydroalkenylation of Alkynes through C–F Bond Activation: Synthesis of 2-Fluoro-1,3-dienes

• Full Text
• HTML
• PDF (357 kb)

Xiao, Jian; Wang, Ya-Wen; Peng, Yu: Nickel-Promoted Reductive Cyclization Cascade: A Short Synthesis of a New Aromatic Strigolactone Analogue

• Full Text
• HTML
• PDF (740 kb)

Barday, Manuel; Janot, Christopher; Clare, Daniel; Carr-Knox, Caitlin; Higginson, Bradley; Ho, Kelvin Y. T.; Aïssa, Christophe: On the Regioselectivity of the Nickel-Catalyzed Insertion of Alkynes into the Carbon–Carbon Bond of Oxetan-3-one

• Full Text
• HTML
• PDF (213 kb)

Sumida, Yuto; Sumida, Tomoe; Hosoya, Takamitsu: Nickel-Catalyzed Reductive Cross-Coupling of Aryl Triflates and Nonaflates with Alkyl Iodides

• Full Text
• HTML
• PDF (285 kb)

Shi, Shicheng; Szostak, Michal: Nickel-Catalyzed Negishi Cross-Coupling of N-Acylsuccinimides: Stable, Amide-Based, Twist-Controlled Acyl-Transfer Reagents via N–C Activation

• Full Text
• HTML
• PDF (684 kb)

Current Issue 13/2017

Special Topic Cover Page

• Full Text
• PDF (574 kb)

Parmeggiani, Camilla; Matassini, Camilla; Cardona, Francesca; Goti, Andrea: On the Oxidation of Hydroxylamines with o-Iodoxybenzoic Acid (IBX)

• Full Text
• HTML
• PDF (1437 kb)

Muñiz, Kilian; Fra, Laura: Enantioselective 4-Hydroxylation of Phenols under Chiral Organoiodine(I/III) Catalysis

• Full Text
• HTML
• PDF (365 kb)

Kiyokawa, Kensuke; Takemoto, Kenta; Yahata, Shunsuke; Kojima, Takumi; Minakata, Satoshi: Oxidative Cyclization of β,γ-Unsaturated Carboxylic Acids Using Hypervalent Iodine Reagents: An Efficient Synthesis of 4-Substituted Furan-2-ones

• Full Text
• HTML
• PDF (204 kb)

Fujita, Morifumi; Lee, Hee Jin; Ichihara, Chisaki; Sugimura, Takashi: E/Z-Selectivity Controlled by Participation of Internal Oxy Group During Electrophilic Substitution of Alk-1-enylboronate with Bis(2,4,6-trimethylpyridine)iodonium Salt

• Full Text
• HTML
• PDF (163 kb)

Li, Guangchen; Zhang-Negrerie, Daisy; Du, Yunfei: Synthesis of N-Substituted 2-Amino-3,4-diiodofurans from Allenes via NIS-Mediated Intramolecular Electrophilic Iodocyclization

• Full Text
• HTML
• PDF (353 kb)

Dagenais, Robin; Lauriers, Antoine Jobin-Des; Legault, Claude Y.: Iodine(III)-Mediated Oxidative Hydrolysis of Haloalkenes: Investigation of the Effect of Iodine(III) Reagents

• Full Text
• HTML
• PDF (182 kb)

Current Issue 17/2016

Shaw, Subrata; White, James D.: Asymmetric Catalysis with Iron–Salen Complexes

• Full Text
• HTML
• PDF (323 kb)

Liu, Cheng-Yuan; Chen, Ying-Ho; Chen, Chih-Hao; Yu, Ming-Shiuan; Tsai, Fu-Yu; Ong, Tiow-Gan: Selective C(8)–H Activation of Imidazopyridines Mediated by Cooperative Nickel–Aluminum Catalysis

• Full Text
• HTML
• PDF (219 kb)

Kumar, Ravindra; Tamai, Eri; Ohnishi, Akira; Nishimura, Akira; Hoshimoto, Yoichi; Ohashi, Masato; Ogoshi, Sensuke: Nickel-Catalyzed Enantioselective Synthesis of Cyclobutenes via [2+2] Cycloaddition of α,β-Unsaturated Carbonyls with 1,3-Enynes

• Full Text
• HTML
• PDF (223 kb)

Malineni, Jagadeesh; Jezorek, Ryan L.; Zhang, Na; Percec, Virgil: An Indefinitely Air-Stable σ-Ni^II Precatalyst for Quantitative Cross-Coupling of Unreactive Aryl Halides and Mesylates with Aryl Neopentylglycolboronates

• Full Text
• HTML
• PDF (1114 kb)

Malineni, Jagadeesh; Jezorek, Ryan L.; Zhang, Na; Percec, Virgil: Ni^IICl(1-Naphthyl)(PCy₃)₂, An Air-Stable σ-Ni^II Precatalyst for Quantitative Cross-Coupling of Aryl C–O Electrophiles with Aryl Neopentylglycolboronates

• Full Text
• HTML
• PDF (729 kb)

Moragas, Toni; Martin, Ruben: Nickel-Catalyzed Reductive Carboxylation of Cyclopropyl Motifs with Carbon Dioxide

• Full Text
• HTML
• PDF (1041 kb)

Sugiyama, Yu-ki; Heigozono, Shiori; Tamura, Kazuhiro; Okamoto, Sentaro: Iron-Catalyzed Reductive Metalation–Allylation and Metalative Cyclization of 2,3-Disubstituted Oxetanes and Their Stereoselectivity

• Full Text
• HTML
• PDF (203 kb)

Zhang, Qingchen; Wang, Xuan; Qian, Qun; Gong, Hegui: Nickel-Catalyzed Reductive Cross-Coupling of Benzyl Halides with Aryl Halides

• Full Text
• HTML
• PDF (191 kb)

Xi, Tuo; Chen, Xu; Zhang, Heyi; Lu, Zhan: Reductive Cyclization of 1,6- and 1,7-Enynes Catalyzed by Iron Complexes

• Full Text
• HTML
• PDF (203 kb)

Current Issue 16/2016

Cai, Pin-Wen; You, Zhi-Hao; Xie, Liang-Hui; Tan, Rui; Tong, Zhi-Ping; Liu, Yan-Kai: The Attractive Application of Lactol Chemistry: From Racemic Lactol to Natural Product Skeleton

• Full Text
• HTML
• PDF (891 kb)

Su, Lin; Xu, Ming-Hua: Asymmetric Reformatsky-Type Reaction of Isatin-Derived N-Sulfinyl Ketimines: Efficient and Practical Synthesis of Enantiopure Chiral 2-Oxoindolinyl-β^3,3-Amino Esters

• Full Text
• HTML
• PDF (906 kb)

Gao, Xing; Han, Jianwei; Wang, Limin: Chiral Iminophosphorane Organocatalyzed Asymmetric Sulfenyl­ation of 3-Substituted Oxindoles: Substrate-Interrelated Enantio­selectivities

• Full Text
• HTML
• PDF (216 kb)

Nishimura, Takahiro; Nagai, Tomotaka; Takechi, Ryosuke; Ebe, Yusuke: Rhodium-Catalyzed Enantioselective Addition of Tricyclopropylboroxin to N-Sulfonylimines

• Full Text
• HTML
• PDF (199 kb)

Chen, Shi; Mondal, Mukulesh; Ibrahim, Ahmad A.; Wheeler, Kraig A.; Kerrigan, Nessan J.: Asymmetric Synthesis of Dipropionate Derivatives through Catalytic Hydrogenation of Enantioenriched E-Ketene Heterodimers

• Full Text
• HTML
• PDF (218 kb)

Sun, Shutao; Liu, Lei: Catalytic Enantioselective Alkynylation of Tetrahydroisoquinoline-Based N-Acyl Hemiaminals

• Full Text
• HTML
• PDF (248 kb)

Feng, Yangyang; Huang, Ruofeng; Hu, Liangzhen; Xiong, Yan; Coeffard, Vincent: Chiral C₂-Symmetric Iodoarene-Catalyzed Asymmetric α-Oxidation of β-Keto Esters

• Full Text
• HTML
• PDF (226 kb)

Berti, Francesco; Favero, Lucilla; Pineschi, Mauro: Asymmetric Synthesis of Methylphenidate and Quinolizidinones by Addition of Aldehydes to Piperidine-Based Conjugated N-Acyl­iminium Ions

• Full Text
• HTML
• PDF (217 kb)

Dai, Wen; Mi, Yuan; Lv, Ying; Shang, Sensen; Li, Guosong; Chen, Guangwen; Gao, Shuang: Development of a Continuous-Flow Microreactor for Asymmetric Epoxidation of Electron-Deficient Olefins

• Full Text
• HTML
• PDF (1267 kb)

Salomó, Ernest; Orgué, Sílvia; Riera, Antoni; Verdaguer, Xavier: Efficient Preparation of (S)- and (R)-tert-Butylmethylphosphine–Borane: A Novel Entry to Important P-Stereogenic Ligands

• Full Text
• HTML
• PDF (195 kb)

Shibata, Takanori; Fukai, Miku; Sekine, Ryosuke; Hazra, Madhurima; Kanyiva, Kyalo Stephen: Enantioselective Synthesis of Planar-Chiral 1,n-Dioxa[n]paracyclophane-Based Phosphites and Their Application as Chiral Ligands

• Full Text
• HTML
• PDF (211 kb)

Vishwanath, Manjunatha; Prakash, Muthuraj; Vinayagam, Poopathy; Kesavan, Venkitasamy: Construction of Polycyclic Fused Pyrrolidines with Three Contiguous Stereocenters via Michael Addition of Vinylmalononitriles to Nitrostyrenes­ Using l-Proline-Derived Thiourea

• Full Text
• HTML
• PDF (198 kb)

Current Issue 12/2016

Wildermuth, Raphael; Speck, Klaus; Magauer, Thomas: Gold(I)-Catalyzed Enyne Cyclizations: Studies Toward the Total Synthesis of (+)-Aureol

• Full Text
• HTML
• PDF (262 kb)

Shi, Shicheng; Lalancette, Roger; Szostak, Michal: Cyclization of Imides to 2-Azabicycles via Aminoketyl Radicals by Using Samarium(II) Iodide–Water: Reaction Development, Synthetic Scope, and Mechanistic Studies

• Full Text
• HTML
• PDF (1362 kb)

Sugimoto, Kenji; Hoshiba, Yuya; Tsuge, Kiyoshi; Matsuya, Yuji: Synthesis of Substituted Pyrrolo[2,1-a]isoquinolines by Gold-Catalyzed Domino Cyclization of Alkynyl Iminoesters

• Full Text
• HTML
• PDF (1173 kb)

Shirke, Rajendra P.; Reddy, Virsinha; Anand, R. Vijaya; Ramasastry, S. S. V.: Furans to Benzofurans: Intramolecular Cross-Benzoin Reactions Catalysed by N-Heterocyclic Carbenes

• Full Text
• HTML
• PDF (1183 kb)

Gandeepan, Parthasarathy; Rajamalli, Pachaiyappan; Cheng, Chien-Hong: Palladium-Catalyzed C–H Activation and Cyclization of Anilides with 2-Iodoacetates and 2-Iodobenzoates: An Efficient Method toward Oxindoles and Phenanthridones

• Full Text
• HTML
• PDF (324 kb)

Malkina, Anastasiya G.; Stepanov, Anton V.; Sobenina, Lyubov N.; Shemyakina, Olesya A.; Ushakov, Igor A.; Smirnov, Vladimir I.; Trofimov, Boris A.: Organocatalyzed Microwave-Assisted Competing Cyclization of Cyanopropargylic Alcohols with Carboxylic Acids: 4-Cyano-3(2H)-furanones versus 4-Cyano-[(Z)-3-cyanomethylene]-2,3-dihydro­furans

• Full Text
• HTML
• PDF (913 kb)

Nambu, Hisanori; Ono, Naoki; Yakura, Takayuki: Acid-Catalyzed Ring-Opening Cyclization of Spirocyclopropanes for the Construction of a 2-Arylbenzofuran Skeleton: Total Synthesis of Cuspidan B

• Full Text
• HTML
• PDF (255 kb)

Parker, Patrick D.; Pierce, Joshua G.: Synthesis of 1,2,4-Oxadiazoles via DDQ-Mediated Oxidative Cyclization of Amidoximes

• Full Text
• HTML
• PDF (196 kb)

Cavitt, Marchello A.; France, Stefan: Aluminum(III)-Catalyzed, Formal Homo-Nazarov-Type Ring-Opening Cyclizations toward the Synthesis of Functionalized Tetrahydroindolizines

• Full Text
• HTML
• PDF (253 kb)

Ren, Zhi-Hui; Zhao, Mi-Na; Yi, Yukun; Wang, Yao-Yu; Guan, Zheng-Hui: Copper-Catalyzed Aerobic Oxidative Cyclization of Ketoxime Acetates with Pyridines for the Synthesis of Imidazo[1,2-a]pyridines

• Full Text
• HTML
• PDF (204 kb)

Morita, Nobuyoshi; Mashiko, Rie; Hakuta, Dai; Eguchi, Daisuke; Ban, Shintaro; Hashimoto, Yoshimitsu; Okamoto, Iwao; Tamura, Osamu: Gold-Catalyzed Dimeric Cyclization of Isoeugenol and Related 1-Phenylpropenes in Ionic Liquid: Environmentally Friendly and Stereoselective Synthesis of 1,2,3-Trisubstituted 2,3-Dihydro-1H-indenes

• Full Text
• HTML
• PDF (236 kb)

Yu, Mangfei; Zhang, Qian; Wang, Jia; Huang, Peng; Yan, Pengfei; Zhang, Rui; Dong, Dewen: Triflic Anhydride Mediated Ring-Opening/Recyclization Reaction of α-Carbamoyl α-Oximyl Cyclopropanes with DMF: Synthetic Route to 5-Aminoisoxazoles

• Full Text
• HTML
• PDF (255 kb)

Current Issue 11/2016

Li, Zhilong; Tong, Rongbiao: Asymmetric Total Syntheses of the trans-2-Aryl-6-alkyltetrahydropyrans Diospongin B and Parvistones D and E from a Common Precursor

• Full Text
• HTML
• PDF (1319 kb)

Kousara, Mohammad; Bideau, Franck Le; Ibrahim, Rama; Ferry, Angélique; Venot, Pierre-Etienne; Dejean, Camille; Raingeaud, Joël; Dubois, Joëlle; Retailleau, Pascal; Dumas, Françoise: Suberosanes as Potential Antitumor Agents: First Enantioselective Total Synthesis of (1S)-Suberosanone and Configurational Assignment of Suberosenol A

• Full Text
• HTML
• PDF (1245 kb)

Nakayama, Yasuaki; Maeda, Yuichiro; Hama, Naoto; Sato, Takaaki; Chida, Noritaka: Total Synthesis of (–)-Stemoamide by Sequential Overman/Claisen Rearrangement

• Full Text
• HTML
• PDF (210 kb)

García-Ruiz, Cristina; Cheng-Sánchez, Iván; Sarabia, Francisco: Synthesis of (–)- and (+)-Gummiferol via Asymmetric Synthesis of Glycidic Amides

• Full Text
• HTML
• PDF (324 kb)

Konda, Saidulu; Khatravath, Mahender; Mallurwar, Naveen Kumar; Rao, Pallavi; Sripelly, Shivashankar; Iqbal, Javed; Arya, Prabhat: Stereoselective Synthesis of the C27–C35 Eribulin Fragment and Its Utilization in Building Structurally Diverse Macrocycles

• Full Text
• HTML
• PDF (391 kb)

Ye, Jian-Liang; Liu, Yang; Zhang, Yu-Feng; Yang, Zhi-Ping; Huang, Pei-Qiang: Studies on the Second-Generation Approach to Loline Alkaloids: Synthesis of N-Bus-norloline through N-tert-Butanesulfinyl Imine Based Asymmetric Vinylogous Mannich Reaction

• Full Text
• HTML
• PDF (632 kb)

Yang, Xiaoyu; Yu, Biao: Synthesis of Landomycin D: Studies on the Saccharide Assembly

• Full Text
• HTML
• PDF (218 kb)

Hunter, Thomas J.; Wang, Yanping; Zheng, Jiamin; O’Doherty, George A.: Asymmetric Iterative Hydration of Polyene Strategy to Cryptocaryols A and B

• Full Text
• HTML
• PDF (267 kb)

Current Issue 19/2015

Liu, Le; Zhang-Negrerie, Daisy; Du, Yunfei; Zhao, Kang: Hypervalent Iodine Mediated C–C Double Bond Activation: A Cascade Access to α-Keto Diacetates from Readily Available Cinnamic Acids

• Full Text
• HTML
• PDF (234 kb)

Sun, Gui-Jun; Wang, Yong; Kang, Qiang: Palladium-Catalyzed Allylic Amination of Homoallylic Alcohols with Amines via Carbon–Carbon Bond Cleavage

• Full Text
• HTML
• PDF (160 kb)

Okuma, Kentaro; Horigami, Kenta; Nagahora, Noriyoshi; Shioji, Kosei: Enantioselective Synthesis of 4,4′-Biaryl-BINOLs from Arynes and β-Diketones

• Full Text
• HTML
• PDF (218 kb)

Aoyama, Tadashi; Hayakawa, Mamiko; Kubota, Sho; Ogawa, Sumire; Nakajima, Erika; Mitsuyama, Emi; Iwabuchi, Taku; Kaneko, Haruki; Obara, Rina; Takido, Toshio; Kodomari, Mitsuo; Ouchi, Akihiko: Simple Method for sp²–sp³ and sp³–sp³ Carbon–Carbon Bond Activation in 2-Substituted 1,3-Diketones

• Full Text
• HTML
• PDF (265 kb)

Choi, Jeongae; Jung, Hyunuk; Yeo, Jeong-Eun; Koo, Sangho: Synthesis of Tribenzotropone by Ring Expansion of Phenanthrene-9,10-dione

• Full Text
• HTML
• PDF (160 kb)

Shadrin, Ivan A.; Rzhevskii, Sergey A.; Rybakov, Victor B.; Babaev, Eugene V.: Sonogashira Reaction of the Indolizine Ring

• Full Text
• HTML
• PDF (450 kb)

Parida, Amarchand; Sharique, Mohd.; Kakde, Badrinath N.; Ghosh, Santanu; Bisai, Alakesh: Efficient Synthesis of 3-Alkynyl-2-(hydroxymethyl)cyclohex-2-en-1-ones by a Stork–Danheiser Sequence from Vinylogous Esters and Terminal Alkynes

• Full Text
• HTML
• PDF (189 kb)

Ou, Yang; Qin, Chong; Song, Song; Jiao, Ning: An Iron-Catalyzed Direct Approach to Amides from Benzyl Azides via C–C Bond Cleavage

• Full Text
• HTML
• PDF (879 kb)

Current Issue 18/2015

Luo, Guo-Ying; Wu, Hao; Tang, Yu; Li, Hui; Yeom, Hyun-Suk; Yang, Ka; Hsung, Richard P.: A Total Synthesis of (±)-Rhododaurichromanic Acid A via an Oxa-[3+3] Annulation of Resorcinols

• Full Text
• HTML
• PDF (219 kb)

Kumar, Raju Suresh; Almansour, Abdulrahman I.; Arumugam, Natarajan; Menéndez, J. Carlos; Osman, Hasnah; Kumar, Raju Ranjith: Dipolar Cycloaddition-Based Multicomponent Reactions in Ionic Liquids: A Green, Fully Stereoselective Synthesis of Novel Polycyclic Cage Systems with the Generation of Two New Azaheterocyclic Rings

• Full Text
• HTML
• PDF (936 kb)

Zhao, Yating; Huang, Binbin; Yang, Chao; Li, Bing; Xia, Wujiong: Metal-Free [3+2] Oxidative Coupling of Phenols with Alkenes: Synthesis of Dihydrobenzofurans

• Full Text
• HTML
• PDF (208 kb)

Cserép, Gergely B.; Demeter, Orsolya; Bätzner, Effi; Kállay, Mihály; Wagenknecht, Hans-Achim; Kele, Péter: Synthesis and Evaluation of Nicotinic Acid Derived Tetrazines for Bioorthogonal Labeling

• Full Text
• HTML
• PDF (319 kb)

Islam, Kobirul; Das, Deb K.; Akram, Ejaz; Khan, Abu T.: Exploration of C5–C6-Unsubstituted 1,4-Dihydropyridines for the Construction of exo-Hexahydro-1H-chromeno[3,4-h][1,6]naphthyridine-3-carboxylates Using a Stereoselective Povarov Reaction

• Full Text
• HTML
• PDF (971 kb)

Olson, Christopher A.; Shaner, Courtnay E.; Roche, Sydney C.; Ferrence, Gregory M.; Mitchell, T. Andrew: Hexahydro-1H-Isoindolinone-Like Scaffolds from Electronically Deactivated and Sterically Hindered Dienes: Synthesis in the Context­ of Muironolide A

• Full Text
• HTML
• PDF (1001 kb)

Högermeier, Jens; Trawny, Daniel; Zimmer, Reinhold; Reissig, Hans-Ulrich: Diels–Alder Reactions of 1,3-Dienes Incorporated into 8-Oxa- and 8-Thiabicyclo[3.2.1]octane Skeletons: A Convenient Access to Complex Tri- and Tetracyclic Compounds

• Full Text
• HTML
• PDF (807 kb)

Lopchuk, Justin M.; Song, Mia; Butler, Blythe; Gribble, Gordon W.: Synthesis of Heteroaryl-Substituted Pyrroles via the 1,3-Dipolar Cycloaddition of Unsymmetrical Münchnones and Nitrovinylheterocycles

• Full Text
• HTML
• PDF (180 kb)

Ribeiro Laia, Fernanda M.; Pinho e Melo, Teresa M. V. D.: Synthesis and Reactivity of Aziridines with Internal Dipolarophiles: An Approach to 1,4-Dihydrochromeno[4,3-b]pyrroles and 3-Methylenechromano[4,3-b]pyrroles

• Full Text
• HTML
• PDF (349 kb)

Miller, Daniel K.; Bailey, Christopher A.; Sammelson, Robert E.: Synthesis of Isoxazolines and Isoxazoles Inspired by Fipronil

• Full Text
• HTML
• PDF (210 kb)

Pop, Lidia; Golban, Mirabela Ligia; Hădade, Niculina D.; Socaci, Crina; Grosu, Ion: CuAAC Synthesis of Tetragonal Building Blocks Decorated with Nucleobases

• Full Text
• HTML
• PDF (201 kb)

Kratzer, Philipp; Gerster, Holger; Maas, Gerhard: Cycloaddition Reactions of Propyne Iminium Salts and Enol Ethers

• Full Text
• HTML
• PDF (397 kb)

Yamaoka, Yousuke; Taniguchi, Marie; Yamada, Ken-ichi; Takasu, Kiyosei: Asymmetric Total Synthesis of Tylophorine through a Formal [2+2] Cycloaddition Followed by Migrative Ring Opening of a Cyclobutane

• Full Text
• HTML
• PDF (209 kb)

Seck, Insa; Fall, Alioune; Lago, Carmen; Sène, Massène; Gaye, Mohamed; Seck, Matar; Gómez, Generosa; Fall, Yagamare: Synthesis of a Cholesterol Side-Chain Triazole Analogue via ‘Click’ Chemistry

• Full Text
• HTML
• PDF (177 kb)

Current Issue 17/2015

Dobrydnev, Alexey V.; Popova, Maria V.; Saffon-Merceron, Nathalie; Listunov, Dymytrii; Volovenko, Yulian M.: Synthesis of the First Representatives of Spiro-1λ⁶-isothiazolidine-1,1,4-triones

• Full Text
• HTML
• PDF (271 kb)

Zhang, Shuang; Hu, Xiu-Qin; Wang, Zhu-Yin; Xu, Peng-Fei: Reactions of Sulfonium Salts with 2,3-Dioxopyrrolidine Derivatives: A Concise Synthesis of Spirocyclopropane

• Full Text
• HTML
• PDF (320 kb)

Peng, Jing; Ran, Guang-Yao; Du, Wei; Chen, Ying-Chun: Tertiary-Amine-Catalyzed Asymmetric [3+2] Annulations of Morita–Baylis–Hillman Carbonates of Isatins with Nitroolefins to Construct Spirooxindoles

• Full Text
• HTML
• PDF (881 kb)

Xiao, Fenfen; Zhang, Qing; Wang, Yunxia; Hu, Xiangdong: Synthetic Studies toward Bi-linderone Lead To Unexpected 6π-Electrocyclization Reactions: A Facile Construction of Highly Congested Spiro Compounds

• Full Text
• HTML
• PDF (1349 kb)

Cormier, Morgan; Chardon, Aurélien; Blanchet, Jérôme; Rouden, Jacques; Maddaluno, Jacques; De Paolis, Michaël: An Organocatalytic Access to Spiro[4.5]decanes and Spiro[4.6]undecanes Containing Aminolactones and 3-Aminopyrrolidines

• Full Text
• HTML
• PDF (165 kb)

Current Issue 16/2015

Philipps, Arne R.; Fritze, Lars; Erdmann, Nico; Enders, Dieter: An Asymmetric Organocatalytic Quadruple Domino Reaction Employing a Vinylogous Friedel–Crafts/Michael/Michael/Aldol Condensation Sequence

• HTML
• PDF (257 kb)

Garbarino, Silvia; Protti, Stefano; Basso, Andrea: Toward a Green Atom Economy: Development of a Sustainable Multicomponent Reaction

• Full Text
• HTML
• PDF (999 kb)

Firth, James D.; Zhang, Rong; Morgentin, Rémy; Guilleux, Rachel; Kalliokoski, Tuomo; Warriner, Stuart; Foster, Richard; Marsden, Stephen P.; Nelson, Adam: Exploitation of the Ugi–Joullié Reaction in the Synthesis of Libraries of Drug-Like Bicyclic Hydantoins

• Full Text
• HTML
• PDF (1829 kb)

Neochoritis, Constantinos G.; Zhang, Ji; Dömling, Alexander: Leuckart–Wallach Approach to Sugar Isocyanides and Its IMCRs

• Full Text
• HTML
• PDF (330 kb)

Xu, Shibo; Su, Shikuan; Zhang, Huiting; Tian, Lumin; Liang, Pengcheng; Chen, Jiawen; Zhang, Yuan; Li, Chunju; Jia, Xueshun; Li, Jian: Isocyanide-Based Multicomponent Reactions: Rapid Synthesis of a 5,5-Fused Bicyclic Skeleton from α,β-Unsaturated Ketones and Allenoates

• Full Text
• HTML
• PDF (579 kb)

Neo, Ana G.; Castellano, Teresa G.; Marcos, Carlos F.: Enol-Ugi Reaction of Hydroxycoumarins: Straightforward Synthesis of Amino Acid Derived Coumarin Enamines

• Full Text
• HTML
• PDF (274 kb)

Carboni, Aude; Dagousset, Guillaume; Magnier, Emmanuel; Masson, Géraldine: Three-Component Photoredox-Mediated Chloro-, Bromo-, or Iodotrifluoromethylation of Alkenes

• Full Text
• HTML
• PDF (1375 kb)

Qureshi, Zafar; Schlundt, Waldemar; Lautens, Mark: Introduction of Hindered Electrophiles via C–H Functionalization in a Palladium-Catalyzed Multicomponent Domino Reaction

• Full Text
• HTML
• PDF (232 kb)

Current Issue 15/2015

Du, Haiying; Rodriguez, Jean; Bugaut, Xavier; Constantieux, Thierry: Michael Addition Initiated Substrate- or Catalyst-Controlled Chemodivergent Three-Component Construction of Fused and Bridged Polycyclic Heterocycles

• Full Text
• HTML
• PDF (301 kb)

Vízcaíno-Milla, Pascuala; Sansano, José M.; Nájera, Carmen; Fiser, Béla; Gómez-Bengoa, Enrique: Primary Amine–2-Aminopyrimidine Chiral Organocatalysts for the Enantioselective Conjugate Addition of Branched Aldehydes to Maleimides

• Full Text
• HTML
• PDF (285 kb)

Fu, Niankai; Guo, Yinliang; Zhang, Long; Luo, Sanzhong: Chiral Primary Amine Catalyzed Asymmetric Tandem Reduction–Michael Addition–Protonation Reaction between Alkylidene Meldrum’s Acid and α-Substituted Vinyl Ketones

• Full Text
• HTML
• PDF (233 kb)

Rideau, Emeline; Mäsing, Florian; Fletcher, Stephen P.: Asymmetric Conjugate Addition of Alkylzirconocenes to Cyclopent-4-ene-1,3-dione Monoacetals

• Full Text
• HTML
• PDF (189 kb)

Tai, Hung-Che; Chavan, Arjun S.; Chuang, Shih-Ching: Nucleophilic Conjugate 1,5-Addition of Gilman Reagents to (E)-Hex-2-en-4-ynedioates: An Access to β(γ′)-Substituted Muconates

• Full Text
• HTML
• PDF (230 kb)

Roscales, Silvia; Sancho, Ainhoa; Csákÿ, Aurelio G.: Metal-Free Conjugate Addition of Alkenylboronic Acids to Enedicarbonyl Compounds towards the Synthesis of Pyridazine Derivatives

• Full Text
• HTML
• PDF (226 kb)

Peck, Cheryl L.; Calderone, Joseph A.; Santos, Webster L.: Copper(II)-Catalyzed β-Borylation of Acetylenic Esters in Water

• Full Text
• HTML
• PDF (214 kb)

Witte, Swjatoslaw N. R.; Voigt, Benjamin; Mahrwald, Rainer: Amine-Catalyzed Cascade Reactions of Unprotected and Unactivated­ Carbohydrates: Direct Access to C-Glycosides

• Full Text
• HTML
• PDF (204 kb)

Nishimura, Katsumi; Fukuyama, Naoshi; Yamashita, Mitsuaki; Sumiyoshi, Takaaki; Yamamoto, Yasutomo; Yamada, Ken-ichi; Tomioka, Kiyoshi: Cyclic Model for the Asymmetric Conjugate Addition of Organolithiums with Enoates

• Full Text
• HTML
• PDF (242 kb)

Sugiura, Masaharu; Ishikawa, Wakoto; Kuboyama, Yukinobu; Nakajima, Makoto: Conjugate Addition of Diboron Catalyzed by O-Monoacyltartaric Acids

• Full Text
• HTML
• PDF (190 kb)

Current Issue 17/2014

Mori, Yasuyuki; Mori, Takamichi; Onodera, Gen; Kimura, Masanari: Nickel-Catalyzed Multicomponent Coupling of Alkyne, Buta-1,3-diene, and Dimethylzinc under Carbon Dioxide

• Full Text
• HTML
• PDF (208 kb)

Strack, Martin; Metzler-Nolte, Nils; Albada, H. Bauke: Copper-Free Cleavage-Sonogashira Conjugation of Silylacetylene Immobilized Peptides

• Full Text
• HTML
• PDF (190 kb)

Ma, Wenbo; Ackermann, Lutz: Silver-Mediated Alkyne Annulations by C–H/P–H Functionalizations: Step-Economical Access to Benzophospholes

• Full Text
• HTML
• PDF (237 kb)

Park, Youngchul; Kang, Dongjin; Jeon, Woo Hyung; Ryu, Taekyu; Lee, Phil Ho: Synthesis of Ethyl Arylpropiolates through Palladium-Catalyzed Cross-Coupling­ Reactions of Aryl Iodides with In Situ Generated Lithium Tetrakis(ethoxycarbonylethynyl)indates

• Full Text
• HTML
• PDF (214 kb)

Current Issue 16/2014

Guo, Wei; Xia, Yuanzhi: THF Solvent as a Proton Shuttle in the AuCl₃-Catalyzed Cycloisomerization of a Bromoallenyl Ketone: A Mechanistic DFT Study

• Full Text
• HTML
• PDF (264 kb)

Lee, Ji Hyung; Jeong, Wook; Rhee, Young Ho: Unique Divergent Reactivity of Boc-Protected Homopropargylic Alkoxyalkylamines in the Gold(I)-Catalyzed Domino Catalytic Reactions: Application to the Formal Synthesis of (–)-Pseudodistomin B

• Full Text
• HTML
• PDF (206 kb)

Liu, Meng-Qi; Zhou, Ai-Hua; Jiang, Shuang; Wang, Jia-Qi; Ye, Long-Wu: Highly Diastereoselective Synthesis of Cyclopentenones via a One-Pot Gold Catalysis, Nazarov Cyclization and Alkylation Cascade

• Full Text
• HTML
• PDF (208 kb)

Wei, Fang; Wang, Xianghua; Peng, Shasha; Jia, Qiuhui; Jiang, Chao; Liu, Shili; Xu, Zhenghu: Direct Gold-Catalyzed Regioselective Tetrafunctionalization of Nonactivated Alkynes

• Full Text
• HTML
• PDF (239 kb)

Current Issue 14/2014

Zhou, Mingxin; Song, Qiuling: Synthesis of α-Ketoamides from Aryl Methyl Ketones and N,N-Dimethylformamide via Copper-Catalyzed Aerobic Oxidative Coupling

• Full Text
• HTML
• PDF (193 kb)

Belhomme, Marie-Charlotte; Dru, Delphine; Xiong, Heng-Ying; Cahard, Dominique; Besset, Tatiana; Poisson, Thomas; Pannecoucke, Xavier: Copper-Mediated Direct Functionalization of Unsaturated C–C Bonds with Ethyl Bromo(difluoro)acetate: A Straightforward Access to Highly Valuable Difluoromethylated Alkenes

• Full Text
• HTML
• PDF (295 kb)

Székely, Anna; Sinai, Ádám; Tóth, Edina B.; Novák, Zoltán: Utilization of a Copper on Iron Catalyst for the Synthesis of Biaryl Systems and Benzoxazines via Oxidative Arylation of Anilide Derivatives

• Full Text
• HTML
• PDF (241 kb)

Duong, Hung A.; Nguyen, Tuan Minh; Rosman, Nurul Zubaidah Binte; Tan, Lionel Jia Liang: Carboxylation of Organoboronic Esters with Potassium Methyl Carbonate under Copper Catalysis

• Full Text
• HTML
• PDF (184 kb)

Sahoo, Santosh K.; Jena, Himanshu Sekhar; Majji, Ganesh; Patel, Bhisma K.: Formation of Imidazolidine-benzothiazole–Copper(II) Complexes via a Copper-Mediated Room-Temperature C–H Activation of Imidazolidinecarbothioamides

• Full Text
• HTML
• PDF (1057 kb)

Zhao, Chenglong; Tan, Zhuozhen; Liang, Zhuye; Deng, Wei; Gong, Hegui: Nickel-Catalyzed Reductive Allylation of Ketones with Allylic Carbonates

• Full Text
• HTML
• PDF (234 kb)

Luo, Long; Zhang, Jian-Jian; Ling, Wei-Jian; Shao, Yong-Liang; Wang, Ya-Wen; Peng, Yu: Unified Synthesis of (–)-Folicanthine and (–)-Ditryptophenaline Enabled by a Room Temperature Nickel-Mediated Reductive Dimerization

• Full Text
• HTML
• PDF (362 kb)

Liu, Jiangguang; Yan, Jiajie; Qin, Dongguang; Cai, Qian: An Unexpected Inversion of Enantioselectivity in a Copper-Catalyzed Intramolecular­ Desymmetric Aryl C–N Coupling Reaction

• Full Text
• HTML
• PDF (209 kb)

Kageyuki, Ikuo; Yoshida, Hiroto; Takaki, Ken: Three-Component Carboboration of Alkenes under Copper Catalysis

• Full Text
• HTML
• PDF (228 kb)

Gurung, Santosh K.; Thapa, Surendra; Shrestha, Bijay; Giri, Ramesh: Copper-Catalyzed Cross-Coupling of Aryl- and Heteroaryltriethoxysilanes with Aryl and Heteroaryl Iodides and Bromides

• Full Text
• HTML
• PDF (227 kb)

Ambler, Brett R.; Peddi, Santosh; Altman, Ryan A.: Copper-Catalyzed Decarboxylative Trifluoromethylation of Propargyl Bromodifluoroacetates

• Full Text
• HTML
• PDF (233 kb)

Current Issue 10/2014

Tang, Weijun; Xiao, Jianliang: Asymmetric Hydrogenation of Imines via Metal–Organo Cooperative Catalysis

• Full Text
• HTML
• PDF (220 kb)

Deiana, Luca; Ghisu, Lorenza; Córdova, Oscar; Afewerki, Samson; Zhang, Renyun; Córdova, Armando: Efficient and Highly Enantioselective Aerobic Oxidation–Michael–Carbocyclization Cascade Transformations by Integrated Pd(0)-CPG Nanoparticle/Chiral Amine Relay Catalysis

• Full Text
• HTML
• PDF (227 kb)

Diezel, Sonja; Breit, Bernhard: Tandem Regioselective Rhodium-Catalyzed Hydroformylation–Enantioselective Aminocatalytic anti-Mannich Reaction

• Full Text
• HTML
• PDF (280 kb)

Gualandi, Andrea; Mengozzi, Luca; Wilson, Claire Margaret; Cozzi, Pier Giorgio: Synergistic Stereoselective Organocatalysis with Indium(III) Salts

• Full Text
• HTML
• PDF (238 kb)

Lee, Hwa-Jung; Shyam, Pranab Kumar; Yoon, Woojin; Yun, Hoseop; Jang, Hye-Young: Diastereo- and Enantioselective Synthesis of Hexasubstituted Cyclohexanes via a Metal–Organocatalytic Quadruple Cascade Sequence

• Full Text
• HTML
• PDF (232 kb)

Praveen, Chandrasekaran; Levêque, Sabine; Vitale, Maxime R.; Michelet, Véronique; Ratovelomanana-Vidal, Virginie: Synergistic Iron-and-Amine Catalysis in Carbocyclizations

• Full Text
• HTML
• PDF (204 kb)

Liu, Lu; Daka, Philias; Sarkisian, Ryan; Deng, Yongming; Wheeler, Kraig; Wang, Hong: Oxa-Diels–Alder Reaction of Isatins and Acyclic α,β-Unsaturated Methyl Ketones through Cooperative Dienamine and Metal Lewis Acid Catalysis

• Full Text
• HTML
• PDF (259 kb)

Jing, Changcheng; Xing, Dong; Qian, Yu; Hu, Wenhao: Rh₂(OAc)₄ and Chiral Phosphoric Acid Cocatalyzed Highly Diastereo- and Enantioselective Four-Component Reactions: Facile Synthesis of Chiral α,β-Diamino Acid Derivatives

• Full Text
• HTML
• PDF (220 kb)

Li, Nan; Chen, Dian-Feng; Wang, Pu-Sheng; Han, Zhi-Yong; Gong, Liu-Zhu: Relay Catalytic Cascade Hydrosiloxylation and Asymmetric Hetero-Diels–Alder Reaction

• Full Text
• HTML
• PDF (253 kb)

Yang, Jinming; Yu, Xingxin; Wu, Jie: A Facile Route to H-Pyrazolo[5,1-a]isoquinolines through a Multicomponent Reaction of 2-Alkynylbenzaldehyde, Sulfonylhydrazine, and Benzyne

• Full Text
• HTML
• PDF (229 kb)

Yoshida, Masanori; Masaki, Erika; Terumine, Tatsuaki; Hara, Shoji: Asymmetric α-Allylation of α-Branched Aldehydes with Allyl Alcohols by Synergistic Catalysis Using an Achiral Palladium Complex and a Chiral Primary Amino Acid

• Full Text
• HTML
• PDF (214 kb)

Current Issue 19/2013

Reboredo, Silvia; Vicario, Jose L.; Carrillo, Luisa; Reyes, Efraím; Uria, Uxue: A Simple Synthesis of Polysubstituted Pyrrolidines by an Organocatalytic Three-Component Approach Featuring a One-Pot Condensation and [3+2]-Cycloaddition Reaction in Aqueous Medium

• Full Text
• HTML
• PDF (245 kb)

Reitel, Kärt; Lippur, Kristin; Järving, Ivar; Kudrjašova, Marina; Lopp, Margus; Kanger, Tõnis: Asymmetric Aminocatalytic Michael Addition of Cyclopropane-Containing Aldehydes to Nitroalkenes

• Full Text
• HTML
• PDF (175 kb)

Shimada, Yoshiko; Hattori, Kasumi; Tada, Norihiro; Miura, Tsuyoshi; Itoh, Akichika: Facile Aerobic Photooxidation of Alcohols Using 2-Chloroanthraquinone under Visible Light Irradiation

• Full Text
• HTML
• PDF (187 kb)

Paria, Suva; Pirtsch, Michael; Kais, Viktor; Reiser, Oliver: Visible-Light-Induced Intermolecular Atom-Transfer Radical Addition of Benzyl Halides to Olefins: Facile Synthesis of Tetrahydroquinolines

• Full Text
• HTML
• PDF (244 kb)

Cismesia, Megan A.; Ischay, Michael A.; Yoon, Tehshik P.: Reductive Cyclizations of Nitroarenes to Hydroxamic Acids by Visible Light Photoredox Catalysis

• Full Text
• HTML
• PDF (209 kb)

Current Issue 15/2013

Mochizuki, Katsufumi; Sakai, Kazunori; Kochi, Takuya; Kakiuchi, Fumitoshi: Rhodium-Catalyzed Dimerization of Arylacetylenes and Addition of Malonates­ to 1,3-Enynes

• Full Text
• HTML
• PDF (179 kb)

Yamada, Yoichi M. A.; Ohta, Hidetoshi; Yuyama, Yoshinari; Uozumi, Yasuhiro: Polymeric Bimetallic Catalyst-Promoted In-Water Dehydrative Alkylation of Ammonia and Amines with Alcohols

• Full Text
• HTML
• PDF (339 kb)

Arnold, Jeffrey S.; Nguyen, Hien M.: Rhodium-Catalyzed Asymmetric Amination of Allylic Trichloroacetimidates

• Full Text
• HTML
• PDF (278 kb)

Ye, Ke-Yin; Zhao, Zhuo-An; Lai, Zeng-Wei; Dai, Li-Xin; You, Shu-Li: Highly Regioselective Allylic Substitution Reactions Catalyzed by an Air-Stable (π-Allyl)iridium Complex Derived from Dinaphthocyclooctatetraene and a Phosphoramidite Ligand

• Full Text
• HTML
• PDF (189 kb)

Obora, Yasushi; Sawaguchi, Takuya; Tsubakimoto, Keiko; Yoshida, Hiroshi; Ogawa, Shinji; Hatanaka, Shintaro: Iridium-Catalyzed Synthesis of ω-Hydroxy Homoallylic Alcohols

• Full Text
• HTML
• PDF (182 kb)

Apsunde, Tushar Dattu; Trudell, Mark L.: Microwave-Assisted Iridium-Catalyzed Synthesis of Nicotine and Anabasine Derivatives

• Full Text
• HTML
• PDF (184 kb)

Wang, Hui; Xu, Ming-Hua: Rhodium-Catalyzed Highly Enantioselective Addition of Arylboronic Acids to Cyclic Aldimines: Practical Asymmetric Synthesis of Cyclic Sulfamidates

• Full Text
• HTML
• PDF (253 kb)

Suzuki, Takeyuki; Ishizaka, Yuka; Ghozati, Kazem; Zhou, Da-Yang; Asano, Kaori; Sasai, Hiroaki: Enantioselective Multicatalytic Synthesis of α-Benzyl-β-hydroxyindan-1-ones

• Full Text
• HTML
• PDF (221 kb)

Liu, Wenting; Hong, Xiaohu; Xu, Bin: Rhodium-Catalyzed Oxidative Coupling of Aryl Hydrazones with Internal Alkynes: Efficient Synthesis of Multisubstituted Isoquinolines

• Full Text
• HTML
• PDF (345 kb)

Current Issue 12/2013

Fukata, Yukihiro; Miyaji, Ryota; Okamura, Takaaki; Asano, Keisuke; Matsubara, Seijiro: Asymmetric Cycloetherifications by Bifunctional Aminothiourea Catalysts: The Importance of Hydrogen Bonding

• Full Text
• HTML
• PDF (251 kb)

Jakab, Gergely; Hosseini, Abolfazl; Hausmann, Heike; Schreiner, Peter R.: Mild and Selective Organocatalytic Iodination of Activated Aromatic Compounds

• Full Text
• HTML
• PDF (259 kb)

Kumar, Vikas; Ray, Bidisha; Rathi, Preeti; Mukherjee, Santanu: Catalytic Asymmetric Direct Vinylogous Michael Addition of γ-Aryl-Substituted Deconjugated Butenolides to Nitroolefins and N-Phenylmaleimide

• Full Text
• HTML
• PDF (201 kb)

Duan, Shu-Wen; Liu, Yi-Yin; Ding, Wei; Li, Tian-Ren; Shi, De-Qing; Chen, Jia-Rong; Xiao, Wen-Jing: Chiral Squaramide Catalyzed Asymmetric Conjugate Additions of 3-Substituted Oxindoles to Vinylphosphonates

• Full Text
• HTML
• PDF (235 kb)

Chen, Guo-Ying; Lu, Yixin: Highly Enantioselective Michael Addition of α-Substituted Nitrophosphonates to a Vinyl Sulfone

• Full Text
• HTML
• PDF (229 kb)

Raimondi, Wilfried; Sanchez Duque, Maria del Mar; Goudedranche, Sébastien; Quintard, Adrien; Constantieux, Thierry; Bugaut, Xavier; Bonne, Damien; Rodriguez, Jean: Activation of 1,2- and 1,3-Ketoamides with Thiourea Organocatalyst for the Enantioselective Domino Synthesis of Functionalized Cyclohexanes

• Full Text
• HTML
• PDF (227 kb)

Current Issue 18/2012

Hassink, Matthew D.; Fox, Joseph M.: Functionalized Cyclopropenes and Methylenecyclopropenes from Dianions of 3-Hydroxymethylcyclopropenes

• Full Text
• HTML
• PDF (216 kb)

Rotstein, Benjamin H.; Yudin, Andrei K.: Aziridine-2-carboxaldehyde Dimers Undergo Homo-Ugi 4-Component-5-center Reactions

• Full Text
• HTML
• PDF (279 kb)

Walker, Daniel P.; Eklov, Brian M.; Bedore, Matthew W.: Practical Synthesis of 3-Oxa-6-azabicyclo[3.1.1]heptane Hydrotosylate; A Novel Morpholine-Based Building Block

• Full Text
• HTML
• PDF (191 kb)

Di Bussolo, Valeria; Frau, Ileana; Pineschi, Mauro; Crotti, Paolo: d-Allal- and d-Galactal-Derived Vinyl N-Mesylaziridines: Regio- and Stereoselectivity in Addition Reactions of O-, C-, N-, and S-Nucleophiles

• Full Text
• HTML
• PDF (265 kb)

Florio, Saverio: Unraveling the Synthetic Utility of the Regio- and Stereoselective Lithiation of Aziridines

• Full Text
• HTML
• PDF (352 kb)

Current Issue 16/2012

Lei, Ming; Tian, Wan; Hu, Ruijun; Li, Wei; Zhang, Hong: An Efficient Synthesis of 2-(Trifluoromethyl)-2H-[1,3]oxazino[2,3-a]isoquinolines via a Three-Component Cascade Approach Using a Continuous-Flow Microreactor

• Full Text
• HTML
• PDF (236 kb)

Rodriguez, Antonio M.; Juan, Alberto; Gómez, M. Victoria; Moreno, Andres; de la Hoz, Antonio: Continuous-Flow Microliter Microwave Irradiation in the Synthesis of Isoxazole Derivatives: An Optimization Procedure

• Full Text
• HTML
• PDF (180 kb)

Slocum, D. W.; Reinscheld, Thomas K.; Austin, Nick D.; Kusmic, Damir; Whitley, Paul E.: Near-Ambient Temperature Halogen–Lithium Exchange of p-Bromoanisole and Related Substrates: Flow/Batch Studies

• Full Text
• HTML
• PDF (191 kb)

Pagano, Nicholas; Heil, Marintha L.; Cosford, Nicholas D. P.: Automated Multistep Continuous Flow Synthesis of 2-(1H-Indol-3-yl)thiazole Derivatives

• Full Text
• HTML
• PDF (256 kb)

Ullah, Farman; Zang, Qin; Javed, Salim; Porubsky, Patrick; Neuenswander, Benjamin; Lushington, Gerald H.; Hanson, Paul R.; Organ, Michael G.: Synthesis of an Isoindoline-Annulated, Tricyclic Sultam Library via Microwave-Assisted, Continuous-Flow Organic Synthesis (MACOS)

• Full Text
• HTML
• PDF (241 kb)

Fukuyama, Takahide; Kajihara, Yoshito; Ryu, Ilhyong; Studer, Armido: Nitroxide-Mediated Polymerization of Styrene, Butyl Acrylate, or Methyl Methacrylate by Microflow Reactor Technology

• Full Text
• HTML
• PDF (187 kb)

Current Issue 14/2012

Wu, Xingxing; Zhang, Junliang: Y(OTf)₃-Catalyzed Diastereoselective [3+2] Cycloaddition of N-Tosyl­aziridines and Imines; Efficient Synthesis of Multisubstituted Imidazolidines

• Full Text
• HTML
• PDF (234 kb)

Yamazaki, Shoko; Fukushima, Yugo; Ukai, Tetsuma; Tatsumi, Kohei; Ogawa, Akiya: Lewis Acid Promoted Reactions of 1,1-Diarylallenes and Ketone Derivatives: Synthesis of Indenes by an Addition/Cyclization Reaction

• Full Text
• HTML
• PDF (303 kb)

Beckendorf, Stephan; Mancheño, Olga García: 'Click'-BINOLs: A New Class of Tunable Ligands for Asymmetric Catalysis

• Full Text
• HTML
• PDF (396 kb)

Auvil, Tyler J.; Mattson, Anita E.: Internal Lewis Acid Assisted Benzoic Acid Catalysis

• Full Text
• HTML
• PDF (230 kb)

Lanari, Daniela; Piermatti, Oriana; Pizzo, Ferdinando; Vaccaro, Luigi: Copper(II) Triflate–Sodium Dodecyl Sulfate Catalyzed Preparation of 1,2-Diphenyl-2,3-dihydro-4-pyridones in Aqueous Acidic Medium

• Full Text
• HTML
• PDF (175 kb)

Komai, Hirotomo; Yoshino, Tatsuhiko; Matsunaga, Shigeki; Kanai, Motomu: Lewis Acid Catalyzed Benzylic C–H Bond Functionalization of Azaarenes; Addition to Imines and Enones

• Full Text
• HTML
• PDF (249 kb)

Schweighauser, Luca; Bodoky, Ina; Kessler, Simon N.; Häussinger, Daniel; Wegner, Hermann A.: Bidentate Lewis Acid Catalyzed Inverse-Electron-Demand Diels–Alder Reaction for the Selective Functionalization of Aldehydes

• Full Text
• HTML
• PDF (204 kb)

Current Issue 12/2012

Shao, Jun; Huang, Xiaomei; Hong, Xiaohu; Liu, Bingxin; Xu, Bin: Synthesis of N-Alkyl-Substituted 4-Quinolones via Tandem Alkenyl and Aryl C–N Bond Formation

• Full Text
• HTML
• PDF (248 kb)

Kim, Ju Hyun; Chun, Yu Sung; Shin, Hyunik; Lee, Sang-gi: Tandem Transformations of Nitriles into N-Heterocyclic Compounds by Electrophilic Trapping of Blaise Reaction Intermediates

• Full Text
• HTML
• PDF (292 kb)

Batsomboon, Paratchata; Gold, Brian A.; Alabugin, Igor V.; Dudley, Gregory B.: Tandem Nucleophilic Addition/Fragmentation of Vinylogous Acyl Nonaflates for the Synthesis of Functionalized Alkynes, with New Mechanistic Insight

• Full Text
• HTML
• PDF (251 kb)

Kusakabe, Taichi; Sekiyama, Emika; Ishino, Yukari; Motodate, Satoshi; Kato, Shigeki; Mochida, Tomoyuki; Kato, Keisuke: Cyclization–Carbonylation–Cyclization Coupling Reactions of N-Propargylanilines and o-Alkynylphenols with Palladium(II)–Bisoxazoline Catalysts

• Full Text
• HTML
• PDF (257 kb)

Barriault, Louis; Denissova, Irina; Goulet, Nathalie: Mechanistic Investigation of the Domino Oxy-Cope/Ene/Claisen Reaction and Its Application to the Synthesis of Desdimethyl Ambliol B

• Full Text
• HTML
• PDF (247 kb)

Palanichamy, Kalanidhi; Suravarapu, Sankar R.; Kaliappan, Krishna P.: An Efficient Copper-Catalyzed Three-Component Synthesis of 3-C-Linked Glycosyl Iminocoumarins

• Full Text
• HTML
• PDF (244 kb)

Chen, Jian-Ming; Fang, Yin-Zhi; Wei, Zhong-lin; Liao, Wei-Wei: A Novel Multicomponent Tandem Phosphine-Catalyzed Umpolung Reaction: Facile Access to Highly Functionalized α-Aminonitriles

• Full Text
• HTML
• PDF (193 kb)

Davy, Jason A.; Moreau, Benoît; Wulff, Jeremy E.: Tandem Dihydroxylation, Hemiketalization and Conjugate Addition Leading to a Singly Anomeric Spiroketal

• Full Text
• HTML
• PDF (265 kb)

Fustero, Santos; Báez, Claribel; Sánchez-Roselló, María; Asensio, Amparo; Miro, Javier; del Pozo, Carlos: A New Tandem Cross Metathesis–Intramolecular Aza-Michael Reaction for the Synthesis of α,α-Difluorinated Lactams

• Full Text
• HTML
• PDF (266 kb)

Álvarez, Estela; Miguel, Delia; García-García, Patricia; Fernández-Rodríguez, Manuel A.; Rodríguez, Félix; Sanz, Roberto: Synthesis of 2-Indol-3-ylbenzofulvenes through a Tandem Reaction Catalyzed by Cationic Gold(I) Complexes

• Full Text
• HTML
• PDF (255 kb)

Rosa, David; Chtchemelinine, Andrei; Orellana, Arturo: Tandem Decarboxylative Allylation and Fragmentation of Allyl Benzocyclobutenyl Carbonates: Access to ortho-Functionalized Aryls from Aryl Bromides

• Full Text
• HTML
• PDF (215 kb)

Current Issue 10/2012

Sequeira, Fatima C.; Bovino, Michael T.; Chipre, Anthony J.; Chemler, Sherry R.: Multigram Synthesis of a Chiral Substituted Indoline Via Copper-Catalyzed Alkene Aminooxygenation

• Full Text
• HTML
• PDF (184 kb)

Park, Jin Kyoon; McQuade, D. Tyler: Chiral 6-NHC Ligand and Copper Complex: Properties, Application, and Mechanism

• Full Text
• HTML
• PDF (320 kb)

Laouiti, Anouar; Jouvin, Kévin; Bourdreux, Flavien; Rammah, Mohamed M.; Rammah, Mohamed B.; Evano, Gwilherm: Oxidative Alkynylation of Imines with Alkynylcopper Reagents: A Straightforward and Practical Entry to Ynimines

• Full Text
• HTML
• PDF (322 kb)

Zhao, Mi-Na; Liang, Hao; Ren, Zhi-Hui; Guan, Zheng-Hui: Copper-Catalyzed N–N Bond Formation by Homocoupling of Ketoximes via N–O Bond Cleavage: Facile, Mild, and Efficient Synthesis of Azines

• Full Text
• HTML
• PDF (217 kb)

Tsai, Wen-Ting; Lin, Yun-Yung; Wang, Yu-Jen; Lee, Chin-Fa: Microwave-Assisted Copper-Catalyzed Cross-Coupling Reaction of Alkynes with Aryl Iodides and Vinyl Halides

• Full Text
• HTML
• PDF (162 kb)

Crotti, Stefano; Di Bussolo, Valeria; Pineschi, Mauro: Regio- and Stereoselective Copper-Catalyzed Ring Opening of Dihetero­bicyclic Alkenes with Grignard Reagents

• Full Text
• HTML
• PDF (180 kb)

Oda, Yoshiro; Matsuyama, Naoto; Hirano, Koji; Satoh, Tetsuya; Miura, Masahiro: Dehydrogenative Synthesis of C3-Azolylindoles via Copper-Promoted Annulative Direct Coupling of o-Alkynylanilines

• Full Text
• HTML
• PDF (213 kb)

Chu, Lingling; Qing, Feng-Ling: Copper-Catalyzed Aerobic Oxidative Trifluoromethylation of H-Phospho­nates Using Trimethyl(trifluoromethyl)silane

• Full Text
• HTML
• PDF (174 kb)

Wang, Yi-Feng; Zhang, Feng-Lian; Chiba, Shunsuke: Copper-Catalyzed Aerobic Methyl/Methylene Oxygenation and C–H Formylation with a DABCO–DMSO System for the Synthesis of Carbonyl Indoles and Pyrroles

• Full Text
• HTML
• PDF (249 kb)

Nagao, Kazunori; Ohmiya, Hirohisa; Sawamura, Masaya: Functional Group Tolerable Synthesis of Allylsilanes through Copper-Catalyzed γ-Selective Allyl–Alkyl Coupling between Allylic Phosphates and Alkylboranes

• Full Text
• HTML
• PDF (226 kb)

Nakamura, Itaru; Kudo, Yu; Araki, Toshiharu; Zhang, Dong; Kwon, Eunsang; Terada, Masahiro: Copper-Catalyzed Skeletal Rearrangement of O-Propargylic Aryloximes into Four-Membered Cyclic Nitrones – Chirality Transfer and Mechanistic Insight

• Full Text
• HTML
• PDF (249 kb)

Zhao, Jiaji; Wang, Yong; Zhu, Qiang: Copper-Catalyzed Regioselective C–H Aerobic Oxidative Cycloetherification of o-Arylphenols Bearing an Additional Directing Group

• Full Text
• HTML
• PDF (197 kb)

Current Issue 08/2012

Brand, Jonathan P.; Waser, Jérôme: Synthesis of 1-[(Triisopropylsilyl)ethynyl]-1λ³,2-benziodoxol-3(1H)-one and Alkynylation of Indoles, Thiophenes, and Anilines

• Full Text
• HTML
• PDF (194 kb)

Kitamura, Tsugio; Tazawa, Yui; Morshed, Mohammad Hasan; Kobayashi, Soichi: Convenient Chlorination with Concentrated Hydrochloric Acid in the Presence of Iodosylbenzene

• Full Text
• HTML
• PDF (190 kb)

Yoshimura, Yuichi; Kan-no, Hiroya; Kiran, Y. B.; Natori, Yoshihiro; Saito, Yukako; Takahata, Hiroki: A New Route to N¹-Substituted Uracil Derivatives Using Hypervalent Iodine

• Full Text
• HTML
• PDF (242 kb)

Singh, Fateh V.; Wirth, Thomas: Hypervalent Iodine Mediated Oxidative Cyclization of o-Hydroxystilbenes into Benzo- and Naphthofurans

• Full Text
• HTML
• PDF (202 kb)

Rodríguez, Arantxa; Moran, Wesley J.: Chiral Aryl Iodide-Catalyzed Enantioselective α-Oxidation of Ketones

• Full Text
• HTML
• PDF (244 kb)

Dohi, Toshifumi; Nakae, Tomofumi; Takenaga, Naoko; Uchiyama, Teruyoshi; Fukushima, Kei-ichiro; Fujioka, Hiromichi; Kita, Yasuyuki: μ-Oxo-Bridged Hypervalent Iodine(III) Compound as an Extreme Oxidant for Aqueous Oxidations

• Full Text
• HTML
• PDF (240 kb)

Kong, Aidi; Blakey, Simon B.: Intramolecular Olefin Diamination for the Stereoselective Synthesis of 3-Aminopiperidines

• Full Text
• HTML
• PDF (255 kb)

Wardrop, Duncan J.; Yermolina, Maria V.; Bowen, Edward G.: Iodine(III)-Mediated Cyclization of Unsaturated O-Alkyl Hydroxamates: Silyl-Assisted Access to α-Vinyl and α-(2-Silylvinyl) Lactams

• Full Text
• HTML
• PDF (259 kb)

Current Issue 17/2011

van Delft, Pieter; van Schie, Evert; Meeuwenoord, Nico J.; Overkleeft, Herman S.; van der Marel, Gijsbert A.; Filippov, Dmitri V.: Oligonucleotide Conjugates by Means of Copper-Free Click Chemistry - Expanding the Repertoire of Strained Cyclooctyne Phosphoramidites

• Full Text
• HTML
• PDF (277 kb)

Walter, Miriam; Kottke, Tim; Weizel, Lilia; Schwed, J. Stephan; Stark, Holger: Synthesis of 1,2,3-Triazole Elements in Histamine H₃ Receptor Ligands

• Full Text
• HTML
• PDF (88 kb)

Aizpurua, Jesus M.; Sagartzazu-Aizpurua, Maialen; Azcune, Itxaso; Miranda, José I.; Monasterio, Zaira; García-Lecina, Eva; Fratila, Raluca M.: ‘Click’ Synthesis of Nonsymmetrical 4,4′-Bis(1,2,3-triazolium) Salts

• Full Text
• HTML
• PDF (122 kb)

Zang, Qin; Javed, Salim; Ullah, Farman; Zhou, Aihua; Knudtson, Christopher A.; Bi, Danse; Basha, Fatima Z.; Organ, Michael G.; Hanson, Paul R.: Application of a Double Aza-Michael Reaction in a ‘Click, Click, Cy-Click’ Strategy: From Bench to Flow

• Full Text
• HTML
• PDF (145 kb)

Current Issue 16/2011

Beladhria, Anissa; Beydoun, Kassem; Ammar, Hamed Ben; Salem, Ridha Ben; Doucet, Henri: Pd-Catalysed Direct 5-Arylation of 1-Methylpyrazole with Aryl Bromides

• Full Text
• HTML
• PDF (172 kb)

Ding, Zhenhua; Yoshikai, Naohiko: Cobalt-Catalyzed Alkenylation of Thiazoles with Alkynes via C-H Bond Functionalization

• Full Text
• HTML
• PDF (116 kb)

Ohno, Hiroaki; Yamamoto, Mio; Iuchi, Mutsumi; Fujii, Nobutaka; Tanaka, Tetsuaki: Palladium-Catalyzed Construction of Polycyclic Heterocycles by an Alkyne Insertion and Direct Arylation Cascade

• Full Text
• HTML
• PDF (207 kb)

Kubota, Asako; Sanford, Melanie S.: Palladium-Catalyzed Ligand-Directed Oxidative Functionalization of Cyclopropanes

• Full Text
• HTML
• PDF (183 kb)

Wang, Cong; Ge, Haibo: Palladium-Mediated Olefination of 2-(tert-Butyldimethylsilyl)pyridine by sp^³ C-H Activation

• Full Text
• HTML
• PDF (97 kb)

Lu, Zhiyao; Cui, Yuxin; Jia, Yanxing: Palladium-Catalyzed Domino Heck/C-H Activation/Intermolecular Direct Arylation Reactions

• Full Text
• HTML
• PDF (110 kb)

Ahlsten, Nanna; Bartoszewicz, Agnieszka; Agrawal, Santosh; Martín-Matute, Belén: A Facile Synthesis of α-Fluoro Ketones Catalyzed by [Cp*IrCl₂]₂

• Full Text
• HTML
• PDF (179 kb)

Current Issue 15/2011

Yin, Bin; Inagi, Shinsuke; Fuchigami, Toshio: Selective Electrochemical Fluorodesulfurization of Benzo- and Pyrido-Fused Oxazine Derivatives Using Ex-cell Halogen Mediators

• Full Text
• HTML
• PDF (138 kb)

Kutsumura, Noriki; Kubokawa, Keisuke; Saito, Takao: TBAF-Promoted Elimination of Vicinal Dibromides Having an Adjacent O-Functional Group: Syntheses of 2-Bromoalk-1-enes and Alkynes

• Full Text
• HTML
• PDF (125 kb)

Wang, Weibo; Xu, Bo; Hammond, Gerald B.: Synthesis of Fluorohydrins through Electrophilic Fluorination of Allyl Silanes

• Full Text
• HTML
• PDF (92 kb)

Tovar, John D.: Organic Halogenation Chemistry as a Vital Tool for the Construction of Functional π-Conjugated Materials

• Full Text
• HTML
• PDF (114 kb)

Chiappe, Cinzia; Sanzone, Angelo: Using the ‘Chemical Tunability’ of Ionic Liquids to Increase Sustainability in the Electrophilic Bromination of Unsaturated Compounds

• Full Text
• HTML
• PDF (91 kb)

Current Issue 14/2011

Salman, Ghazwan Ali; Ali, Asad; Hussain, Munawar; Khera, Rasheed Ahmad; Langer, Peter: Synthesis of Functionalized Benzofurans by a Double Heck Reaction of 2,3-Dibromofurans and Subsequent 6π-Electrocyclization/Dehydrogenation

• Full Text
• HTML
• PDF (122 kb)

Srivastava, Ajay Kumar; Song, Heebum; Park, Seung Bum: Diversity-Oriented Synthesis of Functionalized Polyheterocycles from Garner Aldehyde

• Full Text
• HTML
• PDF (158 kb)

Zhu, Mingzhao; Zheng, Nan: Photoinduced Cleavage of N-N Bonds of Aromatic Hydrazines and Hydrazides by Visible Light