Synthesis

Issue eFirst

Philkhana, Satish Chandra; Badmus, Fatimat O.; Dos Reis, Isaac C.; Kartika, Rendy: Recent Advancements in Pyrrole Synthesis

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Badart, Michael P.; Hawkins, Bill C.: Synthetic Strategies to Access Heteroatomic Spirocentres Embedded in Natural Products

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Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.: IntraMolecular Diels–Alder Reactions of Vinylarenes and Alkynyl Arenes (the IMDAV Reaction)

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Mamedov, Vakhid A.; Zhukova, Nataliya A.: Recent Developments Towards Synthesis of (Het)arylbenzimidazoles

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Cullen, Stephen T. J.; Friestad, Gregory K.: Synthesis of Chiral Amines by C–C Bond Formation with Photoredox Catalysis

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Issue Accepted Manuscripts

Bellina, Fabio: Real Metal-Free C-H Arylation of (Hetero)arenes: The Radical Way

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Issue 08/2021

Pellissier, Hélène: Enantioselective Indium-Catalyzed Transformations

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Issue 07/2021

Nguyen, Thanh T.; Wipf, Peter: Intramolecular Diels–Alder Reactions of Oxazoles, Imidazoles, and Thiazoles

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Issue 06/2021

Juhász, Kinga; Magyar, Ágnes; Hell, Zoltán: Transition-Metal-Catalyzed Cross-Coupling Reactions of Grignard Reagents

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Ung, Sosthène P.-M.; Mechrouk, Victoria Atica; Li, Chao-Jun: Shining Light on the Light-Bearing Element: A Brief Review of Photomediated C–H Phosphorylation Reactions

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Issue 05/2021

Bernardi, Eric; Colombo, Lino; Serra, Massimo: Recent Advances in One-Pot Enyne Metathesis Processes for the Preparation of Biologically and Medicinally Relevant Compounds

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Vijayan, Ajesh; Rao, Desaboini Nageswara; Radhakrishnan, K. V.; Lam, Patrick Y. S.; Das, Parthasarathi: Advances in Carbon–Element Bond Construction under Chan–Lam Cross-Coupling Conditions: A Second Decade

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Issue 04/2021

Huang, Jiuzhong; Yu, Fuchao: Recent Advances in Organic Synthesis Based on N,N-Dimethyl Enaminones

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Issue 03/2021

Moreira, Ryan; Noden, Michael; Taylor, Scott D.: Synthesis of Azido Acids and Their Application in the Preparation of Complex Peptides

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Pharande, Shrikant G.: Synthesis of Lactams via Isocyanide-Based Multicomponent Reactions

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Issue 02/2021

Ponra, Sudipta; Boudet, Bernard; Phansavath, Phannarath; Ratovelomanana-Vidal, Virginie: Recent Developments in Transition-Metal-Catalyzed Asymmetric Hydrogenation of Enamides

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Carceller-Ferrer, Laura; Blay, Gonzalo; Pedro, José R.; Vila, Carlos: Recent Advances in Catalytic Enantioselective Synthesis of Pyrazolones with a Tetrasubstituted Stereogenic Center at the 4-Position

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Issue 01/2021

Chen, Hui; Liu, Yahu A; Liao, Xuebin: Recent Progress in Radical Decarboxylative Functionalizations Enabled by Transition-Metal (Ni, Cu, Fe, Co or Cr) Catalysis

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Molina Betancourt, Ricardo; Echeverria, Pierre-Georges; Ayad, Tahar; Phansavath, Phannarath; Ratovelomanana-Vidal, Virginie: Recent Progress and Applications of Transition-Metal-Catalyzed Asymmetric Hydrogenation and Transfer Hydrogenation of Ketones and Imines through Dynamic Kinetic Resolution

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Issue 24/2020

Dimitrov, Ivaylo V.; Suonio, Elina E. K.: Syntheses of Analogues of Propofol: A Review

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Issue 23/2020

Zhu, Da-Liang; Young, David James; Li, Hong-Xi: Carbonyl-Photoredox/Metal Dual Catalysis: Applications in Organic Synthesis

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Markovič, Martin; Lopatka, Pavol; Gracza, Tibor; Koóš, Peter: Recent Applications of Continuous Flow in Homogeneous Palladium Catalysis

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Issue 22/2020

Grover, Nitika; Senge, Mathias O.: Synthetic Advances in the C–H Activation of Rigid Scaffold Molecules

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Issue 21/2020

Loska, Rafał; Mąkosza, Mieczysław: Introduction of Carbon Substituents into Nitroarenes via Nucleophilic Substitution of Hydrogen: New Developments

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Issue 20/2020

Chan, Chun-Ming; Chow, Yip-Chi; Yu, Wing-Yiu: Recent Advances in Photocatalytic C–N Bond Coupling Reactions

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Issue 19/2020

Christodoulou, Michael S.; Beccalli, Egle M.; Foschi, Francesca; Giofrè, Sabrina: Pd-Catalyzed Domino Reactions Involving Alkenes To Access Substituted Indole Derivatives

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Issue 18/2020

Li, Guangchen; Szostak, Michal: Non-Classical Amide Bond Formation: Transamidation and Amidation of Activated Amides and Esters by Selective N–C/O–C Cleavage

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Issue 17/2020

Lam, Heather; Lautens, Mark: Recent Advances in Transition-Metal-Catalyzed (4+3)-Cycloadditions

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Issue 16/2020

Idris, Muhammad Aliyu; Lee, Sunwoo: Recent Advances in Decarboxylative Reactions of Alkynoic Acids

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Issue 15/2020

Xie, Wen-Bin; Li, Zhi: Asymmetric Synthesis of Ethers by Catalytic Alkene Hydro­alkoxy­lation

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Issue 14/2020

Abdul-Rashed, Shukree; Holt, Connor; Frontier, Alison J.: Alkynyl Prins and Alkynyl Aza-Prins Annulations: Scope and Synthetic Applications

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Issue 13/2020

Teixeira, Wystan K. O.; de Albuquerque, Danilo Yano; Narayanaperumal, Senthil; Schwab, Ricardo S.: Recent Advances in the Synthesis of Enantiomerically Enriched Diaryl, Aryl Heteroaryl, and Diheteroaryl Alcohols through Addition of Organometallic Reagents to Carbonyl Compounds

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Issue 12/2020

McMurray, Lindsay; McGuire, Thomas M.; Howells, Rachel L.: Recent Advances in Photocatalytic Decarboxylative Coupling Reactions in Medicinal Chemistry

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Issue 11/2020

Xiao, Tiebo; Huang, Hongtai; Anand, Devireddy; Zhou, Lei: Iminyl-Radical-Triggered C–C Bond Cleavage of Cycloketone Oxime Derivatives: Generation of Distal Cyano-Substituted Alkyl Radicals and Their Functionalization

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Issue 10/2020

Laurita, Teresa; D’Orsi, Rosarita; Chiummiento, Lucia; Funicello, Maria; Lupattelli, Paolo: Recent Advances in Synthetic Strategies to 2,3-Dihydrobenzofurans

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Issue 09/2020

Časar, Zdenko: Synthetic Approaches to Contemporary Drugs that Contain the Cyclopropyl Moiety

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Issue 08/2020

Zambroń, Bartosz K.: Internal Chelation within Functionalized Organoindium Reagents: Prospects for Regio- and Stereocontrol in the Allylation, Propargylation and Allenylation of Carbonyl Compounds

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Issue 07/2020

DaBell, Peter; Thomas, Stephen P.: Iron Catalysis in Target Synthesis

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Issue 06/2020

Reznikov, Alexander N.; Klimochkin, Yuri N.: Recent Developments in Highly Stereoselective Michael Addition Reactions Catalyzed by Metal Complexes

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Issue 05/2020

Liu, Heng; Eisen, Moris S.: Organo-f-Complexes for Efficient and Selective Hydroborations

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Issue 02/2020

Kletskov, Alexey V.; Bumagin, Nikolay A.; Zubkov, Fedor I.; Grudinin, Dmitry G.; Potkin, Vladimir I.: Isothiazoles in the Design and Synthesis of Biologically Active Substances and Ligands for Metal Complexes

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Issue 01/2020

Sheng, Xia; Chen, Kaijun; Shi, Chengjin; Huang, Dayun: Recent Advances in Reactions of Propargylamines

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Issue 24/2019

Bao, Xiazhen; Li, Jun; Jiang, Wei; Huo, Congde: Radical-Mediated Difunctionalization of Styrenes

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Issue 23/2019

Dénès, Fabrice; Farard, Julien; Lebreton, Jacques: Synthesis of ¹³C-Labeled Steroids

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Issue 22/2019

Monika, Monika; Selvakumar, Sermadurai: Recent Developments in Direct C–H Functionalization of Quinoxalin-2(1H)-ones via Radical Addition Processes

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Issue 21/2019

Dank, Christian; Sanichar, Randy; Choo, Ken-Loon; Olsen, Madeline; Lautens, Mark: Recent Advances Towards Syntheses of Diterpenoid Alkaloids

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Issue 20/2019

Mittal, Rupali; Awasthi, Satish K.: Recent Advances in the Synthesis of 5-Substituted 1H-Tetrazoles: A Complete Survey (2013–2018)

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Issue 19/2019

Wu, Ronghai; Huang, Keke; Qiu, Guanyinsheng; Liu, Jin-Biao: Synthesis of Thioethers from Sulfonyl Chlorides, Sodium Sulfinates, and Sulfonyl Hydrazides

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Issue 18/2019

Sośnicki, Jacek G.; Idzik, Tomasz J.: Pyridones – Powerful Precursors for the Synthesis of Alkaloids, Their Derivatives, and Alkaloid-Inspired Compounds

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Issue 17/2019

Antermite, Daniele; Bull, James A.: Transition Metal-Catalyzed Directed C(sp³)–H Functionalization of Saturated Heterocycles

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Issue 16/2019

Wei, Yi; Zhou, Quan-Quan; Tan, Fen; Lu, Liang-Qiu; Xiao, Wen-Jing: Visible-Light-Driven Organic Photochemical Reactions in the Absence of External Photocatalysts

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Issue 15/2019

Le Bras, Jean; Muzart, Jacques: Carbonylated Indoles from Pd^II-Catalyzed Intermolecular Reactions of Indolyl Cores

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Issue 14/2019

Lim, Hyeonggeun; Seong, Sikwang; Han, Sunkyu: Syntheses of Post-Iboga Alkaloids

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Liu, Jian-Quan; Shatskiy, Andrey; Matsuura, Bryan S.; Kärkäs, Markus D.: Recent Advances in Photoredox Catalysis Enabled Functionalization of α-Amino Acids and Peptides: Concepts, Strategies and Mechanisms

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Issue 13/2019

Thoke, Mahesh Bhagwan; Kang, Qiang: Rhodium-Catalyzed Allylation Reactions

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Issue 12/2019

Stratakis, Manolis; Lykakis, Ioannis N.: Nanogold(0)-Catalyzed Addition of Heteroelement σ Linkages to Functional Groups

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Issue 11/2019

Ruan, Zhuwei; Li, Cheng; Shen, Defeng; Huang, Sha-Hua; Hong, Ran: FR901483: Synthetic Efficiency Remains a Challenge

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Issue 10/2019

Noack, Florian; Heinze, Robert C.; Heretsch, Philipp: Contemporary Synthetic Strategies towards Secosteroids, abeo-Steroids, and Related Triterpenes

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Yong, Xuefeng; Thurston, Ryan; Ho, Chun-Yu: Electronic Effects on Chiral NHC–Transition-Metal Catalysis

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Issue 09/2019

de Andrade, Vitor S.C.; de Mattos, Marcio C.S.: N-Halo Reagents: Modern Synthetic Approaches for Heterocyclic Synthesis

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De Risi, Carmela; Bortolini, Olga; Di Carmine, Graziano; Ragno, Daniele; Massi, Alessandro: Kinetic Resolution, Dynamic Kinetic Resolution and Asymmetric Desymmetrization by N-Heterocyclic Carbene Catalysis

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Issue 08/2019

Czerwiński, Paweł J.; Michalak, Michał: Synthetic Approaches to Chiral Non-C₂-symmetric N-Heterocyclic Carbene Precursors

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Engesser, Tobias; Brückner, Reinhard: Stereoselective Aldol Additions of Glycolic Acid and Its Derivatives

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Issue 07/2019

Macha, Lingamurthy; D’hooghe, Matthias; Ha, Hyun-Joon: Deployment of Aziridines for the Synthesis of Alkaloids and Their Derivatives

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Issue 06/2019

Liu, Xufang; Li, Bin; Liu, Qiang: Base-Metal-Catalyzed Olefin Isomerization Reactions

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Issue 05/2019

Kurandina, Daria; Chuentragool, Padon; Gevorgyan, Vladimir: Transition-Metal-Catalyzed Alkyl Heck-Type Reactions

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Issue 04/2019

Trushkov, Igor V.; Uchuskin, Maxim G.; Abaev, Vladimir T.; Serdyuk, Olga V.: Indolylvinyl Ketones: Building Blocks for the Synthesis of Natural Products and Bioactive Compounds

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Issue 03/2019

Pomarański, Piotr; Czarnocki, Zbigniew: Arylpyridines: A Review from Selective Synthesis to Atropisomerism

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Issue 02/2019

Banerjee, Arghya; Lei, Zhen; Ngai, Ming-Yu: Acyl Radical Chemistry via Visible-Light Photoredox Catalysis

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Esguerra, Kenneth Virgel N.; Lumb, Jean-Philip: Cu(III)-Mediated Aerobic Oxidations

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Issue 01/2019

Trost, Barry M.; Schultz, Johnathan E.: Palladium-Catalyzed Asymmetric Allylic Alkylation Strategies for the Synthesis of Acyclic Tetrasubstituted Stereocenters

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Issue 24/2018

O’Duill, Miriam L.; Engle, Keary M.: Protodepalladation as a Strategic Elementary Step in Catalysis

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Petsi, Marina; Zografos, Alexandros L.: Advances in Catalytic Aerobic Oxidations by Activation of Dioxygen-Monooxygenase Enzymes and Biomimetics

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Issue 23/2018

Grošelj, Uroš; Požgan, Franc; Štefane, Bogdan; Svete, Jurij: Copper-Catalyzed Azomethine Imine–Alkyne Cycloadditions (CuAIAC)

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El-Sawy, Eslam R.; Abdelwahab, Ahmed B.; Kirsch, Gilbert: Utilization of 1H-Indole-3-carboxaldehyde as a Precursor for the Synthesis of Bioactive Indole Alkaloids

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Issue 21/2018

Brahmachari, Goutam; Nayek, Nayana; Nurjamal, Khondekar; Karmakar, Indrajit; Begam, Sanchari: Triethylamine — A Versatile Organocatalyst in Organic Transformations: A Decade Update

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Li, Zhao-Kun; Jia, Xue-Shun; Yin, Liang: Recent Advances in Copper(II)-Mediated or -Catalyzed C–H Functionalization

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Issue 20/2018

Yavari, Issa; Khajeh-Khezri, Aliyeh: Recent Advances in the Synthesis of Hetero- and Carbocyclic Compounds­ and Complexes Based on Acenaphthylene-1,2-dione

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O’Neill, Matthew; Cornella, Josep: Retaining Alkyl Nucleophile Regiofidelity in Transition-Metal-Mediated Cross-Couplings to Aryl Electrophiles

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Issue 19/2018

Cheng-Sánchez, Iván; Sarabia, Francisco: Recent Advances in Total Synthesis via Metathesis Reactions

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Butenschön, Holger: Haloferrocenes: Syntheses and Selected Reactions

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Issue 18/2018

Giustiniano, Mariateresa; Moni, Lisa; Sangaletti, Luca; Pelliccia, Sveva; Basso, Andrea; Novellino, Ettore; Tron, Gian Cesare: Interrupted Ugi and Passerini Reactions: An Underexplored Treasure Island

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Kiss, Loránd; Kardos, Márton; Vass, Csaba; Fülöp, Ferenc: Application of Metathesis Reactions in the Synthesis and Transformations of Functionalized β-Amino Acid Derivatives

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Issue 17/2018

Oger, Camille; Cuyamendous, Claire; de la Torre, Aurélien; Candy, Mathieu; Guy, Alexandre; Bultel-Poncé, Valérie; Durand, Thierry; Galano, Jean-Marie: History of Chemical Routes towards Cyclic Non-Enzymatic Oxygenated Metabolites of Polyunsaturated Fatty Acids

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Blay, Gonzalo; Pedro, José R.; Sanz-Marco, Amparo: Conjugate Alkynylation of Electrophilic Double Bonds. From Regioselectivity to Enantioselectivity

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Issue 16/2018

Makarov, Anton S.; Uchuskin, Maxim G.; Trushkov, Igor V.: Furan Oxidation Reactions in the Total Synthesis of Natural Products

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Gilbert, Nicolas; Casault, Paméla; Ladouceur, François; Ricard, Simon; Daoust, Benoit: 1,2-Dihaloalkenes in Metal-Catalyzed Reactions

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Issue 15/2018

Li, Caifeng; Liu, Liu; Fu, Xuegang; Huang, Jianhui: Norbornene in Organic Synthesis

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Hoff, B. H.: Acetonitrile as a Building Block and Reactant

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Issue 14/2018

Boilevin, Jérémy M.; Reymond, Jean-Louis: Synthesis of Lipid-Linked Oligosaccharides (LLOs) and Their Phosphonate Analogues as Probes To Study Protein Glycosylation Enzymes

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Kumar, Inder; Kumar, Rakesh; Sharma, Upendra: Recent Advances in the Regioselective Synthesis of Indoles via C–H Activation/Functionalization

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Issue 13/2018

Larson, Gerald L.: Some Aspects of the Chemistry of Alkynylsilanes

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Issue 12/2018

Wang, Hui; Deng, Yu-Hua; Shao, Zhihui: An Update of N-Tosylhydrazones: Versatile Reagents for Metal-Catalyzed and Metal-Free Coupling Reactions

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Issue 11/2018

Khajuria, Rajni; Rasheed, Sk.; Khajuria, Chhavi; Kapoor, Kamal K.; Das, Parthasarathi: Recent Developments in the Synthesis of Pyrido[1,2-a]benzimidazoles

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Issue 10/2018

Sedgwick, Daniel M.; Grayson, Matthew N.; Fustero, Santos; Barrio, Pablo: Recent Developments and Applications of the Chiral Brønsted Acid Catalyzed Allylboration of Carbonyl Compounds

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Issue 09/2018

Fujihara, Tetsuaki; Tsuji, Yasushi: Cu-Catalyzed Borylative and Silylative Transformations of Allenes: Use of β-Functionalized Allyl Copper Intermediates in Organic Synthesis

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Burns, Jed M.; Krenske, Elizabeth H.; McGeary, Ross P.: Claisen Rearrangements of Benzyl Vinyl Ethers and Heterobenzyl Vinyl Ethers

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Issue 08/2018

Stateman, Leah M.; Nakafuku, Kohki M.; Nagib, David A.: Remote C–H Functionalization via Selective Hydrogen Atom Transfer

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Issue 07/2018

Balci, Metin: Acyl Azides: Versatile Compounds in the Synthesis of Various Heterocycles­

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Issue 06/2018

Mardjan, Muhammad Idham Darussalam; Parrain, Jean-Luc; Commeiras, Laurent: Strategies To Access γ-Hydroxy-γ-butyrolactams

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Issue 05/2018

Drouin, Myriam; Hamel, Jean-Denys; Paquin, Jean-François: Synthesis of Monofluoroalkenes: A Leap Forward

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Issue 04/2018

Kaga, Atsushi; Chiba, Shunsuke: Synthesis of Tricyclic Marine Alkaloids, Cylindricines, Lepadiformines, Fasicularin, and Polycitorols: A Recent Update

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Issue 03/2018

Dastan, Arif; Kilic, Haydar; Saracoglu, Nurullah: The Dibenzosuberenone Scaffold as a Privileged Substructure: From Synthesis to Application

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Chen, Long: Recent Advances in the Catalytic Asymmetric Construction of Phosphorus-Substituted Quaternary Carbon Stereocenters

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Issue 02/2018

Verbitskiy, Egor V.; Rusinov, Gennady L.; Chupakhin, Oleg N.; Charushin, Valery N.: Recent Advances in Direct C–H Functionalization of Pyrimidines

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Issue 01/2018

Dhokale, Ranjeet A.; Mhaske, Santosh B.: Transition-Metal-Catalyzed Reactions Involving Arynes

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Issue 24/2017

Li, Yajun; Ge, Liang; Muhammad, Munira Taj; Bao, Hongli: Recent Progress on Radical Decarboxylative Alkylation for Csp³–C Bond Formation

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Issue 23/2017

Cao, Chengyao Kimmy; Sheng, Jinyu; Chen, Chao: Cu-Catalyzed Cascade Annulation of Diaryliodonium Salts and Nitriles: Synthesis of Nitrogen-Containing Heterocycles

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Issue 22/2017

Zhang, Zhihong; Tong, Rongbiao: Synthetic Approaches to 2,6-trans-Tetrahydropyrans

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Issue 21/2017

Chen, Kai; Wang, Linghua; Meng, Ge; Li, Pengfei: Recent Advances in Transition-Metal-Free Aryl C–B Bond Formation

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Issue 20/2017

Puerto Galvis, Carlos E.; Kouznetsov, Vladimir V.: Recent Advances for the C–C and C–N Bond Formation in the Synthesis­ of 1-Phenethyl-tetrahydroisoquinoline, Aporphine, Homoaporphine­, and β-Carboline Alkaloids

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Issue 19/2017

Bian, Ming; Li, Lekai; Ding, Hanfeng: Recent Advances on the Application of Electrocyclic Reactions in Complex Natural Product Synthesis

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Issue 18/2017

Hervin, Vincent O.; Coutant, Eloi P.; Gagnot, Glwadys; Janin, Yves L.: Synthesis of α-Amino Esters via α-Nitro or α-Oxime Esters: A Review

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Issue 17/2017

Listratova, Anna V.; Voskressensky, Leonid G.: Recent Advances in the Synthesis of Hydrogenated Azocine-Containing­ Molecules

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Issue 16/2017

Taniguchi, Tsuyoshi: Recent Advances in Reactions of Heteroatom-Centered Radicals

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Issue 15/2017

Evano, Gwilherm; Lecomte, Morgan; Thilmany, Pierre; Theunissen, Cédric: Keteniminium Ions: Unique and Versatile Reactive Intermediates for Chemical Synthesis

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Issue 14/2017

Su, Bochao; Kinjo, Rei: Construction of Boron-Containing Aromatic Heterocycles

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Issue 13/2017

Sánchez-Roselló, María; Miró, Javier; del Pozo, Carlos: Cross-Metathesis/Intramolecular (Hetero-)Michael Addition: A Convenient Sequence for the Generation of Carbo- and Heterocycles

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Issue 12/2017

Gettys, Kristen E.; Ye, Zhishi; Dai, Mingji: Recent Advances in Piperazine Synthesis

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Issue 11/2017

Battistini, Lucia; Curti, Claudio; Rassu, Gloria; Sartori, Andrea; Zanardi, Franca: Enolizable Alkylidene Heterocyclic and Carbocyclic Carbonyl Systems­: Valuable Vinylogous Donor Substrates in Synthesis

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Issue 10/2017

Hachem, Ali; Grée, Danielle; Chandrasekhar, Srivari; Grée, René: Synthesis of Propargylic Fluorides toward Carbo- and Heterocycles with Mono- and gem-Difluorinated Side Chains

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Issue 09/2017

Fañanás-Mastral, Martín: Copper-Catalyzed Arylation with Diaryliodonium Salts

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Issue 08/2017

Gagnon, Alexandre; Dansereau, Julien; Le Roch, Adrien: Organobismuth Reagents: Synthesis, Properties and Applications in Organic Synthesis

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Issue 07/2017

Usman, Muhammad; Ren, Zhi-Hui; Wang, Yao-Yu; Guan, Zheng-Hui: Recent Developments in Cobalt Catalyzed Carbon–Carbon and Carbon–Heteroatom Bond Formation via C–H Bond Functionalization

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Issue 06/2017

Miyamura, Shin; Itami, Kenichiro; Yamaguchi, Junichiro: Syntheses of Biologically Active 2-Arylcyclopropylamines

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Issue 05/2017

Jiao, Yan-Xiao; Ma, Xiao-Pan; Su, Gui-Fa; Mo, Dong-Liang: Recent Advances in the Arylation and Alkenylation of N–O Bonds

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Issue 04/2017

Undheim, Kjell: Spirocyclic Orthoesters, Orthothioesters and Orthoaminals in the Synthesis and Structural Modification of Natural Products

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Issue 03/2017

Reyes, Efraím; Uria, Uxue; Carrillo, Luisa; Vicario, Jose L.: Enantioselective Cascade Reactions under N-Heterocyclic Carbene Catalysis

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Issue 24/2016

Sakhuja, Rajeev; Pericherla, Kasiviswanadharaju; Bajaj, Kiran; Khungar, Bharti; Kumar, Anil: Ytterbium Triflate Catalyzed Synthesis of Heterocycles

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Issue 23/2016

Gao, Yangguang; He, Xianran; Ding, Fei; Zhang, Yongmin: Recent Progress in Chemical Syntheses of Sphingosines and Phytosphingosines

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Issue 22/2016

Rossi, Renzo; Lessi, Marco; Manzini, Chiara; Marianetti, Giulia; Bellina, Fabio: Direct (Hetero)arylation Reactions of (Hetero)arenes as Tools for the Step- and Atom-Economical Synthesis of Biologically Active Unnatural Compounds Including Pharmaceutical Targets

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Issue 21/2016

Vincent-Rocan, Jean-François; Beauchemin, André M.: N-Isocyanates, N-Isothiocyanates and Their Masked/Blocked Derivatives: Synthesis and Reactivity

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Issue 20/2016

Littleson, Mairi M.; Russell, Claire J.; Frye, Elizabeth C.; Ling, Kenneth B.; Jamieson, Craig; Watson, Allan J. B.: Synthetic Approaches to Coronafacic Acid, Coronamic Acid, and Coronatine

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Issue 18/2016

Grange, Rebecca L.; Clizbe, Elizabeth A.; Evans, P. Andrew: Recent Developments in Asymmetric Allylic Amination Reactions

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Issue 17/2016

Gmach, Joanna; Joachimiak, Łukasz; Błażewska, Katarzyna M.: Aza-Michael Addition of Imidazole Analogues

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Issue 16/2016

Chen, Yantao: Recent Functionalizations of Primary Sulfonamides

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Issue 15/2016

Priyanka; Sharma, Rajesh Kumar; Katiyar, Diksha: Recent Advances in Transition-Metal-Catalyzed Synthesis of Coumarins

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Issue 13/2016

Liu, Nai-Wei; Liang, Shuai; Manolikakes, Georg: Recent Advances in the Synthesis of Sulfones

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Issue 12/2016

Nikolaev, Andrei; Orellana, Arturo: Transition-Metal-Catalyzed C–C and C–X Bond-Forming Reactions Using Cyclopropanols

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Issue 11/2016

Gehrtz, Paul H.; Hirschbeck, Vera; Ciszek, Benjamin; Fleischer, Ivana: Carbonylations of Alkenes in the Total Synthesis of Natural Compounds

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Issue 10/2016

Jones-Mensah, Ebenezer; Karki, Megha; Magolan, Jakob: Dimethyl Sulfoxide as a Synthon in Organic Chemistry

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Issue 09/2016

Rohokale, Rajendra S.; Kshirsagar, Umesh A.: Advanced Synthetic Strategies for Constructing Quinazolinone Scaffolds

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Issue 08/2016

Shintani, Ryo: Recent Progress in Copper-Catalyzed Asymmetric Allylic Substitution Reactions Using Organoboron Nucleophiles

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Issue 07/2016

Dryzhakov, Marian; Richmond, Edward; Moran, Joseph: Recent Advances in Direct Catalytic Dehydrative Substitution of Alcohols

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Issue 06/2016

Barniol-Xicota, Marta; Leiva, Rosana; Escolano, Carmen; Vázquez, Santiago: Syntheses of Cinacalcet: An Enantiopure Active Pharmaceutical Ingredient (API)

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Issue 05/2016

Voskressensky, Leonid G.; Golantsov, Nikita E.; Maharramov, Abel M.: Recent Advances in Bromination of Aromatic and Heteroaromatic Compounds

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Issue 04/2016

Röse, Philipp; Hilt, Gerhard: Cobalt-Catalysed Bond Formation Reactions; Part 2

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Issue 03/2016

Catti, Lorenzo; Zhang, Qi; Tiefenbacher, Konrad: Self-Assembled Supramolecular Structures as Catalysts for Reactions Involving Cationic Transition States

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Issue 02/2016

Whittaker, Rachel E.; Dermenci, Alpay; Dong, Guangbin: Synthesis of Ynones and Recent Application in Transition-Metal-Catalyzed Reactions

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Issue 01/2016

Brant, Michael G.; Wulff, Jeremy E.: 3-Sulfolenes and Their Derivatives: Synthesis and Applications

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Issue 24/2015

Kuninobu, Yoichiro; Sueki, Shunsuke: C–H Bond Transformations Leading to the Synthesis of Organic Functional Materials

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Issue 23/2015

Wang, Zhaobin; Sun, Jianwei: Recent Advances in Catalytic Asymmetric Reactions of o-Quinone Methides

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Issue 22/2015

Deska, Jan; Thiel, Daniel; Gianolio, Eleonora: The Achmatowicz Rearrangement – Oxidative Ring Expansion of Furfuryl Alcohols

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Issue 21/2015

Hong, Bor-Cherng; Raja, Arun; Sheth, Vishal M.: Asymmetric Synthesis of Natural Products and Medicinal Drugs through One-Pot-Reaction Strategies

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Issue 20/2015

Mann, Sam E.; Benhamou, L.; Sheppard, Tom D.: Palladium(II)-Catalysed Oxidation of Alkenes

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Issue 19/2015

Reck, Bernhard; Spiteller, Peter: Synthesis of Secondary Metabolites from Higher Fungi

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Issue 18/2015

Zhu, Guili; Liu, Rong; Liu, Bo: Total Synthesis of Atisane-Type Diterpenoids and Related Diterpenoid Alkaloids

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Issue 17/2015

Undheim, Kjell: Stereoselective Reactions in Preparation of Chiral α-Hetera­spiro[m.n]alkanes

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Issue 16/2015

Zhang, Lin; Fang, Guichun; Kumar, Rapolu Kiran; Bi, Xihe: Coinage-Metal-Catalyzed Reactions of Propargylic Alcohols

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Issue 15/2015

Vetica, Fabrizio; de Figueiredo, Renata Marcia; Orsini, Monica; Tofani, Daniela; Gasperi, Tecla: Recent Advances in Organocatalytic Cascade Reactions toward the Formation of Quaternary Stereocenters

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Issue 14/2015

Singh, Sarbjit; Chimni, Swapandeep Singh: Recent Advances in Iodine Monochloride Mediated Electrophilic Cyclizations

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Issue 13/2015

Courant, Thibaut; Dagousset, Guillaume; Masson, Géraldine: Enamide Derivatives: Versatile Building Blocks for Total Synthesis

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Issue 12/2015

Toma, Štefan; Šebesta, Radovan: Applications of Ferrocenium Salts in Organic Synthesis

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Issue 11/2015

Han, Jianguang; Jones, Alexander X.; Lei, Xiaoguang: Recent Advances in the Total Synthesis of Prenylflavonoid and Related Diels–Alder Natural Products

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Issue 10/2015

Yetra, Santhivardhana Reddy; Patra, Atanu; Biju, Akkattu T.: Recent Advances in the N-Heterocyclic Carbene (NHC)-Organocatalyzed Stetter Reaction and Related Chemistry

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Issue 09/2015

Song, Ren-Jie; Liu, Yu; Xie, Ye-Xiang; Li, Jin-Heng: Difunctionalization of Acrylamides through C–H Oxidative Radical Coupling: New Approaches to Oxindoles

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Issue 08/2015

Cao, Derong; Meier, Herbert: Synthesis of Pillar[6]arenes and Their Host–Guest Complexes

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Issue 07/2015

Pericherla, Kasiviswanadharaju; Kaswan, Pinku; Pandey, Khima; Kumar, Anil: Recent Developments in the Synthesis of Imidazo[1,2-a]pyridines

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Issue 06/2015

Cai, Xiao-hua; Xie, Bing: Carbon–Hydrogen Bond Functionalizations Mediated by Copper

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Issue 05/2015

Berthiol, Florian: Reagent and Catalyst Design for Asymmetric Hypervalent Iodine Oxidations

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Issue 04/2015

Mo, Jiayu; Wang, Lianhui; Liu, Yunqi; Cui, Xiuling: Transition-Metal-Catalyzed Direct C–H Functionalization under External-Oxidant-Free Conditions

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Issue 03/2015

Wang, Youliang; Zhang, Liming: Recent Developments in the Chemistry of Heteroaromatic N-Oxides

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Issue 02/2015

Ameen, Dana; Snape, Timothy J.: Mechanism and Application of Baker–Venkataraman O→C Acyl Migration Reactions

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Issue 01/2015

Mackay, Emily G.; Sherburn, Michael S.: The Diels–Alder Reaction in Steroid Synthesis

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Issue 24/2014

Schmidt, Andrea-Katharina C.; Stark, Christian B. W.: The Glycol Cleavage in Natural Product Synthesis: Reagent Classics and Recent Advances

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Issue 23/2014

Dagousset, Guillaume; François, Cyril; Leόn, Thierry; Blanc, Romain; Sansiaume-Dagousset, Elodie; Knochel, Paul: Preparation of Functionalized Lithium, Magnesium, Aluminum, Zinc, Manganese­, and Indium Organometallics from Functionalized Organic Halides

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Issue 22/2014

Zhou, Feng; Liao, Fu-Min; Yu, Jin-Sheng; Zhou, Jian: Catalytic Asymmetric Electrophilic Amination Reactions To Form Nitrogen-Bearing Tetrasubstituted Carbon Stereocenters

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Issue 21/2014

Rossi, Renzo; Bellina, Fabio; Lessi, Marco; Manzini, Chiara; Perego, Luca A.: Synthesis of Multiply Arylated Heteroarenes, Including Bioactive Derivatives, via Palladium-Catalyzed Direct C–H Arylation of Heteroarenes with (Pseudo)Aryl Halides or Aryliodonium Salts

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Issue 20/2014

Deore, Prashant S.; Haval, Kishan P.; Gadre, Smita R.; Argade, Narshinha P.: A Concise Account of the Chemistry of Valuable Alkyl(methyl)maleic Anhydrides

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Issue 19/2014

De Houwer, Johan; Maes, Bert U. W.: Synthesis of Aryl(di)azinylmethanes and Bis(di)azinylmethanes via Transition-Metal-Catalyzed Cross-Coupling Reactions

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Issue 18/2014

Windler, G. Kenneth; Pagoria, Philip F.; Vollhardt, K. Peter C.: Nitroalkynes: A Unique Class of Energetic Materials

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Issue 17/2014

Liu, Xiaohua; Zheng, Ke; Feng, Xiaoming: Advancements in Catalytic Asymmetric Intermolecular Ene-Type Reactions

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Issue 16/2014

Sen, Subhabrata; Prabhu, Ganesh; Bathula, Chandramohan; Hati, Santanu: Diversity-Oriented Asymmetric Synthesis

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Issue 15/2014

Undheim, Kjell: Preparation and Structure Classification of Heteraspiro[m.n]alkanes

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Issue 14/2014

Candish, Lisa; Nakano, Yuji; Lupton, David W.: Lewis Base Catalysis of Three n–π* Mediated Reactions with N-Heterocyclic Carbenes (NHCs), Isothioureas, Bicyclic Tertiary Amines, and Electron-Rich Pyridyls

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Issue 13/2014

Fang, Weiwei; Zhu, Haibo; Deng, Qinyue; Liu, Shuangliang; Liu, Xiyu; Shen, Yajing; Tu, Tao: Design and Development of Ligands for Palladium-Catalyzed Carbonylation Reactions

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Issue 12/2014

Le Bras, Jean; Muzart, Jacques: Dehydrogenative Heck Annelations of Internal Alkynes

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Issue 11/2014

Dastbaravardeh, Navid; Christakakou, Maria; Haider, Maximilian; Schnürch, Michael: Recent Advances in Palladium-Catalyzed C(sp³)–H Activation for the Formation of Carbon–Carbon and Carbon–Heteroatom Bonds

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Issue 10/2014

Hugelshofer, Cedric L.; Magauer, Thomas: High-Pressure Transformations in Natural Product Synthesis

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Issue 09/2014

Rodriguez, Juan B.: Tetraethyl Vinylidenebisphosphonate: A Versatile Synthon for the Preparation of Bisphosphonates

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Issue 08/2014

Bartoli, Giuseppe; Bencivenni, Giorgio; Dalpozzo, Renato: Asymmetric Cyclopropanation Reactions

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Issue 07/2014

La Spisa, Fabio; Tron, Gian Cesare; El Kaïm, Laurent: The Nef Reaction of Isocyanides

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Ni, Chuanfa; Hu, Jinbo: Recent Advances in the Synthetic Application of Difluorocarbene

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Issue 06/2014

Abbiati, Giorgio; Arcadi, Antonio; Marinelli, Fabio; Rossi, Elisabetta: Sequential Addition and Cyclization Processes of α,β-Ynones and α,β-Ynoates Containing Proximate Nucleophiles

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Issue 05/2014

Neochoritis, Constantinos G.; Zarganes-Tzitzikas, Tryfon; Stephanidou-Stephanatou, Julia: Dimethyl Acetylenedicarboxylate: A Versatile Tool in Organic Synthesis

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Issue 04/2014

Olszewski, Tomasz K.: Environmentally Benign Syntheses of α-Substituted Phosphonates: Preparation of α-Amino- and α-Hydroxyphosphonates in Water, in Ionic Liquids, and under­ Solvent-Free Conditions

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Issue 03/2014

Palmer, Leoni I.; Frazier, Charles P.; Read de Alaniz, Javier: Developments in Nitrosocarbonyl Chemistry: Mild Oxidation of N-Substituted Hydroxylamines Leads to New Discoveries

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Issue 02/2014

Fochi, Mariafrancesca; Caruana, Lorenzo; Bernardi, Luca: Catalytic Asymmetric Aza-Diels–Alder Reactions: The Povarov Cycloaddition Reaction

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Issue 01/2014

Aitken, David J.; Eijsberg, Hendrik; Frongia, Angelo; Ollivier, Jean; Piras, Pier Paolo: Recent Progress in the Synthetic Assembly of 2-Cyclopentenones

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Issue 24/2013

Cai, Xiaohua; Xie, Bing: Direct Carboxylative Reactions for the Transformation of Carbon Dioxide into Carboxylic Acids and Derivatives

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Issue 23/2013

Oliver, Samuel; Evans, P. Andrew: Transition-Metal-Catalyzed Allylic Substitution Reactions: Stereoselective Construction of α- and β-Substituted Carbonyl Compounds

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Issue 22/2013

Silva, Eduarda M. P.; Varandas, Pedro A. M. M.; Silva, Artur M. S.: Developments in the Synthesis of 1,2-Dihydropyridines

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Issue 21/2013

Chen, Pinhong; Liu, Guosheng: Recent Advances in Transition-Metal-Catalyzed Trifluoromethylation and Related Transformations

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Issue 20/2013

Karimi, Babak; Enders, Dieter; Jafari, Ehsan: Recent Advances in Metal-Catalyzed Asymmetric Mannich Reactions

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Issue 19/2013

Aitken, Lewis S.; Arezki, Natasha R.; Dell’Isola, Antonio; Cobb, Alexander J. A.: Asymmetric Organocatalysis and the Nitro Group Functionality

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Issue 18/2013

Bandar, Jeffrey S.; Lambert, Tristan H.: Aminocyclopropenium Ions: Synthesis, Properties, and Applications

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Issue 17/2013

Ila, Hiriyakkanavar; Markiewicz, John T.; Malakhov, Vladimir; Knochel, Paul: Metalated Indoles, Indazoles, Benzimidazoles, and Azaindoles and Their Synthetic Applications

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Issue 16/2013

Weidmann, Verena; Maison, Wolfgang: Allylic Oxidations of Olefins to Enones

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Issue 15/2013

Liu, Wei; Zhao, Xiaoming: Carbon–Sulfur Bond Formation via Metal-Catalyzed Allylations of Sulfur Nucleophiles

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Issue 14/2013

Goudedranche, Sébastien; Raimondi, Wilfried; Bugaut, Xavier; Constantieux, Thierry; Bonne, Damien; Rodriguez, Jean: Enantioselective Organocatalyzed Domino Synthesis of Six-Membered Carbocycles

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Issue 12/2013

Basavaprabhu; Vishwanatha, T. M.; Panguluri, Nageswara Rao; Sureshbabu, Vommina V.: Propanephosphonic Acid Anhydride (T3P^®) - A Benign Reagent for Diverse Applications Inclusive of Large-Scale Synthesis

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Issue 11/2013

Nakamura, Akihiko; Nakada, Masahisa: Allylic Oxidations in Natural Product Synthesis

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Issue 10/2013

Majumdar, K. C.; Sinha, Biswajit: Palladium-Mediated Total Synthesis of Bioactive Natural Products

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Issue 09/2013

Rehbein, Julia; Hiersemann, Martin: Claisen Rearrangement of Aliphatic Allyl Vinyl Ethers from 1912 to 2012: 100 Years of Electrophilic Catalysis

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Issue 08/2013

Finkbeiner, Peter; Nachtsheim, Boris J.: Iodine in Modern Oxidation Catalysis

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Issue 07/2013

Nguyen, Thanh Vinh; Hartmann, Jan Marc; Enders, Dieter: Recent Synthetic Strategies to Access Seven-Membered Carbocycles in Natural Product Synthesis

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Issue 06/2013

Selig, Philipp: Guanidine Organocatalysis

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Issue 05/2013

Flores-Gaspar, Areli; Martin, Ruben: Recent Advances in the Synthesis and Application of Benzocyclobutenones and Related Compounds

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Issue 04/2013

Matsunaga, Shigeki; Shibasaki, Masakatsu: Multimetallic Schiff Base Complexes as Cooperative Asymmetric Catalysts

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Issue 03/2013

Streuff, Jan: The Electron-Way: Metal-Catalyzed Reductive Umpolung Reactions of Saturated and α,β-Unsaturated Carbonyl Derivatives

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Issue 02/2013

Sorochinsky, Alexander E.; Aceña, José Luis; Soloshonok, Vadim A.: Self-Disproportionation of Enantiomers of Chiral, Non-Racemic Fluoroorganic Compounds: Role of Fluorine as Enabling Element

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Issue 01/2013

Ding, Qiuping; Ye, Yang; Fan, Renhua: Recent Advances in Phenol Dearomatization and Its Application in Complex Syntheses

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Issue 24/2012

Palmes, Jean A.; Aponick, Aaron: Strategies for Spiroketal Synthesis Based on Transition-Metal Catalysis

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Issue 23/2012

Trstenjak, Uroš; Ilaš, Janez; Kikelj, Danijel: Advances in the Synthesis of Morpholin-3-ones and Morpholin-2-ones

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Issue 22/2012

Adcock, Holly V.; Davies, Paul W.: π-Acid Mediated Insertion of Alkynes into Carbon–Heteroatom σ-Bonds

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Issue 21/2012

Schmidt, Andreas; Guan, Zong: Mesomeric Betaines and N-Heterocyclic Carbenes of Pyrazole and Indazole

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Issue 20/2012

Silva, Eduarda M. P.; Silva, Artur M. S.: 1,6-Conjugate Addition of Nucleophiles to α,β,γ,δ-Diunsaturated Systems

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Issue 19/2012

Tang, Pei; Qin, Yong: Recent Applications of Cyclopropane-Based Strategies to Natural Product Synthesis

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Issue 18/2012

Liu, Tao; Fu, Hua: Copper-Catalyzed Synthesis of N-Heterocyclic Compounds

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Issue 17/2012

Broere, Daniël L. J.; Ruijter, Eelco: Recent Advances in Transition-Metal-Catalyzed [2+2+2]-Cyclo(co)trimerization Reactions

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Issue 16/2012

Majumdar, K. C.; Karunakar, Galla V.; Sinha, Biswajit: Formation of Five- and Six-Membered Heterocyclic Rings under Radical Cyclization Conditions

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Issue 15/2012

Douglas, James; Churchill, Gwydion; Smith, Andrew D.: NHCs in Asymmetric Organocatalysis: Recent Advances in Azolium Enolate Generation and Reactivity

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Issue 14/2012

Serdyuk, Olga V.; Muzalevskiy, Vasiliy M.; Nenajdenko, Valentine G.: Synthesis and Properties of Fluoropyrroles and Their Analogues

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Issue 13/2012

Cant, Alastair A.; Sutherland, Andrew: Asymmetric Synthesis of Pipecolic Acid and Derivatives

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Issue 12/2012

Stolze, Sara C.; Kaiser, Markus: Challenges in the Syntheses of Peptidic Natural Products

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Issue 11/2012

Aceña, José Luis; Sorochinsky, Alexander E.; Soloshonok, Vadim A.: Recent Advances in the Asymmetric Synthesis of α-(Trifluoromethyl)-Containing α-Amino Acids

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Issue 10/2012

Endo, Kohei; Shibata, Takanori: Detour and Direct Induction of Methyl-Containing Chiral Centers via Catalytic C–H or C–C Bond Formation

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Issue 09/2012

Larraufie, Marie-Hélène; Maestri, Giovanni; Malacria, Max; Ollivier, Cyril; Fensterbank, Louis; Lacôte, Emmanuel: The Cyanamide Moiety, Synthesis and Reactivity

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Issue 08/2012

Bauer, Eike B.: Transition-Metal-Catalyzed Functionalization of Propargylic Alcohols and Their Derivatives

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Issue 07/2012

Lim, Diane S. W.; Anderson, Edward A.: Synthesis of Vinylsilanes

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Issue 06/2012

Majumdar, K. C.; Samanta, Srikanta; Sinha, Biswajit: Recent Developments in Palladium-Catalyzed Formation of Five- and Six-Membered Fused Heterocycles

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Issue 05/2012

Cornella, Josep; Larrosa, Igor: Decarboxylative Carbon-Carbon Bond-Forming Transformations of (Hetero)aromatic Carboxylic Acids

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Pan, Changduo; Jia, Xiaofei; Cheng, Jiang: Transition-Metal-Catalyzed Synthesis of Aromatic Ketones via Direct C-H Bond Activation

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Issue 04/2012

Nishibayashi, Yoshiaki: Transition-Metal-Catalyzed Enantioselective Propargylic Substitution Reactions of Propargylic Alcohol Derivatives with Nucleophiles

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Bandini, Marco; Cera, Gianpiero; Chiarucci, Michel: Catalytic Enantioselective Alkylations with Allylic Alcohols

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Issue 03/2012

Shibata, Yu; Tanaka, Ken: Rhodium-Catalyzed [2+2+2] Cycloaddition of Alkynes for the Synthesis of Substituted Benzenes: Catalysts, Reaction Scope, and Synthetic Applications

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Schultz, Danielle M.; Wolfe, John P.: Recent Developments in Palladium-Catalyzed Alkene Aminoarylation Reactions for the Synthesis of Nitrogen Heterocycles

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Issue 02/2012

Müller, Thomas J. J.: Synthesis of Carbo- and Heterocycles via Coupling-Isomerization Reactions

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Huang, Xueliang; Klimczyk, Sebastian; Maulide, Nuno: Charge-Accelerated Sulfonium [3,3]-Sigmatropic Rearrangements

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Issue 01/2012

Zhang, Ming; Zhang, Aiqin: Non-Cyclizing Direct Transformation of Arene Carbon-Hydrogen Bonds into Carbon-Nitrogen Bonds

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Kandepi, V. V. Krishna Mohan; Narender, Nama: Ecofriendly Oxidative Nuclear Halogenation of Aromatic Compounds Using Potassium and Ammonium Halides

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Issue 24/2011

Boldon, Sophie; Stenhagen, Ida S. R.; Moore, Jane E.; Luthra, Sajinder K.; Gouverneur, Véronique: Supported Synthesis of Halogenated Organic Compounds

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Barker, Timothy J.; Jarvo, Elizabeth R.: Developments in Transition-Metal-Catalyzed Reactions Using Electrophilic Nitrogen Sources

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Issue 23/2011

Paradies, Jan: [2.2]Paracyclophane Derivatives: Synthesis and Application in Catalysis

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Majumdar, Krishna C.; Ray, Krishanu: Synthesis of 1,2,3-Triazole-Fused Heterocycles via Intramolecular Azide-Alkyne Cycloaddition Reactions

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Issue 22/2011

Sperry, Jonathan: The Oxidation of Amides to Imides: A Powerful Synthetic Transformation

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Le Bras, Jean; Muzart, Jacques: Heck Arylations of Baylis-Hillman Adducts

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Issue 21/2011

Aïssa, Christophe: Transition-Metal-Catalyzed Rearrangements of Small Cycloalkanes: Regioselectivity Trends in β-Carbon Elimination Reactions

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Zhang, Ming: Advances in the Direct Amination of Azole C-H Bonds

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Issue 20/2011

Nakao, Yoshiaki: Transition-Metal-Catalyzed C-H Functionalization for the Synthesis of Substituted Pyridines

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Issue 19/2011

Mikami, Koichi; Fustero, Santos; Sánchez-Roselló, Maria; Aceña, José Luis; Soloshonok, Vadim; Sorochinsky, Alexander: Synthesis of Fluorinated β-Amino Acids

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Issue 18/2011

Sharma, Pallavi; Powell, Kimberley J.; Burnley, James; Awaad, Amani S.; Moses, John E.: Total Synthesis of Polypropionate-Derived γ-Pyrone Natural Products

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Issue 17/2011

Lehnert, Tobias; Özüduru, Gülsüm; Grugel, Holger; Albrecht, Fabian; Telligmann, Susanne M.; Boysen, Mike M. K.: More Than Just Sweet - Sugar-Derived Stereodifferentiating Agents for Asymmetric Synthesis

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Issue 16/2011

Serdyuk, Olga V.; Abaev, Vladimir T.; Butin, Alexander V.; Nenajdenko, Valentine G.: Synthesis of Fluorinated Thiophenes and Their Analogues

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de Haro, Teresa; Nevado, Cristina: On Gold-Mediated C-H Activation Processes

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Issue 15/2011

Mąkosza, Mieczysław: Nucleophilic Substitution of Hydrogen in Nitroarenes: A New Chapter of Aromatic Chemistry

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Issue 14/2011

Ariza, Xavier; Garcia, Jordi; Romea, Pedro; Urpí, Fèlix: Stereoselective Acetate Aldol Reactions from Metal Enolates

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Issue 13/2011

Lam, Hon Wai: TADDOL-Derived Phosphonites, Phosphites, and Phosphoramidites in Asymmetric Catalysis

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Pan, Yuanhang; Tan, Choon-Hong: Catalytic Decarboxylative Reactions: Biomimetic Approaches Inspired by Polyketide Biosynthesis

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Issue 12/2011

Bhanushali, Mayur; Zhao, Cong-Gui: Developing Novel Organocatalyzed Aldol Reactions for the Enantioselective Synthesis of Biologically Active Molecules

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Issue 11/2011

Verendel, J. Johan; Church, Tamara L.; Andersson, Pher G.: Catalytic One-Pot Production of Small Organics from Polysaccharides

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Su, Yijin; Jia, Wei; Jiao, Ning: Inexpensive Copper/Iron-Cocatalyzed Reactions

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Issue 10/2011

Pradal, Alexandre; Toullec, Patrick Y.; Michelet, Véronique: Recent Developments in Asymmetric Catalysis in the Presence of Chiral Gold Complexes

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Issue 09/2011

Ramadhar, Timothy R.; Batey, Robert A.: Allylation of Imines and Their Derivatives with Organoboron Reagents: Stereocontrolled Synthesis of Homoallylic Amines

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Issue 08/2011

O’Brien, Matthew; Denton, Ross; Ley, Steven V.: Lesser-Known Enabling Technologies for Organic Synthesis

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Issue 07/2011

Bonjoch, Josep; Diaba, Faïza; Bradshaw, Ben: Synthesis of 2-Azabicyclo[3.3.1]nonanes

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Issue 06/2011

Qiao, Jennifer X.; Lam, Patrick Y. S.: Copper-Promoted Carbon-Heteroatom Bond Cross-Coupling with Boronic Acids and Derivatives

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Issue 05/2011

Burns, Alan R.; Taylor, Richard J. K.: Synthetic Approaches to Enantiomerically Enriched 4-Hydroxycyclohex-2-en-1-one - A Key Chiral Building Block in Complex Natural Product Synthesis

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Issue 04/2011

Merritt, Eleanor A.; Olofsson, Berit: α-Functionalization of Carbonyl Compounds Using Hypervalent Iodine Reagents

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Issue 03/2011

Klussmann, Martin; Sureshkumar, Devarajulu: Catalytic Oxidative Coupling Reactions for the Formation of Carbon-Carbon Bonds without Carbon-Metal Intermediates

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Issue 02/2011

Höfling, Sarah B.; Heinrich, Markus R.: Nitrogen-Centered Radical Scavengers

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Issue 01/2011

Sadig, Jessie E. R.; Willis, Michael C.: Palladium- and Copper-Catalyzed Aryl Halide Amination, Etherification and Thioetherification Reactions in the Synthesis of Aromatic Heterocycles

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Issue 24/2010

Rossi, Renzo; Bellina, Fabio; Lessi, Marco: Alkenylation Reactions of Heteroarenes by Transition-Metal Catalysts

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Issue 23/2010

Wan, Jie-Ping; Liu, Yunyun: Synthesis of Dihydropyrimidinones and Thiones by Multicomponent Reactions: Strategies Beyond the Classical Biginelli Reaction

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Issue 22/2010

Rinner, Uwe; Lentsch, Christoph; Aichinger, Christian: Syntheses of Galbulimima Alkaloids

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Issue 21/2010

Yin, Biaolin; Zhang, Yuanxiu; Xu, Li-Wen: Recent Applications of α-Amido Sulfones as in situ Equivalents of Activated Imines for Asymmetric Catalytic Nucleophilic Addition Reactions

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Issue 20/2010

Satoh, Tetsuya; Miura, Masahiro: Transition-Metal-Catalyzed Regioselective Arylation and Vinylation of Carboxylic Acids

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Issue 19/2010

Koester, Dennis C.; Holkenbrink, Annika; Werz, Daniel B.: Recent Advances in the Synthesis of Carbohydrate Mimetics

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Issue 18/2010

Tappe, Florian M. J.; Trepohl, Verena T.; Oestreich, Martin: Transition-Metal-Catalyzed C-P Cross-Coupling Reactions

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Issue 17/2010

Dömling, Alexander; Huang, Yijun: Piperazine Scaffolds via Isocyanide-Based Multicomponent Reactions

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Issue 16/2010

Shibatomi, Kazutaka: Alternative Synthetic Strategies for Enantioselective Construction of Halogenated Chiral Carbon Centers

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Issue 15/2010

Winternheimer, David J.; Shade, Ryan E.; Merlic, Craig A.: Methods for Vinyl Ether Synthesis

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Issue 14/2010

Soloshonok, Vadim A.; Sorochinsky, Alexander E.: Practical Methods for the Synthesis of Symmetrically α,α-Disubstituted α-Amino Acids

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Issue 13/2010

Schlosser, Manfred; Ruzziconi, Renzo: Nucleophilic Substitutions of Nitroarenes and Pyridines: New Insight and New Applications

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Issue 12/2010

Terada, Masahiro: Chiral Phosphoric Acids as Versatile Catalysts for Enantioselective Transformations

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Issue 11/2010

Pigge, F. Christopher: Metal-Catalyzed Allylation of Organoboranes and Organoboronic Acids

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Issue 10/2010

Boncel, Sławomir; Gondela, Andrzej; Walczak, Krzysztof: Michael-type Addition as a Convenient Method for Regioselective N-Alkylation of Ambident Uracils

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Issue 09/2010

Karimi, Babak; Behzadnia, Hesam; Elhamifar, Dawood; Akhavan, Pari Fadavi; Esfahani, Farhad Kabiri; Zamani, Asghar: Transition-Metal-Catalyzed Oxidative Heck Reactions

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Issue 08/2010

Marcelli, Tommaso; Hiemstra, Henk: Cinchona Alkaloids in Asymmetric Organocatalysis

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Issue 07/2010

Silva, Jr., Luiz F.; Carneiro, Vânia M. T.: Thallium(III) in Organic Synthesis

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Issue 06/2010

Elford, Tim G.; Hall, Dennis G.: Advances in 2-(Alkoxycarbonyl)allylboration of Carbonyl Compounds and Other Direct Methods for the Preparation of α-Exo-Alkylidene γ-Lactones

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Issue 05/2010

Küchenthal, Christian-H.; Maison, Wolfgang: Synthesis of Cyclic Hydrazino α-Carboxylic Acids

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Issue 04/2010

Czekelius, Constantin; Tzschucke, Carl Christoph: Synthesis of Halogenated Carboxylic Acids and Amino Acids

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Issue 03/2010

Jautze, Sascha; Peters, René: Catalytic Asymmetric Michael Additions of α-Cyanoacetates

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Issue 02/2010

Hentschel, Fabia; Lindel, Thomas: Synthesis of Oximinotyrosine-Derived Marine Natural Products

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Issue 01/2010

Merino, Pedro; Marqués-López, Eugenia; Tejero, Tomás; Herrera, Raquel P.: Enantioselective Organocatalytic Diels-Alder Reactions

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Issue 24/2009

Kulkarni, Amol A.; Daugulis, Olafs: Direct Conversion of Carbon-Hydrogen into Carbon-Carbon Bonds by First-Row Transition-Metal Catalysis

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Issue 23/2009

Muzalevskiy, Vasiliy M.; Shastin, Aleksey V.; Balenkova, Elizabeth S.; Haufe, Günter; Nenajdenko, Valentine G.: Synthesis of Trifluoromethyl Pyrroles and Their Benzo Analogues

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Issue 22/2009

Volochnyuk, Dmitriy M.; Ryabukhin, Sergey V.; Plaskon, Andrey S.; Grygorenko, Oleksandr O.: Organosilicon Compounds as Water Scavengers in Reactions of Carbonyl Compounds

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Issue 21/2009

Semeniuchenko, Volodymyr; Groth, Ulrich; Khilya, Volodymyr: Synthesis of Chroman-2-ones by Reduction of Coumarins

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Issue 20/2009

De Simone, Filippo; Waser, Jérôme: Cyclization and Cycloaddition Reactions of Cyclopropyl Carbonyls and Imines

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Issue 19/2009

Kajimoto, Tetsuya; Node, Manabu: Synthesis of Glycosyltransferase Inhibitors

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Issue 18/2009

Trost, Barry M.; Brennan, Megan K.: Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural Products

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Issue 16/2009

Rosenberg, Sara; Leino, Reko: Synthesis of Spirocyclic Ethers

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Issue 15/2009

Singh, Rohit; Kaur, Harneet: Advances in Synthetic Approaches for the Preparation of Combretastatin-Based Anti-Cancer Agents

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Issue 14/2009

Li, Jun; Menche, Dirk: Direct Methods for Stereoselective Polypropionate Synthesis: A Survey

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Issue 13/2009

Majumdar, K. C.; Bhattacharyya, Trijit; Chattopadhyay, Buddhadeb; Sinha, Biswajit: Recent Advances in the Aza-Claisen Rearrangement

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Issue 12/2009

Opatz, Till: The Chemistry of Deprotonated α-Aminonitriles

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Issue 11/2009

Ogasawara, Masamichi; Watanabe, Susumu: Transition-Metal-Catalyzed Enantioselective Synthesis of Compounds with Non-Centrochirality

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Issue 10/2009

Bella, Marco; Gasperi, Tecla: Organocatalytic Formation of Quaternary Stereocenters

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Issue 09/2009

Wang, Jia-Rui; Manabe, Kei: Transition-Metal-Catalyzed Site-Selective Cross-Coupling of Di- and Polyhalogenated Compounds

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Issue 08/2009

Janecki, Tomasz; Kędzia, Jacek; Wąsek, Tomasz: Michael Additions to Activated Vinylphosphonates

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Issue 07/2009

Kuwano, Ryoichi: Catalytic Transformations of Benzylic Carboxylates and Carbonates

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Issue 06/2009

Bournaud, Chloée; Chung, Florence; Luna, Alejandro Pérez; Pasco, Morgane; Errasti, Gauthier; Lecourt, Thomas; Micouin, Laurent: Stereoselective Transformations of meso Bicyclic Hydrazines: Versatile Access to Functionalized Aminocyclopentanes

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Issue 05/2009

Clarke, Paul A.; Reeder, Andrew T.; Winn, Joby: Transannulation Reactions in the Synthesis of Natural Products

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Issue 04/2009

Yazici, Arife; Pyne, Stephen G.: Intermolecular Addition Reactions of N-Acyliminium Ions (Part II)

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Issue 03/2009

Yazici, Arife; Pyne, Stephen G.: Intermolecular Addition Reactions of N-Acyliminium Ions (Part I)

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Issue 02/2009

Kotha, Sambasivarao; Deb, Ashoke Chandra; Lahiri, Kakali; Manivannan, Ethirajan: Selected Synthetic Strategies to Spirocyclics

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Issue 01/2009

Seebach, Dieter; Beck, Albert K.; Capone, Stefania; Deniau, Gildas; Grošelj, Uroš; Zass, Engelbert: Enantioselective Preparation of β^²-Amino Acid Derivatives for β-Peptide Synthesis

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Issue 24/2008

Feist, Holger; Langer, Peter: One-Pot Cyclizations of (2,4-Dioxobutylidene)phosphoranes and (2-Alkoxy-4-oxobut-2-enylidene)phosphoranes

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Issue 23/2008

Balasubramaniam, Sivaraman; Aidhen, Indrapal Singh: The Growing Synthetic Utility of the Weinreb Amide

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Issue 22/2008

Hess, Wilfried; Treutwein, Jonas; Hilt, Gerhard: Cobalt-Catalysed Carbon-Carbon Bond-Formation Reactions

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Issue 21/2008

Tanaka, Takanori; Hayashi, Masahiko: New Approach for Complete Reversal of Enantioselectivity Using a Single Chiral Source

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Issue 20/2008

Kirsch, Stefan F.: Construction of Heterocycles by the Strategic Use of Alkyne π-Activation in Catalyzed Cascade Reactions

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Issue 19/2008

Kakiuchi, Fumitoshi; Kochi, Takuya: Transition-Metal-Catalyzed Carbon-Carbon Bond Formation via Carbon-Hydrogen Bond Cleavage

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Issue 18/2008

Breuning, Matthias; Steiner, Melanie: Chiral Bispidines

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Issue 17/2008

Han, Soo Bong; Hassan, Abbas; Krische, Michael J.: Diastereo- and Enantioselective Reductive Aldol Addition of Vinyl Ketones via Catalytic Hydrogenation

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Issue 16/2008

Witt, Dariusz: Recent Developments in Disulfide Bond Formation

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Issue 15/2008

Kwong, Cathy Kar-Wing; Fu, Michael Yunyi; Lam, Cynthia Sze-Lok; Toy, Patrick H.: The Phosphine-Catalyzed Alkyne to 1,3-Diene Isomerization Reaction

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Issue 13/2008

Vogler, Thomas; Studer, Armido: Applications of TEMPO in Synthesis

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Issue 12/2008

von Zezschwitz, Paultheo: Selectivity Control in 1,2- and 1,4-Additions of Aluminum Organyls to Carbonyl Compounds

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Issue 11/2008

Hatano, Manabu; Ishihara, Kazuaki: Recent Progress in the Catalytic Synthesis of Tertiary Alcohols from Ketones with Organometallic Reagents

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Issue 10/2008

Stavber, Stojan; Jereb, Marjan; Zupan, Marko: Electrophilic Iodination of Organic Compounds Using Elemental Iodine or Iodides

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Issue 09/2008

Christie, Steven D. R.; Warrington, Adam D.: Osmium and Palladium: Complementary Metals in Alkene Activation and Oxidation

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Issue 08/2008

Vorbrüggen, Helmut: The Conversion of Primary or Secondary Alcohols with Nonaflyl Fluoride into Their Corresponding Inverted Fluorides

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Issue 07/2008

Winkel, Andreas; Reddy, Peddiahgari Vasu Govardhana; Wilhelm, René: Recent Advances in the Synthesis and Application of Chiral Ionic Liquids

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Issue 06/2008

Smitha, Gouni; Chandrasekhar, Srivari; Reddy, Cherkupally Sanjeeva: Applications of Zirconium(IV) Chloride in Organic Synthesis

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Issue 05/2008

Lloyd-Jones, Guy C.; Moseley, Jonathan D.; Renny, Joseph S.: Mechanism and Application of the Newman-Kwart O→S Rearrangement of O-Aryl Thiocarbamates

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Issue 04/2008

Kouznetsov, Vladimir V.; Vargas Méndez, Leonor Yamile: Recent Developments in Three-Component Grignard-Barbier-Type Reactions

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Issue 03/2008

Lawrence, Adrien K.; Gademann, Karl: Aza-Annulation Strategies in Alkaloid Total Synthesis

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Issue 02/2008

Kostyuk, Aleksandr N.; Volochnyuk, Dmitriy M.; Sibgatulin, Dmitriy A.: Reaction of Linear Push-Pull Enamines at the β′-Position

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Issue 01/2008

Shestopalov, Anatoliy M.; Shestopalov, Alexander A.; Rodinovskaya, Lyudmila A.: Multicomponent Reactions of Carbonyl Compounds and Derivatives of Cyanoacetic Acid: Synthesis of Carbo- and Heterocycles

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Issue 24/2007

Ciufolini, Marco A.; Braun, Norbert A.; Canesi, Sylvain; Ousmer, Malika; Chang, Jonah; Chai, David: Oxidative Amidation of Phenols through the Use of Hypervalent Iodine Reagents: Development and Applications

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Issue 23/2007

Gołebiewski, W. Marek; Gucma, Mirosław: Applications of N-Chlorosuccinimide in Organic Synthesis

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Issue 22/2007

Banert, Klaus: Hexadecyltributylphosphonium Azide - A Highly Potent Reagent for the Synthesis of Unusual Azides

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Issue 21/2007

Ferraz, Helena M. C.; Bombonato, Fernanda I.; Longo Jr, Luiz S.: Synthetic Approaches to Naturally Occurring Ten-Membered-Ring Lactones

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Issue 20/2007

Schmuck, Carsten; Rupprecht, Daniel: The Synthesis of Highly Functionalized Pyrroles: A Challenge in Regioselectivity and Chemical Reactivity

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Issue 19/2007

Shuklov, Ivan A.; Dubrovina, Natalia V.; Börner, Armin: Fluorinated Alcohols as Solvents, Cosolvents and Additives in Homogeneous Catalysis

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