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Carreira, E. M.  et al.: 2017 Science of Synthesis: Knowledge Updates 2017/3 DOI: 10.1055/sos-SD-112-00112
Knowledge Updates 2017/3

12.1.5 Pyrazoles (Update 2017)

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Book

Editors: Carreira, E. M. ; Christmann, M.; Reißig, H.-U.

Authors: Bartels, F.; Christmann, M.; Götzinger, A. C.; Müller, T. J. J.; Schneider, C.; Sickert, M.; Zimmer, R.

Title: Knowledge Updates 2017/3

Print ISBN: 9783132414181; Online ISBN: 9783132414211; Book DOI: 10.1055/b-005-143665

1st edition © 2017 Thieme. All rights reserved.
Georg Thieme Verlag, Stuttgart

Subjects: Organic Chemistry;Chemical Reactions, Catalysis;Organometallic Chemistry;Laboratory Techniques, Stoichiometry

Science of Synthesis Knowledge Updates



Parent publication

Title: Science of Synthesis

DOI: 10.1055/b-00000101

Series Editors: Carreira, E. M.; Decicco, C. P.; Fürstner, A.; Koch, G.; Molander, G.; Schaumann, E.; Shibasaki, M.; Thomas, E. J.; Trost, B. M.

Type: Multivolume Edition

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Abstract

This review presents an overview of the developments in pyrazole synthesis since the beginning of the 21st century. It includes the synthesis of the pyrazole core by ring-closing reactions, ring expansion or contraction, and aromatization. The introduction of substituents onto the pyrazole ring is also covered. Novel synthetic methods that have been developed since the original Science of Synthesis review on pyrazoles (Section 12.1) include various multicomponent approaches in which multiple bonds are formed, cross coupling, and C—H activation reactions of pyrazole derivatives.

Key words

pyrazoles - nitrogen heterocycles - ring-closing reactions - condensation reactions - multicomponent reactions - ring expansion - ring contraction - aromatization - regioselectivity - 1,3-dicarbonyl compounds - hydrazines - hydrazones - diazo compounds - cross-coupling reactions - C—H activation
 
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