DOI: 10.1055/s-00000131

Synfacts

Issue 09 · Volume 2006 · September 2006 DOI: 10.1055/s-002-5078

Synthesis of Natural Products and Potential Drugs

0863
Yue, T.-Y.; McLeod, D. D.; Albertson, K. B.; Beck, S. R.; Deerberg, J.; Fortunak, J. M.; Nugent, W. A.; Radesca, L. A.; Tang, L.; Xiang, C. D.: Synthesis of a CCR3 Antagonist
0864
Chapsal, B. D.; Ojima, I.: Total Synthesis of (+)-γ-Lycorane
0865
Pettigrew, J. D.; Wilson, P. D.: Synthesis of (-)-Xyloketal A
0866
Heuser, S.; Barrett, D. G.; Berg, M.; Bonnier, B.; Kahl, A.; De La Puente, M. L.; Oram, N.; Riedl, R.; Roettig, U.; Gil, G. S.; Seger, E.; Steggles, D. J.; Wanner, J.; Wiechert, A. G.: Synthesis of Glucokinase Activators
0867
Scott, J. P.; Oliver, S. F.; Brands, K. M. J.; Brewer, S. E.; Davies, A. J.; Gibb, A. D.; Hands, D.; Keen, S. P.; Sheen, F. J.; Reamer, R. A.; Wilson, R. D.; Dolling, U.-H.: Synthesis of a γ-Secretase Inhibitor
0868
Meketa, M. L.; Weinreb, S. M.: Synthesis of Ageladine A
0869
Yu, C.-M.; Youn, J.; Jung, J.: Synthesis of (-)-Avenaciolide
0870
Fleming, J. J.; Bois, J. Du: Synthesis of (+)-Saxitoxin
0871
Bardhan, S.; Schmitt, D. C.; Porco, J. A.: Total Synthesis of (+)-Calafianin
0872
Nichols, P. J.; DeMattei, J. A.; Barnett, B. R.; LeFur, N. A.; Chuang, T.-H.; Piscopio, A. D.; Koch, K.: Synthesis of IC86518
0873
Saikawa, Y.; Moriya, K.; Hashimoto, K.; Nakata, M.: Synthesis of Hipposudoric Acid
0874
Hu, S.; Kelly, S.; Lee, S.; Tao, J.; Flahive, E.: Synthesis of Pelitrexol
0875
Damon, D. B.; Dugger, R. W.; Hubbs, S. E.; Scott, J. M.; Scott, R. W.: Synthesis of Torcetrapib
0876
Lu, C. V.; Chen, J. J.; Perrault, W. R.; Conway, B. G.; Maloney, M. T.; Wang, Y.: Synthesis of PNU-288034
0877
Han, Z.; Krishnamurthy, D.; Senanayake, C. H.: Synthesis of (R)-Sibutramine

Synthesis of Heterocycles

0879
de Figueiredo, R. M.; Fröhlich, R.; Christmann, M.: Synthesis of Chiral Azetidines
0880
Inada, Y.; Yoshikawa, M.; Milton, M. D.; Nishibayashi, Y.; Uemura, S.: Ru-Catalyzed Propargylation of Aromatics and Heteroaromatics
0881
Karpov, A. S.; Merkul, E.; Oeser, T.; Müller, T. J. J.: Multicomponent Synthesis of Substituted 3-Halofurans
0882
Kim, H.; Lee, C.: Synthesis of Fused Piperidines by Rhodium-Catalyzed Cyclization
0883
Oh, C. H.; Reddy, V. R.; Kim, A.; Rhim, C. Y.: Synthesis of Substituted Furans by Pt-Catalyzed Cyclization of Enynones
0884
Ambrogio, I.; Cacchi, S.; Fabrizi, G.: Pd-Catalyzed Synthesis of 2-(Aminomethyl)indoles
0885
Natarajan, S. R.; Chen, M.-H.; Heller, S. T.; Tynebor, R. M.; Crawford, E. M.; Minxiang, C.; Kaizheng, H.; Dong, J.; Hu, B.; Hao, W.; Chen, S.-H.: Lateral Metallation-Cycloannulation Synthesis of 2H-quinolizin-2-ones
0886
Jurík, V.; Wilhelm, R.: Chiral Imidazolinium Salts: Lewis Acids, Shift Reagents and Ionic Liquids
0887
Sakai, N.; Ridder, A.; Hartwig, J. F.: Synthesis of Tropenes by Pd-Catalyzed Double Hydroamination
0888
De Benassuti, L.; Buttero, P. Del; Molteni, G.: Stereoselective Synthesis of Enantiopure Pyrrolo[3,4-c]pyrazoles
0889
Smith III, A. B.; Kürti, L.; Davulcu, A. H.: Modular Synthesis of Fused Indole Derivatives
0890
Lin, L.; Fan, Q.; Qin, B.; Feng, X.: Enantioselective Cu-Catalyzed Hetero-Diels-Alder Synthesis of δ-Lactones
0891
Rosiak, A.; Christoffers, J.: A Short Synthesis of Unsymmetrical 2,3-Dihydrothiopyran-4-ones
0892
Patil, N. T.; Lutete, L. M.; Wu, H.; Pahadi, N. K.; Gridnev, I. D.; Yamamoto, Y.: Asymmetric Synthesis of O- and N-Heterocycles by Intramolecular Hydroamination and -alkoxylation
0893
Stanislawski, P. C.; Willis, A. C.; Banwell, M. G.: Synthesis of 1,1-Spirocyclic Tetrahydroisoquinoline Systems

Synthesis of Materials and Unnatural Products

0895
Yoshimura, T.; Inaba, A.; Sonoda, M.; Tahara, K.; Tobe, Y.; Williams, R. V.: Synthesis of a tris[12]DBA
0896
Vets, N.; Diliën, H.; Toppet, S.; Dehaen, W.: Preparation of 5,7,12,14-Tetraarylpentacenes
0897
Hennrich, G.; Alonso, B.; Monge, A.; Gutierrez-Puebla, E.; Echavarren, A. M.; Gómez-Lor, B.: A Redox-Active Triazacyclophane
0898
Ito, H.; Ishida, Y.; Saigo, K.: Fullerene-Centered Dissymmetric Molecular Triads
0899
Yamamoto, Y.; Hattori, K.; Nishiyama, H.: Synthesis of p-Diiodobenzenes by [2+2+2] Cycloaddition
0900
Katz, J. L.; Geller, B. J.; Conry, R. R.: Synthesis of Oxacalixarenes with Nitrogen Heterocycles
0901
Ishida, T.; Morisaki, Y.; Chujo, Y.: A Porphyrin Molecular Tube
0902
Leontiev, A. V.; Dias, H. V. Rasika; Rudkevich, D. M.: Synthesis of a Poly(sulfamide) from Sulfur Dioxide
0903
Jung, S.; Pisula, W.; Rouhanipour, A.; Räder, H. J.; Jacob, J.; Müllen, K.: Template-Assisted Synthesis of a Polycarbazole Macrocycle
0904
Xie, L.-H.; Liu, F.; Tang, C.; Hou, X.-Y.; Hua, Y.-R.; Fan, Q.-L.; Huang, W.: An Efficient One-Pot Synthesis of Spiro[fluorene-9,9′-xanthene]

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

0905
Yang, Q.; Shang, G.; Gao, W.; Deng, J.; Zhang, X.: Pd-TangPhos-Catalyzed Hydrogenation of N-Tosylimines
0906
Hashmi, A. S. K.; Haufe, P.; Schmid, C.; Nass, A. Rivas; Frey, W.: Enantioselective Synthesis of 8-Hydroxytetrahydroisoquinolines
0907
Fang, T.; Xu, J.; Du, D.-M.: C3-Symmetric Tripodal β-Hydroxy Amide Mediated Borane Reduction
0908
Lu, S.-F.; Du, D.-M.; Xu, J.; Zhang, S.-W.: Catalyzed Michael Addition of Nitroalkanes to Nitroalkenes
0909
Lauzon, C.; Charette, A. B.: Copper-Catalyzed Synthesis of α,α,α-Trifluoromethylamines
0910
Bisai, A.; Singh, V. K.: Enantioselective Multicomponent Synthesis of Propargylamines
0911
Nanchen, S.; Pfaltz, A.: Iridium-Catalyzed Hydrogenation
0912
Liang, C.; Robert-Peillard, F.; Fruit, C.; Müller, P.; Dodd, R. H.; Dauban, P.: Rhodium-Catalyzed Diastereoselective Intermolecular C-H Amination
0913
Lee, K.-S.; Brown, M. K.; Hird, A. W.; Hoveyda, A. H.: Enantioselective Conjugate Addition of Organozinc Reagents to Enones
0914
Basra, S.; Fennie, M. W.; Kozlowski, M. C.: Addition of Dialkylzinc Reagents toα-Aldiminoesters
0915
Gonzalez, A. S.; Arrayas, R. G.; Carretero, J. C.: Enantioselective Mannich-Type Reaction of N-Sulfonyl Imines
0916
Oisaki, K.; Zhao, D.; Kanai, M.; Shibasaki, M.: Catalytic Enantioselective Addition of Silyl Ketene Acetals to Ketones
0917
Yan, Y.; Zhang, X.: Rh(I)/YanPhos-Catalyzed Asymmetric Hydroformylation
0918
Kiyooka, S.-i; Takeshita, Y.; Tanaka, Y.; Higaki, T.; Wada, Y.: Pd(II)/Sparteine-Catalyzed Mukaiyama Aldol Reaction
0919
Fukuzumi, T.; Shibata, N.; Sugiura, M.; Yasui, H.; Nakamura, S.; Toru, T.: Catalytic Enantioselective Allylic Monofluoromethylation
0920
Du, H.; Long, J.; Shi, Y.: Simmons-Smith Cyclopropanation of Silyl Enol Ethers
0921
Mouhtady, O.; Gaspard-Iloughmane, H.; Laporterie, A.; Roux, C. Le: (R)-6,6′-Bis(CF3SO2)-binaphthol: A New Ligand for Asymmetric Synthesis
0922
Onodera, G.; Nishibayashi, Y.; Uemura, S.: Asymmetric α-Alkylative Reduction of Ketones with Alcohols
0923
Moteki, S. A.; Wu, D.; Chandra, K. L.; Reddy, D. S.; Takacs, J. M.: Efficient Rhodium-Catalyzed Asymmetric Hydroboration
0924
Matsubara, R.; Kawai, N.; Kobayashi, S.: Addition of Aldehyde-Derived Enecarbamates to α-Oxo Aldehydes
0925
Hansen, E. C.; Lee, D.: Regiochemical Controlled Transposition of Allylic Silyl Ethers
0926
Li, Q.; Liu, X.; Wang, J.; Shen, K.; Feng, X.: Ti(IV)/N-Oxide-Catalyzed Cyanosilylation of Ketones
0927
Kobayashi, Y.; Takeuchi, A.; Wang, Y.-G.: Cannabidiols via Alkenylation of Cyclohexenyl Monoacetate
0928
Park, B.-M.; Mun, S.; Yun, J.: Zinc-Catalyzed Enantioselective Hydrosilylation of Imines
0929
El-Awa, A.; Fuchs, P.: Diastereoselective Strategy for Stereotetrads Synthesis
0930
Babu, S. A.; Yasuda, M.; Okabe, Y.; Shibata, I.; Baba, A.: Stereoselective Reformatsky Reaction of Indium Enolates
0931
Biermann, U.; Lützen, A.; Metzger, J. O.: 2,3,4,6-Tetrasubstituted Tetrahydropyrans by Prins-Type Cyclization

Metal-Mediated Synthesis

0933
Tobisu, M.; Kita, Y.; Chatani, N.: Rh(I)-Catalyzed Synthesis of Aryl and Alkenyl Silanes from Nitriles
0934
Baati, R.; Mioskowski, C.; Barma, D.; Kache, R.; Falck, J. R.: Reductive Olefination of Aldehydes via Chromium Brook Rearrangement
0935
Lipshutz, B. H.; Lower, A.; Kucejko, R. J.; Noson, K.: Cu-Catalyzed Asymmetric Hydrosilylations of Ketones
0936
Martin, D.; Kehrli, S.; d’Augustin, M.; Clavier, H.; Mauduit, M.; Alexakis, A.: Asymmetric Conjugate Addition of Grignard Reagents to Enones
0937
Wang, Z.; Cheng, M.; Wu, P.; Wei, S.; Sun, J.: Organocatalytic Enantioselective Hydrosilylation of N-Aryl Imines
0938
Takahashi, H.; Inagaki, S.; Nishihara, Y.; Shibata, T.; Takagi, K.: Rh-Catalyzed Coupling of Alkyl Halides with o-Substituted Arylzinc Compounds
0939
Sebelius, S.; Olsson, V. J.; Wallner, O. A.; Szabó, K. J.: γ-Selective Pd-Catalyzed Cross-Coupling of Allylboronic Acids with Iodobenzenes
0940
Denhez, C.; Médégan, S.; Hélion, F.; Namy, J.-L.; Vasse, J.-L.; Szymoniak, J.: Cp2ZrCl2-Mischmetall as a New ‘Cp2Zr’ Equivalent
0941
Marshall, J. A.; Eidam, P.; Eidam, H. S.: Chiral Allenylzinc and Indium Reagents for Asymmetric Propargylation
0942
Sakai, T.; Kawamoto, Y.; Tomioka, K.: Ligand-Controlled Asymmetric Conjugate Addition of Lithium Amides
0943
Ohmiya, H.; Yorimitsu, H.; Oshima, K.: Co-Mediated Synthesis of Alkenyl- and Alkynyl Silanes from Alkyl Halides
0944
Chedid, R. B.; Fröhlich, R.; Hoppe, D.: Asymmetric Homoaldol Reactions of Metallated Dienyl Carbamates
0945
Yao, Q.; Sheets, M.: An Efficient Catalyst for Allylation of Aldehydes with Allyltributyltin

Organo- and Biocatalysis

0947
But, T. Y. S.; Toy, P. H.: Catalytic Mitsunobu Reaction
0948
Itoh, J.; Fuchibe, K.; Akiyama, T.: Enantioselective Aza-Diels-Alder Reaction of Brassard’s Diene with Imines
0949
Chen, Y. K.; Yoshida, M.; MacMillan, D. W. C.: Enantioselective Amine Conjugate Addition
0950
Nair, V.; Vellalath, S.; Poonoth, M.; Suresh, E.: N-Heterocyclic Carbene Catalyzed Synthesis of 1,3,4-Trisubstituted Cyclopentenes
0951
Shibuguchi, T.; Mihara, H.; Kuramochi, A.; Sakuraba, S.; Ohshima, T.; Shibasaki, M.: Total Synthesis of (+)-Cylindricine C Using an Organocatalytic Michael Reaction
0952
Nakashima, D.; Yamamoto, H.: A Phosphoramide Catalyzed Asymmetric Diels-Alder Reaction
0953
Bartoli, G.; Bosco, M.; Carlone, A.; Cavalli, A.; Locatelli, M.; Mazzanti, A.; Ricci, P.; Sambri, L.; Melchiorre, P.: Organocatalytic Asymmetric Addition of 1,3-Dicarbonyl Compounds to Maleimides
0954
Rodgen, S. A.; Schaus, S. E.: Clerodane-Derivatives by Catalytic Morita-Baylis-Hillman Reaction
0955
Pansare, S. V.; Pandya, K.: Amine/Protonic Acid Catalyzed Michael Addition
0956
Zhang, H.; Mifsud, M.; Tanaka, F.; Barbas III, C. F.: Organocatalytic anti-Mannich Reaction of Ketones
0957
Inokuma, T.; Hoashi, Y.; Takemoto, Y.: Organocatalytic Asymmetric Michael Reaction of α,β-Unsaturated Imides

Polymer-Supported Synthesis

0959
Maegawa, T.; Akashi, A.; Sajiki, H.: Rh/C-Catalyzed Hydrogenation of Aromatic Compounds in Water
0960
Qian, H.; Huang, X.: Solid-Phase Synthesis of β-Keto Sulfones
0961
Barluenga, S.; Dakas, P.-Y.; Ferandin, Y.; Meijer, L.; Winssinger, N.: Polymer-Supported Synthesis of Aigialomycin D
0962
McEleney, K.; Allen, D. P.; Holliday, A. E.; Crudden, C. M.: Mesoporous Silicates as Grubbs Catalyst Scavengers
0963
Mukhopadhyay, B.: H2SO4-Silica-Promoted One-Pot Protection of Sugars
0964
Solodenko, W.; Mennecke, K.; Vogt, C.; Gruhl, S.; Kirschning, A.: Polyvinylpyridine-Supported Palladacycle for the Suzuki Coupling Reaction
0965
Bouillon, C.; Meyer, A.; Vidal, S.; Jochum, A.; Chevolot, Y.; Cloarec, J.-P.; Praly, J.-P.; Vasseur, J.-J.; Morvan, F.: Microwave-Assisted ‘Click’ Chemistry on Solid Support
0966
Lu, F.; Liu, J.; Xu, J.: Hydrogenation Catalyzed by PVP-Ru Nanoparticles
0967
He, Y.; Wilkins, J. P.; Kiessling, L. L.: N-Acylsulfonamide Linker Activation by Pd-Catalyzed Allylation
0968
Fujita, N.; Motokura, K.; Mori, K.; Mizugaki, T.; Ebitani, K.; Jitsukawa, K.; Kaneda, K.: A Rhodium-Grafted Hydrotalcite as an Efficient Heterogeneous Catalyst
0969
Yang, Q.; Ma, S.; Li, J.; Xiao, F.; Xiong, H.: PEG-Coated Mesoporous Silica-Supported Pd for the Suzuki-Miyaura Coupling Reaction
0970
Shi, L.; Wang, X.; Sandoval, C. A.; Li, M.; Qi, Q.; Li, Z.; Ding, K.: An Orthogonal Self-Assembled Heterogeneous Catalyst for Asymmetric Hydrogenation
0971
Röttger, S.; Waldmann, H.: Solid-Phase Synthesis of Decalin Scaffolds by Robinson Annulation